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—— 5,7-dimethyl-6-[3-[methyl-[(2R)-1-(4-methylphenyl)butan-2-yl]amino]-3-oxopropyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H31N5O2
5,7-dimethyl-6-[3-[methyl-[(2R)-1-(4-methylphenyl)butan-2-yl]amino]-3-oxopropyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [5-(2-chloro-4-nitrophenyl)furan-2-yl]-[(2R,5R)-5-methyl-2-(2-methylphenyl)morpholin-4-yl]methanone —— C23H21ClN2O5
[5-(2-chloro-4-nitrophenyl)furan-2-yl]-[(2R,5R)-5-methyl-2-(2-methylphenyl)morpholin-4-yl]methanone
—— 5-bromo-6-oxo-N-[(1S,2S)-2-phenylcyclopropyl]-1H-pyridine-3-carboxamide —— C15H13BrN2O2
5-bromo-6-oxo-N-[(1S,2S)-2-phenylcyclopropyl]-1H-pyridine-3-carboxamide
—— [5-(2-chloro-4-nitrophenyl)furan-2-yl]-[(2S,5R)-5-methyl-2-(2-methylphenyl)morpholin-4-yl]methanone —— C23H21ClN2O5
[5-(2-chloro-4-nitrophenyl)furan-2-yl]-[(2S,5R)-5-methyl-2-(2-methylphenyl)morpholin-4-yl]methanone
—— 5-bromo-N-[(1R)-1-naphthalen-1-ylethyl]-6-oxo-1H-pyridine-3-carboxamide —— C18H15BrN2O2
5-bromo-N-[(1R)-1-naphthalen-1-ylethyl]-6-oxo-1H-pyridine-3-carboxamide
—— 5-chloro-N-methyl-N-[(2R)-1-phenylbutan-2-yl]-6-(2,2,2-trifluoroethoxy)pyridine-3-carboxamide —— C19H20ClF3N2O2
5-chloro-N-methyl-N-[(2R)-1-phenylbutan-2-yl]-6-(2,2,2-trifluoroethoxy)pyridine-3-carboxamide
—— (5-chloro-1,3-dimethylpyrazol-4-yl)methyl (1S,2S)-2-pyridin-3-ylcyclopropane-1-carboxylate —— C15H16ClN3O2
(5-chloro-1,3-dimethylpyrazol-4-yl)methyl (1S,2S)-2-pyridin-3-ylcyclopropane-1-carboxylate
—— (5-chloro-1,3-dimethylpyrazol-4-yl)methyl (1R,2S)-2-pyridin-3-ylcyclopropane-1-carboxylate —— C15H16ClN3O2
(5-chloro-1,3-dimethylpyrazol-4-yl)methyl (1R,2S)-2-pyridin-3-ylcyclopropane-1-carboxylate
—— (5-Ethoxycarbonyl-4-methyl-1,3-thiazol-2-yl)methyl-methyl-[2-oxo-2-(propan-2-ylamino)ethyl]azanium —— C14H24N3O3S+
(5-Ethoxycarbonyl-4-methyl-1,3-thiazol-2-yl)methyl-methyl-[2-oxo-2-(propan-2-ylamino)ethyl]azanium
—— 5-bromo-2-fluoro-N-[(2R)-1-(2-methoxyphenyl)propan-2-yl]-N-methylbenzamide —— C18H19BrFNO2
5-bromo-2-fluoro-N-[(2R)-1-(2-methoxyphenyl)propan-2-yl]-N-methylbenzamide
—— 5-chloro-N-methyl-N-[(2S)-1-phenylbutan-2-yl]-6-(2,2,2-trifluoroethoxy)pyridine-3-carboxamide —— C19H20ClF3N2O2
5-chloro-N-methyl-N-[(2S)-1-phenylbutan-2-yl]-6-(2,2,2-trifluoroethoxy)pyridine-3-carboxamide
—— 5-hydroxy-2-[[methyl-[(2S)-1-phenylbutan-2-yl]amino]methyl]pyran-4-one —— C17H21NO3
5-hydroxy-2-[[methyl-[(2S)-1-phenylbutan-2-yl]amino]methyl]pyran-4-one
—— (5-chloro-1,3-dimethylpyrazol-4-yl)methyl (1S,2R)-2-pyridin-3-ylcyclopropane-1-carboxylate —— C15H16ClN3O2
(5-chloro-1,3-dimethylpyrazol-4-yl)methyl (1S,2R)-2-pyridin-3-ylcyclopropane-1-carboxylate
—— (5-chloro-1,3-dimethylpyrazol-4-yl)methyl (1R,2R)-2-pyridin-3-ylcyclopropane-1-carboxylate —— C15H16ClN3O2
(5-chloro-1,3-dimethylpyrazol-4-yl)methyl (1R,2R)-2-pyridin-3-ylcyclopropane-1-carboxylate
—— 5-(3-cyanophenoxy)-N-[(S)-(1-methylbenzimidazol-2-yl)-phenylmethyl]pentanamide —— C27H26N4O2
5-(3-cyanophenoxy)-N-[(S)-(1-methylbenzimidazol-2-yl)-phenylmethyl]pentanamide
—— 5-bromo-2-fluoro-N-[(2S)-1-(2-methoxyphenyl)propan-2-yl]-N-methylbenzamide —— C18H19BrFNO2
5-bromo-2-fluoro-N-[(2S)-1-(2-methoxyphenyl)propan-2-yl]-N-methylbenzamide
—— 5-hydroxy-2-[[methyl-[(2R)-1-phenylbutan-2-yl]amino]methyl]pyran-4-one —— C17H21NO3
5-hydroxy-2-[[methyl-[(2R)-1-phenylbutan-2-yl]amino]methyl]pyran-4-one
—— 5-(3-cyanophenoxy)-N-[(R)-(1-methylbenzimidazol-2-yl)-phenylmethyl]pentanamide —— C27H26N4O2
5-(3-cyanophenoxy)-N-[(R)-(1-methylbenzimidazol-2-yl)-phenylmethyl]pentanamide
—— 5-[2-(4-fluoroanilino)-1,3-thiazol-4-yl]-1-methyl-3H-indol-2-one —— C18H14FN3OS
5-[2-(4-fluoroanilino)-1,3-thiazol-4-yl]-1-methyl-3H-indol-2-one
—— 5-(3-cyanophenoxy)-N-[[2-[[(2S)-2-methylpiperidin-1-yl]methyl]phenyl]methyl]pentanamide —— C26H33N3O2
5-(3-cyanophenoxy)-N-[[2-[[(2S)-2-methylpiperidin-1-yl]methyl]phenyl]methyl]pentanamide
—— 5-(3-cyanophenoxy)-N-[2-[(3S,5R)-3,5-dimethylpiperidine-1-carbonyl]phenyl]pentanamide —— C26H31N3O3
5-(3-cyanophenoxy)-N-[2-[(3S,5R)-3,5-dimethylpiperidine-1-carbonyl]phenyl]pentanamide
—— 5-(3-cyanophenoxy)-N-[2-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]phenyl]pentanamide —— C26H31N3O3
5-(3-cyanophenoxy)-N-[2-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]phenyl]pentanamide
—— 5-(3-cyanophenoxy)-N-[2-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]phenyl]pentanamide —— C26H31N3O3
5-(3-cyanophenoxy)-N-[2-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]phenyl]pentanamide
—— 5-(3-cyanophenoxy)-N-[(2S)-3-methyl-2-(4-methylpiperidin-1-yl)butyl]pentanamide —— C23H35N3O2
5-(3-cyanophenoxy)-N-[(2S)-3-methyl-2-(4-methylpiperidin-1-yl)butyl]pentanamide
—— 5-methyl-N-[(1S)-1-phenylethyl]-1-pyridin-2-ylpyrazole-4-sulfonamide —— C17H18N4O2S
5-methyl-N-[(1S)-1-phenylethyl]-1-pyridin-2-ylpyrazole-4-sulfonamide
—— 5-(3-cyanophenoxy)-N-[3-[[(2R)-2-pyrazol-1-ylpropanoyl]amino]phenyl]pentanamide —— C24H25N5O3
5-(3-cyanophenoxy)-N-[3-[[(2R)-2-pyrazol-1-ylpropanoyl]amino]phenyl]pentanamide
—— 5-(3-cyanophenoxy)-N-[3-[[(2S)-2-pyrazol-1-ylpropanoyl]amino]phenyl]pentanamide —— C24H25N5O3
5-(3-cyanophenoxy)-N-[3-[[(2S)-2-pyrazol-1-ylpropanoyl]amino]phenyl]pentanamide
—— 5-(3-cyanophenoxy)-N-[(2S)-2-(3-methylphenyl)-2-morpholin-4-ylethyl]pentanamide —— C25H31N3O3
5-(3-cyanophenoxy)-N-[(2S)-2-(3-methylphenyl)-2-morpholin-4-ylethyl]pentanamide
—— 5-(3-cyanophenoxy)-N-[[2-[[(2R)-2-methylpiperidin-1-yl]methyl]phenyl]methyl]pentanamide —— C26H33N3O2
5-(3-cyanophenoxy)-N-[[2-[[(2R)-2-methylpiperidin-1-yl]methyl]phenyl]methyl]pentanamide
—— 5-[2-(3-fluoro-4-methylanilino)-1,3-thiazol-4-yl]-1-methyl-3H-indol-2-one —— C19H16FN3OS
5-[2-(3-fluoro-4-methylanilino)-1,3-thiazol-4-yl]-1-methyl-3H-indol-2-one
—— 5-methyl-N-[(1R)-1-phenylethyl]-1-pyridin-2-ylpyrazole-4-sulfonamide —— C17H18N4O2S
5-methyl-N-[(1R)-1-phenylethyl]-1-pyridin-2-ylpyrazole-4-sulfonamide
—— 5-(3-cyanophenoxy)-N-[(2R)-3-methyl-2-(4-methylpiperidin-1-yl)butyl]pentanamide —— C23H35N3O2
5-(3-cyanophenoxy)-N-[(2R)-3-methyl-2-(4-methylpiperidin-1-yl)butyl]pentanamide
—— 5-(3-cyanophenoxy)-N-[(2R)-2-(3-methylphenyl)-2-morpholin-4-ylethyl]pentanamide —— C25H31N3O3
5-(3-cyanophenoxy)-N-[(2R)-2-(3-methylphenyl)-2-morpholin-4-ylethyl]pentanamide
—— 5-[(E)-3-[[(1S)-1-(2,5-dimethylphenyl)ethyl]amino]-3-oxoprop-1-enyl]-N-methylpyridine-3-carboxamide —— C20H23N3O2
5-[(E)-3-[[(1S)-1-(2,5-dimethylphenyl)ethyl]amino]-3-oxoprop-1-enyl]-N-methylpyridine-3-carboxamide
—— 5-[(E)-3-[[(1R)-1-(2,5-dimethylphenyl)ethyl]amino]-3-oxoprop-1-enyl]-N-methylpyridine-3-carboxamide —— C20H23N3O2
5-[(E)-3-[[(1R)-1-(2,5-dimethylphenyl)ethyl]amino]-3-oxoprop-1-enyl]-N-methylpyridine-3-carboxamide
—— 5-bromo-N-[(2R)-1-(4-fluoro-2-prop-2-ynoxyanilino)-1-oxopropan-2-yl]thiophene-2-carboxamide —— C17H14BrFN2O3S
5-bromo-N-[(2R)-1-(4-fluoro-2-prop-2-ynoxyanilino)-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-cyano-N-[(1R,3S)-3-ethoxyspiro[3.5]nonan-1-yl]-N-methylpyridine-2-carboxamide —— C19H25N3O2
5-cyano-N-[(1R,3S)-3-ethoxyspiro[3.5]nonan-1-yl]-N-methylpyridine-2-carboxamide
—— 5-cyano-N-[(1S,3S)-3-ethoxyspiro[3.5]nonan-1-yl]-N-methylpyridine-2-carboxamide —— C19H25N3O2
5-cyano-N-[(1S,3S)-3-ethoxyspiro[3.5]nonan-1-yl]-N-methylpyridine-2-carboxamide
—— 5-cyano-N-[(1S,3R)-3-ethoxyspiro[3.5]nonan-1-yl]-N-methylpyridine-2-carboxamide —— C19H25N3O2
5-cyano-N-[(1S,3R)-3-ethoxyspiro[3.5]nonan-1-yl]-N-methylpyridine-2-carboxamide
—— 5-cyano-N-[(1R,3R)-3-ethoxyspiro[3.5]nonan-1-yl]-N-methylpyridine-2-carboxamide —— C19H25N3O2
5-cyano-N-[(1R,3R)-3-ethoxyspiro[3.5]nonan-1-yl]-N-methylpyridine-2-carboxamide
—— (5S)-5-[[5-[(2-chloro-6-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-1,3-oxazolidin-2-one —— C13H11ClFN3O3S
(5S)-5-[[5-[(2-chloro-6-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-1,3-oxazolidin-2-one
—— (5R)-5-[[5-[(2-chloro-6-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-1,3-oxazolidin-2-one —— C13H11ClFN3O3S
(5R)-5-[[5-[(2-chloro-6-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-1,3-oxazolidin-2-one
—— 5-bromo-N-[(2S)-1-(4-fluoro-2-prop-2-ynoxyanilino)-1-oxopropan-2-yl]thiophene-2-carboxamide —— C17H14BrFN2O3S
5-bromo-N-[(2S)-1-(4-fluoro-2-prop-2-ynoxyanilino)-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(3S)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]-2-fluorobenzamide —— C17H13BrClFN2O2
5-bromo-N-[(3S)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]-2-fluorobenzamide
—— 5-bromo-N-[(3R)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]pyridine-3-carboxamide —— C16H13BrClN3O2
5-bromo-N-[(3R)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]pyridine-3-carboxamide
—— 5-bromo-N-[(3R)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]-2-fluorobenzamide —— C17H13BrClFN2O2
5-bromo-N-[(3R)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]-2-fluorobenzamide
—— 5-[[4-[(2R)-butan-2-yl]-3-oxo-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-5-yl]sulfanyl]-N,N-dimethylpentanamide —— C22H33N3O2S2
5-[[4-[(2R)-butan-2-yl]-3-oxo-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-5-yl]sulfanyl]-N,N-dimethylpentanamide
—— 5-bromo-2-chloro-N-[(3R)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]benzamide —— C17H13BrCl2N2O2
5-bromo-2-chloro-N-[(3R)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]benzamide
—— 5-[[4-[(2S)-butan-2-yl]-3-oxo-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-5-yl]sulfanyl]-N,N-dimethylpentanamide —— C22H33N3O2S2
5-[[4-[(2S)-butan-2-yl]-3-oxo-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-5-yl]sulfanyl]-N,N-dimethylpentanamide
—— 5-bromo-N-[(3S)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]pyridine-3-carboxamide —— C16H13BrClN3O2
5-bromo-N-[(3S)-1-(2-chlorophenyl)-2-oxopyrrolidin-3-yl]pyridine-3-carboxamide