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—— 5-[2-[(3R,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]-2-oxoethyl]-7,8-dihydro-6H-thieno[3,2-c]azepin-4-one —— C17H25N3O2S
5-[2-[(3R,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]-2-oxoethyl]-7,8-dihydro-6H-thieno[3,2-c]azepin-4-one
—— 5-[2-[(3S,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]-2-oxoethyl]-7,8-dihydro-6H-thieno[3,2-c]azepin-4-one —— C17H25N3O2S
5-[2-[(3S,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]-2-oxoethyl]-7,8-dihydro-6H-thieno[3,2-c]azepin-4-one
—— (5-chloro-1-benzofuran-2-yl)-[(3R,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone —— C16H19ClN2O2
(5-chloro-1-benzofuran-2-yl)-[(3R,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone
—— (5-Chloro-1-benzofuran-2-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone —— C18H18ClN2O2S+
(5-Chloro-1-benzofuran-2-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone
—— 5-acetyl-N-[2-(3-fluorophenyl)ethyl]thiophene-2-carboxamide —— C15H14FNO2S
5-acetyl-N-[2-(3-fluorophenyl)ethyl]thiophene-2-carboxamide
—— 5-fluoro-N-[2-(3-fluorophenyl)ethyl]-3-methyl-1-benzofuran-2-carboxamide —— C18H15F2NO2
5-fluoro-N-[2-(3-fluorophenyl)ethyl]-3-methyl-1-benzofuran-2-carboxamide
—— 5-(4-fluorophenyl)-N-[(Z)-furan-2-ylmethylideneamino]thiophene-2-carboxamide —— C16H11FN2O2S
5-(4-fluorophenyl)-N-[(Z)-furan-2-ylmethylideneamino]thiophene-2-carboxamide
—— 5-(1,3-benzothiazol-2-yl)-N-[2-(3-fluorophenyl)ethyl]furan-2-carboxamide —— C20H15FN2O2S
5-(1,3-benzothiazol-2-yl)-N-[2-(3-fluorophenyl)ethyl]furan-2-carboxamide
—— 5-(4-fluorophenyl)-N-[(Z)-thiophen-2-ylmethylideneamino]thiophene-2-carboxamide —— C16H11FN2OS2
5-(4-fluorophenyl)-N-[(Z)-thiophen-2-ylmethylideneamino]thiophene-2-carboxamide
—— [5-(2-Fluorophenyl)furan-2-yl]-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone —— C20H20FN2O2S+
[5-(2-Fluorophenyl)furan-2-yl]-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone
—— 5-(4-Fluorophenyl)-3-[2-oxo-2-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]ethyl]-1,3,4-oxadiazol-2-one —— C19H20FN4O3S+
5-(4-Fluorophenyl)-3-[2-oxo-2-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]ethyl]-1,3,4-oxadiazol-2-one
—— (5-Fluoro-3-methyl-1-benzofuran-2-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone —— C19H20FN2O2S+
(5-Fluoro-3-methyl-1-benzofuran-2-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone
—— 5-[2-Oxo-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]ethyl]-2,3-dihydro-1,5-benzoxazepin-4-one —— C20H23N3O3S
5-[2-Oxo-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]ethyl]-2,3-dihydro-1,5-benzoxazepin-4-one
—— [(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone —— C19H25N2OS2+
[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone
—— (5-Methyl-3-phenyl-1,2-oxazol-4-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone —— C20H22N3O2S+
(5-Methyl-3-phenyl-1,2-oxazol-4-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone
—— (5-Methyl-3-phenyl-1,2-oxazol-4-yl)-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone —— C20H21N3O2S
(5-Methyl-3-phenyl-1,2-oxazol-4-yl)-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone
—— (5-Ethoxy-3-methyl-1-benzofuran-2-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone —— C21H25N2O3S+
(5-Ethoxy-3-methyl-1-benzofuran-2-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone
—— 5-fluoro-2-[[(2S)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methyl]benzonitrile —— C17H20FN5O
5-fluoro-2-[[(2S)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methyl]benzonitrile
—— (5-Methoxy-3-methyl-1-benzofuran-2-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone —— C20H23N2O3S+
(5-Methoxy-3-methyl-1-benzofuran-2-yl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone
—— 5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone —— C19H24N2OS2
5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone
—— 5-fluoro-2-[[(2R)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methyl]benzonitrile —— C17H20FN5O
5-fluoro-2-[[(2R)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methyl]benzonitrile
—— (5-Chloro-2-nitrophenyl)-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone —— C16H16ClN3O3S
(5-Chloro-2-nitrophenyl)-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone —— C17H20N2OS2
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone
—— 5-cyclopropyl-3-[(2S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole —— C13H17N5O
5-cyclopropyl-3-[(2S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-chloro-N',N'-dimethyl-1-benzofuran-2-carbohydrazide —— C11H11ClN2O2
5-chloro-N',N'-dimethyl-1-benzofuran-2-carbohydrazide
—— 5-fluoro-2-[[(3R)-3-[methyl-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino]pyrrolidin-1-yl]methyl]benzonitrile —— C17H20FN5O
5-fluoro-2-[[(3R)-3-[methyl-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino]pyrrolidin-1-yl]methyl]benzonitrile
—— (5-Chloro-2-nitrophenyl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone —— C16H17ClN3O3S+
(5-Chloro-2-nitrophenyl)-[4-(thiophen-3-ylmethyl)piperazin-4-ium-1-yl]methanone
—— (5-Bromo-2-chlorophenyl)-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone —— C16H16BrClN2OS
(5-Bromo-2-chlorophenyl)-[4-(thiophen-3-ylmethyl)piperazin-1-yl]methanone
—— 5-cyclopropyl-3-[(3R)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl]-1,2,4-oxadiazole —— C15H20N4OS
5-cyclopropyl-3-[(3R)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1,2,4-oxadiazole —— C16H20N4O
5-cyclopropyl-3-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-(1,3-benzothiazol-2-yl)-N-(4-methylsulfanylphenyl)pentanamide —— C19H20N2OS2
5-(1,3-benzothiazol-2-yl)-N-(4-methylsulfanylphenyl)pentanamide
—— 5-chloro-2-fluoro-N-(4-methylsulfanylphenyl)benzamide —— C14H11ClFNOS
5-chloro-2-fluoro-N-(4-methylsulfanylphenyl)benzamide
—— 5-cyclopropyl-3-[(2R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole —— C13H17N5O
5-cyclopropyl-3-[(2R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-fluoro-2-[[(3S)-3-[methyl-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino]pyrrolidin-1-yl]methyl]benzonitrile —— C17H20FN5O
5-fluoro-2-[[(3S)-3-[methyl-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino]pyrrolidin-1-yl]methyl]benzonitrile
—— (5-propan-2-yl-1,3-oxazol-4-yl)-[(2S)-2-(5-propyl-1H-1,2,4-triazol-3-yl)morpholin-4-yl]methanone —— C16H23N5O3
(5-propan-2-yl-1,3-oxazol-4-yl)-[(2S)-2-(5-propyl-1H-1,2,4-triazol-3-yl)morpholin-4-yl]methanone
—— 5-[(2R)-2-(5-propyl-1H-1,2,4-triazol-3-yl)morpholine-4-carbonyl]thiophene-3-carboxamide —— C15H19N5O3S
5-[(2R)-2-(5-propyl-1H-1,2,4-triazol-3-yl)morpholine-4-carbonyl]thiophene-3-carboxamide
—— (5R)-5-[(2R)-2-(3-tert-butyl-1H-1,2,4-triazol-5-yl)morpholine-4-carbonyl]pyrrolidin-2-one —— C15H23N5O3
(5R)-5-[(2R)-2-(3-tert-butyl-1H-1,2,4-triazol-5-yl)morpholine-4-carbonyl]pyrrolidin-2-one
—— 5-(2-chlorophenyl)-N-(4-methylsulfanylphenyl)furan-2-carboxamide —— C18H14ClNO2S
5-(2-chlorophenyl)-N-(4-methylsulfanylphenyl)furan-2-carboxamide
—— (5-ethyl-1,3-oxazol-4-yl)-[(2R)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone —— C15H21N5O3
(5-ethyl-1,3-oxazol-4-yl)-[(2R)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone
—— 5-[(2S)-2-(5-propyl-1H-1,2,4-triazol-3-yl)morpholine-4-carbonyl]thiophene-3-carboxamide —— C15H19N5O3S
5-[(2S)-2-(5-propyl-1H-1,2,4-triazol-3-yl)morpholine-4-carbonyl]thiophene-3-carboxamide
—— (5-propan-2-yl-1,3-oxazol-4-yl)-[(2R)-2-(5-propyl-1H-1,2,4-triazol-3-yl)morpholin-4-yl]methanone —— C16H23N5O3
(5-propan-2-yl-1,3-oxazol-4-yl)-[(2R)-2-(5-propyl-1H-1,2,4-triazol-3-yl)morpholin-4-yl]methanone
—— (5S)-5-[(2S)-2-(3-tert-butyl-1H-1,2,4-triazol-5-yl)morpholine-4-carbonyl]pyrrolidin-2-one —— C15H23N5O3
(5S)-5-[(2S)-2-(3-tert-butyl-1H-1,2,4-triazol-5-yl)morpholine-4-carbonyl]pyrrolidin-2-one
—— (5R)-5-[(2S)-2-(3-tert-butyl-1H-1,2,4-triazol-5-yl)morpholine-4-carbonyl]pyrrolidin-2-one —— C15H23N5O3
(5R)-5-[(2S)-2-(3-tert-butyl-1H-1,2,4-triazol-5-yl)morpholine-4-carbonyl]pyrrolidin-2-one
—— (5S)-5-[(2R)-2-(3-tert-butyl-1H-1,2,4-triazol-5-yl)morpholine-4-carbonyl]pyrrolidin-2-one —— C15H23N5O3
(5S)-5-[(2R)-2-(3-tert-butyl-1H-1,2,4-triazol-5-yl)morpholine-4-carbonyl]pyrrolidin-2-one
—— 5-(2-fluorophenyl)-N-(4-methylsulfanylphenyl)furan-2-carboxamide —— C18H14FNO2S
5-(2-fluorophenyl)-N-(4-methylsulfanylphenyl)furan-2-carboxamide
—— (5-ethyl-1,3-oxazol-4-yl)-[(2S)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone —— C15H21N5O3
(5-ethyl-1,3-oxazol-4-yl)-[(2S)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone
—— (5-propan-2-yl-1,3-oxazol-4-yl)-[(2S)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone —— C16H23N5O3
(5-propan-2-yl-1,3-oxazol-4-yl)-[(2S)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone
—— 5-(diethylsulfamoyl)-2-fluoro-N-(4-methylsulfanylphenyl)benzamide —— C18H21FN2O3S2
5-(diethylsulfamoyl)-2-fluoro-N-(4-methylsulfanylphenyl)benzamide
—— (5-propan-2-yl-1,3-oxazol-4-yl)-[(2R)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone —— C16H23N5O3
(5-propan-2-yl-1,3-oxazol-4-yl)-[(2R)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone
—— (5-methyl-1,2-oxazol-3-yl)-[(2S)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone —— C14H19N5O3
(5-methyl-1,2-oxazol-3-yl)-[(2S)-2-(3-propan-2-yl-1H-1,2,4-triazol-5-yl)morpholin-4-yl]methanone