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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-5-[(2,6-dimethylpyridin-4-yl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H26N4O2
(5S)-5-[(2,6-dimethylpyridin-4-yl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[2-[(2S)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C19H22N4O4
5-[2-[(2S)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— 5-[(2R)-2-[2-(1,3-benzoxazol-2-ylamino)ethyl]morpholin-4-yl]-2-methylpyridazin-3-one —— C18H21N5O3
5-[(2R)-2-[2-(1,3-benzoxazol-2-ylamino)ethyl]morpholin-4-yl]-2-methylpyridazin-3-one
—— 5-[2-[(2R)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C19H22N4O4
5-[2-[(2R)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— 5-[(2R)-1-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C20H24N4O2
5-[(2R)-1-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(2S)-1-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C20H24N4O2
5-[(2S)-1-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(2R)-2-[2-(cyclopentylamino)ethyl]morpholin-4-yl]-2-methylpyridazin-3-one —— C16H26N4O2
5-[(2R)-2-[2-(cyclopentylamino)ethyl]morpholin-4-yl]-2-methylpyridazin-3-one
—— 5-[(2S)-1-[(4-methoxypyridin-2-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C19H20N4O2
5-[(2S)-1-[(4-methoxypyridin-2-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(2S)-2-[2-(cyclopentylamino)ethyl]morpholin-4-yl]-2-methylpyridazin-3-one —— C16H26N4O2
5-[(2S)-2-[2-(cyclopentylamino)ethyl]morpholin-4-yl]-2-methylpyridazin-3-one
—— (5R)-7-(5-acetylthiophene-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione —— C14H14N2O4S
(5R)-7-(5-acetylthiophene-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
—— 5-[(2R)-1-[(4-methoxypyridin-2-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C19H20N4O2
5-[(2R)-1-[(4-methoxypyridin-2-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-[[(6R)-2-(2-methoxyethyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-N,N-dimethylfuran-2-carboxamide —— C20H31N3O4
5-[[(6R)-2-(2-methoxyethyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-N,N-dimethylfuran-2-carboxamide
—— (5S)-7-(5-acetylthiophene-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione —— C14H14N2O4S
(5S)-7-(5-acetylthiophene-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
—— 5-[(3S)-3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H19N3O5
5-[(3S)-3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-[[(6S)-2-(2-methoxyethyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-N,N-dimethylfuran-2-carboxamide —— C20H31N3O4
5-[[(6S)-2-(2-methoxyethyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-N,N-dimethylfuran-2-carboxamide
—— (5R)-1-(3-chlorophenyl)-4-(2-hydroxy-3-methylbenzoyl)-5-methylpiperazin-2-one —— C19H19ClN2O3
(5R)-1-(3-chlorophenyl)-4-(2-hydroxy-3-methylbenzoyl)-5-methylpiperazin-2-one
—— [5-(hydroxymethyl)furan-2-yl]-[(3S)-3-(3-methoxypropyl)piperidin-1-yl]methanone —— C15H23NO4
[5-(hydroxymethyl)furan-2-yl]-[(3S)-3-(3-methoxypropyl)piperidin-1-yl]methanone
—— 5-[(2S)-1-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C18H23N5O
5-[(2S)-1-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyrazin-2-one —— C14H17N5O3
5-[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyrazin-2-one
—— [5-(hydroxymethyl)furan-2-yl]-[(3R)-3-(3-methoxypropyl)piperidin-1-yl]methanone —— C15H23NO4
[5-(hydroxymethyl)furan-2-yl]-[(3R)-3-(3-methoxypropyl)piperidin-1-yl]methanone
—— (5S)-1-(3-chlorophenyl)-4-(2-hydroxy-3-methylbenzoyl)-5-methylpiperazin-2-one —— C19H19ClN2O3
(5S)-1-(3-chlorophenyl)-4-(2-hydroxy-3-methylbenzoyl)-5-methylpiperazin-2-one
—— 5-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyrazin-2-one —— C14H17N5O3
5-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-[[(2R)-2-butyl-4-methyl-3-oxopiperazin-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide —— C14H23N5O3
5-[[(2R)-2-butyl-4-methyl-3-oxopiperazin-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
—— 5-[[(2S)-2-butyl-4-methyl-3-oxopiperazin-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide —— C14H23N5O3
5-[[(2S)-2-butyl-4-methyl-3-oxopiperazin-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
—— 5-[(2S)-1-(2-propan-2-ylsulfanylethyl)pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C16H22N4OS
5-[(2S)-1-(2-propan-2-ylsulfanylethyl)pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-[(3R)-3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H19N3O5
5-[(3R)-3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-[(2R)-1-(2-propan-2-ylsulfanylethyl)pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C16H22N4OS
5-[(2R)-1-(2-propan-2-ylsulfanylethyl)pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-[(2R)-1-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C18H23N5O
5-[(2R)-1-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(3S)-3-benzoylpiperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C22H21N3O3
5-[(3S)-3-benzoylpiperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— 5-[(3R)-3-benzoylpiperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C22H21N3O3
5-[(3R)-3-benzoylpiperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— 5-methyl-3-[(5-thiophen-2-yl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-1,2-oxazole —— C11H10N4OS2
5-methyl-3-[(5-thiophen-2-yl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-1,2-oxazole
—— (5-Methyl-1,2-oxazol-3-yl)methyl 2-butyl-1,3-dioxoisoindole-5-carboxylate —— C18H18N2O5
(5-Methyl-1,2-oxazol-3-yl)methyl 2-butyl-1,3-dioxoisoindole-5-carboxylate
—— (5-methyl-1H-pyrazol-3-yl)-[(2R)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methanone —— C16H26N4O2
(5-methyl-1H-pyrazol-3-yl)-[(2R)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methanone
—— 5-[(6S)-2-(cyclopropylmethyl)-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]pyridine-2-carbonitrile —— C20H24N4O2
5-[(6S)-2-(cyclopropylmethyl)-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]pyridine-2-carbonitrile
—— 5-[(1R)-1-[2-(2-cyclohexylpyrimidin-5-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole —— C19H24N6O
5-[(1R)-1-[2-(2-cyclohexylpyrimidin-5-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole
—— [5-(imidazol-1-ylmethyl)furan-2-yl]-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone —— C17H19N5O2
[5-(imidazol-1-ylmethyl)furan-2-yl]-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone
—— 5-methoxy-3-methyl-2-[[(2S)-2-[2-(2-methylimidazol-1-yl)ethyl]piperidin-1-yl]methyl]-1H-indole —— C22H30N4O
5-methoxy-3-methyl-2-[[(2S)-2-[2-(2-methylimidazol-1-yl)ethyl]piperidin-1-yl]methyl]-1H-indole
—— (5-methyl-1H-pyrazol-3-yl)-[(2S)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methanone —— C16H26N4O2
(5-methyl-1H-pyrazol-3-yl)-[(2S)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methanone
—— 5-methoxy-3-methyl-2-[[(2R)-2-[2-(2-methylimidazol-1-yl)ethyl]piperidin-1-yl]methyl]-1H-indole —— C22H30N4O
5-methoxy-3-methyl-2-[[(2R)-2-[2-(2-methylimidazol-1-yl)ethyl]piperidin-1-yl]methyl]-1H-indole
—— 5-[(2S)-1-[(1-methylindol-2-yl)methyl]pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C21H21N5O
5-[(2S)-1-[(1-methylindol-2-yl)methyl]pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-[(1S)-1-[2-(2-cyclohexylpyrimidin-5-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole —— C19H24N6O
5-[(1S)-1-[2-(2-cyclohexylpyrimidin-5-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole
—— 5-[(2R)-1-[(1-methylindol-2-yl)methyl]pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C21H21N5O
5-[(2R)-1-[(1-methylindol-2-yl)methyl]pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— [5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone —— C17H20N6O2
[5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone
—— [5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone —— C17H20N6O2
[5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone
—— 5-methyl-1-[2-oxo-2-[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]ethyl]pyrimidine-2,4-dione —— C17H23N5O3
5-methyl-1-[2-oxo-2-[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]ethyl]pyrimidine-2,4-dione
—— (5-propan-2-yl-1,2-oxazol-3-yl)-[(2S)-2-(2-pyridin-2-ylethyl)piperidin-1-yl]methanone —— C19H25N3O2
(5-propan-2-yl-1,2-oxazol-3-yl)-[(2S)-2-(2-pyridin-2-ylethyl)piperidin-1-yl]methanone
—— (5-propan-2-yl-1,2-oxazol-3-yl)-[(2R)-2-(2-pyridin-2-ylethyl)piperidin-1-yl]methanone —— C19H25N3O2
(5-propan-2-yl-1,2-oxazol-3-yl)-[(2R)-2-(2-pyridin-2-ylethyl)piperidin-1-yl]methanone
—— 5-[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C18H19N5O3
5-[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C18H19N5O3
5-[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-butyl-4-ethyl-2-[2-oxo-2-[(3R)-3-phenylpiperazin-1-yl]ethyl]-1,2,4-triazol-3-one —— C20H29N5O2
5-butyl-4-ethyl-2-[2-oxo-2-[(3R)-3-phenylpiperazin-1-yl]ethyl]-1,2,4-triazol-3-one