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—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 3-(methylsulfonylmethyl)benzoate —— C16H14N2O5S2
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 3-(methylsulfonylmethyl)benzoate
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]pyridine-3-carboxylate —— C21H17N3O4S
(5-Phenyl-1,3-oxazol-2-yl)methyl 2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]pyridine-3-carboxylate
—— 5-[2-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C19H26N4O2
5-[2-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-bromo-N-[(1S,3S)-3-methylsulfonylcyclohexyl]pyrimidin-2-amine —— C11H16BrN3O2S
5-bromo-N-[(1S,3S)-3-methylsulfonylcyclohexyl]pyrimidin-2-amine
—— 5-[2-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C19H26N4O2
5-[2-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— (5-Methyl-1,2-oxazol-3-yl)methyl 2-(2-oxo-5-phenyl-1,3,4-oxadiazol-3-yl)acetate —— C15H13N3O5
(5-Methyl-1,2-oxazol-3-yl)methyl 2-(2-oxo-5-phenyl-1,3,4-oxadiazol-3-yl)acetate
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]pyridine-3-carboxylate —— C20H16N4O4S
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]pyridine-3-carboxylate
—— 5-chloro-6-[[(2R)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]pyridine-3-carbonitrile —— C11H14ClN3OS
5-chloro-6-[[(2R)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]pyridine-3-carbonitrile
—— 5-bromo-N-[(1S,3R)-3-methylsulfonylcyclohexyl]pyrimidin-2-amine —— C11H16BrN3O2S
5-bromo-N-[(1S,3R)-3-methylsulfonylcyclohexyl]pyrimidin-2-amine
—— 5-bromo-N-[(1R,3R)-3-methylsulfonylcyclohexyl]pyrimidin-2-amine —— C11H16BrN3O2S
5-bromo-N-[(1R,3R)-3-methylsulfonylcyclohexyl]pyrimidin-2-amine
—— 5-bromo-N-[(1R,3S)-3-methylsulfonylcyclohexyl]pyrimidin-2-amine —— C11H16BrN3O2S
5-bromo-N-[(1R,3S)-3-methylsulfonylcyclohexyl]pyrimidin-2-amine
—— 5-chloro-2-[[(2S)-4-hydroxybutan-2-yl]amino]benzonitrile —— C11H13ClN2O
5-chloro-2-[[(2S)-4-hydroxybutan-2-yl]amino]benzonitrile
—— (5-Acetyl-2-methoxyphenyl)methyl 2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]pyridine-3-carboxylate —— C21H20N2O5S
(5-Acetyl-2-methoxyphenyl)methyl 2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]pyridine-3-carboxylate
—— 5-chloro-2-[[(2R)-4-hydroxybutan-2-yl]amino]benzonitrile —— C11H13ClN2O
5-chloro-2-[[(2R)-4-hydroxybutan-2-yl]amino]benzonitrile
—— 5-bromo-N-[3-[[(3R)-oxolan-3-yl]methoxy]propyl]pyrimidin-2-amine —— C12H18BrN3O2
5-bromo-N-[3-[[(3R)-oxolan-3-yl]methoxy]propyl]pyrimidin-2-amine
—— 5-nitro-N-[3-[[(3R)-oxolan-3-yl]methoxy]propyl]pyridin-2-amine —— C13H19N3O4
5-nitro-N-[3-[[(3R)-oxolan-3-yl]methoxy]propyl]pyridin-2-amine
—— 5,6-dimethyl-N-[2-[(R)-phenylsulfinyl]ethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H17N5OS
5,6-dimethyl-N-[2-[(R)-phenylsulfinyl]ethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-nitro-N-[3-[[(3S)-oxolan-3-yl]methoxy]propyl]pyridin-2-amine —— C13H19N3O4
5-nitro-N-[3-[[(3S)-oxolan-3-yl]methoxy]propyl]pyridin-2-amine
—— 5,6-dimethyl-N-[2-[(S)-phenylsulfinyl]ethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H17N5OS
5,6-dimethyl-N-[2-[(S)-phenylsulfinyl]ethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-bromo-N-[3-[[(3S)-oxolan-3-yl]methoxy]propyl]pyrimidin-2-amine —— C12H18BrN3O2
5-bromo-N-[3-[[(3S)-oxolan-3-yl]methoxy]propyl]pyrimidin-2-amine
—— (5-ethyl-1-pyridin-2-ylpyrazol-4-yl)-[(3R)-3-methyl-2,3-dihydroindol-1-yl]methanone —— C20H20N4O
(5-ethyl-1-pyridin-2-ylpyrazol-4-yl)-[(3R)-3-methyl-2,3-dihydroindol-1-yl]methanone
—— (5-Fluoro-2-methoxyphenyl)methyl 2-(2-oxo-5-phenyl-1,3,4-oxadiazol-3-yl)acetate —— C18H15FN2O5
(5-Fluoro-2-methoxyphenyl)methyl 2-(2-oxo-5-phenyl-1,3,4-oxadiazol-3-yl)acetate
—— (5-ethyl-1-pyridin-2-ylpyrazol-4-yl)-[(3S)-3-methyl-2,3-dihydroindol-1-yl]methanone —— C20H20N4O
(5-ethyl-1-pyridin-2-ylpyrazol-4-yl)-[(3S)-3-methyl-2,3-dihydroindol-1-yl]methanone
—— 5-(2,5-dimethoxyphenyl)-N-[(2R)-2-hydroxy-3-phenylpropyl]-2-methylpyrazole-3-carboxamide —— C22H25N3O4
5-(2,5-dimethoxyphenyl)-N-[(2R)-2-hydroxy-3-phenylpropyl]-2-methylpyrazole-3-carboxamide
—— 5-(4-fluorophenyl)-N-[(2R)-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]-2-methylpyrazole-3-carboxamide —— C20H17F4N3O2
5-(4-fluorophenyl)-N-[(2R)-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]-2-methylpyrazole-3-carboxamide
—— 5-(2,5-dimethoxyphenyl)-N-[(2S)-2-(dimethylamino)-2-(1-methylindol-3-yl)ethyl]-2-methylpyrazole-3-carboxamide —— C26H31N5O3
5-(2,5-dimethoxyphenyl)-N-[(2S)-2-(dimethylamino)-2-(1-methylindol-3-yl)ethyl]-2-methylpyrazole-3-carboxamide
—— 5-(2,5-dimethoxyphenyl)-N-[(2R)-2-hydroxy-2-phenylpropyl]-2-methylpyrazole-3-carboxamide —— C22H25N3O4
5-(2,5-dimethoxyphenyl)-N-[(2R)-2-hydroxy-2-phenylpropyl]-2-methylpyrazole-3-carboxamide
—— 5-(2,5-dimethoxyphenyl)-N-[(2S)-2-hydroxy-2-phenylpropyl]-2-methylpyrazole-3-carboxamide —— C22H25N3O4
5-(2,5-dimethoxyphenyl)-N-[(2S)-2-hydroxy-2-phenylpropyl]-2-methylpyrazole-3-carboxamide
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 4-methyl-2-thiophen-2-yl-1,3-thiazole-5-carboxylate —— C18H13N3O3S2
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 4-methyl-2-thiophen-2-yl-1,3-thiazole-5-carboxylate
—— [5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-chloro-1-benzothiophen-2-yl)prop-2-enoate —— C18H11ClN2O4S
[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-chloro-1-benzothiophen-2-yl)prop-2-enoate
—— 5-(2,5-dimethoxyphenyl)-N-[(2R)-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]-2-methylpyrazole-3-carboxamide —— C22H22F3N3O4
5-(2,5-dimethoxyphenyl)-N-[(2R)-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]-2-methylpyrazole-3-carboxamide
—— [5-(1-ethylbenzimidazol-2-yl)-1H-pyrrol-3-yl]-(2-hydroxy-5-methoxyphenyl)methanone —— C21H19N3O3
[5-(1-ethylbenzimidazol-2-yl)-1H-pyrrol-3-yl]-(2-hydroxy-5-methoxyphenyl)methanone
—— [5-(1-ethylbenzimidazol-2-yl)-1H-pyrrol-3-yl]-(2-hydroxyphenyl)methanone —— C20H17N3O2
[5-(1-ethylbenzimidazol-2-yl)-1H-pyrrol-3-yl]-(2-hydroxyphenyl)methanone
—— 5-(2,5-dimethoxyphenyl)-N-[(2S)-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]-2-methylpyrazole-3-carboxamide —— C22H22F3N3O4
5-(2,5-dimethoxyphenyl)-N-[(2S)-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]-2-methylpyrazole-3-carboxamide
—— 5-(4-fluorophenyl)-N-[(2R)-2-(3-methoxyphenyl)-2-morpholin-4-ylethyl]-2-methylpyrazole-3-carboxamide —— C24H27FN4O3
5-(4-fluorophenyl)-N-[(2R)-2-(3-methoxyphenyl)-2-morpholin-4-ylethyl]-2-methylpyrazole-3-carboxamide
—— 5-(2,5-dimethoxyphenyl)-N-[(2S)-2-hydroxy-3-phenylpropyl]-2-methylpyrazole-3-carboxamide —— C22H25N3O4
5-(2,5-dimethoxyphenyl)-N-[(2S)-2-hydroxy-3-phenylpropyl]-2-methylpyrazole-3-carboxamide
—— 5-(4-fluorophenyl)-2-methyl-N-[2-[(2R)-1-thiophen-2-ylsulfonylpiperidin-2-yl]ethyl]pyrazole-3-carboxamide —— C22H25FN4O3S2
5-(4-fluorophenyl)-2-methyl-N-[2-[(2R)-1-thiophen-2-ylsulfonylpiperidin-2-yl]ethyl]pyrazole-3-carboxamide
—— 5-(2,5-dimethoxyphenyl)-N-[[(3S)-1,4-dioxaspiro[4.5]decan-3-yl]methyl]-2-methylpyrazole-3-carboxamide —— C22H29N3O5
5-(2,5-dimethoxyphenyl)-N-[[(3S)-1,4-dioxaspiro[4.5]decan-3-yl]methyl]-2-methylpyrazole-3-carboxamide
—— 5-(2,5-dimethoxyphenyl)-N-[(2S)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-2-methylpyrazole-3-carboxamide —— C21H26N4O4
5-(2,5-dimethoxyphenyl)-N-[(2S)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-2-methylpyrazole-3-carboxamide
—— 5-(2,5-dimethoxyphenyl)-N-[(2R)-2-(dimethylamino)-2-(1-methylindol-3-yl)ethyl]-2-methylpyrazole-3-carboxamide —— C26H31N5O3
5-(2,5-dimethoxyphenyl)-N-[(2R)-2-(dimethylamino)-2-(1-methylindol-3-yl)ethyl]-2-methylpyrazole-3-carboxamide
—— [5-(2,5-dimethoxyphenyl)-2-methylpyrazol-3-yl]-[(2S)-2-phenylmorpholin-4-yl]methanone —— C23H25N3O4
[5-(2,5-dimethoxyphenyl)-2-methylpyrazol-3-yl]-[(2S)-2-phenylmorpholin-4-yl]methanone
—— 5-(4-fluorophenyl)-2-methyl-N-[(2S)-3,3,3-trifluoro-2-hydroxy-2-phenylpropyl]pyrazole-3-carboxamide —— C20H17F4N3O2
5-(4-fluorophenyl)-2-methyl-N-[(2S)-3,3,3-trifluoro-2-hydroxy-2-phenylpropyl]pyrazole-3-carboxamide
—— 5-(4-fluorophenyl)-N-[(2S)-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]-2-methylpyrazole-3-carboxamide —— C20H17F4N3O2
5-(4-fluorophenyl)-N-[(2S)-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]-2-methylpyrazole-3-carboxamide
—— 5-(4-fluorophenyl)-2-methyl-N-[(2R)-2-morpholin-4-yl-2-thiophen-3-ylethyl]pyrazole-3-carboxamide —— C21H23FN4O2S
5-(4-fluorophenyl)-2-methyl-N-[(2R)-2-morpholin-4-yl-2-thiophen-3-ylethyl]pyrazole-3-carboxamide
—— 5-(4-fluorophenyl)-2-methyl-N-[(2S)-2-morpholin-4-yl-2-thiophen-3-ylethyl]pyrazole-3-carboxamide —— C21H23FN4O2S
5-(4-fluorophenyl)-2-methyl-N-[(2S)-2-morpholin-4-yl-2-thiophen-3-ylethyl]pyrazole-3-carboxamide
—— 5-(4-fluorophenyl)-2-methyl-N-[(2R)-3,3,3-trifluoro-2-hydroxy-2-phenylpropyl]pyrazole-3-carboxamide —— C20H17F4N3O2
5-(4-fluorophenyl)-2-methyl-N-[(2R)-3,3,3-trifluoro-2-hydroxy-2-phenylpropyl]pyrazole-3-carboxamide
—— 5-(4-fluorophenyl)-N-[(2R)-2-hydroxy-3-(4-methoxyphenyl)-2-methylpropyl]-2-methylpyrazole-3-carboxamide —— C22H24FN3O3
5-(4-fluorophenyl)-N-[(2R)-2-hydroxy-3-(4-methoxyphenyl)-2-methylpropyl]-2-methylpyrazole-3-carboxamide
—— [5-(2,5-dimethoxyphenyl)-2-methylpyrazol-3-yl]-[(3S)-3-phenylpyrrolidin-1-yl]methanone —— C23H25N3O3
[5-(2,5-dimethoxyphenyl)-2-methylpyrazol-3-yl]-[(3S)-3-phenylpyrrolidin-1-yl]methanone
—— 5-(4-fluorophenyl)-N-[(2S)-2-hydroxy-3-(4-methoxyphenyl)-2-methylpropyl]-2-methylpyrazole-3-carboxamide —— C22H24FN3O3
5-(4-fluorophenyl)-N-[(2S)-2-hydroxy-3-(4-methoxyphenyl)-2-methylpropyl]-2-methylpyrazole-3-carboxamide
—— 5-(4-fluorophenyl)-2-methyl-N-[2-[(2S)-1-thiophen-2-ylsulfonylpiperidin-2-yl]ethyl]pyrazole-3-carboxamide —— C22H25FN4O3S2
5-(4-fluorophenyl)-2-methyl-N-[2-[(2S)-1-thiophen-2-ylsulfonylpiperidin-2-yl]ethyl]pyrazole-3-carboxamide