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—— (5-chlorofuran-2-yl)-[(3S)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C13H14ClN3O3
(5-chlorofuran-2-yl)-[(3S)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— 5-[4-[(1R)-1-hydroxy-2-phenylethyl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one —— C20H24N2O3
5-[4-[(1R)-1-hydroxy-2-phenylethyl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one
—— (5-Methyl-1,2-oxazol-3-yl)methyl 4-methyl-3-piperidin-1-ylsulfonylbenzoate —— C18H22N2O5S
(5-Methyl-1,2-oxazol-3-yl)methyl 4-methyl-3-piperidin-1-ylsulfonylbenzoate
—— (5S)-N,5-dimethyl-N-[(3-pyrazol-1-ylphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide —— C20H23N5O
(5S)-N,5-dimethyl-N-[(3-pyrazol-1-ylphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
—— 5-[1-[(2R)-2-(3,5-dimethylpyrazol-1-yl)propyl]imidazol-2-yl]-6-methylquinoline —— C21H23N5
5-[1-[(2R)-2-(3,5-dimethylpyrazol-1-yl)propyl]imidazol-2-yl]-6-methylquinoline
—— 5-[(3R)-3-[(1,3-benzoxazol-2-ylamino)methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one —— C17H19N5O2
5-[(3R)-3-[(1,3-benzoxazol-2-ylamino)methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one
—— 5-[2-[4-[(1S)-1-hydroxy-2-phenylethyl]piperidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one —— C21H27N3O3
5-[2-[4-[(1S)-1-hydroxy-2-phenylethyl]piperidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one
—— 5-[(3S)-3-[(1,3-benzoxazol-2-ylamino)methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one —— C17H19N5O2
5-[(3S)-3-[(1,3-benzoxazol-2-ylamino)methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one
—— 5-[2-[4-[(1R)-1-hydroxy-2-phenylethyl]piperidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one —— C21H27N3O3
5-[2-[4-[(1R)-1-hydroxy-2-phenylethyl]piperidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one
—— (5-methoxy-1H-indazol-3-yl)-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methanone —— C20H22N4O3
(5-methoxy-1H-indazol-3-yl)-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methanone
—— 5-[(2R)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C14H20N4OS
5-[(2R)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5R)-N,5-dimethyl-N-[(3-pyrazol-1-ylphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide —— C20H23N5O
(5R)-N,5-dimethyl-N-[(3-pyrazol-1-ylphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
—— 5-[(2S)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C14H20N4OS
5-[(2S)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[2-[(2S)-2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C19H23N3O4
5-[2-[(2S)-2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— 5-[1-[(2S)-2-(3,5-dimethylpyrazol-1-yl)propyl]imidazol-2-yl]-6-methylquinoline —— C21H23N5
5-[1-[(2S)-2-(3,5-dimethylpyrazol-1-yl)propyl]imidazol-2-yl]-6-methylquinoline
—— (5-ethyl-1H-pyrazol-4-yl)-[(2S)-2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl]methanone —— C19H25N3O2
(5-ethyl-1H-pyrazol-4-yl)-[(2S)-2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl]methanone
—— (5S)-7-(2-methyl-1,3-benzothiazole-5-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione —— C16H15N3O3S
(5S)-7-(2-methyl-1,3-benzothiazole-5-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
—— 5-[4-[(1S)-1-hydroxy-2-phenylethyl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one —— C20H24N2O3
5-[4-[(1S)-1-hydroxy-2-phenylethyl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one
—— (5R)-7-(2-methyl-1,3-benzothiazole-5-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione —— C16H15N3O3S
(5R)-7-(2-methyl-1,3-benzothiazole-5-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
—— (5S)-7-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione —— C18H18FN3O3
(5S)-7-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
—— (5-ethyl-1H-pyrazol-4-yl)-[(2R)-2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl]methanone —— C19H25N3O2
(5-ethyl-1H-pyrazol-4-yl)-[(2R)-2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl]methanone
—— (5R)-7-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione —— C18H18FN3O3
(5R)-7-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
—— 5-[2-[(3R)-3-benzoylpiperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C18H19N3O4
5-[2-[(3R)-3-benzoylpiperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— 5-[2-[(3S)-3-benzoylpiperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C18H19N3O4
5-[2-[(3S)-3-benzoylpiperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— (5-ethyl-1,3-oxazol-4-yl)-[(3S)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C16H22N4O2
(5-ethyl-1,3-oxazol-4-yl)-[(3S)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methanone —— C21H25N5O
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methanone
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methanone —— C21H25N5O
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methanone
—— 5-[(3R)-3-benzoylpiperidine-1-carbonyl]-4-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H19N3O3
5-[(3R)-3-benzoylpiperidine-1-carbonyl]-4-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— (5-chlorothiophen-2-yl)-[(3R)-3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methanone —— C15H21ClN2O2S
(5-chlorothiophen-2-yl)-[(3R)-3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methanone
—— (5-ethyl-1,3-oxazol-4-yl)-[(3R)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C16H22N4O2
(5-ethyl-1,3-oxazol-4-yl)-[(3R)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— 5-butyl-2-[2-[(2S)-2-(furan-2-yl)pyrrolidin-1-yl]-2-oxoethyl]-4-phenyl-1,2,4-triazol-3-one —— C22H26N4O3
5-butyl-2-[2-[(2S)-2-(furan-2-yl)pyrrolidin-1-yl]-2-oxoethyl]-4-phenyl-1,2,4-triazol-3-one
—— 5-[3-[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C19H22N4O3
5-[3-[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-[3-[(3S)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C19H22N4O3
5-[3-[(3S)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— [5-[(dimethylamino)methyl]furan-2-yl]-[(3S)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]methanone —— C20H25FN2O3
[5-[(dimethylamino)methyl]furan-2-yl]-[(3S)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]methanone
—— 5-(methoxymethyl)-3-[[(2R)-2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H18N6O3
5-(methoxymethyl)-3-[[(2R)-2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[(3S)-3-benzoylpiperidine-1-carbonyl]-4-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H19N3O3
5-[(3S)-3-benzoylpiperidine-1-carbonyl]-4-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— [5-[(dimethylamino)methyl]furan-2-yl]-[(3R)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]methanone —— C20H25FN2O3
[5-[(dimethylamino)methyl]furan-2-yl]-[(3R)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]methanone
—— 5-(methoxymethyl)-3-[[(2S)-2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H18N6O3
5-(methoxymethyl)-3-[[(2S)-2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-acetyl-3-[(2R)-2-(2-imidazol-1-ylethyl)piperidine-1-carbonyl]-6-methyl-1H-pyridin-2-one —— C19H24N4O3
5-acetyl-3-[(2R)-2-(2-imidazol-1-ylethyl)piperidine-1-carbonyl]-6-methyl-1H-pyridin-2-one
—— (5S)-7-[3-(3-hydroxy-3-methylbutyl)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione —— C19H24N2O4
(5S)-7-[3-(3-hydroxy-3-methylbutyl)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
—— 5-[[(3S)-3-(3-methoxypropyl)piperidin-1-yl]methyl]-2-thiophen-2-ylpyrimidine —— C18H25N3OS
5-[[(3S)-3-(3-methoxypropyl)piperidin-1-yl]methyl]-2-thiophen-2-ylpyrimidine
—— 5-[[(3R)-3-(3-methoxypropyl)piperidin-1-yl]methyl]-2-thiophen-2-ylpyrimidine —— C18H25N3OS
5-[[(3R)-3-(3-methoxypropyl)piperidin-1-yl]methyl]-2-thiophen-2-ylpyrimidine
—— 5-butyl-2-[2-[(2R)-2-(furan-2-yl)pyrrolidin-1-yl]-2-oxoethyl]-4-phenyl-1,2,4-triazol-3-one —— C22H26N4O3
5-butyl-2-[2-[(2R)-2-(furan-2-yl)pyrrolidin-1-yl]-2-oxoethyl]-4-phenyl-1,2,4-triazol-3-one
—— 5-[(1R)-1-[2-(5-ethylpyridin-2-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole —— C16H19N5O
5-[(1R)-1-[2-(5-ethylpyridin-2-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole
—— 5-[(1S)-1-[2-(5-ethylpyridin-2-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole —— C16H19N5O
5-[(1S)-1-[2-(5-ethylpyridin-2-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole
—— 5-acetyl-3-[(2S)-2-(2-imidazol-1-ylethyl)piperidine-1-carbonyl]-6-methyl-1H-pyridin-2-one —— C19H24N4O3
5-acetyl-3-[(2S)-2-(2-imidazol-1-ylethyl)piperidine-1-carbonyl]-6-methyl-1H-pyridin-2-one
—— (5R)-7-[3-(3-hydroxy-3-methylbutyl)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione —— C19H24N2O4
(5R)-7-[3-(3-hydroxy-3-methylbutyl)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
—— (5-phenyl-1,2-oxazol-3-yl)-[(3S)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]methanone —— C21H21N3O3
(5-phenyl-1,2-oxazol-3-yl)-[(3S)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]methanone
—— 5-[(2S)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C18H20N4O2
5-[(2S)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(2R)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C18H20N4O2
5-[(2R)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole