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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(3R)-1-(1,3-benzothiazole-2-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C22H21N5O2S
5-[(3R)-1-(1,3-benzothiazole-2-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-(2,6-difluorophenyl)sulfonylpiperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C20H20F2N4O3S
5-[(3R)-1-(2,6-difluorophenyl)sulfonylpiperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3S)-1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C19H19ClN4O2S
5-[(3S)-1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3S)-1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C21H20N6O2S
5-[(3S)-1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-bromo-N-[[(4R)-4-hydroxy-2,3-dihydrochromen-4-yl]methyl]thiophene-2-sulfonamide —— C14H14BrNO4S2
5-bromo-N-[[(4R)-4-hydroxy-2,3-dihydrochromen-4-yl]methyl]thiophene-2-sulfonamide
—— 5-[(4,5-Dimethoxy-2-methylphenyl)methylsulfanyl]-1-(3,5-dimethylphenyl)tetrazole —— C19H22N4O2S
5-[(4,5-Dimethoxy-2-methylphenyl)methylsulfanyl]-1-(3,5-dimethylphenyl)tetrazole
—— 5-[(3R)-1-[2-(2-chlorophenyl)acetyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C22H23ClN4O2
5-[(3R)-1-[2-(2-chlorophenyl)acetyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C24H23FN6O2
5-[(3R)-1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C20H23N5O2S
5-[(3R)-1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-(2-ethylsulfanylbenzoyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C23H26N4O2S
5-[(3R)-1-(2-ethylsulfanylbenzoyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3S)-1-[5-(furan-2-yl)-1H-pyrazole-3-carbonyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C22H22N6O3
5-[(3S)-1-[5-(furan-2-yl)-1H-pyrazole-3-carbonyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-bromo-N-[(2R)-2-hydroxy-2-methyl-4-methylsulfanylbutyl]thiophene-2-sulfonamide —— C10H16BrNO3S3
5-bromo-N-[(2R)-2-hydroxy-2-methyl-4-methylsulfanylbutyl]thiophene-2-sulfonamide
—— 5-[(3S)-1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C20H23N5O2S
5-[(3S)-1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-(2-methoxybenzoyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C22H24N4O3
5-[(3R)-1-(2-methoxybenzoyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C21H25N5O3
5-[(3R)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-[(3-fluorophenyl)methylsulfonyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C21H23FN4O3S
5-[(3R)-1-[(3-fluorophenyl)methylsulfonyl]piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3S)-1-(4-acetylphenyl)sulfonylpiperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C22H24N4O4S
5-[(3S)-1-(4-acetylphenyl)sulfonylpiperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C21H24N4O3
5-[(3R)-1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-(4-acetylphenyl)sulfonylpiperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C22H24N4O4S
5-[(3R)-1-(4-acetylphenyl)sulfonylpiperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-[(3S)-1-(3-methoxy-1-methylpyrazole-4-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C20H24N6O3
5-[(3S)-1-(3-methoxy-1-methylpyrazole-4-carbonyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-(4-fluorophenyl)-N-[[(4S)-4-hydroxy-2,3-dihydrochromen-4-yl]methyl]-2-methylpyrazole-3-carboxamide —— C21H20FN3O3
5-(4-fluorophenyl)-N-[[(4S)-4-hydroxy-2,3-dihydrochromen-4-yl]methyl]-2-methylpyrazole-3-carboxamide
—— 5,6-dimethyl-3-[2-[(3S)-3-(1-methyl-5-oxo-4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl]pyrimidin-4-one —— C22H26N6O3
5,6-dimethyl-3-[2-[(3S)-3-(1-methyl-5-oxo-4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl]pyrimidin-4-one
—— 5-chloro-N-[(2S)-2-cyclopropyl-2-hydroxy-2-thiophen-2-ylethyl]-2-methoxybenzenesulfonamide —— C16H18ClNO4S2
5-chloro-N-[(2S)-2-cyclopropyl-2-hydroxy-2-thiophen-2-ylethyl]-2-methoxybenzenesulfonamide
—— 5-[(Z)-N-[(2-fluorophenyl)carbamothioylamino]-C-methylcarbonimidoyl]thiophene-2-carboxylate —— C14H11FN3O2S2-
5-[(Z)-N-[(2-fluorophenyl)carbamothioylamino]-C-methylcarbonimidoyl]thiophene-2-carboxylate
—— 5-bromo-N-[[(2S)-oxolan-2-yl]methyl]-N-[4-(trifluoromethyl)-1,3-benzothiazol-2-yl]thiophene-2-carboxamide —— C18H14BrF3N2O2S2
5-bromo-N-[[(2S)-oxolan-2-yl]methyl]-N-[4-(trifluoromethyl)-1,3-benzothiazol-2-yl]thiophene-2-carboxamide
—— 5-[(Z)-N-[(4-tert-butylbenzoyl)amino]-C-methylcarbonimidoyl]thiophene-2-carboxylate —— C18H19N2O3S-
5-[(Z)-N-[(4-tert-butylbenzoyl)amino]-C-methylcarbonimidoyl]thiophene-2-carboxylate
—— 5-[3-[(2R)-butan-2-yl]oxyphenyl]-2-ethylthiophene-3-carbaldehyde —— C17H20O2S
5-[3-[(2R)-butan-2-yl]oxyphenyl]-2-ethylthiophene-3-carbaldehyde
—— 5-(4-tert-butylphenyl)-2-[(1R)-1-chloroethyl]-6-methyl-3H-thieno[2,3-d]pyrimidin-4-one —— C19H21ClN2OS
5-(4-tert-butylphenyl)-2-[(1R)-1-chloroethyl]-6-methyl-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-(3-chlorophenyl)-2-(hydroxymethylidene)thiophen-3-one —— C11H7ClO2S
5-(3-chlorophenyl)-2-(hydroxymethylidene)thiophen-3-one
—— 5-(furan-2-yl)-N-[[(2R)-oxolan-2-yl]methyl]-N-[4-(trifluoromethyl)-1,3-benzothiazol-2-yl]-1,2-oxazole-3-carboxamide —— C21H16F3N3O4S
5-(furan-2-yl)-N-[[(2R)-oxolan-2-yl]methyl]-N-[4-(trifluoromethyl)-1,3-benzothiazol-2-yl]-1,2-oxazole-3-carboxamide
—— 5-[(Z)-N-[(4-ethoxybenzoyl)amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid —— C16H16N2O4S
5-[(Z)-N-[(4-ethoxybenzoyl)amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid
—— 5-[(Z)-N-[[(3S)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid —— C16H14N2O5S
5-[(Z)-N-[[(3S)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid
—— 5-[(Z)-C-methyl-N-[(6-phenylthieno[2,3-d]pyrimidin-4-yl)amino]carbonimidoyl]thiophene-2-carboxylate —— C19H13N4O2S2-
5-[(Z)-C-methyl-N-[(6-phenylthieno[2,3-d]pyrimidin-4-yl)amino]carbonimidoyl]thiophene-2-carboxylate
—— 5-[(Z)-C-methyl-N-[[(1R,2S)-2-methylcyclohexyl]carbamothioylamino]carbonimidoyl]thiophene-2-carboxylate —— C15H20N3O2S2-
5-[(Z)-C-methyl-N-[[(1R,2S)-2-methylcyclohexyl]carbamothioylamino]carbonimidoyl]thiophene-2-carboxylate
—— (5R)-2-[(5-benzyl-1,3-thiazol-2-yl)amino]-5-methyl-1,3-thiazol-4-one —— C14H13N3OS2
(5R)-2-[(5-benzyl-1,3-thiazol-2-yl)amino]-5-methyl-1,3-thiazol-4-one
—— (5S)-5-methyl-2-(1,3-thiazol-2-ylamino)-1,3-thiazol-4-one —— C7H7N3OS2
(5S)-5-methyl-2-(1,3-thiazol-2-ylamino)-1,3-thiazol-4-one
—— 5-[(Z)-C-methyl-N-[[(1S,2R)-2-methylcyclohexyl]carbamothioylamino]carbonimidoyl]thiophene-2-carboxylate —— C15H20N3O2S2-
5-[(Z)-C-methyl-N-[[(1S,2R)-2-methylcyclohexyl]carbamothioylamino]carbonimidoyl]thiophene-2-carboxylate
—— 5-chloro-N-[(2R)-2-cyclopropyl-2-hydroxy-2-thiophen-2-ylethyl]-2-methoxybenzenesulfonamide —— C16H18ClNO4S2
5-chloro-N-[(2R)-2-cyclopropyl-2-hydroxy-2-thiophen-2-ylethyl]-2-methoxybenzenesulfonamide
—— 5-[(Z)-N-[[2-(1,3-benzothiazol-2-ylsulfanyl)acetyl]amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid —— C16H13N3O3S3
5-[(Z)-N-[[2-(1,3-benzothiazol-2-ylsulfanyl)acetyl]amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid
—— 5-[(Z)-N-(5,6-dihydro-4H-cyclopenta[b]thiophene-2-carbonylamino)-C-methylcarbonimidoyl]thiophene-2-carboxylate —— C15H13N2O3S2-
5-[(Z)-N-(5,6-dihydro-4H-cyclopenta[b]thiophene-2-carbonylamino)-C-methylcarbonimidoyl]thiophene-2-carboxylate
—— 5-[(Z)-N-[[2-(4-chlorophenyl)sulfanylacetyl]amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid —— C15H13ClN2O3S2
5-[(Z)-N-[[2-(4-chlorophenyl)sulfanylacetyl]amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid
—— 5-[(Z)-N-(cyclopropanecarbonylamino)-C-methylcarbonimidoyl]thiophene-2-carboxylic acid —— C11H12N2O3S
5-[(Z)-N-(cyclopropanecarbonylamino)-C-methylcarbonimidoyl]thiophene-2-carboxylic acid
—— 5-[(Z)-C-methyl-N-[[(1R,2R)-2-methylcyclohexyl]carbamothioylamino]carbonimidoyl]thiophene-2-carboxylic acid —— C15H21N3O2S2
5-[(Z)-C-methyl-N-[[(1R,2R)-2-methylcyclohexyl]carbamothioylamino]carbonimidoyl]thiophene-2-carboxylic acid
—— 5-[(Z)-N-[(4-methoxybenzoyl)amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid —— C15H14N2O4S
5-[(Z)-N-[(4-methoxybenzoyl)amino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid
—— 5-[(Z)-C-methyl-N-[[(1S,2S)-2-methylcyclohexyl]carbamothioylamino]carbonimidoyl]thiophene-2-carboxylic acid —— C15H21N3O2S2
5-[(Z)-C-methyl-N-[[(1S,2S)-2-methylcyclohexyl]carbamothioylamino]carbonimidoyl]thiophene-2-carboxylic acid
—— (5R)-3,3-dimethyl-5-(2-methylpropyl)morpholine —— C10H21NO
(5R)-3,3-dimethyl-5-(2-methylpropyl)morpholine
—— 5-bromo-2-chloro-N-[(2R)-2-cyclopropyl-2-hydroxy-2-thiophen-2-ylethyl]benzamide —— C16H15BrClNO2S
5-bromo-2-chloro-N-[(2R)-2-cyclopropyl-2-hydroxy-2-thiophen-2-ylethyl]benzamide
—— 5-[(Z)-C-methyl-N-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-ylamino)carbonimidoyl]thiophene-2-carboxylate —— C16H13N4O2S2-
5-[(Z)-C-methyl-N-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-ylamino)carbonimidoyl]thiophene-2-carboxylate
—— 5-bromo-N-[(2S)-2-hydroxy-2-methyl-4-methylsulfanylbutyl]thiophene-2-sulfonamide —— C10H16BrNO3S3
5-bromo-N-[(2S)-2-hydroxy-2-methyl-4-methylsulfanylbutyl]thiophene-2-sulfonamide
—— 5-[(2R)-2-methyl-2,3-dihydroindole-1-carbonyl]-3-(thiophen-2-ylmethyl)-1H-pyrimidine-2,4-dione —— C19H17N3O3S
5-[(2R)-2-methyl-2,3-dihydroindole-1-carbonyl]-3-(thiophen-2-ylmethyl)-1H-pyrimidine-2,4-dione