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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-chloro-N-[(3R)-1-(2-fluorophenyl)-2-oxopyrrolidin-3-yl]thiophene-2-sulfonamide —— C14H12ClFN2O3S2
5-chloro-N-[(3R)-1-(2-fluorophenyl)-2-oxopyrrolidin-3-yl]thiophene-2-sulfonamide
—— (5R)-3-[3-(tert-butylsulfonylmethyl)phenyl]-5-methyl-2-sulfanylideneimidazolidin-4-one —— C15H20N2O3S2
(5R)-3-[3-(tert-butylsulfonylmethyl)phenyl]-5-methyl-2-sulfanylideneimidazolidin-4-one
—— 5-chloro-N-[(2R)-2-hydroxy-2-(2-methylphenyl)ethyl]thiophene-2-carboxamide —— C14H14ClNO2S
5-chloro-N-[(2R)-2-hydroxy-2-(2-methylphenyl)ethyl]thiophene-2-carboxamide
—— [5-(Phenoxymethyl)furan-2-yl]-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone —— C22H24N3O3+
[5-(Phenoxymethyl)furan-2-yl]-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone —— C18H22N3OS+
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone
—— (5-Chloro-2-methoxyphenyl)-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone —— C18H21ClN3O2+
(5-Chloro-2-methoxyphenyl)-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone
—— [(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(pyridin-4-ylmethyl)piperazin-1-yl]methanone —— C20H25N3OS
[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(pyridin-4-ylmethyl)piperazin-1-yl]methanone
—— (5-Methyl-3-phenyl-1,2-oxazol-4-yl)-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone —— C21H23N4O2+
(5-Methyl-3-phenyl-1,2-oxazol-4-yl)-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone
—— [5-[4-(2-Chlorophenyl)sulfonylpiperazin-1-yl]-5-oxopentyl]urea —— C16H23ClN4O4S
[5-[4-(2-Chlorophenyl)sulfonylpiperazin-1-yl]-5-oxopentyl]urea
—— [(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone —— C20H26N3OS+
[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(pyridin-4-ylmethyl)piperazin-4-ium-1-yl]methanone
—— 5-bromo-N-[(2S)-1-[2-(4-methoxypiperidin-1-yl)ethylamino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C16H24BrN3O3S
5-bromo-N-[(2S)-1-[2-(4-methoxypiperidin-1-yl)ethylamino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-[[(1R)-1-(5-benzyl-1,2,4-oxadiazol-3-yl)ethyl]amino]-4-chloro-2-methylpyridazin-3-one —— C16H16ClN5O2
5-[[(1R)-1-(5-benzyl-1,2,4-oxadiazol-3-yl)ethyl]amino]-4-chloro-2-methylpyridazin-3-one
—— 5-[[(1S)-1-(5-benzyl-1,2,4-oxadiazol-3-yl)ethyl]amino]-4-chloro-2-methylpyridazin-3-one —— C16H16ClN5O2
5-[[(1S)-1-(5-benzyl-1,2,4-oxadiazol-3-yl)ethyl]amino]-4-chloro-2-methylpyridazin-3-one
—— 5-[[4-[(3R)-thiolan-3-yl]piperazin-1-yl]methyl]-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C18H21F3N4OS
5-[[4-[(3R)-thiolan-3-yl]piperazin-1-yl]methyl]-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— 5-methyl-N'-[2-(3-oxo-1,4-benzoxazin-4-yl)acetyl]-4-propylthiophene-2-carbohydrazide —— C19H21N3O4S
5-methyl-N'-[2-(3-oxo-1,4-benzoxazin-4-yl)acetyl]-4-propylthiophene-2-carbohydrazide
—— 5-[[4-[(3S)-thiolan-3-yl]piperazin-1-yl]methyl]-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C18H21F3N4OS
5-[[4-[(3S)-thiolan-3-yl]piperazin-1-yl]methyl]-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— 5-bromo-N-[(2R)-1-[2-(4-methoxypiperidin-1-yl)ethylamino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C16H24BrN3O3S
5-bromo-N-[(2R)-1-[2-(4-methoxypiperidin-1-yl)ethylamino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— (5R)-5-[2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C16H19N3O3S
(5R)-5-[2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— 5-chloro-N-[2-(4-methoxyphenoxy)ethyl]-N-methyl-1-benzofuran-2-carboxamide —— C19H18ClNO4
5-chloro-N-[2-(4-methoxyphenoxy)ethyl]-N-methyl-1-benzofuran-2-carboxamide
—— 5-[(R)-(4-methyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole —— C22H17N5OS2
5-[(R)-(4-methyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline-2-carbonyl]-2-prop-2-enylisoindole-1,3-dione —— C21H24N2O3
5-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline-2-carbonyl]-2-prop-2-enylisoindole-1,3-dione
—— 5-[(S)-[5-(furan-2-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole —— C24H19N5O2S
5-[(S)-[5-(furan-2-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(R)-[5-(furan-2-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole —— C24H19N5O2S
5-[(R)-[5-(furan-2-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[4-(2-Methylphenyl)piperazine-1-carbonyl]-2-prop-2-enylisoindole-1,3-dione —— C23H23N3O3
5-[4-(2-Methylphenyl)piperazine-1-carbonyl]-2-prop-2-enylisoindole-1,3-dione
—— (5S)-5-[2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C16H19N3O3S
(5S)-5-[2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— 5-[(S)-(4-methyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole —— C22H17N5OS2
5-[(S)-(4-methyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[1-[(2S)-1-(1,3-benzothiazol-2-yl)propan-2-yl]piperidin-4-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C22H23N5OS
5-[1-[(2S)-1-(1,3-benzothiazol-2-yl)propan-2-yl]piperidin-4-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-[1-[(2R)-1-(1,3-benzothiazol-2-yl)propan-2-yl]piperidin-4-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C22H23N5OS
5-[1-[(2R)-1-(1,3-benzothiazol-2-yl)propan-2-yl]piperidin-4-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— (5S)-N-(oxan-4-yl)-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H18N2O3
(5S)-N-(oxan-4-yl)-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-(cyclohexylsulfamoyl)-N-[2-(ethylamino)-2-oxoethyl]-2-methylbenzamide —— C18H27N3O4S
5-(cyclohexylsulfamoyl)-N-[2-(ethylamino)-2-oxoethyl]-2-methylbenzamide
—— 5-methoxy-N'-(2-methylbenzoyl)-2,3-dihydro-1,4-benzodioxine-7-carbohydrazide —— C18H18N2O5
5-methoxy-N'-(2-methylbenzoyl)-2,3-dihydro-1,4-benzodioxine-7-carbohydrazide
—— 5-chloro-N-[2-(3-methylphenoxy)ethyl]-1-benzofuran-2-carboxamide —— C18H16ClNO3
5-chloro-N-[2-(3-methylphenoxy)ethyl]-1-benzofuran-2-carboxamide
—— 5-methoxy-N-[4-[methyl(propan-2-yl)sulfamoyl]phenyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide —— C20H24N2O6S
5-methoxy-N-[4-[methyl(propan-2-yl)sulfamoyl]phenyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide
—— (5S)-5-methyl-N-[4-[methyl(propan-2-yl)sulfamoyl]phenyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H26N2O3S2
(5S)-5-methyl-N-[4-[methyl(propan-2-yl)sulfamoyl]phenyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-5-[2-[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C17H17N3O3S2
(5R)-5-[2-[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— 5-ethyl-4-methyl-N-[4-[methyl(propan-2-yl)sulfamoyl]phenyl]thiophene-2-carboxamide —— C18H24N2O3S2
5-ethyl-4-methyl-N-[4-[methyl(propan-2-yl)sulfamoyl]phenyl]thiophene-2-carboxamide
—— (5S)-5-[2-[(3R)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C17H17N3O3S2
(5S)-5-[2-[(3R)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— [5-[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-5-oxopentyl]urea —— C18H24N4O2S
[5-[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-5-oxopentyl]urea
—— (5R)-N-(oxan-4-yl)-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H18N2O3
(5R)-N-(oxan-4-yl)-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5-fluoro-2-methylphenyl)-[(3R)-3-(pyridin-3-ylmethoxy)pyrrolidin-1-yl]methanone —— C18H19FN2O2
(5-fluoro-2-methylphenyl)-[(3R)-3-(pyridin-3-ylmethoxy)pyrrolidin-1-yl]methanone
—— 5-[2-[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-2-oxoethyl]-2,3-dihydro-1,5-benzoxazepin-4-one —— C23H23N3O3S
5-[2-[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-2-oxoethyl]-2,3-dihydro-1,5-benzoxazepin-4-one
—— 5-bromo-N-[2-[[(1S,3R)-3-[(S)-ethylsulfinyl]cyclohexyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C16H23BrN2O3S2
5-bromo-N-[2-[[(1S,3R)-3-[(S)-ethylsulfinyl]cyclohexyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— (5-fluoro-2-methylphenyl)-[(3S)-3-(pyridin-3-ylmethoxy)pyrrolidin-1-yl]methanone —— C18H19FN2O2
(5-fluoro-2-methylphenyl)-[(3S)-3-(pyridin-3-ylmethoxy)pyrrolidin-1-yl]methanone
—— 5-bromo-N-[2-[[(1S,3R)-3-[(R)-ethylsulfinyl]cyclohexyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C16H23BrN2O3S2
5-bromo-N-[2-[[(1S,3R)-3-[(R)-ethylsulfinyl]cyclohexyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-[[4-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-1,4-diazepan-1-yl]methyl]-3-[(1S)-1-methoxyethyl]-1,2,4-oxadiazole —— C21H29ClN4O4
5-[[4-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-1,4-diazepan-1-yl]methyl]-3-[(1S)-1-methoxyethyl]-1,2,4-oxadiazole
—— 5-bromo-N-[2-[[(1S,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C16H23BrN2O3S2
5-bromo-N-[2-[[(1S,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-methyl-3-nitro-2-[4-[[(2S)-oxan-2-yl]methoxy]piperidin-1-yl]pyridine —— C17H25N3O4
5-methyl-3-nitro-2-[4-[[(2S)-oxan-2-yl]methoxy]piperidin-1-yl]pyridine
—— 5-[[4-(2,6-dimethylpyrimidin-4-yl)-1,4-diazepan-1-yl]methyl]-3-[(1R)-1-methoxyethyl]-1,2,4-oxadiazole —— C17H26N6O2
5-[[4-(2,6-dimethylpyrimidin-4-yl)-1,4-diazepan-1-yl]methyl]-3-[(1R)-1-methoxyethyl]-1,2,4-oxadiazole
—— 5-chloro-2-[[(2R)-2-(hydroxymethyl)-3-pyridin-2-ylpropyl]amino]benzonitrile —— C16H16ClN3O
5-chloro-2-[[(2R)-2-(hydroxymethyl)-3-pyridin-2-ylpropyl]amino]benzonitrile
—— 5-bromo-N-[2-[[(1S,3S)-3-[(R)-ethylsulfinyl]cyclohexyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C16H23BrN2O3S2
5-bromo-N-[2-[[(1S,3S)-3-[(R)-ethylsulfinyl]cyclohexyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide