中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
propan-2-yl (2S)-2-[[(2-benzylphenoxy)-[[(3R,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-4-fluoro-3-hydroxy-4-methyloxolan-2-yl]methoxy]phosphoryl]amino]propanoate |
—— |
C29H35FN3O9P |
|
—— |
1-[(2R,4R,5R)-3,4-dihydroxy-5-(hydroxymethyl)-4-methyloxolan-2-yl]pyrimidine-2,4-dione |
—— |
C10H14N2O6 |
|
—— |
S-[2-[dimethylamino-[[(2R,3S,5R)-4-ethynyl-4-fluoro-3-hydroxy-5-(2-methylidene-4-methyliminopyrimidin-1-yl)oxolan-2-yl]methoxy]phosphoryl]oxyethyl] ethanethioate |
—— |
C19H28FN4O6PS |
|
—— |
S-[2-[dimethylamino-[[(2R,3S,5R)-4-fluoro-3-hydroxy-4-methyl-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methoxy]phosphoryl]oxyethyl] ethanethioate |
—— |
C17H27FN3O8PS |
|
—— |
S-[2-[[(2S,5S)-5-(4-amino-2-oxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy-(benzylamino)phosphoryl]oxyethyl] 2,2-dimethylbutanethioate |
—— |
C24H35N4O7PS |
|
—— |
S-[2-[dimethylamino-[[(2R,3S,5R)-4-ethynyl-4-fluoro-3-hydroxy-5-(2-methylidene-4-oxopyrimidin-1-yl)oxolan-2-yl]methoxy]phosphoryl]oxyethyl] ethanethioate |
—— |
C18H25FN3O7PS |
|
—— |
[2-[[(3R,5R)-4,4-difluoro-3-hydroxy-5-(4-methyl-2-oxopyrimidin-1-yl)oxolan-2-yl]methoxy]-2-oxoethyl] butanoate |
—— |
C16H20F2N2O7 |
|
—— |
[(2R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-2-(hydroxymethyl)-4-tri(propan-2-yl)silyloxyoxolan-3-yl] (3E)-3-(1-butyl-5-oxopyrrolidin-2-ylidene)propanoate |
—— |
C29H47N3O8Si |
|
—— |
[(2R,3S,5R)-5-(5-bromo-2,4-dioxopyrimidin-1-yl)-2-(hydroxymethyl)-4-tri(propan-2-yl)silyloxyoxolan-3-yl] 7-(butylamino)-4,7-dioxoheptanoate |
—— |
C29H48BrN3O9Si |
|
—— |
propan-2-yl (2S)-2-[[[(2S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-4-methyl-4-(1-sulfanyloxycyclopentyl)oxyoxolan-2-yl]methoxy-phenoxyphosphinothioyl]amino]propanoate |
—— |
C27H38N3O9PS2 |
|
—— |
[(2S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-4-fluoro-4-methyloxolan-2-yl]methoxy-oxo-[[(2S)-1-oxo-1-propan-2-yloxypropan-2-yl]amino]phosphanium |
—— |
C16H24FN3O7P+ |
|
—— |
N-(2-aminoethyl)-2-[(2R,3S,5R)-2-(2,4-dioxopyrimidin-1-yl)-4-hydroxy-5-(hydroxymethyl)oxolan-3-yl]oxyacetamide |
—— |
C13H20N4O7 |
|
—— |
propan-2-yl 2-[[[(2S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-4-fluoro-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate |
—— |
C22H29FN3O8P |
|
—— |
[3-[(2R,3S,5R)-3-[2-(2-aminoethylamino)-2-oxoethoxy]-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-2,6-dioxopyrimidin-1-yl]methyl 2,2-dimethylpropanoate |
—— |
C19H30N4O9 |
|
—— |
propan-2-yl (2S)-2-[[[(2R,3R,4R,5R)-4-chloro-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-propylsulfanylphosphoryl]amino]propanoate |
—— |
C19H31ClN3O8PS |
|
—— |
propan-2-yl (2S)-2-[[chloro-[[(2R,3R,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxy-4-methyloxolan-2-yl]methoxy]phosphoryl]amino]propanoate |
—— |
C16H25ClN3O9P |
|
—— |
propan-2-yl (2R)-2-[[[(2R,3R,4R,5R)-4-chloro-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(2-methoxy-2-oxoethyl)sulfanylphosphoryl]amino]propanoate |
—— |
C19H29ClN3O10PS |
|
—— |
propan-2-yl (2S)-2-[[[(2R,3R,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxy-4-methyloxolan-2-yl]methoxy-(2-methoxy-2-oxoethyl)sulfanylphosphoryl]amino]propanoate |
—— |
C19H30N3O11PS |
|
—— |
propan-2-yl (2S)-2-[[[(2R,3R,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxy-4-methyloxolan-2-yl]methoxy-(3-ethoxy-3-oxopropyl)sulfanylphosphoryl]amino]propanoate |
—— |
C21H34N3O11PS |
|
—— |
propan-2-yl 2-[[[(2S,4R,5R)-5-(4-amino-2-methylidenepyrimidin-1-yl)-4-fluoro-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate |
—— |
C23H32FN4O6P |
|
—— |
propan-2-yl (2S)-2-[[[(2R,3R,4R,5R)-4-chloro-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-cyclopentylsulfanylphosphoryl]amino]propanoate |
—— |
C21H33ClN3O8PS |
|
—— |
propan-2-yl (2S)-2-[[[(2S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-4-fluoro-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate |
—— |
C22H29FN3O8P |
|
—— |
4-amino-5-(2-hydroxyethylsulfanylmethyl)-1-[(2R,4R,5R)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one |
—— |
C12H19N3O5S |
|
—— |
(2R)-2-amino-3-[[4-amino-1-[(2R,4R,5R)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-2-oxopyrimidin-5-yl]methylsulfanyl]propanoic acid |
—— |
C13H20N4O6S |
|
—— |
4-amino-5-[(2,3-dihydroxy-4-sulfanylbutyl)sulfanylmethyl]-1-[(2R,4R,5R)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one |
—— |
C14H23N3O6S2 |
|
—— |
2-[(2R,3R,4R,5R)-2-(4-amino-5-methyl-2-oxopyrimidin-1-yl)-4-hydroxy-5-(hydroxymethyl)oxolan-3-yl]oxy-N-ethylacetohydrazide |
—— |
C14H23N5O6 |
|
—— |
2-[(2R,3R,4R,5R)-2-(4-amino-2-oxopyrimidin-1-yl)-4-hydroxy-5-(hydroxymethyl)oxolan-3-yl]oxy-N-ethylacetohydrazide |
—— |
C13H21N5O6 |
|
—— |
1-[(2R,3R,5S)-3-[2-[hydroxy(dimethyl)silyl]-2-methylpropyl]-5-(hydroxymethyl)oxolan-2-yl]-5-methylpyrimidine-2,4-dione |
—— |
C16H28N2O5Si |
|
—— |
[(2S,3R,5R)-3-methyl-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methyl 2-bromoacetate |
—— |
C13H17BrN2O5 |
|
—— |
4-amino-1-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-5-propanoylpyrimidin-2-one |
—— |
C12H17N3O6 |
|
—— |
[[1-[(2R,4S,5R)-3-fluoro-4-hydroxy-5-(hydroxymethyl)-3-methyloxolan-2-yl]-2-oxopyrimidin-4-yl]amino] octanoate |
—— |
C18H28FN3O6 |
|
—— |
US10874683, Example 56.5 |
—— |
C10H15N3O6 |
|
—— |
N-[1-[(2R,5R)-3,3-difluoro-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-2-oxopyrimidin-4-yl]-4-phenylbutanamide |
—— |
C19H21F2N3O5 |
|
—— |
N-[1-[(2R,5R)-3,3-difluoro-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-2-oxopyrimidin-4-yl]butanamide |
—— |
C13H17F2N3O5 |
|
—— |
5-[(E)-2-cyclohexylethenyl]-1-[(4R,5R)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidine-2,4-dione |
—— |
C17H24N2O5 |
|
—— |
1-[(2R,3S,4R,5R)-3-fluoro-4-hydroxy-5-(hydroxymethyl)-3-methyloxolan-2-yl]-4-(hydroxyamino)pyrimidin-2-one |
—— |
C10H14FN3O5 |
|
—— |
2-[[[(2R,3R,4R,5R)-4-fluoro-3-hydroxy-4-methyl-5-[2-oxo-4-(phenylmethoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoic acid |
—— |
C26H30FN4O9P |
|
—— |
propan-2-yl (2S)-2-[[[(2R,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-4-fluoro-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate |
—— |
C22H29FN3O9P |
|
—— |
(E)-3-[4-amino-1-[(2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-2-oxopyrimidin-5-yl]prop-2-enamide |
—— |
C12H16N4O5 |
|
—— |
2-cyanoethyl [(2R,3R,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-4-fluoro-3-hydroxy-4-methyloxolan-2-yl]methyl 3-hexadecoxypropyl phosphite |
—— |
C32H55FN3O8P |
|
—— |
4-amino-1-[(2R,3S,5R)-4-butoxy-5-(butoxymethyl)-3-fluorooxolan-2-yl]-5-(butoxymethyl)pyrimidin-2-one |
—— |
C22H38FN3O5 |
|
—— |
1-[(2R,3R,4R,5R)-3-benzyl-3,4-dihydroxy-2,5-bis(hydroxymethyl)oxolan-2-yl]pyrimidine-2,4-dione |
—— |
C17H20N2O7 |
|
—— |
1-[(2R,3S,5R)-4-hydroxy-5-(hydroxymethyl)-3-naphthalen-1-yloxyoxolan-2-yl]pyrimidine-2,4-dione |
—— |
C19H18N2O6 |
|
—— |
propyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(2-chlorophenoxy)phosphoryl]amino]propanoate |
—— |
C22H28ClN6O9P |
|
—— |
propan-2-yl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate |
—— |
C22H29N6O9P |
|
—— |
2-methylpropyl (2S)-2-[[[(2R,3S,4R)-5-(4-amino-2-oxopyrimidin-1-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate |
—— |
C23H32N7O8P |
|
—— |
methyl (2S)-2-[[[(2R,3S,4R,5R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate |
—— |
C20H25N6O9P |
|
—— |
ethyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(4-fluorophenoxy)phosphoryl]amino]propanoate |
—— |
C21H26FN6O9P |
|
—— |
ethyl 3-[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-[[(2S)-1-methoxy-1-oxopropan-2-yl]amino]phosphoryl]oxybenzoate |
—— |
C23H29N6O11P |
|
—— |
[(1S)-1-phenylethyl] (2S)-2-[[[(2R,3S,4R,5R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate |
—— |
C27H31N6O9P |
|