中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
(4S)-2-[1-(cyclopropylcarbonyl)piperidin-3-yl]-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine |
—— |
C28H29N5O3 |
|
—— |
2-{[7-(3,5-dimethylisoxazol-4-yl)-4-phenyl-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl](methyl)amino}ethanol |
—— |
C23H24N4O3 |
|
—— |
US9624241, Example 87 |
—— |
C24H23N5O3 |
|
—— |
4-[7-(3,5-dimethylisoxazol-4-yl)-2-oxo-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazin-4-yl]benzonitrile |
—— |
C21H16N4O3 |
|
—— |
(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-5-(2-methylpyrazol-3-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7-trien-2-one;2,2,2-trifluoroacetic acid |
—— |
C25H21F3N6O5 |
|
—— |
US9624241, Example 70 |
—— |
C21H20N4O3 |
|
—— |
N-{[5-nitro-3-(pyridin-2-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]methyl}acetamide |
—— |
C16H16N4O4 |
|
—— |
4-(piperidin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C14H17N3O2 |
|
—— |
7-bromo-4-methyl-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C15H12BrN3O2 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-N-ethyl-2-oxo-4-phenyl-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazine-5-carboxamide |
—— |
C23H22N4O4 |
|
—— |
Azane;7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-piperidin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7-trien-2-one |
—— |
C19H25N5O3 |
|
—— |
N-{1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]azetidin-3-yl}-2-methylpropanamide |
—— |
C26H28N6O3 |
|
—— |
7-(3,5-Dimethylisoxazol-4-yl)-4-(1-oxidopyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C19H16N4O4 |
|
—— |
(3S)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]-N,N-dimethylpyrrolidin-3-amine |
—— |
C25H28N6O2 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-5-methyl-4-phenyl-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C21H19N3O3 |
|
—— |
N-{(3R)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]pyrrolidin-3-yl}propane-2-sulfonamide |
—— |
C26H30N6O4S |
|
—— |
tert-butyl 5-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]-3,6-dihydropyridine-1(2H)-carboxylate |
—— |
C29H31N5O4 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-4-phenyl-2-(pyrrolidin-1-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine |
—— |
C24H24N4O2 |
|
—— |
2-{[7-(3,5-dimethylisoxazol-4-yl)-4-phenyl-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]amino}propan-1-ol |
—— |
C23H24N4O3 |
|
—— |
(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraene-2-carboxylic acid |
—— |
C20H16N4O4 |
|
—— |
[1-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]azetidin-3-yl]carbamic acid |
—— |
C23H22N6O4 |
|
—— |
US9624241, Example 71 |
—— |
C21H19N5O4 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-4-(1,3-thiazol-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C17H14N4O3S |
|
—— |
11-[[(2S)-6-amino-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methylamino]-8-(2-fluorophenyl)-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C24H21FN8O2 |
|
—— |
10-Pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7-trien-2-one |
—— |
C14H11N3O2 |
|
—— |
(4S)-2-[1-(cyclopropylcarbonyl)piperidin-4-yl]-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine |
—— |
C28H29N5O3 |
|
—— |
2-{2-[7-(3,5-dimethylisoxazol-4-yl)-2-oxo-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazin-4-yl]phenoxy}-N-(2-hydroxyethyl)acetamide |
—— |
C24H24N4O6 |
|
—— |
3-Pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7-trien-2-one |
—— |
C14H11N3O2 |
|
—— |
5-amino-11-[[(2R)-7-fluoro-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl-methylamino]-8-phenyl-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C25H23FN8O2 |
|
—— |
8-(2-Fluorophenyl)-11-[methyl-[[4-(2,2,2-trifluoroethyl)-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]amino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C26H21F4N7O2 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-4-methyl-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C20H18N4O3 |
|
—— |
N-{(3R)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]pyrrolidin-3-yl}-2,2,2-trifluoroacetamide |
—— |
C25H23F3N6O3 |
|
—— |
11-[(4-Methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-8-[3-(trifluoromethyl)phenyl]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C25H20F3N7O2 |
|
—— |
7-(4-chloro-1-methyl-1H-pyrazol-5-yl)-4-phenyl-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C19H15ClN4O2 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-9-methyl-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C20H18N4O3 |
|
—— |
7-bromo-N-methyl-2-oxo-4-(pyridin-2-yl)-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazine-4-carboxamide |
—— |
C16H13BrN4O3 |
|
—— |
US9624241, Example 125 |
—— |
C19H15FN4O3 |
|
—— |
US9624241, Example 137 |
—— |
C20H19N5O3 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-4-(piperidin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C19H22N4O3 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-4,9-diphenyl-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C26H21N3O3 |
|
—— |
(1R)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]ethane-1,2-diol |
—— |
C21H20N4O4 |
|
—— |
US9624241, Example 8 |
—— |
C20H15F2N3O3 |
|
—— |
3-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]piperidine-1-carboxylic acid |
—— |
C25H25N5O4 |
|
—— |
2-[[7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl](methyl)amino]ethanol |
—— |
C22H23N5O3 |
|
—— |
7-(3,5-Dimethyl-1,2-oxazol-4-yl)-2-oxo-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7-triene-5-carbaldehyde |
—— |
C20H16N4O4 |
|
—— |
N-{(3R)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]pyrrolidin-3-yl}-2-methoxyacetamide |
—— |
C26H28N6O4 |
|
—— |
(4S)-7-(3,5-Dimethylisoxazol-4-yl)-N-methyl-4-pyridin-2-yl-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine-2-carboxamide |
—— |
C21H19N5O3 |
|
—— |
(3R)-N-cyclopropyl-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]pyrrolidine-3-carboxamide |
—— |
C27H28N6O3 |
|
—— |
4-ethyl-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C16H15N3O2 |
|
—— |
5-nitro-3-(pyridin-2-yl)-3,4-dihydro-2H-1,4-benzoxazine-3-carboxylic acid |
—— |
C14H11N3O5 |
|