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吡啶并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(2S)-2-(3,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O3
6-[(2S)-2-(3,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 2-(1,3-benzodioxol-5-yl)-1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone —— C21H20N4O3
2-(1,3-benzodioxol-5-yl)-1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone
—— (2-methylpyridin-3-yl)-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C19H19N5O
(2-methylpyridin-3-yl)-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— [(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-(oxan-4-yl)methanone —— C18H22N4O2
[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-(oxan-4-yl)methanone
—— (1-ethenylpyrrol-2-yl)-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C19H19N5O
(1-ethenylpyrrol-2-yl)-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— [(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-pyridin-4-ylmethanone —— C18H17N5O
[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-pyridin-4-ylmethanone
—— (2R)-2-(2-methoxyphenoxy)-1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one —— C22H24N4O3
(2R)-2-(2-methoxyphenoxy)-1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one
—— [(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-(oxan-4-yl)methanone —— C18H22N4O2
[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-(oxan-4-yl)methanone
—— (5-hydroxypyridin-3-yl)-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C18H17N5O2
(5-hydroxypyridin-3-yl)-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— 1-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-2-[(2S)-oxan-2-yl]ethanone —— C19H24N4O2
1-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-2-[(2S)-oxan-2-yl]ethanone
—— 2-(1,3-benzodioxol-5-yl)-1-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone —— C21H20N4O3
2-(1,3-benzodioxol-5-yl)-1-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone
—— [(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-[(2S)-oxolan-2-yl]methanone —— C17H20N4O2
[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-[(2S)-oxolan-2-yl]methanone
—— 6-[(2R)-2-(2,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O3
6-[(2R)-2-(2,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[4-(2,4-Dimethylphenoxy)butanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25N5O3
6-[4-(2,4-Dimethylphenoxy)butanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (4-chloro-1-methylpyrazol-3-yl)-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C17H17ClN6O
(4-chloro-1-methylpyrazol-3-yl)-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— [(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-pyrazin-2-ylmethanone —— C17H16N6O
[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-pyrazin-2-ylmethanone
—— 1-[(2R)-1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-1-oxopropan-2-yl]pyrrolidin-2-one —— C19H23N5O2
1-[(2R)-1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-1-oxopropan-2-yl]pyrrolidin-2-one
—— 6-[(2S)-2-(2,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O3
6-[(2S)-2-(2,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (5-hydroxypyridin-3-yl)-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C18H17N5O2
(5-hydroxypyridin-3-yl)-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— 1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-3-pyrazol-1-ylpropan-1-one —— C18H20N6O
1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-3-pyrazol-1-ylpropan-1-one
—— [(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-pyridin-4-ylmethanone —— C18H17N5O
[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-pyridin-4-ylmethanone
—— 2-(2-methoxy-4-methylphenoxy)-1-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone —— C22H24N4O3
2-(2-methoxy-4-methylphenoxy)-1-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone
—— 6-Imino-11-methyl-5-(4-methylpiperazine-1-carbonyl)-7-(3-propan-2-yloxypropyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaen-2-one —— C24H32N6O3
6-Imino-11-methyl-5-(4-methylpiperazine-1-carbonyl)-7-(3-propan-2-yloxypropyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaen-2-one
—— [(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-pyrazin-2-ylmethanone —— C17H16N6O
[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-pyrazin-2-ylmethanone
—— 1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-2-[(2S)-oxan-2-yl]ethanone —— C19H24N4O2
1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-2-[(2S)-oxan-2-yl]ethanone
—— [5-(1,3-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C21H21N7O2
[5-(1,3-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— 2-(4-chloropyrazol-1-yl)-1-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone —— C17H17ClN6O
2-(4-chloropyrazol-1-yl)-1-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone
—— [5-(1,3-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C21H21N7O2
[5-(1,3-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— (4-chloro-1-methylpyrazol-3-yl)-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C17H17ClN6O
(4-chloro-1-methylpyrazol-3-yl)-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— 7-[2-(4-Methylphenyl)acetyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H19N5O2
7-[2-(4-Methylphenyl)acetyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2,4-dimethyl-1,3-oxazol-5-yl)-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C18H19N5O2
(2,4-dimethyl-1,3-oxazol-5-yl)-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— [(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-[(2S)-oxolan-2-yl]methanone —— C17H20N4O2
[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]-[(2S)-oxolan-2-yl]methanone
—— (2,4-dimethyl-1,3-oxazol-5-yl)-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C18H19N5O2
(2,4-dimethyl-1,3-oxazol-5-yl)-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— (3R)-3-(3,5-dimethylpyrazol-1-yl)-1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one —— C21H26N6O
(3R)-3-(3,5-dimethylpyrazol-1-yl)-1-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one
—— (3-Methyl-1,2-oxazol-5-yl)-[4-(2-propan-2-ylpyrido[2,3-d]pyrimidin-4-yl)piperidin-1-yl]methanone —— C20H23N5O2
(3-Methyl-1,2-oxazol-5-yl)-[4-(2-propan-2-ylpyrido[2,3-d]pyrimidin-4-yl)piperidin-1-yl]methanone
—— 7-(3-Methyl-1,2-oxazole-5-carbonyl)-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C16H14N6O3
7-(3-Methyl-1,2-oxazole-5-carbonyl)-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— ethyl (2Z)-2-{[(4-fluorophenyl)carbonyl]imino}-10-methyl-5-oxo-1-(tetrahydrofuran-2-ylmethyl)-1,5-dihydro-2H-dipyrido[1,2-a:2',3'-d]pyrimidine-3-carboxylate —— C27H25FN4O5
ethyl (2Z)-2-{[(4-fluorophenyl)carbonyl]imino}-10-methyl-5-oxo-1-(tetrahydrofuran-2-ylmethyl)-1,5-dihydro-2H-dipyrido[1,2-a:2',3'-d]pyrimidine-3-carboxylate
—— 6-imino-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C24H30N6O4
6-imino-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— N-cyclohexyl-13-methyl-2-oxo-6-[[(2R)-oxolan-2-yl]methylamino]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C24H29N5O3
N-cyclohexyl-13-methyl-2-oxo-6-[[(2R)-oxolan-2-yl]methylamino]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— N-[1-[1-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]benzimidazol-2-yl]butyl]benzamide —— C28H27N5O2
N-[1-[1-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]benzimidazol-2-yl]butyl]benzamide
—— 9-methyl-2-[[(4S)-4-phenyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methyl]pyrido[1,2-a]pyrimidin-4-one —— C23H21N3OS
9-methyl-2-[[(4S)-4-phenyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 9-methyl-2-[[5-[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C21H20N4O2S2
9-methyl-2-[[5-[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-bromo-2-[[[(1S)-1-(2,4-dichloro-5-fluorophenyl)ethyl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one —— C17H13BrCl2FN3O
7-bromo-2-[[[(1S)-1-(2,4-dichloro-5-fluorophenyl)ethyl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one
—— (E)-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]-2-(4-methylphenyl)sulfonylprop-2-enenitrile —— C25H26N4O4S
(E)-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]-2-(4-methylphenyl)sulfonylprop-2-enenitrile
—— (3Z,5E)-N-[5-cyano-11-methyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaen-6-ylidene]-3-nitroocta-3,5,7-trienamide —— C26H24N6O5
(3Z,5E)-N-[5-cyano-11-methyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaen-6-ylidene]-3-nitroocta-3,5,7-trienamide
—— 6-(2-Hydroxypropyl)-2-[(3-methylphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H23N3O2
6-(2-Hydroxypropyl)-2-[(3-methylphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 7-bromo-2-[[5-[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C20H17BrN4O2S2
7-bromo-2-[[5-[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— (2E,4E)-N-[5-cyano-11-methyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaen-6-ylidene]-5-methylsulfanylpenta-2,4-dienamide —— C24H23N5O3S
(2E,4E)-N-[5-cyano-11-methyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaen-6-ylidene]-5-methylsulfanylpenta-2,4-dienamide
—— ethyl 6-[(2E,4E)-5-methoxypenta-2,4-dienoyl]imino-11-methyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxylate —— C26H28N4O6
ethyl 6-[(2E,4E)-5-methoxypenta-2,4-dienoyl]imino-11-methyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxylate
—— 2-[[[(1R)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylpropyl]amino]methyl]-6-methylpyrido[1,2-a]pyrimidin-4-one —— C23H27N3O3
2-[[[(1R)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylpropyl]amino]methyl]-6-methylpyrido[1,2-a]pyrimidin-4-one