中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
6-imino-13-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C24H30N6O4 |
|
—— |
(5Z)-3-[[(2R)-oxolan-2-yl]methyl]-5-[(4-oxo-2-pyrrolidin-1-ylpyrido[1,2-a]pyrimidin-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C21H22N4O3S2 |
|
—— |
(5Z)-3-[(2S)-butan-2-yl]-5-[[7-methyl-4-oxo-2-[[(1R)-1-phenylethyl]amino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C25H26N4O2S2 |
|
—— |
6-imino-13-methyl-2-oxo-N-[(1R)-1-phenylethyl]-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C24H25N5O2 |
|
—— |
(5Z)-3-[(2S)-butan-2-yl]-5-[(7-methyl-4-oxo-2-piperidin-1-ylpyrido[1,2-a]pyrimidin-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C22H26N4O2S2 |
|
—— |
2-[(5Z)-5-[[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid |
—— |
C22H24N4O4S2 |
|
—— |
(5Z)-3-[(2R)-butan-2-yl]-5-[[2-(3-morpholin-4-ylpropylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C23H29N5O3S2 |
|
—— |
7-[(2S)-butan-2-yl]-6-imino-13-methyl-2-oxo-N-(2-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C25H27N5O2 |
|
—— |
(5Z)-5-[[2-[[(2S)-2-hydroxypropyl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C18H18N4O3S2 |
|
—— |
6-imino-13-methyl-2-oxo-N-[(1R)-1-phenylethyl]-7-(2-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C29H27N5O2 |
|
—— |
7-ethyl-6-imino-13-methyl-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C23H23N5O2 |
|
—— |
(5Z)-5-[[2-(1,3-benzodioxol-5-ylmethylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(2S)-butan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C24H22N4O4S2 |
|
—— |
(5Z)-5-[[2-[[(2R)-2-hydroxypropyl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C18H18N4O3S2 |
|
—— |
6-imino-13-methyl-N-(2-morpholin-4-ylethyl)-2-oxo-7-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C24H30N6O4 |
|
—— |
6-imino-13-methyl-2-oxo-N-[(1S)-1-phenylethyl]-7-(2-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C29H27N5O2 |
|
—— |
6-imino-13-methyl-N-(2-morpholin-4-ylethyl)-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C24H30N6O4 |
|
—— |
(5Z)-3-[(2R)-butan-2-yl]-5-[[7-methyl-4-oxo-2-[[(1R)-1-phenylethyl]amino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C25H26N4O2S2 |
|
—— |
N-ethyl-6-imino-13-methyl-2-oxo-7-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C20H23N5O3 |
|
—— |
7-[(2R)-butan-2-yl]-6-imino-13-methyl-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C25H27N5O2 |
|
—— |
(5Z)-3-[(4-fluorophenyl)methyl]-5-[[2-[[(2S)-2-hydroxypropyl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C22H19FN4O3S2 |
|
—— |
(5Z)-3-[(2R)-butan-2-yl]-5-[[7-methyl-4-oxo-2-[[(1S)-1-phenylethyl]amino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C25H26N4O2S2 |
|
—— |
(5Z)-3-[(2S)-butan-2-yl]-5-[[7-methyl-4-oxo-2-[[(1S)-1-phenylethyl]amino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C25H26N4O2S2 |
|
—— |
(5Z)-5-[[2-(1,3-benzodioxol-5-ylmethylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(2R)-butan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C24H22N4O4S2 |
|
—— |
(5Z)-3-[(2R)-butan-2-yl]-5-[[7-methyl-2-(3-morpholin-4-ylpropylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C24H31N5O3S2 |
|
—— |
(5Z)-5-[(4-oxo-2-pyrrolidin-1-ylpyrido[1,2-a]pyrimidin-3-yl)methylidene]-3-[(1S)-1-phenylethyl]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C24H22N4O2S2 |
|
—— |
(5Z)-3-[(2S)-2-ethylhexyl]-5-[(4-oxo-2-pyrrolidin-1-ylpyrido[1,2-a]pyrimidin-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C24H30N4O2S2 |
|
—— |
2-[(5Z)-5-[[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid |
—— |
C22H24N4O4S2 |
|
—— |
(5Z)-5-[[2-[[(2S)-2-hydroxypropyl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(2-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C23H22N4O3S2 |
|
—— |
6-imino-13-methyl-2-oxo-N-[(1S)-1-phenylethyl]-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C24H25N5O2 |
|
—— |
(5Z)-3-[(2S)-butan-2-yl]-5-[[7-methyl-2-(4-methylpiperidin-1-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C23H28N4O2S2 |
|
—— |
7-[(2R)-butan-2-yl]-6-imino-13-methyl-2-oxo-N-(2-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C25H27N5O2 |
|
—— |
(5Z)-5-[[2-(1,3-benzodioxol-5-ylmethylamino)-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(2S)-butan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C25H24N4O4S2 |
|
—— |
(5Z)-3-ethyl-5-[[2-[[(2R)-1-hydroxybutan-2-yl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C18H20N4O3S2 |
|
—— |
(5Z)-5-[[2-[[(2R)-2-hydroxypropyl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(2-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C23H22N4O3S2 |
|
—— |
4-[(5Z)-5-[[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoic acid |
—— |
C23H26N4O5S2 |
|
—— |
6-imino-13-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C24H30N6O4 |
|
—— |
6-imino-13-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C27H30N6O3 |
|
—— |
(5Z)-3-[(2S)-butan-2-yl]-5-[[2-(3-morpholin-4-ylpropylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C23H29N5O3S2 |
|
—— |
(5Z)-3-[(2-chlorophenyl)methyl]-5-[[2-[[(2R)-1-hydroxybutan-2-yl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C23H21ClN4O3S2 |
|
—— |
6-imino-N-(3-methoxypropyl)-13-methyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C22H27N5O4 |
|
—— |
(5Z)-3-[(2S)-butan-2-yl]-5-[[7-methyl-2-(3-morpholin-4-ylpropylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C24H31N5O3S2 |
|
—— |
7-ethyl-6-imino-13-methyl-2-oxo-N-[(1R)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C23H23N5O2 |
|
—— |
4-[(5Z)-5-[[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoic acid |
—— |
C23H26N4O5S2 |
|
—— |
(5Z)-3-(3-methoxypropyl)-5-[[9-methyl-4-oxo-2-[[(1R)-1-phenylethyl]amino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C25H26N4O3S2 |
|
—— |
4-[(5Z)-5-[[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoic acid |
—— |
C23H26N4O5S2 |
|
—— |
6-imino-N,13-dimethyl-2-oxo-7-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C19H21N5O3 |
|
—— |
(5Z)-5-[[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(1R)-1-phenylethyl]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C26H26N4O3S2 |
|
—— |
(5Z)-5-[[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-fluorophenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C26H25FN4O2S2 |
|
—— |
(5Z)-5-[[7-methyl-4-oxo-2-[[(2R)-oxolan-2-yl]methylamino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-methylphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one |
—— |
C26H26N4O3S2 |
|
—— |
6-imino-N,13-dimethyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide |
—— |
C19H21N5O3 |
|