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吡啶并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-morpholin-4-yl-1-(2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)propan-1-one —— C19H29N5O2
(2R)-2-morpholin-4-yl-1-(2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)propan-1-one
—— (2R)-2-(3-methoxyphenoxy)-1-[(2S)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C22H28N4O3
(2R)-2-(3-methoxyphenoxy)-1-[(2S)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one
—— 7-acetyl-2-[(2R)-1-[(2S)-2-(3-fluorophenoxy)propanoyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H25FN4O4
7-acetyl-2-[(2R)-1-[(2S)-2-(3-fluorophenoxy)propanoyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2S)-1-[2-[(3S)-1-acetylpyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2-piperidin-1-ylpropan-1-one —— C21H31N5O2
(2S)-1-[2-[(3S)-1-acetylpyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2-piperidin-1-ylpropan-1-one
—— (2S)-2-(2-methoxyphenoxy)-1-[(2S)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C22H28N4O3
(2S)-2-(2-methoxyphenoxy)-1-[(2S)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one
—— (2R)-1-[2-[(2R)-1-acetylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2-piperidin-1-ylpropan-1-one —— C21H31N5O2
(2R)-1-[2-[(2R)-1-acetylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2-piperidin-1-ylpropan-1-one
—— 1-[(2R)-1-oxo-1-[4-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-2-yl]pyrrolidin-2-one —— C19H27N5O2
1-[(2R)-1-oxo-1-[4-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-2-yl]pyrrolidin-2-one
—— (2S)-1-[4-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-pyrrolidin-1-ylpropan-1-one —— C21H31N5O2
(2S)-1-[4-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-pyrrolidin-1-ylpropan-1-one
—— (2S)-2-(3-methoxyphenoxy)-1-[(3R)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C22H28N4O3
(2S)-2-(3-methoxyphenoxy)-1-[(3R)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2S)-2-morpholin-4-yl-1-(2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)propan-1-one —— C19H29N5O2
(2S)-2-morpholin-4-yl-1-(2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)propan-1-one
—— (2S)-2-(3-methoxyphenoxy)-1-[2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2S)-2-(3-methoxyphenoxy)-1-[2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2R)-2-(3-methoxyphenoxy)-1-[2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2R)-2-(3-methoxyphenoxy)-1-[2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— 1-[(2S)-1-[(3S)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]pyrrolidin-2-one —— C20H29N5O2
1-[(2S)-1-[(3S)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]pyrrolidin-2-one
—— (2S)-2-(3-fluorophenoxy)-1-[2-(1-methylpiperidin-4-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H27FN4O2
(2S)-2-(3-fluorophenoxy)-1-[2-(1-methylpiperidin-4-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-1-[2-[(2R)-1-acetylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2-piperidin-1-ylpropan-1-one —— C21H31N5O2
(2S)-1-[2-[(2R)-1-acetylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2-piperidin-1-ylpropan-1-one
—— (2S)-2-(2-methoxyphenoxy)-1-[2-[(2R)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2S)-2-(2-methoxyphenoxy)-1-[2-[(2R)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— 2-(dimethylamino)-7-[(3S)-1-[(2S)-2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl]-6H-pyrido[4,3-d]pyrimidin-5-one —— C21H28N6O3
2-(dimethylamino)-7-[(3S)-1-[(2S)-2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl]-6H-pyrido[4,3-d]pyrimidin-5-one
—— (2R)-1-[2-[(3S)-1-acetylpyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2-piperidin-1-ylpropan-1-one —— C21H31N5O2
(2R)-1-[2-[(3S)-1-acetylpyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2-piperidin-1-ylpropan-1-one
—— (2R)-2-(3-methoxyphenoxy)-1-[2-[(2S)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2R)-2-(3-methoxyphenoxy)-1-[2-[(2S)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2R)-2-(3-methoxyphenoxy)-1-[2-[(3R)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2R)-2-(3-methoxyphenoxy)-1-[2-[(3R)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-2-morpholin-4-yl-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C18H27N5O2
(2S)-2-morpholin-4-yl-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one
—— (2R)-2-(4-fluorophenoxy)-1-[2-(1-methylpiperidin-4-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H27FN4O2
(2R)-2-(4-fluorophenoxy)-1-[2-(1-methylpiperidin-4-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-2-(2-fluorophenoxy)-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C20H23FN4O2
(2S)-2-(2-fluorophenoxy)-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one
—— (2S)-2-(3-methoxyphenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2S)-2-(3-methoxyphenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-2-(3-methoxyphenoxy)-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C22H28N4O3
(2S)-2-(3-methoxyphenoxy)-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— 1-[(2R)-1-[(3R)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]pyrrolidin-2-one —— C20H29N5O2
1-[(2R)-1-[(3R)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]pyrrolidin-2-one
—— (2R)-2-(4-fluorophenoxy)-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C21H25FN4O2
(2R)-2-(4-fluorophenoxy)-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2S)-1-[(3R)-3-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-piperidin-1-ylpropan-1-one —— C21H31N5O2
(2S)-1-[(3R)-3-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-piperidin-1-ylpropan-1-one
—— 7-acetyl-2-[(2R)-1-[(2S)-2-(2-fluorophenoxy)propanoyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H25FN4O4
7-acetyl-2-[(2R)-1-[(2S)-2-(2-fluorophenoxy)propanoyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2S)-2-(3-fluorophenoxy)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C20H23FN4O2
(2S)-2-(3-fluorophenoxy)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one
—— (2R)-2-morpholin-4-yl-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C19H29N5O2
(2R)-2-morpholin-4-yl-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2R)-2-(4-fluorophenoxy)-1-[(2R)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C21H25FN4O2
(2R)-2-(4-fluorophenoxy)-1-[(2R)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one
—— (2R)-2-morpholin-4-yl-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C18H27N5O2
(2R)-2-morpholin-4-yl-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one
—— (2S)-2-(3-methoxyphenoxy)-1-[2-[(2R)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2S)-2-(3-methoxyphenoxy)-1-[2-[(2R)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-1-[(3R)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-morpholin-4-ylpropan-1-one —— C20H31N5O2
(2S)-1-[(3R)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-morpholin-4-ylpropan-1-one
—— (2S)-2-(4-fluorophenoxy)-1-[2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C21H25FN4O2
(2S)-2-(4-fluorophenoxy)-1-[2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2R)-2-(4-fluorophenoxy)-1-[(3R)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C21H25FN4O2
(2R)-2-(4-fluorophenoxy)-1-[(3R)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2R)-2-(3-methoxyphenoxy)-1-[2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2R)-2-(3-methoxyphenoxy)-1-[2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-2-(2-fluorophenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C21H25FN4O2
(2S)-2-(2-fluorophenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2R)-2-(3-methoxyphenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2R)-2-(3-methoxyphenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-2-(2-methoxyphenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H28N4O3
(2S)-2-(2-methoxyphenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-2-(4-fluorophenoxy)-1-[(3R)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C21H25FN4O2
(2S)-2-(4-fluorophenoxy)-1-[(3R)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2R)-2-(2-methoxyphenoxy)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C22H28N4O3
(2R)-2-(2-methoxyphenoxy)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2S)-2-(2-methoxyphenoxy)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C22H28N4O3
(2S)-2-(2-methoxyphenoxy)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2R)-2-(benzimidazol-1-yl)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C22H26N6O
(2R)-2-(benzimidazol-1-yl)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-2-(3-fluorophenoxy)-1-[2-[(3R)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C21H25FN4O2
(2S)-2-(3-fluorophenoxy)-1-[2-[(3R)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2R)-2-(2-fluorophenoxy)-1-[2-[(3R)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C21H25FN4O2
(2R)-2-(2-fluorophenoxy)-1-[2-[(3R)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— 2-(dimethylamino)-7-[(3R)-1-[(2R)-2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl]-6H-pyrido[4,3-d]pyrimidin-5-one —— C21H28N6O3
2-(dimethylamino)-7-[(3R)-1-[(2R)-2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl]-6H-pyrido[4,3-d]pyrimidin-5-one
—— (2R)-2-(3-fluorophenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C21H25FN4O2
(2R)-2-(3-fluorophenoxy)-1-[2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-2-(3-fluorophenoxy)-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C20H23FN4O2
(2S)-2-(3-fluorophenoxy)-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one