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吡啶并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-1-[(2S)-2-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H28N4O2
(2S)-1-[(2S)-2-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— (2R)-1-[4-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H30N4O
(2R)-1-[4-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— 7-(cyclopropanecarbonyl)-2-[(3R)-1-[(2R)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H30N4O3
7-(cyclopropanecarbonyl)-2-[(3R)-1-[(2R)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2S)-2-(4-methylphenyl)-1-[(3R)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C22H28N4O
(2S)-2-(4-methylphenyl)-1-[(3R)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2R)-1-[(3S)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H30N4O
(2R)-1-[(3S)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— (2S)-1-[(2R)-2-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H28N4O2
(2S)-1-[(2R)-2-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— (2R)-2-(4-methylphenyl)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C22H28N4O
(2R)-2-(4-methylphenyl)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2S)-1-[(3S)-3-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H28N4O2
(2S)-1-[(3S)-3-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— (2R)-2-(4-methylphenyl)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C21H26N4O
(2R)-2-(4-methylphenyl)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one
—— (2R)-2-(4-methylphenyl)-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C22H28N4O
(2R)-2-(4-methylphenyl)-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— 6-methyl-2-[(3R)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N4O2
6-methyl-2-[(3R)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 7-methyl-2-[1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O2
7-methyl-2-[1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2S)-1-[(3R)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H30N4O
(2S)-1-[(3R)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— (2R)-2-(4-methylphenyl)-1-[2-[(2S)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one —— C23H30N4O
(2R)-2-(4-methylphenyl)-1-[2-[(2S)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
—— (2S)-1-[(2R)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H30N4O
(2S)-1-[(2R)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— (2R)-1-[(3R)-3-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H28N4O2
(2R)-1-[(3R)-3-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— 1-[(3S)-3-[6-[(2-hydroxy-5-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone —— C22H28N4O2
1-[(3S)-3-[6-[(2-hydroxy-5-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone
—— 1-[(2S)-2-[6-[(2-methoxy-4-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone —— C23H30N4O2
1-[(2S)-2-[6-[(2-methoxy-4-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone
—— 6-methyl-2-[(3R)-1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N4O2
6-methyl-2-[(3R)-1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 7-acetyl-2-[(3S)-1-[(2R)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H28N4O3
7-acetyl-2-[(3S)-1-[(2R)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-(2-methoxy-4-methylphenoxy)-1-[2-[(2R)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]ethanone —— C22H28N4O3
2-(2-methoxy-4-methylphenoxy)-1-[2-[(2R)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]ethanone
—— 1-[(2R)-2-[6-[(2-methoxy-4-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone —— C23H30N4O2
1-[(2R)-2-[6-[(2-methoxy-4-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone
—— 2-(2-methoxy-4-methylphenoxy)-1-[2-[(2S)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]ethanone —— C22H28N4O3
2-(2-methoxy-4-methylphenoxy)-1-[2-[(2S)-1-methylpyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]ethanone
—— (2S)-2-(4-methylphenyl)-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C22H28N4O
(2S)-2-(4-methylphenyl)-1-[(3S)-3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— 7-(cyclopropanecarbonyl)-2-[(3S)-1-[(2S)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H30N4O3
7-(cyclopropanecarbonyl)-2-[(3S)-1-[(2S)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2S)-1-[(3S)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H30N4O
(2S)-1-[(3S)-3-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— 6-methyl-2-[(3S)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N4O2
6-methyl-2-[(3S)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (2R)-1-[(2R)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H30N4O
(2R)-1-[(2R)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]-2-(4-methylphenyl)propan-1-one
—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C26H32N4O3
7-(cyclopropanecarbonyl)-2-[(2R)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-acetyl-2-[(3R)-1-[(2S)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H28N4O3
7-acetyl-2-[(3R)-1-[(2S)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2R)-2-(4-methylphenyl)-1-[4-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one —— C22H28N4O
(2R)-2-(4-methylphenyl)-1-[4-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]propan-1-one
—— (2R)-2-(4-methylphenyl)-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one —— C21H26N4O
(2R)-2-(4-methylphenyl)-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]propan-1-one
—— 7-methyl-2-[1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O2
7-methyl-2-[1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-(2-methoxy-4-methylphenoxy)-1-[(2S)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]ethanone —— C22H28N4O3
2-(2-methoxy-4-methylphenoxy)-1-[(2S)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]ethanone
—— 7-cyclohexyl-2-[(3R)-1-[(2R)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C27H36N4O2
7-cyclohexyl-2-[(3R)-1-[(2R)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 6-[(2-methoxy-4-methylphenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H26N4O
6-[(2-methoxy-4-methylphenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 2-[1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-7-propan-2-yl-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H34N4O2
2-[1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-7-propan-2-yl-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 6-[(2-methoxy-4-methylphenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H26N4O
6-[(2-methoxy-4-methylphenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H32N4O3
7-(cyclobutanecarbonyl)-2-[(3R)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-acetyl-2-[(3S)-1-[(2S)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H28N4O3
7-acetyl-2-[(3S)-1-[(2S)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-(2-methoxy-4-methylphenoxy)-1-[(2R)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]ethanone —— C22H28N4O3
2-(2-methoxy-4-methylphenoxy)-1-[(2R)-2-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]ethanone
—— 1-[(3R)-3-[6-[(2-hydroxy-5-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone —— C22H28N4O2
1-[(3R)-3-[6-[(2-hydroxy-5-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone
—— 7-cyclohexyl-2-[(3S)-1-[(2R)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C27H36N4O2
7-cyclohexyl-2-[(3S)-1-[(2R)-2-(4-methylphenyl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H32N4O3
7-(cyclobutanecarbonyl)-2-[(3S)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-(2-methoxy-4-methylphenoxy)-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]ethanone —— C22H28N4O3
2-(2-methoxy-4-methylphenoxy)-1-[(2R)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]ethanone
—— 2-(2-methoxy-4-methylphenoxy)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]ethanone —— C22H28N4O3
2-(2-methoxy-4-methylphenoxy)-1-[(2S)-2-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)piperidin-1-yl]ethanone
—— 1-[4-[6-[(2-hydroxy-5-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone —— C22H28N4O2
1-[4-[6-[(2-hydroxy-5-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone
—— 2-[1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-7-propan-2-yl-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H34N4O2
2-[1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-7-propan-2-yl-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 1-[(2S)-2-[6-[(2-hydroxy-5-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone —— C22H28N4O2
1-[(2S)-2-[6-[(2-hydroxy-5-methylphenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]piperidin-1-yl]ethanone
—— (2S)-1-[(3R)-3-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one —— C23H28N4O2
(2S)-1-[(3R)-3-(6-acetyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl)pyrrolidin-1-yl]-2-(4-methylphenyl)propan-1-one