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异吲哚及其衍生物

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R,4S)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-(2-hydroxyethoxy)ethoxy]-4-propan-2-yl-3,4-dihydro-2H-pyran-6-carboxamide —— C28H31ClN2O7
(2R,4S)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-(2-hydroxyethoxy)ethoxy]-4-propan-2-yl-3,4-dihydro-2H-pyran-6-carboxamide
—— methyl 4-[(2R,4R)-6-[[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]carbamoyl]-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C33H31ClN2O9
methyl 4-[(2R,4R)-6-[[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]carbamoyl]-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— (2R,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-(2-hydroxyethoxy)ethoxy]-4-phenyl-3,4-dihydro-2H-pyran-6-carboxamide —— C31H29ClN2O7
(2R,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-(2-hydroxyethoxy)ethoxy]-4-phenyl-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-4-(1,3-benzodioxol-5-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide —— C32H29ClN2O8
(2R,4R)-4-(1,3-benzodioxol-5-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-4-phenyl-3,4-dihydro-2H-pyran-6-carboxamide —— C31H29ClN2O6
(2R,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-4-phenyl-3,4-dihydro-2H-pyran-6-carboxamide
—— methyl 4-[(2R,4R)-6-[[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]carbamoyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C33H31ClN2O8
methyl 4-[(2R,4R)-6-[[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]carbamoyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— (2S,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-(2-hydroxyethoxy)ethoxy]-4-propan-2-yl-3,4-dihydro-2H-pyran-6-carboxamide —— C28H31ClN2O7
(2S,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-(2-hydroxyethoxy)ethoxy]-4-propan-2-yl-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,3R,4S)-4-(1,3-benzodioxol-5-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxamide —— C33H31ClN2O8
(2R,3R,4S)-4-(1,3-benzodioxol-5-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-4-propan-2-yl-3,4-dihydro-2H-pyran-6-carboxamide —— C28H31ClN2O6
(2S,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-4-propan-2-yl-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide —— C35H32ClN3O7
(2R,4R)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S,4S)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[[4-(hydroxymethyl)phenyl]methoxy]-4-thiophen-3-yl-3,4-dihydro-2H-pyran-6-carboxamide —— C33H27ClN2O6S
(2S,4S)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[[4-(hydroxymethyl)phenyl]methoxy]-4-thiophen-3-yl-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[[4-(hydroxymethyl)phenyl]methoxy]-4-thiophen-3-yl-3,4-dihydro-2H-pyran-6-carboxamide —— C33H27ClN2O6S
(2R,4R)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[[4-(hydroxymethyl)phenyl]methoxy]-4-thiophen-3-yl-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-4-(1-benzofuran-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide —— C33H29ClN2O7
(2R,4R)-4-(1-benzofuran-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide
—— (3R)-1-(2-methyl-1,3-dioxoisoindol-5-yl)-5-oxopyrrolidine-3-carboxamide —— C14H13N3O4
(3R)-1-(2-methyl-1,3-dioxoisoindol-5-yl)-5-oxopyrrolidine-3-carboxamide
—— (2R,4R)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamide —— C39H32ClN3O7
(2R,4R)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamide
—— (3R)-1-(2-methyl-1,3-dioxoisoindol-5-yl)-5-oxopyrrolidine-3-carbonyl chloride —— C14H11ClN2O4
(3R)-1-(2-methyl-1,3-dioxoisoindol-5-yl)-5-oxopyrrolidine-3-carbonyl chloride
—— (2R,4S)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-4-propan-2-yl-3,4-dihydro-2H-pyran-6-carboxamide —— C28H31ClN2O6
(2R,4S)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-(4-hydroxybutoxy)-4-propan-2-yl-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S,4S)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamide —— C39H32ClN3O7
(2S,4S)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S,4S)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide —— C42H39ClN4O10S
(2S,4S)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S,3R,4R)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C39H40ClN3O9
(2S,3R,4R)-4-(1-acetylindol-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-4-(1,3-benzodioxol-5-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide —— C32H29ClN2O9
(2R,4R)-4-(1,3-benzodioxol-5-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-4-(1-benzofuran-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide —— C40H36ClN3O10S
(2R,4R)-4-(1-benzofuran-3-yl)-N-[4-(5-chloro-1,3-dioxoisoindol-2-yl)-3-methylphenyl]-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide
—— N-cyclopropyl-N-[(1R)-1-(2-fluorophenyl)ethyl]-3-(5-methyl-1,3-dioxoisoindol-2-yl)propanamide —— C23H23FN2O3
N-cyclopropyl-N-[(1R)-1-(2-fluorophenyl)ethyl]-3-(5-methyl-1,3-dioxoisoindol-2-yl)propanamide
—— 2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]acetamide —— C20H26N2O5
2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]acetamide
—— (1R,2S,6S,7S)-4-[2-oxo-2-[(3S)-3-(5-pyridin-4-ylpyrimidin-4-yl)piperidin-1-yl]ethyl]-4-azatricyclo[5.2.1.02,6]decane-3,5-dione —— C25H27N5O3
(1R,2S,6S,7S)-4-[2-oxo-2-[(3S)-3-(5-pyridin-4-ylpyrimidin-4-yl)piperidin-1-yl]ethyl]-4-azatricyclo[5.2.1.02,6]decane-3,5-dione
—— (3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C40H37ClN4O6S
(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— methyl (3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxylate —— C39H33ClN4O8S
methyl (3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxylate
—— 3-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[(4-ethoxyphenyl)methyl]-N-methylpropanamide —— C21H28N2O4
3-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[(4-ethoxyphenyl)methyl]-N-methylpropanamide
—— (3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-hydroxy-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C37H31ClN4O7S
(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-hydroxy-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 3-[(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]propanoic acid —— C40H35ClN4O8S
3-[(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]propanoic acid
—— (3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C44H35Cl2F3N6O6S
(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-ethyl-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C39H35ClN4O6S
(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-ethyl-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 4-[(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]butanoic acid —— C41H37ClN4O8S
4-[(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]butanoic acid
—— 6-[(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid —— C43H41ClN4O8S
6-[(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid
—— (3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-2-[2-(4-hydroxyphenyl)ethyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C45H39ClN4O7S
(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(6-hydroxy-4H-chromen-3-yl)-2-[2-(4-hydroxyphenyl)ethyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-cyclohexyl-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C42H43ClN4O6S
(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-cyclohexyl-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-2,6a-dimethyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C37H35ClN4O6S
(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-2,6a-dimethyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-ethyl-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C38H37ClN4O6S
(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-ethyl-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C36H33ClN4O6S
(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-hydroxy-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C36H33ClN4O7S
(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-hydroxy-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6S,6aS,9aR,10aS,10bR)-2-tert-butyl-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C40H41ClN4O6S
(3aS,6S,6aS,9aR,10aS,10bR)-2-tert-butyl-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6S,6aS,9aR,10aS,10bR)-2-benzyl-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C43H39ClN4O6S
(3aS,6S,6aS,9aR,10aS,10bR)-2-benzyl-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-2-(thiophen-2-ylmethyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C41H37ClN4O6S2
(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-2-(thiophen-2-ylmethyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 3-[(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]propanoic acid —— C39H37ClN4O8S
3-[(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]propanoic acid
—— (3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-2-[2-(4-hydroxyphenyl)ethyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C44H41ClN4O7S
(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[4-(2-hydroxyethoxy)phenyl]-2-[2-(4-hydroxyphenyl)ethyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C43H37Cl2F3N6O6S
(3aS,6S,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-[4-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-[2-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C43H37Cl2F3N6O6S
(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-[2-(2-hydroxyethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (2S)-N-cyclopropyl-2-(1,3-dioxoisoindol-2-yl)-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide —— C22H19F3N2O3
(2S)-N-cyclopropyl-2-(1,3-dioxoisoindol-2-yl)-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide
—— N-[(1R)-1-(2,5-difluorophenyl)ethyl]-N-methyl-2-(1-methylidene-3-oxoisoindol-2-yl)acetamide —— C20H18F2N2O2
N-[(1R)-1-(2,5-difluorophenyl)ethyl]-N-methyl-2-(1-methylidene-3-oxoisoindol-2-yl)acetamide
—— (3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[2-(2-hydroxyethoxy)phenyl]-6a-methyl-2-(thiophen-2-ylmethyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C41H37ClN4O6S2
(3aS,6R,6aS,9aR,10aS,10bR)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[2-(2-hydroxyethoxy)phenyl]-6a-methyl-2-(thiophen-2-ylmethyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone