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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4R)-6-amino-4-(6-chloro-1,3-benzodioxol-5-yl)-3-(2,4-dimethylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C22H17ClN4O3
(4R)-6-amino-4-(6-chloro-1,3-benzodioxol-5-yl)-3-(2,4-dimethylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4R)-6-amino-3-(2-chlorophenyl)-4-(4-cyclopentyloxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C24H21ClN4O2
(4R)-6-amino-3-(2-chlorophenyl)-4-(4-cyclopentyloxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4S)-6-amino-4-(4-cyclopentyloxyphenyl)-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C24H21FN4O2
(4S)-6-amino-4-(4-cyclopentyloxyphenyl)-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4R)-6-amino-4-(4-methoxynaphthalen-1-yl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C25H20N4O3
(4R)-6-amino-4-(4-methoxynaphthalen-1-yl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4S)-6-amino-3-(4-fluorophenyl)-4-(4-hydroxy-3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C20H15FN4O3
(4S)-6-amino-3-(4-fluorophenyl)-4-(4-hydroxy-3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4S)-6-amino-4-(4-cyclopentyloxyphenyl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C25H24N4O3
(4S)-6-amino-4-(4-cyclopentyloxyphenyl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4R)-6-amino-4-(3,5-dimethoxyphenyl)-3-(2,4-dimethylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C23H22N4O3
(4R)-6-amino-4-(3,5-dimethoxyphenyl)-3-(2,4-dimethylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (Z)-1-(azetidin-1-yl)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)prop-2-en-1-one —— C16H16ClN3O
(Z)-1-(azetidin-1-yl)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (4S)-6-amino-4-(4-cyclopentyloxy-3-methoxyphenyl)-3-(2,4-dimethylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C27H28N4O3
(4S)-6-amino-4-(4-cyclopentyloxy-3-methoxyphenyl)-3-(2,4-dimethylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 1-[(3S,3aR)-3-(4-fluorophenyl)-3,3a,4,5-tetrahydrobenzo[g]indazol-2-yl]-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C31H24FN5O2S
1-[(3S,3aR)-3-(4-fluorophenyl)-3,3a,4,5-tetrahydrobenzo[g]indazol-2-yl]-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— (4R)-6-amino-4-(4-cyclopentyloxy-3-methoxyphenyl)-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C25H23FN4O3
(4R)-6-amino-4-(4-cyclopentyloxy-3-methoxyphenyl)-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4R)-6-amino-4-(6-chloro-1,3-benzodioxol-5-yl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C21H15ClN4O4
(4R)-6-amino-4-(6-chloro-1,3-benzodioxol-5-yl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (Z)-3-[1-benzyl-3-(4-ethylphenyl)pyrazol-4-yl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methylprop-2-enamide —— C26H29N3O3S
(Z)-3-[1-benzyl-3-(4-ethylphenyl)pyrazol-4-yl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methylprop-2-enamide
—— (Z)-3-[1-benzyl-3-(4-ethylphenyl)pyrazol-4-yl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-methylprop-2-enamide —— C26H29N3O3S
(Z)-3-[1-benzyl-3-(4-ethylphenyl)pyrazol-4-yl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-methylprop-2-enamide
—— (4R)-6-amino-3-(4-methoxyphenyl)-4-(2-propan-2-yloxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C23H22N4O3
(4R)-6-amino-3-(4-methoxyphenyl)-4-(2-propan-2-yloxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4S)-6-amino-4-(5-bromothiophen-2-yl)-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C17H10BrFN4OS
(4S)-6-amino-4-(5-bromothiophen-2-yl)-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4S)-6-amino-3-(2-chlorophenyl)-4-(4-hydroxy-3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C20H15ClN4O3
(4S)-6-amino-3-(2-chlorophenyl)-4-(4-hydroxy-3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (Z)-1-(azetidin-1-yl)-3-[1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]prop-2-en-1-one —— C23H23N3O2
(Z)-1-(azetidin-1-yl)-3-[1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]prop-2-en-1-one
—— (4S)-6-amino-3-(2,4-dimethylphenyl)-4-(4-methoxynaphthalen-1-yl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C26H22N4O2
(4S)-6-amino-3-(2,4-dimethylphenyl)-4-(4-methoxynaphthalen-1-yl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (Z)-1-(azetidin-1-yl)-3-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]prop-2-en-1-one —— C23H23N3O
(Z)-1-(azetidin-1-yl)-3-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]prop-2-en-1-one
—— (4S)-6-amino-3-(4-methoxyphenyl)-4-quinolin-4-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C23H17N5O2
(4S)-6-amino-3-(4-methoxyphenyl)-4-quinolin-4-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (Z)-N-[(3S)-1-benzylpyrrolidin-3-yl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C23H24N4O
(Z)-N-[(3S)-1-benzylpyrrolidin-3-yl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (Z)-3-[1-benzyl-3-(3,4-dimethylphenyl)pyrazol-4-yl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methylprop-2-enamide —— C26H29N3O3S
(Z)-3-[1-benzyl-3-(3,4-dimethylphenyl)pyrazol-4-yl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methylprop-2-enamide
—— (Z)-1-[4-(4-fluorophenyl)sulfonyl-1,4-diazepan-1-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one —— C23H23FN4O3S
(Z)-1-[4-(4-fluorophenyl)sulfonyl-1,4-diazepan-1-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-1-(azetidin-1-yl)-3-[1-[(4-methylphenyl)methyl]-3-phenylpyrazol-4-yl]prop-2-en-1-one —— C23H23N3O
(Z)-1-(azetidin-1-yl)-3-[1-[(4-methylphenyl)methyl]-3-phenylpyrazol-4-yl]prop-2-en-1-one
—— (Z)-3-[1-[(2-chlorophenyl)methyl]-3-phenylpyrazol-4-yl]-N-(2-morpholin-4-ylethyl)prop-2-enamide —— C25H27ClN4O2
(Z)-3-[1-[(2-chlorophenyl)methyl]-3-phenylpyrazol-4-yl]-N-(2-morpholin-4-ylethyl)prop-2-enamide
—— (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-[4-(4-fluorophenyl)sulfonyl-1,4-diazepan-1-yl]prop-2-en-1-one —— C25H27FN4O3S
(Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-[4-(4-fluorophenyl)sulfonyl-1,4-diazepan-1-yl]prop-2-en-1-one
—— (Z)-N-[(1-benzylpyrazol-4-yl)methyl]-N-methyl-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C24H23N5O
(Z)-N-[(1-benzylpyrazol-4-yl)methyl]-N-methyl-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (8R)-3-(4-chlorophenyl)-2-methyl-8-[(Z)-2-phenylethenyl]-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one —— C25H20ClN3O
(8R)-3-(4-chlorophenyl)-2-methyl-8-[(Z)-2-phenylethenyl]-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one
—— (Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-1-(5-methylfuran-2-yl)prop-2-en-1-one —— C18H14ClFN2O2
(Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-1-(5-methylfuran-2-yl)prop-2-en-1-one
—— 2-[[5-(4-chlorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-hydroxy-4-methylphenyl)acetamide —— C20H19ClN4O2S
2-[[5-(4-chlorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-hydroxy-4-methylphenyl)acetamide
—— (8S)-3-(4-chlorophenyl)-2-methyl-8-[(Z)-2-phenylethenyl]-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one —— C25H20ClN3O
(8S)-3-(4-chlorophenyl)-2-methyl-8-[(Z)-2-phenylethenyl]-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one
—— (8R)-2-methyl-3-phenyl-8-[(Z)-2-phenylethenyl]-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one —— C25H21N3O
(8R)-2-methyl-3-phenyl-8-[(Z)-2-phenylethenyl]-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one
—— 2-[methyl-[(1-phenylpyrazol-4-yl)methyl]amino]-1-[4-[(Z)-2-phenylethenyl]sulfonylpiperazin-1-yl]ethanone —— C25H29N5O3S
2-[methyl-[(1-phenylpyrazol-4-yl)methyl]amino]-1-[4-[(Z)-2-phenylethenyl]sulfonylpiperazin-1-yl]ethanone
—— (6E)-3-(4-chlorophenyl)-6-[(3,4-dimethoxyphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C19H14ClN3O3S
(6E)-3-(4-chlorophenyl)-6-[(3,4-dimethoxyphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— (8S)-2-methyl-3-phenyl-8-[(Z)-2-phenylethenyl]-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one —— C25H21N3O
(8S)-2-methyl-3-phenyl-8-[(Z)-2-phenylethenyl]-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one
—— (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]prop-2-enamide —— C18H21N3O3S
(Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]prop-2-enamide
—— ethyl 2-[(Z)-2-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)ethenyl]-5-nitropyridine-3-carboxylate —— C20H17ClN4O4
ethyl 2-[(Z)-2-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)ethenyl]-5-nitropyridine-3-carboxylate
—— (Z)-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C24H26N4O2
(Z)-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]prop-2-enamide —— C18H21N3O3S
(Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]prop-2-enamide
—— (Z)-1-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one —— C25H24N4O4
(Z)-1-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-3-(1-phenylpyrazol-4-yl)-1-[(4R)-4-thiophen-2-yl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]prop-2-en-1-one —— C23H19N3OS2
(Z)-3-(1-phenylpyrazol-4-yl)-1-[(4R)-4-thiophen-2-yl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]prop-2-en-1-one
—— (Z)-N-[(1R)-2-morpholin-4-yl-1-phenylethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C24H26N4O2
(Z)-N-[(1R)-2-morpholin-4-yl-1-phenylethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— ethyl 2-[(Z)-2-[1-(2-cyanoethyl)-3-(3,4-dimethoxyphenyl)pyrazol-4-yl]ethenyl]-5-nitropyridine-3-carboxylate —— C24H23N5O6
ethyl 2-[(Z)-2-[1-(2-cyanoethyl)-3-(3,4-dimethoxyphenyl)pyrazol-4-yl]ethenyl]-5-nitropyridine-3-carboxylate
—— (Z)-1-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one —— C25H24N4O4
(Z)-1-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-1-[4-(5-methylthiophen-2-yl)sulfonylpiperazin-1-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one —— C21H22N4O3S2
(Z)-1-[4-(5-methylthiophen-2-yl)sulfonylpiperazin-1-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-3-(1-phenylpyrazol-4-yl)-1-[(4S)-4-thiophen-2-yl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]prop-2-en-1-one —— C23H19N3OS2
(Z)-3-(1-phenylpyrazol-4-yl)-1-[(4S)-4-thiophen-2-yl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]prop-2-en-1-one
—— (5Z)-5-[(1-phenylpyrazol-4-yl)methylene]thiazolidine-2,4-dione —— C13H9N3O2S
(5Z)-5-[(1-phenylpyrazol-4-yl)methylene]thiazolidine-2,4-dione
—— (Z)-3-(furan-2-yl)-N-[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]prop-2-enamide —— C16H14N4O3
(Z)-3-(furan-2-yl)-N-[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]prop-2-enamide
—— (Z)-N-[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]-3-thiophen-2-ylprop-2-enamide —— C16H14N4O2S
(Z)-N-[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]-3-thiophen-2-ylprop-2-enamide