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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-methyl-4-(methylsulfonylmethyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide —— C20H22N4O3S
N-methyl-4-(methylsulfonylmethyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide
—— 3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[(2R)-piperidin-2-yl]-1,2,4-oxadiazole —— C12H16N4O2
3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[(2R)-piperidin-2-yl]-1,2,4-oxadiazole
—— 2-(5-methyl-1H-pyrazol-3-yl)-4-piperidin-4-yl-1,3-thiazole —— C12H16N4S
2-(5-methyl-1H-pyrazol-3-yl)-4-piperidin-4-yl-1,3-thiazole
—— 3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(3S)-pyrrolidin-3-yl]methyl]-1,2,4-oxadiazole —— C12H16N4O2
3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(3S)-pyrrolidin-3-yl]methyl]-1,2,4-oxadiazole
—— 3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[(3S)-piperidin-3-yl]-1,2,4-oxadiazole —— C12H16N4O2
3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[(3S)-piperidin-3-yl]-1,2,4-oxadiazole
—— N-(4-methylphenyl)-2-[2-[methyl-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]-2-oxoethyl]sulfanylacetamide —— C22H25N5O2S
N-(4-methylphenyl)-2-[2-[methyl-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]-2-oxoethyl]sulfanylacetamide
—— 3-(2-ethoxyphenyl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide —— C22H26N4O2
3-(2-ethoxyphenyl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide
—— N-methyl-3-(2-methylpropoxy)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide —— C22H26N4O2
N-methyl-3-(2-methylpropoxy)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide
—— 2-(4-methyl-1,3-oxazol-5-yl)-5-[[(3R)-piperidin-3-yl]methyl]-1,3,4-oxadiazole —— C12H16N4O2
2-(4-methyl-1,3-oxazol-5-yl)-5-[[(3R)-piperidin-3-yl]methyl]-1,3,4-oxadiazole
—— 2-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(2S)-pyrrolidin-2-yl]methyl]-1,3,4-oxadiazole —— C12H16N4O2
2-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(2S)-pyrrolidin-2-yl]methyl]-1,3,4-oxadiazole
—— N-(5-methyl-1,2-oxazol-3-yl)-2-[2-[methyl-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]-2-oxoethyl]sulfanylacetamide —— C19H22N6O3S
N-(5-methyl-1,2-oxazol-3-yl)-2-[2-[methyl-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]-2-oxoethyl]sulfanylacetamide
—— N-methyl-2-(thiophen-2-ylmethylsulfanyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C18H20N4OS2
N-methyl-2-(thiophen-2-ylmethylsulfanyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— tert-butyl 4-[methyl-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]carbamoyl]piperidine-1-carboxylate —— C22H31N5O3
tert-butyl 4-[methyl-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]carbamoyl]piperidine-1-carboxylate
—— 5-(2,4-dimethyl-1,3-oxazol-5-yl)-3-[[(3R)-pyrrolidin-3-yl]methyl]-1,2,4-oxadiazole —— C12H16N4O2
5-(2,4-dimethyl-1,3-oxazol-5-yl)-3-[[(3R)-pyrrolidin-3-yl]methyl]-1,2,4-oxadiazole
—— N-methyl-4-(methylsulfonylmethyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide —— C20H22N4O3S
N-methyl-4-(methylsulfonylmethyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide
—— 2-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[(2R)-piperidin-2-yl]-1,3,4-oxadiazole —— C12H16N4O2
2-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[(2R)-piperidin-2-yl]-1,3,4-oxadiazole
—— (1S)-3-methyl-1-(2-pyridin-4-yl-1,3-thiazol-4-yl)butan-1-amine —— C13H17N3S
(1S)-3-methyl-1-(2-pyridin-4-yl-1,3-thiazol-4-yl)butan-1-amine
—— 5-(4-methyl-1,3-oxazol-5-yl)-3-[[(3R)-piperidin-3-yl]methyl]-1,2,4-oxadiazole —— C12H16N4O2
5-(4-methyl-1,3-oxazol-5-yl)-3-[[(3R)-piperidin-3-yl]methyl]-1,2,4-oxadiazole
—— 2-(4-fluorophenoxy)-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C19H19FN4O2
2-(4-fluorophenoxy)-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— 2-(2,3-dihydro-1H-inden-5-yl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C22H24N4O
2-(2,3-dihydro-1H-inden-5-yl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— N-methyl-2-naphthalen-2-yl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C23H22N4O
N-methyl-2-naphthalen-2-yl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— 5-(2-fluorophenyl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]furan-2-carboxamide —— C22H19FN4O2
5-(2-fluorophenyl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]furan-2-carboxamide
—— 3-(4-methyl-1,3-oxazol-5-yl)-5-[[(2R)-piperidin-2-yl]methyl]-1,2,4-oxadiazole —— C12H16N4O2
3-(4-methyl-1,3-oxazol-5-yl)-5-[[(2R)-piperidin-2-yl]methyl]-1,2,4-oxadiazole
—— 2-[(3-chlorophenyl)methylsulfanyl]-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C20H21ClN4OS
2-[(3-chlorophenyl)methylsulfanyl]-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— 2-[(1S)-cyclopent-2-en-1-yl]-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C18H22N4O
2-[(1S)-cyclopent-2-en-1-yl]-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— 7-chloro-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1,3-benzodioxole-5-carboxamide —— C19H17ClN4O3
7-chloro-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1,3-benzodioxole-5-carboxamide
—— (1R)-3-methyl-1-(2-pyridin-4-yl-1,3-thiazol-4-yl)butan-1-amine —— C13H17N3S
(1R)-3-methyl-1-(2-pyridin-4-yl-1,3-thiazol-4-yl)butan-1-amine
—— 2-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C17H22N4O3S
2-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— N-methyl-3-(2-methylpropoxy)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide —— C22H26N4O2
N-methyl-3-(2-methylpropoxy)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide
—— 2-(4-methyl-1,3-oxazol-5-yl)-5-(piperidin-4-ylmethyl)-1,3,4-oxadiazole —— C12H16N4O2
2-(4-methyl-1,3-oxazol-5-yl)-5-(piperidin-4-ylmethyl)-1,3,4-oxadiazole
—— 2-(4-ethoxyphenyl)sulfanyl-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C21H24N4O2S
2-(4-ethoxyphenyl)sulfanyl-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— 3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(2S)-pyrrolidin-2-yl]methyl]-1,2,4-oxadiazole —— C12H16N4O2
3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(2S)-pyrrolidin-2-yl]methyl]-1,2,4-oxadiazole
—— N-methyl-2-(thiophen-2-ylmethylsulfanyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C18H20N4OS2
N-methyl-2-(thiophen-2-ylmethylsulfanyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— 5-(4-methyl-1,3-oxazol-5-yl)-3-[2-[(2S)-pyrrolidin-2-yl]ethyl]-1,2,4-oxadiazole —— C12H16N4O2
5-(4-methyl-1,3-oxazol-5-yl)-3-[2-[(2S)-pyrrolidin-2-yl]ethyl]-1,2,4-oxadiazole
—— 3-(2,5-dioxopyrrolidin-1-yl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide —— C18H21N5O3
3-(2,5-dioxopyrrolidin-1-yl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide
—— 3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide —— C21H24N8O
3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide
—— 2-(4-methyl-1,3-oxazol-5-yl)-5-[2-[(3S)-pyrrolidin-3-yl]ethyl]-1,3,4-oxadiazole —— C12H16N4O2
2-(4-methyl-1,3-oxazol-5-yl)-5-[2-[(3S)-pyrrolidin-3-yl]ethyl]-1,3,4-oxadiazole
—— 5-[[(2S)-piperidin-2-yl]methyl]-2-thiophen-2-yl-1,3-oxazole —— C13H16N2OS
5-[[(2S)-piperidin-2-yl]methyl]-2-thiophen-2-yl-1,3-oxazole
—— 7-chloro-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1,3-benzodioxole-5-carboxamide —— C19H17ClN4O3
7-chloro-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1,3-benzodioxole-5-carboxamide
—— (E)-N-methyl-3-(5-methylthiophen-2-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide —— C19H20N4OS
(E)-N-methyl-3-(5-methylthiophen-2-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide
—— 2-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(3S)-pyrrolidin-3-yl]methyl]-1,3,4-oxadiazole —— C12H16N4O2
2-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(3S)-pyrrolidin-3-yl]methyl]-1,3,4-oxadiazole
—— N-methyl-2-(2-methylphenyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C20H22N4O
N-methyl-2-(2-methylphenyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— (1S)-1-[2-(4-fluorophenyl)-1,3-oxazol-5-yl]-3-methylbutan-1-amine —— C14H17FN2O
(1S)-1-[2-(4-fluorophenyl)-1,3-oxazol-5-yl]-3-methylbutan-1-amine
—— 5-chloro-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiophene-2-carboxamide —— C16H15ClN4OS
5-chloro-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiophene-2-carboxamide
—— (E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide —— C22H27ClN6O
(E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide
—— 3-(2-ethoxyphenyl)-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide —— C22H26N4O2
3-(2-ethoxyphenyl)-N-methyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide
—— 3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(3R)-pyrrolidin-3-yl]methyl]-1,2,4-oxadiazole —— C12H16N4O2
3-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(3R)-pyrrolidin-3-yl]methyl]-1,2,4-oxadiazole
—— 5-(2,4-dimethyl-1,3-oxazol-5-yl)-3-[[(2R)-pyrrolidin-2-yl]methyl]-1,2,4-oxadiazole —— C12H16N4O2
5-(2,4-dimethyl-1,3-oxazol-5-yl)-3-[[(2R)-pyrrolidin-2-yl]methyl]-1,2,4-oxadiazole
—— 2-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(2R)-pyrrolidin-2-yl]methyl]-1,3,4-oxadiazole —— C12H16N4O2
2-(2,4-dimethyl-1,3-oxazol-5-yl)-5-[[(2R)-pyrrolidin-2-yl]methyl]-1,3,4-oxadiazole
—— 5-(4-methyl-1,3-oxazol-5-yl)-3-[2-[(3R)-pyrrolidin-3-yl]ethyl]-1,2,4-oxadiazole —— C12H16N4O2
5-(4-methyl-1,3-oxazol-5-yl)-3-[2-[(3R)-pyrrolidin-3-yl]ethyl]-1,2,4-oxadiazole