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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4-(6-(4-aminopiperidin-1-yl)pyridin-3-ylamino)-6-(3,5-dichloro-4-hydroxyphenyl)quinolin-3-yl)(cyclopropyl)methanone 1356946-65-0 C29H27Cl2N5O2
(4-(6-(4-aminopiperidin-1-yl)pyridin-3-ylamino)-6-(3,5-dichloro-4-hydroxyphenyl)quinolin-3-yl)(cyclopropyl)methanone
—— methyl 6-(4-chloro-3-[3-(dimethylamino)propoxy]phenyl)-5-(2-oxopyrrolidin-1-yl)pyridine-2-carboxylate 1007170-32-2 C22H26ClN3O4
methyl 6-(4-chloro-3-[3-(dimethylamino)propoxy]phenyl)-5-(2-oxopyrrolidin-1-yl)pyridine-2-carboxylate
—— cyclopropyl {6-(3,5-dichloro-4-hydroxyphenyl)-4-[6-(pyrrolidin-1-ylmethyl)pyridin-3-ylamino]quinolin-3-yl}methanone 1356948-03-2 C29H26Cl2N4O2
cyclopropyl {6-(3,5-dichloro-4-hydroxyphenyl)-4-[6-(pyrrolidin-1-ylmethyl)pyridin-3-ylamino]quinolin-3-yl}methanone
—— tert-butyl (3-(1-allylcyclopropanesulfonamido)-1,5-dimethyl-6-oxo-1,6-dihydropyridin-2-yl)(2-fluoro-4-iodophenyl)carbamate 1246443-05-9 C24H29FIN3O5S
tert-butyl (3-(1-allylcyclopropanesulfonamido)-1,5-dimethyl-6-oxo-1,6-dihydropyridin-2-yl)(2-fluoro-4-iodophenyl)carbamate
—— 4-(m-tolylamino)benzaldehyde 1329601-50-4 C14H13NO
4-(m-tolylamino)benzaldehyde
—— 2-(3-Phenylmethoxycyclobutyl)acetic acid 1932186-12-3 C13H16O3
2-(3-Phenylmethoxycyclobutyl)acetic acid
—— 6-((4-(2-hydroxyethyl)piperazin-1-yl)methyl)-2-methyl-2H-benzo[b][1,4]oxazin-3(4H)-one 1246082-61-0 C16H23N3O3
6-((4-(2-hydroxyethyl)piperazin-1-yl)methyl)-2-methyl-2H-benzo[b][1,4]oxazin-3(4H)-one
—— 6-(4-(4-cyanophenoxy)piperidine-1-carbonyl)-N-(1-(4-(pyrrolidin-1-yl)benzyl)piperidin-4-yl)nicotinamide 1356629-60-1 C35H40N6O3
6-(4-(4-cyanophenoxy)piperidine-1-carbonyl)-N-(1-(4-(pyrrolidin-1-yl)benzyl)piperidin-4-yl)nicotinamide
—— tert-butyl (2-fluoro-4-iodophenyl)[3-({[1-(2-hydroxyethyl)cyclopropyl]sulfonyl}amino)-1,5-dimethyl-6-oxo-1 ,6-dihydropyridin-2-yl]carbamate 1246443-10-6 C23H29FIN3O6S
tert-butyl (2-fluoro-4-iodophenyl)[3-({[1-(2-hydroxyethyl)cyclopropyl]sulfonyl}amino)-1,5-dimethyl-6-oxo-1 ,6-dihydropyridin-2-yl]carbamate
—— 8-(4-fluorophenyl)-5,6,7,8-tetrahydroquinazoline-2,4(1H,3H)-dione 1263870-12-7 C14H13FN2O2
8-(4-fluorophenyl)-5,6,7,8-tetrahydroquinazoline-2,4(1H,3H)-dione
—— 5-(1-(furan-3-ylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)-3-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazin-2-amine 1225061-38-0 C21H18N6O4S
5-(1-(furan-3-ylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)-3-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazin-2-amine
—— 8-chloro-4-[(3S)-3-isopropylpiperazin-1-yl][1]benzofuro[3,2-d]pyrimidin-2-amine 1035226-24-4 C17H20ClN5O
8-chloro-4-[(3S)-3-isopropylpiperazin-1-yl][1]benzofuro[3,2-d]pyrimidin-2-amine
—— 5-amino-N-(5-(6,6-difluoro-1,4-diazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,5-difluorophenyl)thiazole-4-carboxamide 1428569-48-5 C19H19F4N7OS
5-amino-N-(5-(6,6-difluoro-1,4-diazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,5-difluorophenyl)thiazole-4-carboxamide
—— 6-chloro-2-isopropyl-4-(2-trifluoromethoxy-benzyl)-quinoline-3-carboxylic acid 1433902-21-6 C21H17ClF3NO3
6-chloro-2-isopropyl-4-(2-trifluoromethoxy-benzyl)-quinoline-3-carboxylic acid
—— 4,5-methylenedioxy-1,3-dihydro-iminoisobenzofuran 1251898-14-2 C9H7NO3
4,5-methylenedioxy-1,3-dihydro-iminoisobenzofuran
—— (+)-(2S)-2-amino-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-N-isobutylpropanamide 1233927-00-8 C17H26N2O3
(+)-(2S)-2-amino-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-N-isobutylpropanamide
—— N-(3-amino-1-([4-(methyloxy)phenyl]methyl)-2,3-dioxopropyl)-2-(3-naphthalen-1-yl-1H-pyrazol-1-yl)pyridine-3-carboxamide 1037827-79-4 C30H25N5O4
N-(3-amino-1-([4-(methyloxy)phenyl]methyl)-2,3-dioxopropyl)-2-(3-naphthalen-1-yl-1H-pyrazol-1-yl)pyridine-3-carboxamide
—— 2-(1-ethyl-1H-indol-3-yl)-2-oxo-N-(2-(piperidin-1-yl)ethyl)acetamide hydrochloride 1228760-83-5 C19H25N3O2*ClH
2-(1-ethyl-1H-indol-3-yl)-2-oxo-N-(2-(piperidin-1-yl)ethyl)acetamide hydrochloride
—— 1-(cyclopropylmethyl)-5-(1-oxa-2-azaspiro[4.4]noN-2-en-3-yl)-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine 1057635-94-5 C22H29N5O2
1-(cyclopropylmethyl)-5-(1-oxa-2-azaspiro[4.4]noN-2-en-3-yl)-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine
—— 1-(4-amino-3-iodophenyl)-2-pyrrolidin-1-yl-pentan-1-one 1170693-27-2 C15H21IN2O
1-(4-amino-3-iodophenyl)-2-pyrrolidin-1-yl-pentan-1-one
—— (4S)-4-(([4-(benzyloxy)-6-phenylpyridin-2-yl]carbonyl)amino)-5-[4-(ethoxycarbonyl)piperazin-1-yl]-5-oxopentanoic acid 1188276-24-5 C31H34N4O7
(4S)-4-(([4-(benzyloxy)-6-phenylpyridin-2-yl]carbonyl)amino)-5-[4-(ethoxycarbonyl)piperazin-1-yl]-5-oxopentanoic acid
—— (S)-N-(6-((R)-2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)-3-hydroxypyrrolidine-1-carboxamide 1218935-01-3 C21H22F2N6O2
(S)-N-(6-((R)-2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)-3-hydroxypyrrolidine-1-carboxamide
—— 5-[4-(azepan-1-yl)-2-[(3-chloro-4-fluorophenyl)amino]pyrimidin-5-yl]pyridine-3-carboxylic acid 1220130-04-0 C22H21ClFN5O2
5-[4-(azepan-1-yl)-2-[(3-chloro-4-fluorophenyl)amino]pyrimidin-5-yl]pyridine-3-carboxylic acid
—— allyl 3-(4-(2,6-difluorobenzamido)phenyl)-4-methyl-5,6-dihydropyridine-1(2H)-carboxylate 1219927-67-9 C23H22F2N2O3
allyl 3-(4-(2,6-difluorobenzamido)phenyl)-4-methyl-5,6-dihydropyridine-1(2H)-carboxylate
—— 3-{[4-(4-trifluoromethyl)benzylpiperazin-1-yl]methylcarboxamido}methyl-5-propyl-1-phenyl-1H-pyrazole 1220347-66-9 C27H32F3N5O
3-{[4-(4-trifluoromethyl)benzylpiperazin-1-yl]methylcarboxamido}methyl-5-propyl-1-phenyl-1H-pyrazole
—— 4-(3-fluoro-azetidine-1-carbonyl)-2-methyl-2H-pyrazole-3-carboxylic acid (2-morpholin-4-yl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-amide 1428746-85-3 C19H21FN8O3
4-(3-fluoro-azetidine-1-carbonyl)-2-methyl-2H-pyrazole-3-carboxylic acid (2-morpholin-4-yl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-amide
—— 2-[2-amino-1-(4-fluorophenyl)ethyl]-5-(1-methyl-1H-pyrazol-5-yl)isoindolin-1-one 1430057-62-7 C20H19FN4O
2-[2-amino-1-(4-fluorophenyl)ethyl]-5-(1-methyl-1H-pyrazol-5-yl)isoindolin-1-one
—— 2-(3-cyano-1-cyclohexyl-5-methyl-1H-indol-2-yl)-N-(propan-2-yl)pyrimidine-5-sulfonamide 1248575-70-3 C23H27N5O2S
2-(3-cyano-1-cyclohexyl-5-methyl-1H-indol-2-yl)-N-(propan-2-yl)pyrimidine-5-sulfonamide
—— N-(2,4-dimethylphenyl)-N-isobutyl-3-(pyridin-4-ylmethoxy)benzenesulfonamide 1429346-87-1 C24H28N2O3S
N-(2,4-dimethylphenyl)-N-isobutyl-3-(pyridin-4-ylmethoxy)benzenesulfonamide
—— N-[4-(3-amino-1H-pyrazolo[3,4-b]pyrazin-6-yl)-2-fluoro-phenyl]-5-chloro-2-fluoro-benzenesulfonamide 1426214-66-5 C17H11ClF2N6O2S
N-[4-(3-amino-1H-pyrazolo[3,4-b]pyrazin-6-yl)-2-fluoro-phenyl]-5-chloro-2-fluoro-benzenesulfonamide
—— 5-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)furo[2,3-b]pyridine 1251728-92-3 C13H16BNO3
5-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)furo[2,3-b]pyridine
—— 6-(5-chloro-3-cyano-1-cyclobutyl-1H-indol-2-yl)-N-[(2R)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide 1248576-86-4 C21H18ClF3N4O2S
6-(5-chloro-3-cyano-1-cyclobutyl-1H-indol-2-yl)-N-[(2R)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide
—— N-[4-(6-chloro-3-cyano-1-cyclohexyl-1H-pyrrolo[3,2-b]pyridin-2-yl)phenyl]-2-methylpropane-2-sulfonamide 1247935-56-3 C24H27ClN4O2S
N-[4-(6-chloro-3-cyano-1-cyclohexyl-1H-pyrrolo[3,2-b]pyridin-2-yl)phenyl]-2-methylpropane-2-sulfonamide
—— 4-(3,5-dicyano-1-cyclobutyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-N-[(2S)-1,1,1-trifluoropropan-2-yl]benzenesulfonamide 1247932-09-7 C22H18F3N5O2S
4-(3,5-dicyano-1-cyclobutyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-N-[(2S)-1,1,1-trifluoropropan-2-yl]benzenesulfonamide
—— 3-bromo-3-(furan-2-ylmethyl)indolin-2-one 1398681-69-0 C13H10BrNO2
3-bromo-3-(furan-2-ylmethyl)indolin-2-one
—— (R)-2-(3-(2-nitrophenyl)-5-oxo-5-phenylpentanoyl)pyridine 1-oxide 1446271-27-7 C22H18N2O5
(R)-2-(3-(2-nitrophenyl)-5-oxo-5-phenylpentanoyl)pyridine 1-oxide
—— 1-O-ethyl 8-O-methyl 3-nitrooct-2-enedioate 1038619-07-6 C11H17NO6
1-O-ethyl 8-O-methyl 3-nitrooct-2-enedioate
—— 4-bromo-2-(α-(3-chloropropoxy)-4-chlorobenzyl)-5-(trifluoromethyl)-1H-pyrrole-3-carbonitrile 1614231-79-6 C16H12BrCl2F3N2O
4-bromo-2-(α-(3-chloropropoxy)-4-chlorobenzyl)-5-(trifluoromethyl)-1H-pyrrole-3-carbonitrile
—— 1-hydroxy-cyclohexanecarboxylic acid (2-bromopyridin-4-yl)amide 1433904-99-4 C12H15BrN2O2
1-hydroxy-cyclohexanecarboxylic acid (2-bromopyridin-4-yl)amide
—— 4-(3-{2-[4-(4-fluorobenzyl)-7,8-dihydropyrido[4,3-d]pyrimidin-6(5H)-yl]-2-oxoethyl}-2-oxoimidazolidin-1-yl)benzonitrile 1430101-37-3 C26H23FN6O2
4-(3-{2-[4-(4-fluorobenzyl)-7,8-dihydropyrido[4,3-d]pyrimidin-6(5H)-yl]-2-oxoethyl}-2-oxoimidazolidin-1-yl)benzonitrile
—— N-[5-(3,5-difluoro-benzenesulfonyl)-1H-indazol-3-yl]-4-[methyl-(2-piperidin-1-yl-ethyl)-amino]-2-nitro-benzamide hydrochloride 1034974-73-6 C28H28F2N6O5S*ClH
N-[5-(3,5-difluoro-benzenesulfonyl)-1H-indazol-3-yl]-4-[methyl-(2-piperidin-1-yl-ethyl)-amino]-2-nitro-benzamide hydrochloride
—— tert-butyl 4-(5-nitro-2-(2-(piperidin-1-yl)ethoxy)pyridin-4-ylamino)piperidine-1-carboxylate 1357922-07-6 C22H35N5O5
tert-butyl 4-(5-nitro-2-(2-(piperidin-1-yl)ethoxy)pyridin-4-ylamino)piperidine-1-carboxylate
—— 4-(3-phenoxyphenyl)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one hydrochloride 1108183-29-4 C30H28N4O2*ClH
4-(3-phenoxyphenyl)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one hydrochloride
—— [4-(4-amino-4-methylcyclohexylamino)-6-(3,5-dichloro-4-hydroxyphenyl)quinolin-3-yl](cyclopropyl)methanone 1356947-84-6 C26H27Cl2N3O2
[4-(4-amino-4-methylcyclohexylamino)-6-(3,5-dichloro-4-hydroxyphenyl)quinolin-3-yl](cyclopropyl)methanone
—— 5-chloro-N-(6,6-dimethyl-5-((3S,8aS)-3-methyl-octahydropyrrolo[1,2-a]pyrazine-2-carbonyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)picolinamide 1072099-98-9 C22H28ClN7O2
5-chloro-N-(6,6-dimethyl-5-((3S,8aS)-3-methyl-octahydropyrrolo[1,2-a]pyrazine-2-carbonyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)picolinamide
—— (13S,16S)-1-cyclopropyl-7-fluoro-16-[2-fluoro-4-((R)-5-hydroxymethyl-2-oxo-oxazolidin-3-yl)-phenoxymethyl]-4-oxo-16-phosphonooxy-1,4,13,15,16,17-hexahydro-12H-11-oxa-1,14-diaza-cyclopenta[a]phenanthrene-3-carboxylic acid benzyl ester 1029429-77-3 C36H34F2N3O12P
(13S,16S)-1-cyclopropyl-7-fluoro-16-[2-fluoro-4-((R)-5-hydroxymethyl-2-oxo-oxazolidin-3-yl)-phenoxymethyl]-4-oxo-16-phosphonooxy-1,4,13,15,16,17-hexahydro-12H-11-oxa-1,14-diaza-cyclopenta[a]phenanthrene-3-carboxylic acid benzyl ester
—— 2-methyl-2H-pyrazole-3,4-dicarboxylic acid 4-(cyclopropyl-methyl-amide) 3-(2-pyrrolidin-1-yl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-amide 1428747-08-3 C20H24N8O2
2-methyl-2H-pyrazole-3,4-dicarboxylic acid 4-(cyclopropyl-methyl-amide) 3-(2-pyrrolidin-1-yl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-amide
—— 2-((1R,2S,4S,5S,6S,8a'R)-5-((tert-butyldimethylsilyl)oxy)-2-hydroxy-4-methylhexahydro-1'H-spiro[cyclohexane-1,8'-indolizin]-6-yl)ethyl pivalate 1417600-81-7 C27H51NO4Si
2-((1R,2S,4S,5S,6S,8a'R)-5-((tert-butyldimethylsilyl)oxy)-2-hydroxy-4-methylhexahydro-1'H-spiro[cyclohexane-1,8'-indolizin]-6-yl)ethyl pivalate
—— (2R,3S)-3-(6-(4-(4-fluorophenoxy)phenyl)pyridin-2-yl)-2,3-dihydroxypropanamide 1433051-09-2 C20H17FN2O4
(2R,3S)-3-(6-(4-(4-fluorophenoxy)phenyl)pyridin-2-yl)-2,3-dihydroxypropanamide
—— ethyl 3-[(4-tert-butylphenyl)amino]-1H-indole-2-carboxylate 1010413-66-7 C21H24N2O2
ethyl 3-[(4-tert-butylphenyl)amino]-1H-indole-2-carboxylate