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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl 4-(3-(1-((1-benzylpiperidin-4-yl)(methyl)carbamoyl)-1H-imidazol-4-yl)benzoyl)piperazine-1-carboxylate 1356960-63-8 C33H42N6O4
tert-butyl 4-(3-(1-((1-benzylpiperidin-4-yl)(methyl)carbamoyl)-1H-imidazol-4-yl)benzoyl)piperazine-1-carboxylate
—— (E)-2-(phenyl(phenylselanyl)methylene)tetrahydroselenophene 1414875-00-5 C17H16Se2
(E)-2-(phenyl(phenylselanyl)methylene)tetrahydroselenophene
—— 2-(difluoromethyl)-5-(methylsulfonyl)pyridine 1574401-82-3 C7H7F2NO2S
2-(difluoromethyl)-5-(methylsulfonyl)pyridine
—— 1-(2,5-difluorobenzyl)-7-methoxy-3-(4-methoxy-phenyl)-2-methyl-1,2,3,4-tetrahydronaphthalene 1245637-15-3 C26H26F2O2
1-(2,5-difluorobenzyl)-7-methoxy-3-(4-methoxy-phenyl)-2-methyl-1,2,3,4-tetrahydronaphthalene
—— 7-(2-chlorophenyl)-6,7-dihydro-3H-benzo[f]pyrazolo[3,4-c]isoquinoline 1234371-51-7 C20H14ClN3
7-(2-chlorophenyl)-6,7-dihydro-3H-benzo[f]pyrazolo[3,4-c]isoquinoline
—— (R)-2-fluoro-5-(6-(2-fluorophenyl)-5,6-dihydrobenzo[h]quinazolin-2-ylamino)phenethyl methanesulfonate 1234352-30-7 C27H23F2N3O3S
(R)-2-fluoro-5-(6-(2-fluorophenyl)-5,6-dihydrobenzo[h]quinazolin-2-ylamino)phenethyl methanesulfonate
—— (S)-2-(8-(5-(hydroxymethyl)thiazol-2-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoic acid 1080639-65-1 C21H20N2O6S2
(S)-2-(8-(5-(hydroxymethyl)thiazol-2-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoic acid
—— —— 1356687-03-0 C13H18O6
—— N-{[4-(3-methoxypropoxy)-2-naphthyl]methyl}cyclopropanamine 1093083-13-6 C18H23NO2
N-{[4-(3-methoxypropoxy)-2-naphthyl]methyl}cyclopropanamine
—— 2-Cyclohexyl-9-(trifluoromethyl)fluoren-9-ol 1220962-47-9 C20H19F3O
2-Cyclohexyl-9-(trifluoromethyl)fluoren-9-ol
—— tert-butyl 3-hexylcyclobut-2-enecarboxylate 1422357-14-9 C15H26O2
tert-butyl 3-hexylcyclobut-2-enecarboxylate
—— Dimethyl 5-[(4-ethynylphenyl)carbamoylamino]benzene-1,3-dicarboxylate 1137673-93-8 C19H16N2O5
Dimethyl 5-[(4-ethynylphenyl)carbamoylamino]benzene-1,3-dicarboxylate
—— (3R,4R)-3-(2,4-dichlorophenyl)-1-oxo-2-[(3R)-2-oxopiperidin-3-yl]-N-phenylmethoxy-3,4-dihydroisoquinoline-4-carboxamide 1091588-96-3 C28H25Cl2N3O4
(3R,4R)-3-(2,4-dichlorophenyl)-1-oxo-2-[(3R)-2-oxopiperidin-3-yl]-N-phenylmethoxy-3,4-dihydroisoquinoline-4-carboxamide
—— 4-(3-Benzoyl-4-cyanopyrrol-1-yl)benzoic acid 1072200-88-4 C19H12N2O3
4-(3-Benzoyl-4-cyanopyrrol-1-yl)benzoic acid
—— 4-methylphenyl 3-(4-fluorophenylthio)-2-methyl-N-(4-methylphenyl)-2-propenimidothioate 1158848-18-0 C24H22FNS2
4-methylphenyl 3-(4-fluorophenylthio)-2-methyl-N-(4-methylphenyl)-2-propenimidothioate
—— N'-[5-bromo-2-methyl-6-[[3-(2-phenylethyl)phenyl]methoxy]pyridin-3-yl]-N-ethyl-N-methylmethanimidamide 1404444-66-1 C25H28BrN3O
N'-[5-bromo-2-methyl-6-[[3-(2-phenylethyl)phenyl]methoxy]pyridin-3-yl]-N-ethyl-N-methylmethanimidamide
—— N-(adamantan-1-ylmethyl)-2-{[4-(2-methoxyethyl)piperazin-1-yl]carbonyl}imidazo[1,2-a]pyridine-5-carboxamide 1031829-87-4 C27H37N5O3
N-(adamantan-1-ylmethyl)-2-{[4-(2-methoxyethyl)piperazin-1-yl]carbonyl}imidazo[1,2-a]pyridine-5-carboxamide
—— 2-bromo-1-[(3S,5R,8R,9R,10S,13S,14S,17S)-3-(fluoromethyl)-3-hydroxy-13-methyl-2,4,5,6,7,8,9,10,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]ethanone 1430063-72-1 C21H32BrFO2
2-bromo-1-[(3S,5R,8R,9R,10S,13S,14S,17S)-3-(fluoromethyl)-3-hydroxy-13-methyl-2,4,5,6,7,8,9,10,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]ethanone
—— (1R,2S,4R,5S,8S,12R)-7-(3,4-dichlorophenyl)-2-hydroxy-4-methyl-9,13-dioxa-7-azatetracyclo[6.3.1.1(1,4).0(5,12)]tridecan-6-one 1095183-31-5 C17H17Cl2NO4
(1R,2S,4R,5S,8S,12R)-7-(3,4-dichlorophenyl)-2-hydroxy-4-methyl-9,13-dioxa-7-azatetracyclo[6.3.1.1(1,4).0(5,12)]tridecan-6-one
—— US10280167, Example 32 1434586-42-1 C15H12N6O2
US10280167, Example 32
—— 1-(3,5-bis(trifluoromethyl)phenyl)-5-(3-chlorophenyl)-1H-pyrazole-3-carboxylic acid methylester 1610952-61-8 C19H11ClF6N2O2
1-(3,5-bis(trifluoromethyl)phenyl)-5-(3-chlorophenyl)-1H-pyrazole-3-carboxylic acid methylester
—— N-methylcarbamate-N-phenyl-O-THP-hydroxylamine 1093102-68-1 C13H17NO4
N-methylcarbamate-N-phenyl-O-THP-hydroxylamine
—— (7R)-7-benzyl-8-[5-fluoro-2-(trifluoromethoxy)phenyl]sulfonyl-2,5,8,11,13-pentazatricyclo[8.4.0.02,6]tetradeca-1(14),3,5,10,12-pentaene 1433992-47-2 C23H17F4N5O3S
(7R)-7-benzyl-8-[5-fluoro-2-(trifluoromethoxy)phenyl]sulfonyl-2,5,8,11,13-pentazatricyclo[8.4.0.02,6]tetradeca-1(14),3,5,10,12-pentaene
—— (+/-)-1-(2-(carboxymethoxy)-5-chlorophenyl)-3,4-dihydro-1H-isoquinoline-2-carboxylic acid 2,3-dimethoxybenzyl ester 1355056-14-2 C27H26ClNO7
(+/-)-1-(2-(carboxymethoxy)-5-chlorophenyl)-3,4-dihydro-1H-isoquinoline-2-carboxylic acid 2,3-dimethoxybenzyl ester
—— 3-(2-chloropyridin-4-yl)-N-[(3R)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-1H-indazole-5-carboxamide 1353246-44-2 C25H23ClFN5O
3-(2-chloropyridin-4-yl)-N-[(3R)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-1H-indazole-5-carboxamide
—— <2-(dimethylaminomethyl)phenyl>tellurium(II) bromide 128543-94-2 C9H12BrNTe
<2-(dimethylaminomethyl)phenyl>tellurium(II) bromide
—— ethyl 6-(9-benzyl-1,3,4,9-tetrahydro-2H-β-carbolin-2-yl)-3,3-dimethyl-6-oxohexanoate 1354803-14-7 C28H34N2O3
ethyl 6-(9-benzyl-1,3,4,9-tetrahydro-2H-β-carbolin-2-yl)-3,3-dimethyl-6-oxohexanoate
—— —— 1010114-96-1 C24H20N2O10
—— 7-methyl-2-(phenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,3-b]indole 1422192-31-1 C19H20N2O2S
7-methyl-2-(phenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,3-b]indole
—— (η(5)-C5Me4H)Fe(CO)(PMe3)I 175162-76-2 C13H22FeIOP
(η(5)-C5Me4H)Fe(CO)(PMe3)I
—— 2-[2-(quinolin-2-yl)ethyl]-8-(thiophen-2-yl)phthalazin-1(2H)-one 1433196-31-6 C23H17N3OS
2-[2-(quinolin-2-yl)ethyl]-8-(thiophen-2-yl)phthalazin-1(2H)-one
—— 5-amino-N-(4-((2R,4R,5S,6R)-4-amino-5-ethyl-5-hydroxy-6-methyltetrahydro-2H-pyran-2-yl)pyridin-3-yl)-2-(2,6-difluorophenyl)pyrimidine-4-carboxamide 1355009-95-8 C24H26F2N6O3
5-amino-N-(4-((2R,4R,5S,6R)-4-amino-5-ethyl-5-hydroxy-6-methyltetrahydro-2H-pyran-2-yl)pyridin-3-yl)-2-(2,6-difluorophenyl)pyrimidine-4-carboxamide
—— [4-[[(3S,4S)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]-[6-[7-(trifluoromethyl)-3,4-dihydro-1H-isoquinolin-2-yl]pyrimidin-4-yl]methanone 1349196-56-0 C26H32F3N5O3
[4-[[(3S,4S)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]-[6-[7-(trifluoromethyl)-3,4-dihydro-1H-isoquinolin-2-yl]pyrimidin-4-yl]methanone
—— N-[(3R)-1-[(3-methoxythiophen-2-yl)methyl]piperidin-3-yl]-3-(2-methylpyridin-4-yl)-1H-indazole-5-carboxamide 1353249-58-7 C25H27N5O2S
N-[(3R)-1-[(3-methoxythiophen-2-yl)methyl]piperidin-3-yl]-3-(2-methylpyridin-4-yl)-1H-indazole-5-carboxamide
—— tert-butyl 2-methoxy-4-{[4-(2-methoxy-2-oxoethyl)isoquinolin-1-yl]methyl}benzoate 1353486-53-9 C25H27NO5
tert-butyl 2-methoxy-4-{[4-(2-methoxy-2-oxoethyl)isoquinolin-1-yl]methyl}benzoate
—— 2-(4-((6-(7-(4-(3-cyclopropylureido)-2-fluorophenoxy)thieno[3.2-b]pyridin-2-yl)pyridin-3-yl)methyl)piperazin-1-yl)-2-oxoethyl 2-(benzyloxycarbonylamino)acetate 1429339-96-7 C39H38FN7O7S
2-(4-((6-(7-(4-(3-cyclopropylureido)-2-fluorophenoxy)thieno[3.2-b]pyridin-2-yl)pyridin-3-yl)methyl)piperazin-1-yl)-2-oxoethyl 2-(benzyloxycarbonylamino)acetate
—— [3-(4-fluoro-3-trifluoromethyl-phenyl)-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazol-5-yl]methanol 1431166-00-5 C14H13F4NO2
[3-(4-fluoro-3-trifluoromethyl-phenyl)-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazol-5-yl]methanol
—— 6-[5-(difluoromethyl)pyridin-3-yl]-N-(2-pyrrolidin-1-ylpyridin-4-yl)imidazo[1,2-b]pyridazine-3-carboxamide 1431643-34-3 C22H19F2N7O
6-[5-(difluoromethyl)pyridin-3-yl]-N-(2-pyrrolidin-1-ylpyridin-4-yl)imidazo[1,2-b]pyridazine-3-carboxamide
—— 3-(2,1,3-benzothiadiazol-5-yl)-N-[(3S,5R)-1-[(2-fluoro-6-methoxyphenyl)methyl]-5-methylpiperidin-3-yl]-1H-indazole-5-carboxamide 1353251-38-3 C28H27FN6O2S
3-(2,1,3-benzothiadiazol-5-yl)-N-[(3S,5R)-1-[(2-fluoro-6-methoxyphenyl)methyl]-5-methylpiperidin-3-yl]-1H-indazole-5-carboxamide
—— 1-(4-fluoro-3-carboxybenzyl)-5,6,7,8-tetrahydroquinazoline-2,4(1H,3H)-dione 1432671-42-5 C16H15FN2O4
1-(4-fluoro-3-carboxybenzyl)-5,6,7,8-tetrahydroquinazoline-2,4(1H,3H)-dione
—— US10280167, Example 25 1434586-03-4 C20H22N8O
US10280167, Example 25
—— (S)-3,5-dichloro-4-(2-(3-(cyclopropylmethoxy)-4-(difluoromethoxy)phenyl)-2-(2-(5-(N-((6-methylpyridin-2-yl)methyl)methylsulfonamido)-1,3-dioxoisoindolin-2-yl)acetoxy)ethyl)pyridine 1-oxide 1431566-54-9 C36H32Cl2F2N4O9S
(S)-3,5-dichloro-4-(2-(3-(cyclopropylmethoxy)-4-(difluoromethoxy)phenyl)-2-(2-(5-(N-((6-methylpyridin-2-yl)methyl)methylsulfonamido)-1,3-dioxoisoindolin-2-yl)acetoxy)ethyl)pyridine 1-oxide
—— 2-[(3-Bromophenyl)methyl]cyclopropane-1-carboxylic acid 1784061-70-6 C11H11BrO2
2-[(3-Bromophenyl)methyl]cyclopropane-1-carboxylic acid
—— tert-butyl 4-(methylamino)-octahydrocyclopenta[c]pyrrole-2-carboxylate, Mixture of diastereomers 1784081-02-2 C13H24N2O2
tert-butyl 4-(methylamino)-octahydrocyclopenta[c]pyrrole-2-carboxylate, Mixture of diastereomers
—— 4-(8-chloro-5H-dibenzo[b,e][1,4]diazepin-11-yl)-N-hydroxybenzamide 1024007-24-6 C20H14ClN3O2
4-(8-chloro-5H-dibenzo[b,e][1,4]diazepin-11-yl)-N-hydroxybenzamide
—— 1,1,4,4-tetrakis(4-bromophenylthio)butatriene 1233711-33-5 C28H16Br4S4
1,1,4,4-tetrakis(4-bromophenylthio)butatriene
—— 2-(4-(trifluoromethyl)phenylamino)benzo[d]oxazol-5-ol 1430331-62-6 C14H9F3N2O2
2-(4-(trifluoromethyl)phenylamino)benzo[d]oxazol-5-ol
—— (Z)-3-(bicyclo[2.2.1]heptan-2-yl)-5-[(5-(4'-methoxy-2',5'-dimethylphenyl)furan-2-yl)methylene]-2-thioxothiazolidin-4-one 1352733-10-8 C24H25NO3S2
(Z)-3-(bicyclo[2.2.1]heptan-2-yl)-5-[(5-(4'-methoxy-2',5'-dimethylphenyl)furan-2-yl)methylene]-2-thioxothiazolidin-4-one
—— 4,4'-bis(trimethylgermyl)-1,1'-biphenyl 1746-53-8 C18H26Ge2
4,4'-bis(trimethylgermyl)-1,1'-biphenyl
—— 3-(5-methoxy-2-pyridin-3-ylindol-1-ylmethyl)benzoic acid 1263299-12-2 C22H18N2O3
3-(5-methoxy-2-pyridin-3-ylindol-1-ylmethyl)benzoic acid