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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(1-ethyl-propyl)-6,7-dimethoxy-1-oxo-1,2-dihydro-isoquinoline-4-carboxylic acid 2-dimethylaminomethyl-benzylamide hydrochloride 1432750-61-2 C27H35N3O4*ClH
2-(1-ethyl-propyl)-6,7-dimethoxy-1-oxo-1,2-dihydro-isoquinoline-4-carboxylic acid 2-dimethylaminomethyl-benzylamide hydrochloride
—— 1-[2-tert-butyl-4-(2-chloropyridin-3-yl)-1H-imidazol-5-yl]-3-[4-(6,7-dimethoxyquinolin-4-yloxy)-2-fluorophenyl]urea 1355347-10-2 C30H28ClFN6O4
1-[2-tert-butyl-4-(2-chloropyridin-3-yl)-1H-imidazol-5-yl]-3-[4-(6,7-dimethoxyquinolin-4-yloxy)-2-fluorophenyl]urea
—— 4-[(7-Benzyl-2,5,8,14-tetrazatricyclo[8.4.0.02,6]tetradeca-1(10),3,5,11,13-pentaen-8-yl)sulfonyl]-2,1,3-benzoxadiazole 1433992-27-8 C23H18N6O3S
4-[(7-Benzyl-2,5,8,14-tetrazatricyclo[8.4.0.02,6]tetradeca-1(10),3,5,11,13-pentaen-8-yl)sulfonyl]-2,1,3-benzoxadiazole
—— 4-[2-(2-ethoxycarbonyl-ethyl)-3-[6-(3-ethoxy-5-pyrimidin-5-yl-phenoxy)-hexyl]-phenoxy]-butyric acid ethyl ester 1246206-52-9 C35H46N2O7
4-[2-(2-ethoxycarbonyl-ethyl)-3-[6-(3-ethoxy-5-pyrimidin-5-yl-phenoxy)-hexyl]-phenoxy]-butyric acid ethyl ester
—— 2-[2-Bis(2,4-ditert-butylphenoxy)phosphanyloxyethoxy]ethyl bis(2,4-ditert-butylphenyl) phosphite 1204513-13-2 C60H92O7P2
2-[2-Bis(2,4-ditert-butylphenoxy)phosphanyloxyethoxy]ethyl bis(2,4-ditert-butylphenyl) phosphite
—— (S)-4-(5-aminothiazolo[5,4-d]pyrimidin-7-yl)-3-methyl-N-[2-methyl-4-(pyrrolidin-1-ylmethyl)phenyl]piperazine-1-carboxamide 1435952-76-3 C23H30N8OS
(S)-4-(5-aminothiazolo[5,4-d]pyrimidin-7-yl)-3-methyl-N-[2-methyl-4-(pyrrolidin-1-ylmethyl)phenyl]piperazine-1-carboxamide
—— 3-(trifluoromethyl)-6-[4-[[3-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]-[1,2,4]triazolo[4,3-b]pyridazine 1166811-04-6 C18H16F6N6
3-(trifluoromethyl)-6-[4-[[3-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]-[1,2,4]triazolo[4,3-b]pyridazine
—— 4-chlorobenzyl 4-{4-[3-(3-oxo-3H-pyrazol-4-yl)propylcarbamoyl]thiazol-2-yl}piperidine-1-carboxylate 1143507-81-6 C23H24ClN5O4S
4-chlorobenzyl 4-{4-[3-(3-oxo-3H-pyrazol-4-yl)propylcarbamoyl]thiazol-2-yl}piperidine-1-carboxylate
—— (2S,4R)-2-{(1R,2S)-1-[2-(7-carboxy-heptanoylamino)-benzenesulfonylaminocarbonyl]-2-vinyl-cyclopropylcarbamoyl}-4-(7-methoxy-2-phenyl-quinolin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester 1051391-75-3 C46H53N5O11S
(2S,4R)-2-{(1R,2S)-1-[2-(7-carboxy-heptanoylamino)-benzenesulfonylaminocarbonyl]-2-vinyl-cyclopropylcarbamoyl}-4-(7-methoxy-2-phenyl-quinolin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester
—— ethyl 4-(((4S,5S)-3-(4-chlorophenyl)-4-(3,5-difluorophenyl)-2-oxooxazolidin-5-yl)methyl)piperazine-1-carboxylate 1035488-98-2 C23H24ClF2N3O4
ethyl 4-(((4S,5S)-3-(4-chlorophenyl)-4-(3,5-difluorophenyl)-2-oxooxazolidin-5-yl)methyl)piperazine-1-carboxylate
—— (8S,10R)-10-[2-(2-isopropylamino-thiazol-4-yl)-7-methoxy-quinolin-4-yloxy]-5-[(1R,2S)-1-carbonylamino-2-vinyl-cyclopropyl]-2,2-dioxo-2λ*6*-thia-3,6,12,22-tetraaza-tricyclo[21.4.0.0*8,12*]heptacosa-1(27),23,25-triene-4,7,13-trione 1051389-05-9 C42H51N7O7S2
(8S,10R)-10-[2-(2-isopropylamino-thiazol-4-yl)-7-methoxy-quinolin-4-yloxy]-5-[(1R,2S)-1-carbonylamino-2-vinyl-cyclopropyl]-2,2-dioxo-2λ*6*-thia-3,6,12,22-tetraaza-tricyclo[21.4.0.0*8,12*]heptacosa-1(27),23,25-triene-4,7,13-trione
—— tert-butyl 2-(diphenylmethyleneamino)-4,4-dimethylpentanoate 1449761-21-0 C24H31NO2
tert-butyl 2-(diphenylmethyleneamino)-4,4-dimethylpentanoate
—— 2-(Pyrimidine-2-carbonylamino)acetic acid 1084331-40-7 C7H7N3O3
2-(Pyrimidine-2-carbonylamino)acetic acid
—— ethyl 8-bromo-2-phenyl-2-(4-piperidinophenyl)-2H-naphtho[1,2-b]pyran-5-carboxylate 1021906-41-1 C33H30BrNO3
ethyl 8-bromo-2-phenyl-2-(4-piperidinophenyl)-2H-naphtho[1,2-b]pyran-5-carboxylate
—— 3-Piperidinecarboxylic acid, 4-phenyl-, hydrochloride (1:1), (3R,4R)-rel- 116140-27-3 C12H16ClNO2
3-Piperidinecarboxylic acid, 4-phenyl-, hydrochloride (1:1), (3R,4R)-rel-
—— N-(2,3-dihydro-1H-inden-2-yl)-2-(piperidin-1-yl)quinazolin-4-amine hydrochloride 1095660-89-1 C22H24N4*ClH
N-(2,3-dihydro-1H-inden-2-yl)-2-(piperidin-1-yl)quinazolin-4-amine hydrochloride
—— (3-tert-butyl-1H-pyrazol-4-ylmethyl)-(3-pyridin-2-yl-phenyl)-amine 1091677-54-1 C19H22N4
(3-tert-butyl-1H-pyrazol-4-ylmethyl)-(3-pyridin-2-yl-phenyl)-amine
—— 3-[2-(2-naphthyl)vinyl]-1-(4-nitrophenyl)cyclohepta[c]pyrazol-8(1H)-one 1205015-51-5 C26H17N3O3
3-[2-(2-naphthyl)vinyl]-1-(4-nitrophenyl)cyclohepta[c]pyrazol-8(1H)-one
—— 4-(benzo[d]thiazol-2-yl)-3-(4-chlorophenyl)butanoic acid 1221964-05-1 C17H14ClNO2S
4-(benzo[d]thiazol-2-yl)-3-(4-chlorophenyl)butanoic acid
—— 3-(6-chloro-2-methyl-1H-indol-3-ylsulfanyl)-5-trifluoromethyl-benzoic acid ethyl ester 1359980-78-1 C19H15ClF3NO2S
3-(6-chloro-2-methyl-1H-indol-3-ylsulfanyl)-5-trifluoromethyl-benzoic acid ethyl ester
—— 4-{1-[3-(4-diethylamino-benzoylamino)phenyl]ethylamino}quinazoline-8-carboxylic acid amide 1240476-31-6 C28H30N6O2
4-{1-[3-(4-diethylamino-benzoylamino)phenyl]ethylamino}quinazoline-8-carboxylic acid amide
—— 5-(4-fluoropyridin-3-yl)-3-methyl-1-{[1-(trifluoromethyl)cyclopropyl]methyl}-1,3-dihydro-2H-benzimidazol-2-one 1359759-04-8 C18H15F4N3O
5-(4-fluoropyridin-3-yl)-3-methyl-1-{[1-(trifluoromethyl)cyclopropyl]methyl}-1,3-dihydro-2H-benzimidazol-2-one
—— 2-(4-((S)-((S)-5-(tert-butyldimethylsilyloxy)-4-iodo-2-isopropyl-7,7-dimethyl-5,6,7,8-tetrahydroquinolin-3-yl)(hydroxy)methyl)phenyl)-2-methylpropanenitrile 1332487-13-4 C31H45IN2O2Si
2-(4-((S)-((S)-5-(tert-butyldimethylsilyloxy)-4-iodo-2-isopropyl-7,7-dimethyl-5,6,7,8-tetrahydroquinolin-3-yl)(hydroxy)methyl)phenyl)-2-methylpropanenitrile
—— [5-(5-methoxy-pyridin-3-yl)-imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-piperidin-4-yl-amine 1360175-53-6 C15H18N6OS
[5-(5-methoxy-pyridin-3-yl)-imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-piperidin-4-yl-amine
—— 4-fluoro-5-(3-fluoropyridin-4-yl)-3-methyl-1-[(1-methylcyclopropyl)methyl]-1,3-dihydro-2H-benzimidazol-2-one 1359760-80-7 C18H17F2N3O
4-fluoro-5-(3-fluoropyridin-4-yl)-3-methyl-1-[(1-methylcyclopropyl)methyl]-1,3-dihydro-2H-benzimidazol-2-one
—— 2-[6-(1-isopropylpyrrolidin-2-yl)pyridin-3-yl]-1H-benzimidazole-4-carboxamide 1103394-29-1 C20H23N5O
2-[6-(1-isopropylpyrrolidin-2-yl)pyridin-3-yl]-1H-benzimidazole-4-carboxamide
—— 3-(1-(4-chloro-2,5-dimethylphenylsulfonyl)piperidin-2-yl)-1-(4-(1-(4-methyl-piperazin-1-yl)-2-phenylethyl)piperidin-1-yl)propan-1-one 1073695-25-6 C34H49ClN4O3S
3-(1-(4-chloro-2,5-dimethylphenylsulfonyl)piperidin-2-yl)-1-(4-(1-(4-methyl-piperazin-1-yl)-2-phenylethyl)piperidin-1-yl)propan-1-one
—— (2R,3R)-4-(2-chlorophenyl)-2-hydroxy-3-({1-[2'-(5-oxo-4,5-dihydrotetrazol-1-yl)biphenyl-4-ylmethyl]-5-propyl-1H-pyrazole-3-carbonyl}amino)butyric acid 1260233-15-5 C31H30ClN7O5
(2R,3R)-4-(2-chlorophenyl)-2-hydroxy-3-({1-[2'-(5-oxo-4,5-dihydrotetrazol-1-yl)biphenyl-4-ylmethyl]-5-propyl-1H-pyrazole-3-carbonyl}amino)butyric acid
—— (1-methanesulfonyl-piperidin-4-yl)-[5-(5-methyl-pyridin-3-yl)-imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-amine 1360174-70-4 C16H20N6O2S2
(1-methanesulfonyl-piperidin-4-yl)-[5-(5-methyl-pyridin-3-yl)-imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-amine
—— N-(2-amino-4,6-dihydroxypyrimidin-5-yl)-3-(3,4-dimethoxyphenyl)propanamide 1245319-70-3 C15H18N4O5
N-(2-amino-4,6-dihydroxypyrimidin-5-yl)-3-(3,4-dimethoxyphenyl)propanamide
—— 1-cyclopropyl-7-[2,5-diazabicyclo(2.2.1)hept-2-yl]-6-fluoro-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid, monohydrochloride 100936-50-3 C17H17FN4O3*ClH
1-cyclopropyl-7-[2,5-diazabicyclo(2.2.1)hept-2-yl]-6-fluoro-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid, monohydrochloride
—— 2-methoxy-3-(2-oxo-propylsulfanyl)-benzoic acid ethyl ester 1359981-26-2 C13H16O4S
2-methoxy-3-(2-oxo-propylsulfanyl)-benzoic acid ethyl ester
—— (R)-1-(4-(6-isobutoxypyrimidin-4-yl)piperazin-1-yl)-2-phenoxypropan-1-one 1359732-53-8 C21H28N4O3
(R)-1-(4-(6-isobutoxypyrimidin-4-yl)piperazin-1-yl)-2-phenoxypropan-1-one
—— 7-chloro-3-oxo-3,4-dihydro-2H-benzo[1,4]thiazine-6-carboxylic acid {1-[2-(7-methoxy-quinoxalin-2-yloxy)-ethyl]-piperidin-4-ylmethyl}-amide 1236220-83-9 C26H28ClN5O4S
7-chloro-3-oxo-3,4-dihydro-2H-benzo[1,4]thiazine-6-carboxylic acid {1-[2-(7-methoxy-quinoxalin-2-yloxy)-ethyl]-piperidin-4-ylmethyl}-amide
—— 4-[({5-[(9-{[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethyl]amino}nonyl)oxy]-2-phenylphenyl}carbamoyl)oxy]-1,1-dimethylpiperidin-1-ium trifluoroacetate 1254098-77-5 C2F3O2*C40H53N4O6
4-[({5-[(9-{[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethyl]amino}nonyl)oxy]-2-phenylphenyl}carbamoyl)oxy]-1,1-dimethylpiperidin-1-ium trifluoroacetate
—— 1-(4-(5-amino-2-(4-fluorophenyl)thiazolo[5,4-d]pyrimidin-7-yl)piperazin-1-yl)-2-(2,4-dichlorophenoxy)ethanone 1245319-43-0 C23H19Cl2FN6O2S
1-(4-(5-amino-2-(4-fluorophenyl)thiazolo[5,4-d]pyrimidin-7-yl)piperazin-1-yl)-2-(2,4-dichlorophenoxy)ethanone
—— 1-(6,7-dihydro-5H-benzo[6,7]cyclohepta[1,2-c]pyridazin-3-yl)-N<sup>3</sup>-(4-((2-pyrrolidin-1-ylethyl)aminocarbonyl)phenyl)-1H-1,2,4-triazole-3,5-diamine 1037624-88-6 C28H31N9O
1-(6,7-dihydro-5H-benzo[6,7]cyclohepta[1,2-c]pyridazin-3-yl)-N<sup>3</sup>-(4-((2-pyrrolidin-1-ylethyl)aminocarbonyl)phenyl)-1H-1,2,4-triazole-3,5-diamine
—— 2-chloro-7-[(E)-2-(2-isobutoxy-3-methoxyphenyl)vinyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one 1192871-99-0 C19H19ClN2O3S
2-chloro-7-[(E)-2-(2-isobutoxy-3-methoxyphenyl)vinyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— PS168 1221962-04-4 C23H19ClN2O2*ClH
PS168
—— (R)-4-(2-chlorophenyl)-3-({1-[2'-(5-oxo-4,5-dihydrotetrazol-1-yl)-biphenyl-4-ylmethyl]-5-propyl-1H-pyrazole-3-carbonyl}amino)butyric acid 1260233-14-4 C31H30ClN7O4
(R)-4-(2-chlorophenyl)-3-({1-[2'-(5-oxo-4,5-dihydrotetrazol-1-yl)-biphenyl-4-ylmethyl]-5-propyl-1H-pyrazole-3-carbonyl}amino)butyric acid
—— (2R,3R)-3-({5-ethoxy-1-[2'-(1H-tetrazol-5-yl)biphenyl-4-ylmethyl]-1H-pyrazole-3-carbonyl}amino)-2-hydroxy-4-phenylbutyric acid 1260231-53-5 C30H29N7O5
(2R,3R)-3-({5-ethoxy-1-[2'-(1H-tetrazol-5-yl)biphenyl-4-ylmethyl]-1H-pyrazole-3-carbonyl}amino)-2-hydroxy-4-phenylbutyric acid
—— 1-cyclohexyl-1H-pyrazole-4-carboxylic acid 1177299-30-7 C10H14N2O2
1-cyclohexyl-1H-pyrazole-4-carboxylic acid
—— (E)-3-(4-((E)-4-fluoro-1-(1H-indazol-5-yl)-2-phenylbut-1-en-1-yl)phenyl)acrylic acid 1365888-72-7 C26H21FN2O2
(E)-3-(4-((E)-4-fluoro-1-(1H-indazol-5-yl)-2-phenylbut-1-en-1-yl)phenyl)acrylic acid
—— (2R)-2-{[4-(6-methoxypyridin-3-yl)phenyl](methylsulfonyl)amino}-4-(4-oxo-1,2,3-benzotriazin-3(4H)-yl)butanoic acid 1369962-67-3 C24H23N5O6S
(2R)-2-{[4-(6-methoxypyridin-3-yl)phenyl](methylsulfonyl)amino}-4-(4-oxo-1,2,3-benzotriazin-3(4H)-yl)butanoic acid
—— —— 1365749-67-2 C44H68N6O8S
—— (methyl 5-acetamido-4,7,8,9-tetra-O-acetyl-3,5-dideoxy-D-glycero-α-D-galacto-2-nonulopyranosonate)-(2->6)-2-O-acetyl-3,4-di-O-benzyl-β-D-glucopyranosyl-(1->1)-(2S,3S,4R)-2-azido-3,4-dibenzylheptadecane-1,3,4-triol 1356164-02-7 C73H98N4O21
(methyl 5-acetamido-4,7,8,9-tetra-O-acetyl-3,5-dideoxy-D-glycero-α-D-galacto-2-nonulopyranosonate)-(2->6)-2-O-acetyl-3,4-di-O-benzyl-β-D-glucopyranosyl-(1->1)-(2S,3S,4R)-2-azido-3,4-dibenzylheptadecane-1,3,4-triol
—— 2-(3,4-dihydro-2H-pyran-6-yl)-4-(4-methylphenyl)sulfonyl-5-(trifluoromethyl)triazole 1343491-93-9 C15H14F3N3O3S
2-(3,4-dihydro-2H-pyran-6-yl)-4-(4-methylphenyl)sulfonyl-5-(trifluoromethyl)triazole
—— 2-((3-chloro-4-((6-(trifluoromethyl)pyridin-3-yl)oxy)benzyl)oxy)-9-methoxy-6,7-dihydro-4H-pyrimido[6,1-a]isoquinolin-4-one 1369253-34-8 C26H19ClF3N3O4
2-((3-chloro-4-((6-(trifluoromethyl)pyridin-3-yl)oxy)benzyl)oxy)-9-methoxy-6,7-dihydro-4H-pyrimido[6,1-a]isoquinolin-4-one
—— methyl N-[(2S)-1-[(2S)-2-[5-[3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6,7-dihydro-[1]benzofuro[3,2-d][1]benzoxepin-9-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1370524-91-6 C44H52N8O8
methyl N-[(2S)-1-[(2S)-2-[5-[3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6,7-dihydro-[1]benzofuro[3,2-d][1]benzoxepin-9-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— ((2R,3S,4R,5S)-5-(4-(cyclopropylamino)thieno[3,2-d]pyrimidin-7-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl sulfamate 1370007-21-8 C14H18N4O6S2
((2R,3S,4R,5S)-5-(4-(cyclopropylamino)thieno[3,2-d]pyrimidin-7-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl sulfamate