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—— 4-(o-tolyl)but-2-yn-1-ol —— C11H12O
4-(o-tolyl)but-2-yn-1-ol
—— N-cyclobutyl-3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C36H40F2N6O2
N-cyclobutyl-3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— N-(cyclopropylmethyl)-3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8 dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C36H40F2N6O2
N-(cyclopropylmethyl)-3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8 dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— 3-{8-(2,6-difluorophenyl)-2-[(1H-imidazol-2-ylmethyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-1,3-thiazol-2-ylbenzamide hydrochloride —— C28H20F2N8O2S*ClH
3-{8-(2,6-difluorophenyl)-2-[(1H-imidazol-2-ylmethyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-1,3-thiazol-2-ylbenzamide hydrochloride
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-methylbenzamide —— C28H30F2N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-methylbenzamide
—— 3-{8-(2,6-difluorophenyl)-2-[(1H-imidazol-2-ylmethyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-1,3-thiazol-2-ylbenzamide methanesulfonate —— CH4O3S*C28H20F2N8O2S
3-{8-(2,6-difluorophenyl)-2-[(1H-imidazol-2-ylmethyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-1,3-thiazol-2-ylbenzamide methanesulfonate
—— N-(2-cyanoethyl)-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C31H33F2N7O2
N-(2-cyanoethyl)-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— 3-(8-(2,6-difluorophenyl)-2-{[2-(dimethylamino)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl)-4-methyl-N-propylbenzamide —— C28H30F2N6O2
3-(8-(2,6-difluorophenyl)-2-{[2-(dimethylamino)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl)-4-methyl-N-propylbenzamide
—— 3-[8-(2,6-difluorophenyl)-2-(methylsulfinyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-(2-phenylethyl)benzamide —— C30H24F2N4O3S
3-[8-(2,6-difluorophenyl)-2-(methylsulfinyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-(2-phenylethyl)benzamide
—— 5,5-bis(4-fluorophenyl)-4,5-dihydro-2-phenylfuran-3-carbonitrile —— C23H15F2NO
5,5-bis(4-fluorophenyl)-4,5-dihydro-2-phenylfuran-3-carbonitrile
—— 3-{8-(2,6-difluorophenyl)-2-[[3-(dimethylamino)propyl](methyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-propylbenzamide —— C30H34F2N6O2
3-{8-(2,6-difluorophenyl)-2-[[3-(dimethylamino)propyl](methyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-propylbenzamide
—— N-cyclopentyl-3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C37H42F2N6O2
N-cyclopentyl-3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— 2-[N-(N-t-Butoxycarbonylsarcosyl)-N-methylamino]ethylbenzene —— C17H26N2O3
2-[N-(N-t-Butoxycarbonylsarcosyl)-N-methylamino]ethylbenzene
—— N-cyclopentyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]benzamide —— C32H36F2N6O2
N-cyclopentyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]benzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methyl-N-phenylbenzamide —— C34H34F2N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methyl-N-phenylbenzamide
—— 1,1-diniethylethyl (2-{[8-(2,6-difluorophenyl)-4-(2-methyl-5-{[(2-phenylethyl)amino]carbonyl}phenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}ethyl)methylcarbamate —— C37H38F2N6O4
1,1-diniethylethyl (2-{[8-(2,6-difluorophenyl)-4-(2-methyl-5-{[(2-phenylethyl)amino]carbonyl}phenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}ethyl)methylcarbamate
—— 1-((6-chloropyridin-3-yl)methyl)-5-phenyl-1H-1,2,3-triazole-4-carbonitrile —— C15H10ClN5
1-((6-chloropyridin-3-yl)methyl)-5-phenyl-1H-1,2,3-triazole-4-carbonitrile
—— 3-{8-(2,6-difluorophenyl)-2-[(1H-imidazol-2-ylmethyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-1,3-thiazol-2-ylbenzamide hydrobromide —— BrH*C28H20F2N8O2S
3-{8-(2,6-difluorophenyl)-2-[(1H-imidazol-2-ylmethyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-1,3-thiazol-2-ylbenzamide hydrobromide
—— N-cyclopentyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C33H38F2N6O2
N-cyclopentyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— N-cyclopropyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methylbenzamide —— C31H34F2N6O2
N-cyclopropyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methylbenzamide
—— 1,1-dimethylethyl {2-[(8-(2,6-difluorophenyl)-4-{2-methyl-5-[(propylamino)carbonyl]phenyl}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]ethyl}methylcarbamate —— C32H36F2N6O4
1,1-dimethylethyl {2-[(8-(2,6-difluorophenyl)-4-{2-methyl-5-[(propylamino)carbonyl]phenyl}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]ethyl}methylcarbamate
—— N-cyclopropyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C31H34F2N6O2
N-cyclopropyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methyl-N-1,3-thiazol-2-ylbenzamide —— C31H31F2N7O2S
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methyl-N-1,3-thiazol-2-ylbenzamide
—— m-fluorophenyl tris(p-methoxyphenyl) orthocarbonate —— C28H25FO7
m-fluorophenyl tris(p-methoxyphenyl) orthocarbonate
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[(1S)-1,2-dimethylpropyl]-4-methylbenzamide —— C33H40F2N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[(1S)-1,2-dimethylpropyl]-4-methylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[(1R)-1,2-dimethylpropyl]-4-methylbenzamide —— C33H40F2N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[(1R)-1,2-dimethylpropyl]-4-methylbenzamide
—— allyl 5-cyano-6-{[2-(diphenylamino)-2-oxoethyl]thio}-4-(furan-2-yl)-2-methyl-1,4-dihydropyridin-3-carboxylate —— C29H25N3O4S
allyl 5-cyano-6-{[2-(diphenylamino)-2-oxoethyl]thio}-4-(furan-2-yl)-2-methyl-1,4-dihydropyridin-3-carboxylate
—— N,N-diphenyl-2,3-epoxy-3-(4-nitrophenyl)-1-propanamide —— C21H16N2O4
N,N-diphenyl-2,3-epoxy-3-(4-nitrophenyl)-1-propanamide
—— N,N'-di{6-[(2-methoxybenzyl)amino]hexyl}-1,1'-biphenyl-4,4'-diyldimethylamine —— C42H58N4O2
N,N'-di{6-[(2-methoxybenzyl)amino]hexyl}-1,1'-biphenyl-4,4'-diyldimethylamine
—— 2-benzoyl-4-(4,5-dimethyl-1,3-dithiol-2-ylidene)but-2-enenitrile —— C16H13NOS2
2-benzoyl-4-(4,5-dimethyl-1,3-dithiol-2-ylidene)but-2-enenitrile
—— 1-(2-methoxy-4-methyl-phenyl)-ethanone oxime —— C10H13NO2
1-(2-methoxy-4-methyl-phenyl)-ethanone oxime
—— 3-amino-N,N,4,6-tetraphenylthieno[2,3-b]pyridine-2-carboxamide —— C32H23N3OS
3-amino-N,N,4,6-tetraphenylthieno[2,3-b]pyridine-2-carboxamide
—— 1-(but-3-enyloxy)-3-fluorobenzene —— C10H11FO
1-(but-3-enyloxy)-3-fluorobenzene
—— 3-fluorophenyl 4-fluorobenzoate —— C13H8F2O2
3-fluorophenyl 4-fluorobenzoate
—— 3-amino-4,4-difluorobut-2-enenitrile —— C4H4F2N2
3-amino-4,4-difluorobut-2-enenitrile
—— 3-fluoro-3-phenylpropylamine —— C9H12FN
3-fluoro-3-phenylpropylamine
—— 7-amino-3-(p-tolyl)-5-phenyl-3H-imidazo[4,5-b]pyridine-6-carbonitrile —— C20H15N5
7-amino-3-(p-tolyl)-5-phenyl-3H-imidazo[4,5-b]pyridine-6-carbonitrile
—— N-methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2-yl)methyl)prop-2-yn-1-amine —— C30H39N3O
N-methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2-yl)methyl)prop-2-yn-1-amine
—— 4-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-1,3-thiazol-2-ylbenzamide —— C30H29F2N7O2S
4-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-1,3-thiazol-2-ylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-1,3-thiazol-2-ylbenzamide —— C30H29F2N7O2S
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-1,3-thiazol-2-ylbenzamide
—— 4-ethyl-2,5,5-triphenyl-4,5-dihydrofuran-3-carbonitrile —— C25H21NO
4-ethyl-2,5,5-triphenyl-4,5-dihydrofuran-3-carbonitrile
—— N-(cyclopropylmethyl)-3-[8-(2,6-difluorophenyl)-2-{[2-hydroxy-1-(hydroxymethyl)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C28H27F2N5O4
N-(cyclopropylmethyl)-3-[8-(2,6-difluorophenyl)-2-{[2-hydroxy-1-(hydroxymethyl)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-phenylbenzamide —— C33H32F2N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-phenylbenzamide
—— 6-methyl-3-phenylquinoxaline-2-carbonitrile 1,4-dioxide —— C16H11N3O2
6-methyl-3-phenylquinoxaline-2-carbonitrile 1,4-dioxide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-4-phenylbenzamide —— C34H34F2N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-4-phenylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-(4-fluorophenyl)-2-methylbenzamide —— C34H33F3N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-(4-fluorophenyl)-2-methylbenzamide
—— N-<(tert-butyloxycarbonyl)sarcosyl>-S-acetylcysteamine —— C12H22N2O4S
N-<(tert-butyloxycarbonyl)sarcosyl>-S-acetylcysteamine
—— 3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N,N,4-trimethylbenzamide —— C34H38F2N6O2
3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N,N,4-trimethylbenzamide
—— 3-cyano-5-methyl-2-phenylfuran —— C12H9NO
3-cyano-5-methyl-2-phenylfuran
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-[(1R)-1-phenylethyl]benzamide —— C36H38F2N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-[(1R)-1-phenylethyl]benzamide