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中文名称 英文名称 CAS号 化学式 结构式图片
—— Thiazoloisoindol-5-one deriv. 69 —— C16H14N2OS
Thiazoloisoindol-5-one deriv. 69
—— Thiazoloisoindol-5-one deriv. 71 —— C14H11N3OS
Thiazoloisoindol-5-one deriv. 71
—— Thiazoloisoindol-5-one deriv. 55 —— C17H12F3NOS
Thiazoloisoindol-5-one deriv. 55
—— Thiazoloisoindol-5-one deriv. 67 —— C15H12N2OS
Thiazoloisoindol-5-one deriv. 67
—— Thiazoloisoindol-5-one deriv. 62 —— C15H12N2OS
Thiazoloisoindol-5-one deriv. 62
—— Thiazoloisoindol-5-one deriv. 59 —— C20H15NOS
Thiazoloisoindol-5-one deriv. 59
—— Thiazoloisoindol-5-one deriv. 68 —— C15H12N2OS
Thiazoloisoindol-5-one deriv. 68
—— Thiazoloisoindol-5-one deriv. 70 —— C16H14N2OS
Thiazoloisoindol-5-one deriv. 70
—— Thiazolobenzimidazole & AZT —— C25H23F2N7O4S
Thiazolobenzimidazole & AZT
—— Thiazoloisoindol-5-one deriv. 51 —— C16H11Cl2NOS
Thiazoloisoindol-5-one deriv. 51
—— Thiazoloisoindol-5-one deriv. 42 —— C17H15NO2
Thiazoloisoindol-5-one deriv. 42
—— Thiazolobenzimidazole & ddI —— C25H22F2N6O3S
Thiazolobenzimidazole & ddI
—— Thiazoloisoindol-5-one deriv. 72 —— C15H13N3OS
Thiazoloisoindol-5-one deriv. 72
—— Thiazoloisoindol-5-one deriv. 50 —— C17H15NO2S
Thiazoloisoindol-5-one deriv. 50
—— Thiazoloisoindol-5-one deriv. 6 —— C20H15NOS
Thiazoloisoindol-5-one deriv. 6
—— Thiazoloisoindol-5-one deriv. 58 —— C16H12ClNOS
Thiazoloisoindol-5-one deriv. 58
—— Thiazoloisoindol-5-one deriv. 48 —— C17H15NOS
Thiazoloisoindol-5-one deriv. 48
—— Toxicol B, p-Qunione deriv. —— C36H52O3
Toxicol B, p-Qunione deriv.
—— Thiazoloisoindol-5-one deriv. 52 —— C17H15NOS
Thiazoloisoindol-5-one deriv. 52
—— Thiazoloisoindol-5-one deriv. 49 —— C16H12ClNOS
Thiazoloisoindol-5-one deriv. 49
—— Thiazoloisoindol-5-one deriv. 57 —— C16H14N2OS
Thiazoloisoindol-5-one deriv. 57
—— Thiazoloisoindol-5-one deriv. 54 —— C17H15NO2S
Thiazoloisoindol-5-one deriv. 54
—— tert-butyl N-[(1S,2S,4S)-1-(cyclohexylmethyl)-2-hydroxy-5-methyl-4-[[(1S)-2-methyl-1-(2-pyridylmethylcarbamoyl)butyl]carbamoyl]hexyl]carbamate —— C32H54N4O5
tert-butyl N-[(1S,2S,4S)-1-(cyclohexylmethyl)-2-hydroxy-5-methyl-4-[[(1S)-2-methyl-1-(2-pyridylmethylcarbamoyl)butyl]carbamoyl]hexyl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate —— C39H49N3O8
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-5-[[4-[2-(1,1-dioxo-1,4-thiazinan-4-yl)ethoxy]phenyl]methyl]-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate —— C39H51N3O8S
tert-butyl N-[(2S,3S,5S)-5-[[4-[2-(1,1-dioxo-1,4-thiazinan-4-yl)ethoxy]phenyl]methyl]-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-5-[[4-[2-[bis(2-methoxyethyl)amino]ethoxy]phenyl]methyl]-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate —— C41H57N3O8
tert-butyl N-[(2S,3S,5S)-5-[[4-[2-[bis(2-methoxyethyl)amino]ethoxy]phenyl]methyl]-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(2-hydroxyethoxy)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate —— C35H44N2O7
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(2-hydroxyethoxy)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenyl-5-[[4-(2-piperidin-1-ylethoxy)phenyl]methyl]hexan-2-yl]carbamate —— C40H53N3O6
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenyl-5-[[4-(2-piperidin-1-ylethoxy)phenyl]methyl]hexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-5-benzyl-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-1-[4-(2-morpholin-4-ylethoxy)phenyl]-6-oxohexan-2-yl]carbamate —— C39H51N3O7
tert-butyl N-[(2S,3S,5S)-5-benzyl-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-1-[4-(2-morpholin-4-ylethoxy)phenyl]-6-oxohexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(3-morpholin-4-ylpropoxy)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate —— C40H53N3O7
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(3-morpholin-4-ylpropoxy)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate
—— Tlnf(NH2) —— C23H36N6O6
Tlnf(NH2)
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenyl-5-[(4-phenylmethoxyphenyl)methyl]hexan-2-yl]carbamate —— C40H46N2O6
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenyl-5-[(4-phenylmethoxyphenyl)methyl]hexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-5-benzyl-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-1-(4-hydroxyphenyl)-6-oxohexan-2-yl]carbamate —— C33H40N2O6
tert-butyl N-[(2S,3S,5S)-5-benzyl-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-1-(4-hydroxyphenyl)-6-oxohexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(2-hydroxyethyl)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate —— C35H44N2O6
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(2-hydroxyethyl)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[(4-iodophenyl)methyl]-6-oxo-1-phenylhexan-2-yl]carbamate —— C33H39IN2O5
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[(4-iodophenyl)methyl]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-5-[[4-[2-(1-oxo-1,4-thiazinan-4-yl)ethoxy]phenyl]methyl]-1-phenylhexan-2-yl]carbamate —— C39H51N3O7S
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-5-[[4-[2-(1-oxo-1,4-thiazinan-4-yl)ethoxy]phenyl]methyl]-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-5-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]carbamoyl]-1-phenyl-7-quinoxalin-2-ylheptan-2-yl]carbamate —— C36H42N4O5
tert-butyl N-[(2S,3S,5S)-3-hydroxy-5-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]carbamoyl]-1-phenyl-7-quinoxalin-2-ylheptan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-5-[[4-[(dimethylamino)methyl]phenyl]methyl]-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate —— C36H47N3O5
tert-butyl N-[(2S,3S,5S)-5-[[4-[(dimethylamino)methyl]phenyl]methyl]-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-5-[(4-aminophenyl)methyl]-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate —— C33H41N3O5
tert-butyl N-[(2S,3S,5S)-5-[(4-aminophenyl)methyl]-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-5-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]carbamoyl]-1-phenylheptan-2-yl]carbamate —— C28H38N2O5
tert-butyl N-[(2S,3S,5S)-3-hydroxy-5-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]carbamoyl]-1-phenylheptan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenyl-5-[[4-(2-thiomorpholin-4-ylethoxy)phenyl]methyl]hexan-2-yl]carbamate —— C39H51N3O6S
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenyl-5-[[4-(2-thiomorpholin-4-ylethoxy)phenyl]methyl]hexan-2-yl]carbamate
—— tert-butyl N-[(1S,2S,4R)-1-benzyl-2-hydroxy-5-[[(1S,2R)-2-hydroxyindan-1-yl]amino]-4-methyl-5-oxo-pentyl]carbamate —— C27H36N2O5
tert-butyl N-[(1S,2S,4R)-1-benzyl-2-hydroxy-5-[[(1S,2R)-2-hydroxyindan-1-yl]amino]-4-methyl-5-oxo-pentyl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-[3-(2-methoxyethoxymethoxy)propyl]phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate —— C40H54N2O8
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-[3-(2-methoxyethoxymethoxy)propyl]phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-1-(4-hydroxyphenyl)-5-[(4-hydroxyphenyl)methyl]-6-oxohexan-2-yl]carbamate —— C33H40N2O7
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-1-(4-hydroxyphenyl)-5-[(4-hydroxyphenyl)methyl]-6-oxohexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[(4-methylsulfonylphenyl)methyl]-6-oxo-1-phenylhexan-2-yl]carbamate —— C34H42N2O7S
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[(4-methylsulfonylphenyl)methyl]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-5-[[4-[2-(dimethylamino)ethoxy]phenyl]methyl]-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate —— C37H49N3O6
tert-butyl N-[(2S,3S,5S)-5-[[4-[2-(dimethylamino)ethoxy]phenyl]methyl]-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-5-[(2,3,4,5,6-pentafluorophenyl)methyl]-1-phenylhexan-2-yl]carbamate —— C33H35F5N2O5
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-5-[(2,3,4,5,6-pentafluorophenyl)methyl]-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-5-[[4-[3-[bis(2-methoxyethyl)amino]propyl]phenyl]methyl]-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate —— C42H59N3O7
tert-butyl N-[(2S,3S,5S)-5-[[4-[3-[bis(2-methoxyethyl)amino]propyl]phenyl]methyl]-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[(4-methylsulfinylphenyl)methyl]-6-oxo-1-phenylhexan-2-yl]carbamate —— C34H42N2O6S
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[(4-methylsulfinylphenyl)methyl]-6-oxo-1-phenylhexan-2-yl]carbamate
—— tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(hydroxymethyl)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate —— C34H42N2O6
tert-butyl N-[(2S,3S,5S)-3-hydroxy-6-[[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]-5-[[4-(hydroxymethyl)phenyl]methyl]-6-oxo-1-phenylhexan-2-yl]carbamate