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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[2-(1',7-Dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-2-oxoethyl]pyrimidin-2-one —— C21H26N4O3
1-[2-(1',7-Dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-2-oxoethyl]pyrimidin-2-one
—— 4-[(3,4-Dimethoxyphenyl)methyl]-1',7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C24H32N2O3
4-[(3,4-Dimethoxyphenyl)methyl]-1',7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— 1'-[3-(4-Chlorophenyl)propanoyl]-7-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H25ClN2O4
1'-[3-(4-Chlorophenyl)propanoyl]-7-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(3,4-Dimethoxyphenyl)acetyl]-7-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H28N2O6
1'-[2-(3,4-Dimethoxyphenyl)acetyl]-7-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 7-Methoxy-1'-[3-(3-methoxy-4-methylphenyl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C25H30N2O5
7-Methoxy-1'-[3-(3-methoxy-4-methylphenyl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-(5-Tert-butyl-3-methylfuran-2-carbonyl)-7-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H30N2O5
1'-(5-Tert-butyl-3-methylfuran-2-carbonyl)-7-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-methoxy-1'-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H29N3O6
8-methoxy-1'-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-(5-Chloro-2-ethoxypyridine-3-carbonyl)-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H24ClN3O4
1'-(5-Chloro-2-ethoxypyridine-3-carbonyl)-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-[[(3R)-1,1-dioxothiolan-3-yl]-methylamino]acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C20H27N3O5S
1'-[2-[[(3R)-1,1-dioxothiolan-3-yl]-methylamino]acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(3,4-Dimethoxyphenyl)acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H28N2O6
1'-[2-(3,4-Dimethoxyphenyl)acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-[(1R,3S)-3-acetyl-2,2-dimethylcyclobutyl]acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H32N2O5
1'-[2-[(1R,3S)-3-acetyl-2,2-dimethylcyclobutyl]acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(3-Chlorophenyl)acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H23ClN2O4
1'-[2-(3-Chlorophenyl)acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 7-Methyl-1'-[2-(4-methylsulfonylphenyl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H26N2O5S
7-Methyl-1'-[2-(4-methylsulfonylphenyl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-[(1S,3R)-3-acetyl-2,2-dimethylcyclobutyl]acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H32N2O5
1'-[2-[(1S,3R)-3-acetyl-2,2-dimethylcyclobutyl]acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(2-Ethoxy-4-methylphenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H28N2O5
1'-[2-(2-Ethoxy-4-methylphenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-(5-Tert-butyl-3-methylfuran-2-carbonyl)-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H30N2O5
1'-(5-Tert-butyl-3-methylfuran-2-carbonyl)-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[3-(3-Methoxy-4-methylphenyl)propanoyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C25H30N2O4
1'-[3-(3-Methoxy-4-methylphenyl)propanoyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-[[(3S)-1,1-dioxothiolan-3-yl]-methylamino]acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C20H27N3O5S
1'-[2-[[(3S)-1,1-dioxothiolan-3-yl]-methylamino]acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[3-(4-Chloro-3,5-dimethylpyrazol-1-yl)propanoyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H27ClN4O3
1'-[3-(4-Chloro-3,5-dimethylpyrazol-1-yl)propanoyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-methoxy-1'-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H29N3O6
8-methoxy-1'-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(2-Oxopyrrolidin-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C19H23N3O4
1'-[2-(2-Oxopyrrolidin-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(2-Chlorophenyl)acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H23ClN2O4
1'-[2-(2-Chlorophenyl)acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-Methoxy-1'-[2-(4-methoxyphenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H26N2O6
8-Methoxy-1'-[2-(4-methoxyphenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(2,4-Dimethoxy-6-methylpyrimidin-5-yl)acetyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H28N4O5
1'-[2-(2,4-Dimethoxy-6-methylpyrimidin-5-yl)acetyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(4-Methylsulfonylphenyl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H24N2O5S
1'-[2-(4-Methylsulfonylphenyl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(2-Methoxy-4-methylphenoxy)acetyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H28N2O5
1'-[2-(2-Methoxy-4-methylphenoxy)acetyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— N-[2-methyl-4-[2-oxo-2-(5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethoxy]phenyl]acetamide —— C24H27N3O5
N-[2-methyl-4-[2-oxo-2-(5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethoxy]phenyl]acetamide
—— 1'-[2-(2,5-Dimethoxyphenyl)acetyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H28N2O5
1'-[2-(2,5-Dimethoxyphenyl)acetyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-(1-Methylsulfonylpiperidine-4-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C20H27N3O5S
1'-(1-Methylsulfonylpiperidine-4-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[3-(3-Acetyl-2,4-dimethylpyrrol-1-yl)propanoyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C25H31N3O4
1'-[3-(3-Acetyl-2,4-dimethylpyrrol-1-yl)propanoyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H30N4O4
1'-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-Methoxy-1'-[3-(2-propan-2-ylimidazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H30N4O4
8-Methoxy-1'-[3-(2-propan-2-ylimidazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— (5R)-3-methyl-5-[2-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C20H23N3O5S
(5R)-3-methyl-5-[2-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— 1'-[3-(4-Ethoxyphenyl)propanoyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C25H30N2O4
1'-[3-(4-Ethoxyphenyl)propanoyl]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-(Cyclopropanecarbonyl)-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C18H22N2O3
1'-(Cyclopropanecarbonyl)-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-(1H-indol-3-yl)acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H25N3O4
1'-[2-(1H-indol-3-yl)acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[2-[(1S,3S)-3-acetyl-2,2-dimethylcyclobutyl]acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H32N2O5
1'-[2-[(1S,3S)-3-acetyl-2,2-dimethylcyclobutyl]acetyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-[(2S)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H30N4O4
1'-[(2S)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-8-methoxyspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 7-Methyl-1'-[2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C19H22N4O3S2
7-Methyl-1'-[2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1-(2,3-dihydro-1,4-benzoxazin-4-yl)-2-(3,4-dihydro-2H-chromen-6-yl)ethanone —— C19H19NO3
1-(2,3-dihydro-1,4-benzoxazin-4-yl)-2-(3,4-dihydro-2H-chromen-6-yl)ethanone
—— 4'-[(6-Chloro-1,3-benzodioxol-5-yl)methyl-methylamino]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C24H27ClN2O4
4'-[(6-Chloro-1,3-benzodioxol-5-yl)methyl-methylamino]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— N-methyl-N-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)pyridine-3-carboxamide —— C22H25N3O3
N-methyl-N-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)pyridine-3-carboxamide
—— N-[5-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-1,3,4-thiadiazol-2-yl]-2-[(2S)-3-oxo-4H-1,4-benzoxazin-2-yl]acetamide —— C23H23N5O3S
N-[5-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-1,3,4-thiadiazol-2-yl]-2-[(2S)-3-oxo-4H-1,4-benzoxazin-2-yl]acetamide
—— 4'-[(2,6-Difluorophenyl)methyl-methylamino]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C23H26F2N2O2
4'-[(2,6-Difluorophenyl)methyl-methylamino]-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— N-methyl-N-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)pentanamide —— C21H30N2O3
N-methyl-N-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)pentanamide
—— (2S)-N-[[1-(dimethylamino)cyclopentyl]methyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C18H27N3O4S
(2S)-N-[[1-(dimethylamino)cyclopentyl]methyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— N-[5-[(4-methoxyphenoxy)methyl]-1,3,4-thiadiazol-2-yl]-2-[(2S)-3-oxo-4H-1,4-benzoxazin-2-yl]acetamide —— C20H18N4O5S
N-[5-[(4-methoxyphenoxy)methyl]-1,3,4-thiadiazol-2-yl]-2-[(2S)-3-oxo-4H-1,4-benzoxazin-2-yl]acetamide
—— (2R)-N-[[1-(dimethylamino)cyclopentyl]methyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C18H27N3O4S
(2R)-N-[[1-(dimethylamino)cyclopentyl]methyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— N-[5-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-1,3,4-thiadiazol-2-yl]-2-[(2R)-3-oxo-4H-1,4-benzoxazin-2-yl]acetamide —— C23H23N5O3S
N-[5-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-1,3,4-thiadiazol-2-yl]-2-[(2R)-3-oxo-4H-1,4-benzoxazin-2-yl]acetamide
—— N-methyl-N-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)butanamide —— C20H28N2O3
N-methyl-N-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)butanamide