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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(3R)-1,1-dioxothiolan-3-yl]-1-[(2S)-1'-prop-2-enylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C23H32N2O4S
2-[(3R)-1,1-dioxothiolan-3-yl]-1-[(2S)-1'-prop-2-enylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— [(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyridin-3-ylmethanone —— C27H29N3O2
[(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyridin-3-ylmethanone
—— 1'-[(2-Ethylpyrimidin-5-yl)methyl]-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C21H28N4O3S
1'-[(2-Ethylpyrimidin-5-yl)methyl]-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— [(2R)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-(6-methylpyridin-3-yl)methanone —— C28H31N3O2
[(2R)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-(6-methylpyridin-3-yl)methanone
—— (2R)-7-methoxy-4-[(4-methoxyphenyl)methyl]-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane] —— C24H32N2O3
(2R)-7-methoxy-4-[(4-methoxyphenyl)methyl]-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]
—— 1'-(Cyclopropylmethyl)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C19H28N2O3S
1'-(Cyclopropylmethyl)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— 4-Methylsulfonyl-1'-[(2-propylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C22H30N4O3S
4-Methylsulfonyl-1'-[(2-propylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— [(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-(6-methylpyridin-3-yl)methanone —— C28H31N3O2
[(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-(6-methylpyridin-3-yl)methanone
—— 1-[(3R)-3-methylpiperidin-1-yl]-2-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone —— C22H33N3O4S
1-[(3R)-3-methylpiperidin-1-yl]-2-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone
—— N,N-dimethyl-2-(7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)acetamide —— C19H29N3O4S
N,N-dimethyl-2-(7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)acetamide
—— 5-[2-[(2S)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione —— C23H30N4O5
5-[2-[(2S)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 4-Imidazol-1-yl-1-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)butan-1-one —— C21H28N4O4S
4-Imidazol-1-yl-1-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)butan-1-one
—— [(2R)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyridin-2-ylmethanone —— C27H29N3O2
[(2R)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyridin-2-ylmethanone
—— 1-(4-Methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-3-(1,2-oxazol-5-yl)propan-1-one —— C20H25N3O5S
1-(4-Methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-3-(1,2-oxazol-5-yl)propan-1-one
—— 4-methylsulfonyl-1'-[[(3R)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C19H28N2O4S
4-methylsulfonyl-1'-[[(3R)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— 1-[1'-[2,2-Dimethyl-3-(4-methylpiperazin-1-yl)propyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C26H42N4O2
1-[1'-[2,2-Dimethyl-3-(4-methylpiperazin-1-yl)propyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— (1'-ethyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-[(3R)-piperidin-3-yl]methanone —— C22H33N3O2
(1'-ethyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-[(3R)-piperidin-3-yl]methanone
—— 1'-[(2-Ethylpyrimidin-5-yl)methyl]-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C22H30N4O3S
1'-[(2-Ethylpyrimidin-5-yl)methyl]-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— 1-[(2R)-2-methylpiperidin-1-yl]-2-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone —— C22H33N3O4S
1-[(2R)-2-methylpiperidin-1-yl]-2-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone
—— 7-Methyl-4-methylsulfonyl-1'-(pyridin-2-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C21H27N3O3S
7-Methyl-4-methylsulfonyl-1'-(pyridin-2-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— Cyclopropyl-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)methanone —— C18H24N2O4S
Cyclopropyl-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)methanone
—— 1-[1'-[(2,3-Dimethylimidazol-4-yl)methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C22H30N4O2
1-[1'-[(2,3-Dimethylimidazol-4-yl)methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— [(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyridin-2-ylmethanone —— C27H29N3O2
[(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyridin-2-ylmethanone
—— [(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyrazin-2-ylmethanone —— C26H28N4O2
[(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyrazin-2-ylmethanone
—— (2S)-7-methoxy-4-[(2-methoxyphenyl)methyl]-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane] —— C24H32N2O3
(2S)-7-methoxy-4-[(2-methoxyphenyl)methyl]-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]
—— 5-[2-[(2R)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione —— C23H30N4O5
5-[2-[(2R)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 6-methyl-5-[2-oxo-2-[(2R)-1'-prop-2-enylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethyl]-1H-pyrimidine-2,4-dione —— C24H30N4O4
6-methyl-5-[2-oxo-2-[(2R)-1'-prop-2-enylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethyl]-1H-pyrimidine-2,4-dione
—— 1-(4-Acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-3-aminopropan-1-one —— C19H27N3O3
1-(4-Acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-3-aminopropan-1-one
—— [(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyridin-4-ylmethanone —— C27H29N3O2
[(2S)-1'-benzylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyridin-4-ylmethanone
—— 1-(4-Methylpiperidin-1-yl)-2-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone —— C22H33N3O4S
1-(4-Methylpiperidin-1-yl)-2-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone
—— 1-[7-Methyl-1'-(2-pyrazol-1-ylethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C21H28N4O2
1-[7-Methyl-1'-(2-pyrazol-1-ylethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— 1-[1'-[(3S)-oxolane-3-carbonyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C20H26N2O4
1-[1'-[(3S)-oxolane-3-carbonyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— 1-[1'-(Oxane-4-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C21H28N2O4
1-[1'-(Oxane-4-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— 4-methylsulfonyl-1'-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C19H28N2O4S
4-methylsulfonyl-1'-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— (2S)-4-[(2,3-dimethoxyphenyl)methyl]-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane] —— C25H34N2O4
(2S)-4-[(2,3-dimethoxyphenyl)methyl]-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]
—— 4-Methylsulfonyl-1'-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C22H30N4O3S
4-Methylsulfonyl-1'-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— 2-Methoxy-1-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone —— C17H24N2O5S
2-Methoxy-1-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone
—— (2R)-7-methoxy-4-[(2-methoxyphenyl)methyl]-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane] —— C24H32N2O3
(2R)-7-methoxy-4-[(2-methoxyphenyl)methyl]-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]
—— 1-[7-Methyl-1'-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C24H32N4O2
1-[7-Methyl-1'-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— 1-[3-[(2R)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-3-oxopropyl]pyridin-2-one —— C24H31N3O4
1-[3-[(2R)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-3-oxopropyl]pyridin-2-one
—— 4-Imidazol-1-yl-1-(7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)butan-1-one —— C22H30N4O4S
4-Imidazol-1-yl-1-(7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)butan-1-one
—— (2R)-7-methoxy-4-[(3-methoxyphenyl)methyl]-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane] —— C24H32N2O3
(2R)-7-methoxy-4-[(3-methoxyphenyl)methyl]-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]
—— 3-Imidazol-1-yl-1-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)propan-1-one —— C20H26N4O4S
3-Imidazol-1-yl-1-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)propan-1-one
—— Cyclopropyl-(1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)methanone —— C18H24N2O2
Cyclopropyl-(1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)methanone
—— 1-(4-Acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-4-imidazol-1-ylbutan-1-one —— C22H28N4O3
1-(4-Acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-4-imidazol-1-ylbutan-1-one
—— (5-Methylpyrazin-2-yl)-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)methanone —— C20H24N4O4S
(5-Methylpyrazin-2-yl)-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)methanone
—— 1-(1',7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-2-[(3S)-1,1-dioxothiolan-3-yl]ethanone —— C21H30N2O4S
1-(1',7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-2-[(3S)-1,1-dioxothiolan-3-yl]ethanone
—— 1',7-Dimethyl-4-(pyridin-4-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C21H27N3O
1',7-Dimethyl-4-(pyridin-4-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— 1-(4-Acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-4-(3,5-dimethylpyrazol-1-yl)butan-1-one —— C24H32N4O3
1-(4-Acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-4-(3,5-dimethylpyrazol-1-yl)butan-1-one
—— 1'-Ethyl-4-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C24H36N4O
1'-Ethyl-4-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]