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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(2R)-1'-(1,5-dimethylpyrazole-4-carbonyl)-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C23H30N4O4
1-[(2R)-1'-(1,5-dimethylpyrazole-4-carbonyl)-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— 1-[(2R)-4-acetyl-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]-4-imidazol-1-ylbutan-1-one —— C24H32N4O4
1-[(2R)-4-acetyl-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]-4-imidazol-1-ylbutan-1-one
—— 1-[(2R)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(2,4-dimethyl-1,3-thiazol-5-yl)ethanone —— C24H34N4O2S
1-[(2R)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(2,4-dimethyl-1,3-thiazol-5-yl)ethanone
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-methylpyrazol-3-yl)methanone —— C17H22N4O2
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-methylpyrazol-3-yl)methanone
—— N-[4-[2-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]-1,3-thiazol-2-yl]methanesulfonamide —— C18H24N4O4S2
N-[4-[2-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]-1,3-thiazol-2-yl]methanesulfonamide
—— 1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(4-methylphenyl)ethanone —— C26H35N3O2
1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(4-methylphenyl)ethanone
—— [(2R)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-(2,4-dimethyl-1,3-oxazol-5-yl)methanone —— C23H32N4O3
[(2R)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-(2,4-dimethyl-1,3-oxazol-5-yl)methanone
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrimidin-5-ylmethanone —— C17H20N4O2
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrimidin-5-ylmethanone
—— 1-[(2S)-1'-[(3,4-dimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C25H32N2O4
1-[(2S)-1'-[(3,4-dimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— 1-[(2R)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2,2-dimethylpropan-1-one —— C22H35N3O2
1-[(2R)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2,2-dimethylpropan-1-one
—— 2-methyl-1-[(2R)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]propan-1-one —— C19H28N2O2
2-methyl-1-[(2R)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]propan-1-one
—— 2-methoxy-1-[(2R)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]ethanone —— C18H26N2O3
2-methoxy-1-[(2R)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]ethanone
—— 1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(2-fluorophenyl)ethanone —— C25H32FN3O2
1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(2-fluorophenyl)ethanone
—— 1-[7-Methyl-1'-(4-phenoxybutyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C26H34N2O3
1-[7-Methyl-1'-(4-phenoxybutyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— N-[4-[2-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]-1,3-thiazol-2-yl]methanesulfonamide —— C18H24N4O4S2
N-[4-[2-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]-1,3-thiazol-2-yl]methanesulfonamide
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-pyridin-2-ylethanone —— C19H23N3O2
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-pyridin-2-ylethanone
—— 1-[(2S)-4-acetyl-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]-4-imidazol-1-ylbutan-1-one —— C24H32N4O4
1-[(2S)-4-acetyl-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]-4-imidazol-1-ylbutan-1-one
—— 1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethanone —— C24H27N3O5
1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethanone
—— 1-[(3S)-4-[[(2S)-1-[(2,3-dimethoxyphenyl)methyl]pyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine —— C26H37N3O3
1-[(3S)-4-[[(2S)-1-[(2,3-dimethoxyphenyl)methyl]pyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine
—— N-[5-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]-4-methyl-1,3-thiazol-2-yl]methanesulfonamide —— C18H24N4O4S2
N-[5-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]-4-methyl-1,3-thiazol-2-yl]methanesulfonamide
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-thiazol-4-yl)methanone —— C16H19N3O2S
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-thiazol-4-yl)methanone
—— 1-[(2R)-4-acetyl-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]-4-(1,2,4-triazol-1-yl)butan-1-one —— C23H31N5O4
1-[(2R)-4-acetyl-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]-4-(1,2,4-triazol-1-yl)butan-1-one
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrimidin-5-ylmethanone —— C17H20N4O2
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrimidin-5-ylmethanone
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1-methylpyrazol-3-yl)methanone —— C17H22N4O2
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1-methylpyrazol-3-yl)methanone
—— N-[5-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]-4-methyl-1,3-thiazol-2-yl]methanesulfonamide —— C18H24N4O4S2
N-[5-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]-4-methyl-1,3-thiazol-2-yl]methanesulfonamide
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-methyl-1,2-oxazol-5-yl)methanone —— C17H21N3O3
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-methyl-1,2-oxazol-5-yl)methanone
—— 1-[(2S)-2-[[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(2-fluorophenyl)ethanone —— C25H32FN3O2
1-[(2S)-2-[[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(2-fluorophenyl)ethanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methoxyethanone —— C15H22N2O3
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methoxyethanone
—— 1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylsulfonylphenyl)ethanone —— C22H23N3O4S
1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylsulfonylphenyl)ethanone
—— cyclopropyl-[(2R)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]methanone —— C19H26N2O2
cyclopropyl-[(2R)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]methanone
—— 1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(3-methylphenyl)ethanone —— C26H35N3O2
1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(3-methylphenyl)ethanone
—— 1-[(2R)-7-methoxy-1'-(piperidine-4-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C23H33N3O4
1-[(2R)-7-methoxy-1'-(piperidine-4-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— 2-methyl-1-[(2S)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]propan-1-one —— C19H28N2O2
2-methyl-1-[(2S)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]propan-1-one
—— [(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3,4,5-trimethoxyphenyl)methanone —— C23H25N3O5
[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3,4,5-trimethoxyphenyl)methanone
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methoxyethanone —— C15H22N2O3
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methoxyethanone
—— 1-[(2R)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(3-methylphenyl)ethanone —— C26H35N3O2
1-[(2R)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(3-methylphenyl)ethanone
—— 1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(2,4-dimethyl-1,3-thiazol-5-yl)ethanone —— C24H34N4O2S
1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(2,4-dimethyl-1,3-thiazol-5-yl)ethanone
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-methyl-1,2-oxazol-5-yl)methanone —— C17H21N3O3
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-methyl-1,2-oxazol-5-yl)methanone
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-methylpyrazol-3-yl)methanone —— C17H22N4O2
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-methylpyrazol-3-yl)methanone
—— 2-[(3R)-1,1-dioxothiolan-3-yl]-1-[(2R)-1'-prop-2-enylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C23H32N2O4S
2-[(3R)-1,1-dioxothiolan-3-yl]-1-[(2R)-1'-prop-2-enylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— 1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(4-fluorophenyl)ethanone —— C25H32FN3O2
1-[(2S)-2-[[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]pyrrolidin-1-yl]-2-(4-fluorophenyl)ethanone
—— (2S)-1'-benzylspiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-azepane] —— C21H26N2O
(2S)-1'-benzylspiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-azepane]
—— 1-[(2S)-1'-(1,5-dimethylpyrazole-4-carbonyl)-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C23H30N4O4
1-[(2S)-1'-(1,5-dimethylpyrazole-4-carbonyl)-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— 1'-(3,6-dihydro-2H-pyran-5-ylmethyl)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C21H30N2O4S
1'-(3,6-dihydro-2H-pyran-5-ylmethyl)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethanone —— C23H30N2O5
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethanone
—— 1-[1'-(3,6-dihydro-2H-pyran-5-ylmethyl)-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C22H30N2O3
1-[1'-(3,6-dihydro-2H-pyran-5-ylmethyl)-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— (2R)-1'-benzylspiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-azepane] —— C21H26N2O
(2R)-1'-benzylspiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-azepane]
—— 2-[(3R)-1,1-dioxothiolan-3-yl]-1-[(2S)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C22H32N2O5S
2-[(3R)-1,1-dioxothiolan-3-yl]-1-[(2S)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— 1-[1'-[[2-(2-Methoxyethyl)pyrimidin-5-yl]methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C24H32N4O3
1-[1'-[[2-(2-Methoxyethyl)pyrimidin-5-yl]methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— N,N-diethyl-2-(7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)acetamide —— C21H33N3O4S
N,N-diethyl-2-(7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)acetamide