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吡啶并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2S)-2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide —— C18H14F3N3O3
N-[(2S)-2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide
—— N-[(2R)-2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide —— C18H14F3N3O3
N-[(2R)-2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide
—— (5E)-3-cyclopentyl-5-[[2-(3-imidazol-1-ylpropylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C23H24N6O2S2
(5E)-3-cyclopentyl-5-[[2-(3-imidazol-1-ylpropylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 2-[(4-tert-butylphenyl)methylsulfanyl]-3-[[(2R)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-4-one —— C23H27N3O2S
2-[(4-tert-butylphenyl)methylsulfanyl]-3-[[(2R)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
—— 3-[[(2S)-oxolan-2-yl]methyl]-2-(3-phenoxypropylsulfanyl)pyrido[2,3-d]pyrimidin-4-one —— C21H23N3O3S
3-[[(2S)-oxolan-2-yl]methyl]-2-(3-phenoxypropylsulfanyl)pyrido[2,3-d]pyrimidin-4-one
—— 7-chloro-2-[[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]pyrido[1,2-a]pyrimidin-4-one —— C17H16ClN3OS
7-chloro-2-[[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 6-Amino-5-(benzenesulfonyl)-7-(3-ethoxypropyl)-11-methyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one —— C23H25N4O4S+
6-Amino-5-(benzenesulfonyl)-7-(3-ethoxypropyl)-11-methyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one
—— methyl (2S)-3-[benzyl-[(4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]amino]-2-methylpropanoate —— C21H23N3O3
methyl (2S)-3-[benzyl-[(4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]amino]-2-methylpropanoate
—— 3-[(2R)-2-hydroxy-2-(2-methoxy-5-methylphenyl)ethyl]pyrido[2,3-d]pyrimidin-4-one —— C17H17N3O3
3-[(2R)-2-hydroxy-2-(2-methoxy-5-methylphenyl)ethyl]pyrido[2,3-d]pyrimidin-4-one
—— 2-[[[(1R)-1-cyclopropylethyl]-methylamino]methyl]pyrido[1,2-a]pyrimidin-4-one —— C15H19N3O
2-[[[(1R)-1-cyclopropylethyl]-methylamino]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 2-[[[(1S)-1-cyclopropylethyl]-methylamino]methyl]pyrido[1,2-a]pyrimidin-4-one —— C15H19N3O
2-[[[(1S)-1-cyclopropylethyl]-methylamino]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 3-[(2S)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]pyrido[2,3-d]pyrimidin-4-one —— C16H13F2N3O3
3-[(2S)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]pyrido[2,3-d]pyrimidin-4-one
—— 2-[[(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl]-7-bromopyrido[1,2-a]pyrimidin-4-one —— C20H17BrN4OS
2-[[(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl]-7-bromopyrido[1,2-a]pyrimidin-4-one
—— 2-[[ethyl-[(3S)-1-[(1S)-1-phenylethyl]pyrrolidin-3-yl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one —— C23H28N4O
2-[[ethyl-[(3S)-1-[(1S)-1-phenylethyl]pyrrolidin-3-yl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one
—— (2R)-2-(4-fluorophenyl)-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one —— C13H10FN3O
(2R)-2-(4-fluorophenyl)-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one
—— (2R)-2-(4-hydroxy-3-methoxyphenyl)-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one —— C14H13N3O3
(2R)-2-(4-hydroxy-3-methoxyphenyl)-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one
—— (2S)-2-(4-hydroxy-3-methoxyphenyl)-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one —— C14H13N3O3
(2S)-2-(4-hydroxy-3-methoxyphenyl)-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one
—— (2S)-2-(4-fluorophenyl)-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one —— C13H10FN3O
(2S)-2-(4-fluorophenyl)-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one
—— Dibutyl-[3-(4-oxopyrido[2,3-d]pyrimidin-3-yl)propyl]azanium —— C18H29N4O+
Dibutyl-[3-(4-oxopyrido[2,3-d]pyrimidin-3-yl)propyl]azanium
—— 2-[[ethyl-[(3R)-1-[(1S)-1-phenylethyl]pyrrolidin-3-yl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one —— C23H28N4O
2-[[ethyl-[(3R)-1-[(1S)-1-phenylethyl]pyrrolidin-3-yl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one
—— N-[(1S)-1-(2,4-difluorophenyl)ethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide —— C17H13F2N3O2
N-[(1S)-1-(2,4-difluorophenyl)ethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide
—— [(Z)-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylideneamino]urea —— C16H20N6O3
[(Z)-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylideneamino]urea
—— 6-amino-N-cyclohexyl-11-methyl-2-oxo-7-propyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C22H28N5O2+
6-amino-N-cyclohexyl-11-methyl-2-oxo-7-propyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— (5S)-5-(3-bromo-4-fluorophenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C17H17BrFN3O2S
(5S)-5-(3-bromo-4-fluorophenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-5-(3-ethoxy-4-methoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C20H25N3O4S
(5S)-5-(3-ethoxy-4-methoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(3,4-diethoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C21H27N3O4S
(5R)-5-(3,4-diethoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-5-(3,4-diethoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C21H27N3O4S
(5S)-5-(3,4-diethoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-1-methyl-5-[4-[(2-methylphenyl)methoxy]phenyl]-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C25H27N3O3S
(5R)-1-methyl-5-[4-[(2-methylphenyl)methoxy]phenyl]-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-1-methyl-5-(4-phenylmethoxyphenyl)-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C24H25N3O3S
(5S)-1-methyl-5-(4-phenylmethoxyphenyl)-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(3-methoxy-4-propan-2-yloxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C21H27N3O4S
(5R)-5-(3-methoxy-4-propan-2-yloxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-1-methyl-5-(4-phenylmethoxyphenyl)-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C24H25N3O3S
(5R)-1-methyl-5-(4-phenylmethoxyphenyl)-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(3-methoxy-4-prop-2-ynoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C21H23N3O4S
(5R)-5-(3-methoxy-4-prop-2-ynoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-1-methyl-5-[4-(2-phenylethoxy)phenyl]-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C25H27N3O3S
(5R)-1-methyl-5-[4-(2-phenylethoxy)phenyl]-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— 2-[4-[(5S)-1-methyl-4,7-dioxo-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidin-5-yl]phenoxy]acetamide —— C19H22N4O4S
2-[4-[(5S)-1-methyl-4,7-dioxo-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidin-5-yl]phenoxy]acetamide
—— (5S)-5-[3-methoxy-4-(2-methylpropoxy)phenyl]-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C22H29N3O4S
(5S)-5-[3-methoxy-4-(2-methylpropoxy)phenyl]-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-1-methyl-5-[4-(2-methylpropoxy)phenyl]-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C21H27N3O3S
(5R)-1-methyl-5-[4-(2-methylpropoxy)phenyl]-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-[3-methoxy-4-(2-methylpropoxy)phenyl]-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C22H29N3O4S
(5R)-5-[3-methoxy-4-(2-methylpropoxy)phenyl]-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(3-methoxy-4-prop-2-enoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C21H25N3O4S
(5R)-5-(3-methoxy-4-prop-2-enoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-5-(3-methoxy-4-prop-2-enoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C21H25N3O4S
(5S)-5-(3-methoxy-4-prop-2-enoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-[4-[(2-fluorophenyl)methoxy]phenyl]-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C24H24FN3O3S
(5R)-5-[4-[(2-fluorophenyl)methoxy]phenyl]-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-5-(3-hydroxy-4-methoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C18H21N3O4S
(5S)-5-(3-hydroxy-4-methoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(3-bromo-4-fluorophenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C17H17BrFN3O2S
(5R)-5-(3-bromo-4-fluorophenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-5-[4-[(2-fluorophenyl)methoxy]phenyl]-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C24H24FN3O3S
(5S)-5-[4-[(2-fluorophenyl)methoxy]phenyl]-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-1-methyl-5-(2-prop-2-enoxyphenyl)-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C20H23N3O3S
(5S)-1-methyl-5-(2-prop-2-enoxyphenyl)-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(3-ethoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C19H23N3O3S
(5R)-5-(3-ethoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(2-ethoxy-3-methoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C20H25N3O4S
(5R)-5-(2-ethoxy-3-methoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-1-methyl-5-(2-prop-2-enoxyphenyl)-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C20H23N3O3S
(5R)-1-methyl-5-(2-prop-2-enoxyphenyl)-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(3-ethoxy-4-methoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C20H25N3O4S
(5R)-5-(3-ethoxy-4-methoxyphenyl)-1-methyl-2-propylsulfanyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-2-ethylsulfanyl-5-(3-hydroxyphenyl)-1-methyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C16H17N3O3S
(5R)-2-ethylsulfanyl-5-(3-hydroxyphenyl)-1-methyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-2-ethylsulfanyl-5-(3-hydroxyphenyl)-1-methyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione —— C16H17N3O3S
(5S)-2-ethylsulfanyl-5-(3-hydroxyphenyl)-1-methyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-4,7-dione