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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-Oxazolamine, 2-phenyl-N-(phenylmethyl)-4-(phenylsulfonyl)- 145317-83-5 C22H18N2O3S
5-Oxazolamine, 2-phenyl-N-(phenylmethyl)-4-(phenylsulfonyl)-
—— 2-(4-Fluoro-3-phenylindazol-1-yl)-1,3-thiazole-4-carboxylic acid 1204771-71-0 C17H10FN3O2S
2-(4-Fluoro-3-phenylindazol-1-yl)-1,3-thiazole-4-carboxylic acid
—— 2-(5-Fluoro-3-phenylindazol-1-yl)-1,3-thiazole-4-carboxylic acid 1204771-72-1 C17H10FN3O2S
2-(5-Fluoro-3-phenylindazol-1-yl)-1,3-thiazole-4-carboxylic acid
—— 1-Methyl-4-trifluoromethyl-5-(p-nitrophenyl)imidazole 129247-50-3 C11H8F3N3O2
1-Methyl-4-trifluoromethyl-5-(p-nitrophenyl)imidazole
—— 3-chloromethyl-5-cyclohexyl-1,2,4-oxadiazole 189130-88-9 C9H13ClN2O
3-chloromethyl-5-cyclohexyl-1,2,4-oxadiazole
—— 5-cyclohexyl-3-[4-methyl-3-(pyrrolidine-1-sulfonyl)-phenyl]-[1,2,4]oxadiazole 1046270-99-8 C19H25N3O3S
5-cyclohexyl-3-[4-methyl-3-(pyrrolidine-1-sulfonyl)-phenyl]-[1,2,4]oxadiazole
—— 5-{3-[4-(5-cyclohexyl-1,2,4-oxadiazol-3-yl)phenoxy]propyl}-3-methylisoxazole 173899-96-2 C21H25N3O3
5-{3-[4-(5-cyclohexyl-1,2,4-oxadiazol-3-yl)phenoxy]propyl}-3-methylisoxazole
—— cyclohexanecarboxylic acid (1-benzyl-3-methyl-5-phenyl-1H-pyrazol-4-yl)-amide 824969-25-7 C24H27N3O
cyclohexanecarboxylic acid (1-benzyl-3-methyl-5-phenyl-1H-pyrazol-4-yl)-amide
—— 4-Methyl-3-thiophen-2-yl-5-trifluoromethyl-isoxazole 1124199-04-7 C9H6F3NOS
4-Methyl-3-thiophen-2-yl-5-trifluoromethyl-isoxazole
—— [4-Chloro-5-methyl-2-(2-phenyl-2H-pyrazol-3-yl)-phenoxy]-acetic acid ethyl ester 293740-20-2 C20H19ClN2O3
[4-Chloro-5-methyl-2-(2-phenyl-2H-pyrazol-3-yl)-phenoxy]-acetic acid ethyl ester
—— cyclohexanecarboxylic acid-{4-[2-(4-nitro-phenyl)-3H-imidazol-4-yl]-phenyl}-amide 783364-08-9 C22H22N4O3
cyclohexanecarboxylic acid-{4-[2-(4-nitro-phenyl)-3H-imidazol-4-yl]-phenyl}-amide
—— N-[2-(4-methoxyphenyl)-6-methyl-2H-benzotriazol-5-yl]-2-methyl-3-nitrobenzamide 6173-62-2 C22H19N5O4
N-[2-(4-methoxyphenyl)-6-methyl-2H-benzotriazol-5-yl]-2-methyl-3-nitrobenzamide
—— Cyclohexanecarboxylic acid [2-(4-nitro-phenyl)-3H-imidazo[4,5-c]pyridine-6-yl]-amide 675200-25-6 C19H19N5O3
Cyclohexanecarboxylic acid [2-(4-nitro-phenyl)-3H-imidazo[4,5-c]pyridine-6-yl]-amide
—— N-((4-bromo-5-(5-bromoselenophen-2-yl)-1-(2,4-dichlorophenyl)-1H-pyrazol-3-yl)methyl)cyclohexanecarboxamide 1003004-57-6 C21H19Br2Cl2N3SSe
N-((4-bromo-5-(5-bromoselenophen-2-yl)-1-(2,4-dichlorophenyl)-1H-pyrazol-3-yl)methyl)cyclohexanecarboxamide
—— Methyl 2-(6-bromo-3-bromomethyl-1H-indazol-1-yl)-6-methoxybenzoate 238756-61-1 C17H14Br2N2O3
Methyl 2-(6-bromo-3-bromomethyl-1H-indazol-1-yl)-6-methoxybenzoate
—— 1-[(4-Bromophenyl)methylideneamino]-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)thiourea 249516-34-5 C19H18BrN5OS
1-[(4-Bromophenyl)methylideneamino]-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)thiourea
—— 4-[2-[2-[4-[(4-Chlorophenyl)methylsulfanyl]phenoxy]propanoyl]-4-methyl-1,3-thiazol-5-yl]butanoic acid 273939-20-1 C24H24ClNO4S2
4-[2-[2-[4-[(4-Chlorophenyl)methylsulfanyl]phenoxy]propanoyl]-4-methyl-1,3-thiazol-5-yl]butanoic acid
—— Methyl 2-(6-bromo-3-methyl-1H-indazol-1-yl)-6-methoxybenzoate 238756-60-0 C17H15BrN2O3
Methyl 2-(6-bromo-3-methyl-1H-indazol-1-yl)-6-methoxybenzoate
—— (VIIb) 41347-39-1 C17H24N2O3
(VIIb)
—— 4-[2-[2-[4-[(4-Chlorophenyl)methylsulfanyl]phenoxy]butanoyl]-4-methyl-1,3-thiazol-5-yl]butanoic acid 273939-21-2 C25H26ClNO4S2
4-[2-[2-[4-[(4-Chlorophenyl)methylsulfanyl]phenoxy]butanoyl]-4-methyl-1,3-thiazol-5-yl]butanoic acid
—— 4-(2-Phenyl-3H-imidazol-4-yl)-piperidine 737766-58-4 C14H17N3
4-(2-Phenyl-3H-imidazol-4-yl)-piperidine
—— 5-(1-ethyl-1H-tetrazol-5-yl)-2-methoxy-N-(2-phenylethyl)benzenesulfonamide 6240-14-8 C18H21N5O3S
5-(1-ethyl-1H-tetrazol-5-yl)-2-methoxy-N-(2-phenylethyl)benzenesulfonamide
—— 2-({[5-Benzyl-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}methyl)-N-[(pyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide 5948-80-1 C27H24N6OS2
2-({[5-Benzyl-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}methyl)-N-[(pyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
—— 1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazole-3-carbaldehyde 1287761-07-2 C17H14N2O3S
1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazole-3-carbaldehyde
—— 3-[1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazol-3-yl]-propionic acid ethyl ester 1287761-09-4 C21H22N2O4S
3-[1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazol-3-yl]-propionic acid ethyl ester
—— 1-isopropyl-4,5-diphenyl-1,2,3-triazole 55324-05-5 C17H17N3
1-isopropyl-4,5-diphenyl-1,2,3-triazole
—— (E)-3-[1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazol-3-yl]-acrylic acid ethyl ester 1287761-08-3 C21H20N2O4S
(E)-3-[1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazol-3-yl]-acrylic acid ethyl ester
—— 1-((4aR,9bS)-2,8-Dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido(4,3-b)indol-5-yl)-2-(1-(4-chlorophenyl)tetrazol-5-yl)sulfanyl-ethanone, 4aR,9bs 1375078-57-1 C22H23ClN6OS
1-((4aR,9bS)-2,8-Dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido(4,3-b)indol-5-yl)-2-(1-(4-chlorophenyl)tetrazol-5-yl)sulfanyl-ethanone, 4aR,9bs
—— 7-tert-butyl 1-methyl 3-phenyl-8,9-dihydro-5H-imidazo[1,5-d][1,4]diazepine-1,7(6H)-dicarboxylate 1229008-01-8 C20H25N3O4
7-tert-butyl 1-methyl 3-phenyl-8,9-dihydro-5H-imidazo[1,5-d][1,4]diazepine-1,7(6H)-dicarboxylate
—— 7-(4-chlorophenyl)-6-(4-bromophenyl)amino-2-methyltriazolo-triazolone 116088-29-0 C16H12Br2N6O
7-(4-chlorophenyl)-6-(4-bromophenyl)amino-2-methyltriazolo-triazolone
—— (4-(1H-1,2,3-triazol-1-yl)phenyl)methanamine 894779-96-5 C9H10N4
(4-(1H-1,2,3-triazol-1-yl)phenyl)methanamine
—— 2-(3-chlorophenyl)-3,4-dimethyl-2,6-dihydro-7H-pyrazolo[3,4-d]pyridazin-7-thione 791824-79-8 C13H11ClN4S
2-(3-chlorophenyl)-3,4-dimethyl-2,6-dihydro-7H-pyrazolo[3,4-d]pyridazin-7-thione
—— 1-Methyl-4-(p-nitrophenyl)-5-trifluoromethylimidazole 129247-44-5 C11H8F3N3O2
1-Methyl-4-(p-nitrophenyl)-5-trifluoromethylimidazole
—— 1-Benzyl-5-phenyl-3-p-tolyl-1H-[1,2,4]triazole 80465-13-0 C22H19N3
1-Benzyl-5-phenyl-3-p-tolyl-1H-[1,2,4]triazole
—— 1-(2,3-dichloro-4-((2-((7-methyl-1H-indazol-5-yl)amino)pyrimidin-4-yl)oxy)phenyl)-3-(1-(p-tolyl)-3-(trimethylsilyl)-1H-pyrazol-5-yl)urea 1571073-71-6 C32H31Cl2N9O2Si
1-(2,3-dichloro-4-((2-((7-methyl-1H-indazol-5-yl)amino)pyrimidin-4-yl)oxy)phenyl)-3-(1-(p-tolyl)-3-(trimethylsilyl)-1H-pyrazol-5-yl)urea
—— 9-Bromo-5-(4-bromoanilino)-2-phenyl-[1,2,4]triazolo[1,2-a][1,2,4]benzotriazine-1,3-dione 1215222-90-4 C21H13Br2N5O2
9-Bromo-5-(4-bromoanilino)-2-phenyl-[1,2,4]triazolo[1,2-a][1,2,4]benzotriazine-1,3-dione
—— 3-((4-(2,3-dichloro-4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)ureido)-phenoxy)pyrimidin-2-yl)amino)-N-(2-(dimethylamino)ethyl)-5-ethynylbenzamide 1562515-84-7 C37H37Cl2N9O3
3-((4-(2,3-dichloro-4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)ureido)-phenoxy)pyrimidin-2-yl)amino)-N-(2-(dimethylamino)ethyl)-5-ethynylbenzamide
—— N-[2-methyl-5-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-2-phenylacetamide 5836-30-6 C23H20N2O2
N-[2-methyl-5-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-2-phenylacetamide
—— diethyl 3-oxo-4-methyl-5-benzyl-1H-pyrazole-1,2(3H)-dicarboxylate 1541204-78-7 C17H20N2O5
diethyl 3-oxo-4-methyl-5-benzyl-1H-pyrazole-1,2(3H)-dicarboxylate
—— diisopropyl 3-oxo-4-methyl-5-benzyl-1H-pyrazole-1,2(3H)-dicarboxylate 1541204-80-1 C19H24N2O5
diisopropyl 3-oxo-4-methyl-5-benzyl-1H-pyrazole-1,2(3H)-dicarboxylate
—— 1-(3-(tert-butyl)-1-(p-tolyl)-1H-pyrazol-5-yl)-3-(2,3-dichloro-4-((2-((3-methoxy-5-(2-(2-(2-methoxyethoxy)ethoxy)ethoxy)phenyl)amino)pyrimidin-4-yl)oxy)phenyl)urea 1610449-78-9 C39H45Cl2N7O7
1-(3-(tert-butyl)-1-(p-tolyl)-1H-pyrazol-5-yl)-3-(2,3-dichloro-4-((2-((3-methoxy-5-(2-(2-(2-methoxyethoxy)ethoxy)ethoxy)phenyl)amino)pyrimidin-4-yl)oxy)phenyl)urea
—— 1-(2,3-dichloro-4-((2-chloropyrimidin-4-yl)oxy)phenyl)-3-(1-(p-tolyl)-3-(trimethylsilyl)-1H-pyrazol-5-yl)urea 1571074-01-5 C24H23Cl3N6O2Si
1-(2,3-dichloro-4-((2-chloropyrimidin-4-yl)oxy)phenyl)-3-(1-(p-tolyl)-3-(trimethylsilyl)-1H-pyrazol-5-yl)urea
—— 1-(3-(tert-butyl)-1-(p-tolyl)-1H-pyrazol-5-yl)-3-(2,3-dichloro-4-((2-((3-methoxy-5-(3-morpholinopropoxy)phenyl)amino)pyrimidin-4-yl)oxy)phenyl)urea 1610449-95-0 C39H44Cl2N8O5
1-(3-(tert-butyl)-1-(p-tolyl)-1H-pyrazol-5-yl)-3-(2,3-dichloro-4-((2-((3-methoxy-5-(3-morpholinopropoxy)phenyl)amino)pyrimidin-4-yl)oxy)phenyl)urea
—— 1-n-butyl-3-<2-<<2-hydroxy-3-<4-(4-methyl-2-imidazolyl)phenoxy>propyl>amino>ethyl>urea 126007-88-3 C20H31N5O3
1-n-butyl-3-<2-<<2-hydroxy-3-<4-(4-methyl-2-imidazolyl)phenoxy>propyl>amino>ethyl>urea
—— 1-(2,3-dichloro-4-((2-((3-(cyclopropylsulfonyl)phenyl)amino)pyrimidin-4-yl)oxy)phenyl)-3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)urea 1610449-46-1 C33H31Cl2N7O4S
1-(2,3-dichloro-4-((2-((3-(cyclopropylsulfonyl)phenyl)amino)pyrimidin-4-yl)oxy)phenyl)-3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)urea
—— S,S-dimethyl-N-(3-((4-(2,3-dichloro-4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)ureido)phenoxy)pyrimidin-2-yl)amino)-5-methoxyphenyl)sulfoximine 1610449-48-3 C33H34Cl2N8O4S
S,S-dimethyl-N-(3-((4-(2,3-dichloro-4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)ureido)phenoxy)pyrimidin-2-yl)amino)-5-methoxyphenyl)sulfoximine
—— 3-((4-(2,3-dichloro-4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)ureido)-phenoxy)pyrimidin-2-yl)amino)-5-ethynylbenzamide 1562515-80-3 C33H28Cl2N8O3
3-((4-(2,3-dichloro-4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)ureido)-phenoxy)pyrimidin-2-yl)amino)-5-ethynylbenzamide
—— 1-(2,3-dichloro-4-((2-((3-methoxy-5-(2-(2-(2-methoxyethoxy)ethoxy)ethoxy)phenyl)amino)pyrimidin-4-yl)oxy)phenyl)-3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)urea 1610449-57-4 C38H43Cl2N7O7
1-(2,3-dichloro-4-((2-((3-methoxy-5-(2-(2-(2-methoxyethoxy)ethoxy)ethoxy)phenyl)amino)pyrimidin-4-yl)oxy)phenyl)-3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)urea
—— N-[4-(1,3-benzoxazol-2-yl)phenyl]-2-(4-bromophenoxy)acetamide 5838-75-5 C21H15BrN2O3
N-[4-(1,3-benzoxazol-2-yl)phenyl]-2-(4-bromophenoxy)acetamide
—— (E)-7-[4-[4-[[(2-Phenoxyethyl)amino]carbonyl]-2-oxazolyl]phenyl]-7-(3-pyridyl)hept-6-enoic Acid 200399-98-0 C30H29N3O5
(E)-7-[4-[4-[[(2-Phenoxyethyl)amino]carbonyl]-2-oxazolyl]phenyl]-7-(3-pyridyl)hept-6-enoic Acid