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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-anilino-4-(1,2-dipropyl-imidazol-5-yl)pyrimidine 600639-32-5 C19H23N5
2-anilino-4-(1,2-dipropyl-imidazol-5-yl)pyrimidine
—— US10138229, Example 17 1558036-44-4 C19H23N5O4S
US10138229, Example 17
—— 5-methyl-4-(N-cyclopropylmethyl-N-propionamido)isoxazole 600699-51-2 C11H16N2O2
5-methyl-4-(N-cyclopropylmethyl-N-propionamido)isoxazole
—— ethyl 3-(4-chlorophenyl)-7-(2-cyanoethyl)-2-(2,4-dichlorophenyl)-6-oxo-6,7-dihydro-2H-pyrazolo[3,4-b]pyridine-5-carboxylate 1174629-87-8 C24H17Cl3N4O3
ethyl 3-(4-chlorophenyl)-7-(2-cyanoethyl)-2-(2,4-dichlorophenyl)-6-oxo-6,7-dihydro-2H-pyrazolo[3,4-b]pyridine-5-carboxylate
—— 7-chloro-3-(4-methoxyphenyl)-2-pentyl-2H-indazole 680611-43-2 C19H21ClN2O
7-chloro-3-(4-methoxyphenyl)-2-pentyl-2H-indazole
—— tert-butyl {3-[3-(4-chloro-phenyl)-5-methyl-[1,2,4]triazol-1-yl]-1,1-dimethyl-propyl}-carbamate 906101-50-6 C19H27ClN4O2
tert-butyl {3-[3-(4-chloro-phenyl)-5-methyl-[1,2,4]triazol-1-yl]-1,1-dimethyl-propyl}-carbamate
—— (2-Dodecyl-2H-tetrazol-5-yl)-fluoro-acetic acid ethyl ester 1027545-17-0 C17H31FN4O2
(2-Dodecyl-2H-tetrazol-5-yl)-fluoro-acetic acid ethyl ester
—— 1-(4-amino-3-methylbenzyl)-N-(propane-2-yl)-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide 1207090-28-5 C16H19F3N4O
1-(4-amino-3-methylbenzyl)-N-(propane-2-yl)-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide
—— 8-chloro-3,4-dimethyl-1-(2-methylphenyl)imidazo[1,5-a]quinoxaline 1159794-30-5 C19H16ClN3
8-chloro-3,4-dimethyl-1-(2-methylphenyl)imidazo[1,5-a]quinoxaline
—— [1-(2-pyrazol-1-yl-ethyl)-1H-pyrazol-4-yl]-{3-[4-(pyrrolidine-1-sulfonyl)-phenyl]-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl}-amine 1448694-10-7 C22H23N11O2S
[1-(2-pyrazol-1-yl-ethyl)-1H-pyrazol-4-yl]-{3-[4-(pyrrolidine-1-sulfonyl)-phenyl]-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl}-amine
—— (3-acetyl-1-(4-chlorophenyl)-1H-[1,2,4]triazol-5-sulfanyl)-acetic acid 1164236-84-3 C12H10ClN3O3S
(3-acetyl-1-(4-chlorophenyl)-1H-[1,2,4]triazol-5-sulfanyl)-acetic acid
—— 2-Bromo-5-(4-chlorophenyl)thiazole 1353856-05-9 C9H5BrClNS
2-Bromo-5-(4-chlorophenyl)thiazole
—— 4-(4-tert-butylphenyl)-3-(4-methylphenyl)-4,5-dihydro-1H-pyrrolo[3,4-c]pyrazol-6-one 901732-24-9 C22H23N3O
4-(4-tert-butylphenyl)-3-(4-methylphenyl)-4,5-dihydro-1H-pyrrolo[3,4-c]pyrazol-6-one
—— 1-benzyl-4-(benzyloxy)-3-phenyl-1H-pyrazole-5-carboxylic acid 1197866-57-1 C24H20N2O3
1-benzyl-4-(benzyloxy)-3-phenyl-1H-pyrazole-5-carboxylic acid
—— 3,4-dichloro-N-methyl-N-thiophen-2-ylsulfonyl-1,2-thiazole-5-carboxamide 367505-59-7 C9H6Cl2N2O3S3
3,4-dichloro-N-methyl-N-thiophen-2-ylsulfonyl-1,2-thiazole-5-carboxamide
—— 2-(1'-methoxy)methyl-1-methylimidazole 1667730-79-1 C6H10N2O
2-(1'-methoxy)methyl-1-methylimidazole
—— 2-(3-(tert-butyl)-1-(3,4-difluorophenyl)-1H-pyrazol-5-yl)-2-oxoacetyl chloride 1087163-05-0 C15H13ClF2N2O2
2-(3-(tert-butyl)-1-(3,4-difluorophenyl)-1H-pyrazol-5-yl)-2-oxoacetyl chloride
—— 2-(4-Chloro-phenoxy)-N-(5-sulfamoyl-[1,3,4]thiadiazol-2-yl)-acetamide 2409-30-5 C10H9ClN4O4S2
2-(4-Chloro-phenoxy)-N-(5-sulfamoyl-[1,3,4]thiadiazol-2-yl)-acetamide
—— 2-[5-(4,6-bis-butylsulfanyl-[1,3,5]triazin-2-ylamino)-benzo[1,2,3]triazol-2-yl]-phenol 100768-87-4 C23H27N7OS2
2-[5-(4,6-bis-butylsulfanyl-[1,3,5]triazin-2-ylamino)-benzo[1,2,3]triazol-2-yl]-phenol
—— (5-<i>sec</i>-butylsulfanyl-[1,3,4]thiadiazol-2-yl)-trimethyl-urea 55693-94-2 C10H18N4OS2
(5-<i>sec</i>-butylsulfanyl-[1,3,4]thiadiazol-2-yl)-trimethyl-urea
—— (7,17-bis(azophenyl)-6,8,15,17-tetramethyldibenzo[b,i][1,4,8,11]-tetraazacyclotetradecinato)nickel(II) 154508-01-7 C34H30N8Ni
(7,17-bis(azophenyl)-6,8,15,17-tetramethyldibenzo[b,i][1,4,8,11]-tetraazacyclotetradecinato)nickel(II)
—— 3-dibutylsulfamoyl-[1,2,4]triazole-1-carboxylic acid diallylamide 43173-64-4 C17H29N5O3S
3-dibutylsulfamoyl-[1,2,4]triazole-1-carboxylic acid diallylamide
—— 1,1,1-trifluoro-4-[5-fluoro-2-(methyloxy)phenyl]-4-methyl-2-[({6-methyl-1-[3-({(2S)-2-[(methyloxy)methyl]-1-pyrrolidinyl}carbonyl)phenyl]-1H-indazol-4-yl}amino)methyl]-2-pentanol 1020169-51-0 C35H40F4N4O4
1,1,1-trifluoro-4-[5-fluoro-2-(methyloxy)phenyl]-4-methyl-2-[({6-methyl-1-[3-({(2S)-2-[(methyloxy)methyl]-1-pyrrolidinyl}carbonyl)phenyl]-1H-indazol-4-yl}amino)methyl]-2-pentanol
—— 1-[3-[4-(p-chlorophenyl)-5-phenyl-([1,2,3]triazol-2-yl)]propyl]-imidazole 1025357-98-5 C20H18ClN5
1-[3-[4-(p-chlorophenyl)-5-phenyl-([1,2,3]triazol-2-yl)]propyl]-imidazole
—— tert-butyl [4-(4-aminosulfonylphenyl)-1-methyl-3-(4-pyridyl)-1H-pyrazol-5-yl]carboxylate 259172-84-4 C20H22N4O4S
tert-butyl [4-(4-aminosulfonylphenyl)-1-methyl-3-(4-pyridyl)-1H-pyrazol-5-yl]carboxylate
—— N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(3-methoxyphenyl)propan-2-yl]pyrimidine-4-carboxamide 1034148-90-7 C28H24FN5O3
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(3-methoxyphenyl)propan-2-yl]pyrimidine-4-carboxamide
—— 3-diethylsulfamoyl-[1,2,4]triazole-1-carboxylic acid allyl-isopropyl-amide 43174-06-7 C13H23N5O3S
3-diethylsulfamoyl-[1,2,4]triazole-1-carboxylic acid allyl-isopropyl-amide
—— 1-cycloheptyl-9-phenyl-1,9-dihydro-purin-6-one 1056634-20-8 C18H20N4O
1-cycloheptyl-9-phenyl-1,9-dihydro-purin-6-one
—— (E)-3-[2-Butyl-1-(2-(2,4-difluorobenzyloxy)-4-methoxy)phenyl-1H-imidazol-5-yl]-2-[(2-methoxy-4,5-methylenedioxyphenyl)methyl]-2-propenoic acid 178533-79-4 C33H32F2N2O7
(E)-3-[2-Butyl-1-(2-(2,4-difluorobenzyloxy)-4-methoxy)phenyl-1H-imidazol-5-yl]-2-[(2-methoxy-4,5-methylenedioxyphenyl)methyl]-2-propenoic acid
—— 4-(2-aminophenyl)-1,3,5-tributyl-1,3-dihydro-2H-imidazol-2-one 1020846-63-2 C21H33N3O
4-(2-aminophenyl)-1,3,5-tributyl-1,3-dihydro-2H-imidazol-2-one
—— 4-((1-(2,6-dichlorophenyl)-4-isopropyl-1H-1,2,3-triazol-5-yl)methoxy)azepane 1103500-57-7 C18H24Cl2N4O
4-((1-(2,6-dichlorophenyl)-4-isopropyl-1H-1,2,3-triazol-5-yl)methoxy)azepane
—— N-benzoyl-N'-[1-(4-nitrophenyl)-3-(4-fluorophenyl)-4-pyrazolylidene]hydrazine 1246443-98-0 C23H16FN5O3
N-benzoyl-N'-[1-(4-nitrophenyl)-3-(4-fluorophenyl)-4-pyrazolylidene]hydrazine
—— 2-[2,6-Dichloro-4-(trifluoromethyl)phenyl]-6-(fluoromethyl)-4-(trifluoromethyl)pyrazolo[4,3-c]pyridin-3-amine 1447806-89-4 C15H7Cl2F7N4
2-[2,6-Dichloro-4-(trifluoromethyl)phenyl]-6-(fluoromethyl)-4-(trifluoromethyl)pyrazolo[4,3-c]pyridin-3-amine
—— 5-[3-({4-[(2,2-difluorocyclopropyl)methyl]-3-oxopiperazin-1-yl}methyl)phenyl]-1-(2,2-dimethylpropyl)-3-methyl-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1352424-44-2 C27H33F2N5O2
5-[3-({4-[(2,2-difluorocyclopropyl)methyl]-3-oxopiperazin-1-yl}methyl)phenyl]-1-(2,2-dimethylpropyl)-3-methyl-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— ethyl 1-[4-(butylcarbamoylsulfamoyl)phenyl]-5-(1-phenylprop-1-en-2-yl)pyrazole-3-carboxylate 81750-33-6 C26H30N4O5S
ethyl 1-[4-(butylcarbamoylsulfamoyl)phenyl]-5-(1-phenylprop-1-en-2-yl)pyrazole-3-carboxylate
—— N-(4-aminothiophen-3-yl)-5-[1-(3-dimethylaminopropyl)-3-phenethylureidomethyl]pyridine-2-carboxylic acid amide 1196981-15-3 C25H32N6O2S
N-(4-aminothiophen-3-yl)-5-[1-(3-dimethylaminopropyl)-3-phenethylureidomethyl]pyridine-2-carboxylic acid amide
—— N-(adamantan-1-ylmethyl)-1-(5-aminopyrazin-2-yl)-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide 1104269-99-9 C20H23F3N6O
N-(adamantan-1-ylmethyl)-1-(5-aminopyrazin-2-yl)-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide
—— 3-(3-chloro-4-cyclohexyloxy-phenyl)-5-o-tolyl-[1,2,4]oxadiazole 1035212-23-7 C21H21ClN2O2
3-(3-chloro-4-cyclohexyloxy-phenyl)-5-o-tolyl-[1,2,4]oxadiazole
—— N-Hydroxy-2-methyl-5-thiazolcarboxamid 60971-68-8 C5H6N2O2S
N-Hydroxy-2-methyl-5-thiazolcarboxamid
—— (rac)-2-(4-{1-[4-(2,6-difluoro-phenyl)-5-oxo-1-(4-trifluoromethyl-phenyl)-4,5-dihydro-1H-[1,2,4]triazol-3-yl]-pentyloxy}-2-methyl-phenoxy)-2-methyl-propionic acid 1050441-33-2 C31H30F5N3O5
(rac)-2-(4-{1-[4-(2,6-difluoro-phenyl)-5-oxo-1-(4-trifluoromethyl-phenyl)-4,5-dihydro-1H-[1,2,4]triazol-3-yl]-pentyloxy}-2-methyl-phenoxy)-2-methyl-propionic acid
—— 5-(3-methoxy-phenyl)-thiazole-4-carboxylic acid methyl ester 1038509-00-0 C12H11NO3S
5-(3-methoxy-phenyl)-thiazole-4-carboxylic acid methyl ester
—— N-benzyl-3-(5-phenyl-1,2,3-triazol-1-yl)pyrrolidine 143699-98-3 C19H20N4
N-benzyl-3-(5-phenyl-1,2,3-triazol-1-yl)pyrrolidine
—— 1,2-diamino-4,5-dimethylimidazole 618439-91-1 C5H10N4
1,2-diamino-4,5-dimethylimidazole
—— 2-phenyl-<i>N</i>-(4-phenyl-[1,2,3]triazol-1-yl)-acetamide 73227-10-8 C16H14N4O
2-phenyl-<i>N</i>-(4-phenyl-[1,2,3]triazol-1-yl)-acetamide
—— 3-(4-methanesulfonyl-phenyl)-1,5-diphenyl-4,5-dihydro-1<i>H</i>-pyrazole 72344-00-4 C22H20N2O2S
3-(4-methanesulfonyl-phenyl)-1,5-diphenyl-4,5-dihydro-1<i>H</i>-pyrazole
—— 1-[4-(8-bromo-6-methyl-3-phenyl-imidazo[1,2-a]pyridin-2-yl)-phenyl]-cyclobutylamine 1355998-75-2 C24H22BrN3
1-[4-(8-bromo-6-methyl-3-phenyl-imidazo[1,2-a]pyridin-2-yl)-phenyl]-cyclobutylamine
—— (2Z)-N-[3-(2-amino-2-oxoethyl)phenyl]-2-{1-[2-chloro-4-(3-methyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}acetamide 530089-77-1 C31H26ClF2N5O3
(2Z)-N-[3-(2-amino-2-oxoethyl)phenyl]-2-{1-[2-chloro-4-(3-methyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}acetamide
—— N-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]-2-[(1R)-1-[[3-methyl-2-(morpholin-4-ylmethyl)imidazole-4-carbonyl]amino]ethyl]-1,3-thiazole-5-carboxamide 1234012-27-1 C22H23ClF3N7O3S
N-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]-2-[(1R)-1-[[3-methyl-2-(morpholin-4-ylmethyl)imidazole-4-carbonyl]amino]ethyl]-1,3-thiazole-5-carboxamide
—— methoxyimino-(1-methyl-1<i>H</i>-imidazol-2-yl)-acetic acid ethyl ester 73213-72-6 C9H13N3O3
methoxyimino-(1-methyl-1<i>H</i>-imidazol-2-yl)-acetic acid ethyl ester
—— 2-Methyl-2-(1,2-oxazol-5-yl)propanoicacid 1784298-21-0 C7H9NO3
2-Methyl-2-(1,2-oxazol-5-yl)propanoicacid