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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(5-fluoropyrimidin-2-yl)-6-(2-(pyridin-2-yl)ethyl)-4,5,6,7-tetrahydropyrazolo[3,4-b]thiazolo[4,5-d]azepin-2-amine 1355993-96-2 C19H17FN8S
N-(5-fluoropyrimidin-2-yl)-6-(2-(pyridin-2-yl)ethyl)-4,5,6,7-tetrahydropyrazolo[3,4-b]thiazolo[4,5-d]azepin-2-amine
—— N-(3-benzoxazol-2-yl-5-bromo-phenyl)-methanesulfonamide 915413-19-3 C14H11BrN2O3S
N-(3-benzoxazol-2-yl-5-bromo-phenyl)-methanesulfonamide
—— (R)-cyclooctyl-(5-dimethylaminomethyl-oxazol-2-yl)-phenyl-methanol 1046820-33-0 C21H30N2O2
(R)-cyclooctyl-(5-dimethylaminomethyl-oxazol-2-yl)-phenyl-methanol
—— diethyl (4-{[4-({4-[1-(4-hydroxybutyl)-1H-pyrazol-4-yl]-2-(methylcarbamoyl)phenyl}amino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-3-methoxybenzyl)phosphonate 1380304-07-3 C32H39F3N7O6P
diethyl (4-{[4-({4-[1-(4-hydroxybutyl)-1H-pyrazol-4-yl]-2-(methylcarbamoyl)phenyl}amino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-3-methoxybenzyl)phosphonate
—— 1-(4-methyl-piperazin-1-yl)-2-(4-phenyl-2-thioxo-2,3-dihydro-imidazol-1-yl)-ethanone 1039746-10-5 C16H20N4OS
1-(4-methyl-piperazin-1-yl)-2-(4-phenyl-2-thioxo-2,3-dihydro-imidazol-1-yl)-ethanone
—— 5-amino-N-(2-((2-chlorophenylcarbonyl)(ethyl)aminomethyl)-3,3,3-trifluoro-2-hydroxypropyl)-1-(4-fluorophenyl)-1H-pyrazole-4-carboxamide 1034141-41-7 C23H22ClF4N5O3
5-amino-N-(2-((2-chlorophenylcarbonyl)(ethyl)aminomethyl)-3,3,3-trifluoro-2-hydroxypropyl)-1-(4-fluorophenyl)-1H-pyrazole-4-carboxamide
—— 1-hydroxy-4,5-dimethyl-2-(3-nitrophenyl)imidazole 29982-12-5 C11H11N3O3
1-hydroxy-4,5-dimethyl-2-(3-nitrophenyl)imidazole
—— 1-[4-(3,4-difluoro-1H-pyrrol-1-yl)-2-(2,2,2-trifluoroethoxy)phenyl]-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one 1357192-05-2 C26H18F5N5O3
1-[4-(3,4-difluoro-1H-pyrrol-1-yl)-2-(2,2,2-trifluoroethoxy)phenyl]-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one
—— N-cyclopropyl-3-(2-isobutyl-2H-pyrazol-3-yl)-5-(5-methyl-pyridin-2-yl)-benzamide 1162643-87-9 C23H26N4O
N-cyclopropyl-3-(2-isobutyl-2H-pyrazol-3-yl)-5-(5-methyl-pyridin-2-yl)-benzamide
—— 5-[5-(3-chloro-4-fluoro-phenyl)-1-(3-chloro-2-fluoro-phenyl)-2-cyclohexyl-1H-imidazol-4-yl]-2H-tetrazole 1268678-17-6 C22H18Cl2F2N6
5-[5-(3-chloro-4-fluoro-phenyl)-1-(3-chloro-2-fluoro-phenyl)-2-cyclohexyl-1H-imidazol-4-yl]-2H-tetrazole
—— 1-[α-(5-phenyl-tetrazol-1-yl)-isobutyryl]-piperidine 131976-46-0 C16H21N5O
1-[α-(5-phenyl-tetrazol-1-yl)-isobutyryl]-piperidine
—— 1-Cyclopropyl-1H-imidazole-4-carbaldehyde hydrochloride 2089257-24-7 C7H9ClN2O
1-Cyclopropyl-1H-imidazole-4-carbaldehyde hydrochloride
—— (2R,3S)-2-((2R,3R)-3-{(2S)-2-methyl-3-[(1-phenyl-1H-tetrazol-5-yl)sulfonyl]propyl}oxiran-2-yl)pentan-3-ol 934497-75-3 C18H26N4O4S
(2R,3S)-2-((2R,3R)-3-{(2S)-2-methyl-3-[(1-phenyl-1H-tetrazol-5-yl)sulfonyl]propyl}oxiran-2-yl)pentan-3-ol
—— 4-benzyl-2-(4-chlorophenyl)-[1,2,4]triazolo[1,5-a]benzimidazole 139954-35-1 C21H15ClN4
4-benzyl-2-(4-chlorophenyl)-[1,2,4]triazolo[1,5-a]benzimidazole
—— 1-[4-(2-phenyl-9H-imidazo[1,2-d]pyrido[2,3-b][1,4]benzodiazepin-3-yl)phenyl]cyclopropanamine 1374261-40-1 C29H23N5
1-[4-(2-phenyl-9H-imidazo[1,2-d]pyrido[2,3-b][1,4]benzodiazepin-3-yl)phenyl]cyclopropanamine
—— 3-sek-Butyl-5-(1-hydroxyaethyl)-1,2-oxazol 71502-38-0 C9H15NO2
3-sek-Butyl-5-(1-hydroxyaethyl)-1,2-oxazol
—— (4-{3-[4-(1-aminocyclobutyl)phenyl]-9H-imidazo[1,2-d]pyrido[2,3-b][1,4]benzodiazepin-2-yl}phenyl)methanol 1374261-09-2 C31H27N5O
(4-{3-[4-(1-aminocyclobutyl)phenyl]-9H-imidazo[1,2-d]pyrido[2,3-b][1,4]benzodiazepin-2-yl}phenyl)methanol
—— 5-(tert-butyl)-2-[5-(4-chloro-2-fluorophenyl)-4,5-diazatricyclo[5.2.1.0(2,6)]deca-2(6),3-dien-3yl]-1,3-oxazole 1024004-29-2 C21H21ClFN3O
5-(tert-butyl)-2-[5-(4-chloro-2-fluorophenyl)-4,5-diazatricyclo[5.2.1.0(2,6)]deca-2(6),3-dien-3yl]-1,3-oxazole
—— 8-(2-chlorophenyl)-N-[(4-fluorophenyl)methyl]-9-(pyrrolidin-3-ylmethyl)purin-2-amine 1021695-56-6 C23H22ClFN6
8-(2-chlorophenyl)-N-[(4-fluorophenyl)methyl]-9-(pyrrolidin-3-ylmethyl)purin-2-amine
—— 3-chloro-5-fluoro-4-((5-(2-(4-fluoro-3-methoxyphenyl)propan-2-yl)-1-(4-fluorophenyl)-1H-imidazol-2-ylthio)methyl)-N-(3-hydroxypropyl)benzenesulfonamide 1311374-47-6 C29H29ClF3N3O4S2
3-chloro-5-fluoro-4-((5-(2-(4-fluoro-3-methoxyphenyl)propan-2-yl)-1-(4-fluorophenyl)-1H-imidazol-2-ylthio)methyl)-N-(3-hydroxypropyl)benzenesulfonamide
—— 5-(4-chlorophenyl)-1-pentyl-4-phenyl-1H-[1,2,3]triazole 1024655-59-1 C19H20ClN3
5-(4-chlorophenyl)-1-pentyl-4-phenyl-1H-[1,2,3]triazole
—— 4-acetyl-5-(2-hydroxyphenyl)-1-phenylpyrazole 104248-19-3 C17H14N2O2
4-acetyl-5-(2-hydroxyphenyl)-1-phenylpyrazole
—— 391953-97-2 C8H8N2NiO2S4*H2O
—— 1453300-11-2 C16H14ClN3O
—— N-[2-[2-[[3-Methoxy-4-(5-oxazolyl)phenyl]amino]-5-oxazolyl]phenyl]-N-methyl-1H-imidazole-1-acetamide 267645-77-2 C25H22N6O4
N-[2-[2-[[3-Methoxy-4-(5-oxazolyl)phenyl]amino]-5-oxazolyl]phenyl]-N-methyl-1H-imidazole-1-acetamide
—— 1-(2-carboxymethyl-5-chloro-phenyl)-5-(3-chloro-4-fluoro-phenyl)-2-cyclohexyl-1H-imidazole-4-carboxylic acid 1268680-21-2 C24H21Cl2FN2O4
1-(2-carboxymethyl-5-chloro-phenyl)-5-(3-chloro-4-fluoro-phenyl)-2-cyclohexyl-1H-imidazole-4-carboxylic acid
—— (S)-3-(3-(4-(1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-1-((S)-2,3-dihydroxypropyl)-4-isopropylimidazolidin-2-one 1269643-71-1 C24H27N7O3
(S)-3-(3-(4-(1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-1-((S)-2,3-dihydroxypropyl)-4-isopropylimidazolidin-2-one
—— 5-methyl-3-(3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)oxazolidin-2-one 1269646-35-6 C25H30N6O3Si
5-methyl-3-(3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)oxazolidin-2-one
—— (alphaS)-3-[(3,5-difluorophenyl)amino]-alpha-ethyl-5-[2-(ethylamino)-4-pyridinyl]-1H-pyrazole-1-ethanol 1195186-23-2 C20H23F2N5O
(alphaS)-3-[(3,5-difluorophenyl)amino]-alpha-ethyl-5-[2-(ethylamino)-4-pyridinyl]-1H-pyrazole-1-ethanol
—— 1-(4-fluorophenyl)-3-({[(1R)-2-hydroxy-1-phenylethyl]amino}carbonyl)imidazo[1,5-a]pyridin-2-ium trifluoroacetate 1039350-90-7 C2HF3O2*C22H18FN3O2
1-(4-fluorophenyl)-3-({[(1R)-2-hydroxy-1-phenylethyl]amino}carbonyl)imidazo[1,5-a]pyridin-2-ium trifluoroacetate
—— 2-Chloromethyl-1-(1-ethoxy-ethyl)-1H-imidazole; hydrochloride 112655-22-8 C8H13ClN2O*ClH
2-Chloromethyl-1-(1-ethoxy-ethyl)-1H-imidazole; hydrochloride
—— 6-(4'-ethoxyphenoxy)-3-methoxy-2-phenylimidazo<1,2-b>pyridazine 121040-61-7 C21H19N3O3
6-(4'-ethoxyphenoxy)-3-methoxy-2-phenylimidazo<1,2-b>pyridazine
—— 5-(2-amino-4-methoxypyrimidin-5-yl)-1-(2-deoxy-3,5-di-O-triisopropylsilyl-β-D-ribofuranosyl)imidazole-4-carbonitrile 597551-32-1 C32H56N6O4Si2
5-(2-amino-4-methoxypyrimidin-5-yl)-1-(2-deoxy-3,5-di-O-triisopropylsilyl-β-D-ribofuranosyl)imidazole-4-carbonitrile
—— 1-methyl-5-(5-nitrofuran-2-yl)-2-phenyl-1H-imidazole 1245794-45-9 C14H11N3O3
1-methyl-5-(5-nitrofuran-2-yl)-2-phenyl-1H-imidazole
—— N,N-dimethyl-5-[2-(methylthio)-4-pyrimidinyl]-4-phenylthiazol-2-amine 1187242-51-8 C16H16N4S2
N,N-dimethyl-5-[2-(methylthio)-4-pyrimidinyl]-4-phenylthiazol-2-amine
—— (2S)-N-(3-{4-[5-(5-formyl-4-methyl-thiophen-2-yl)-[1,2,4]oxadiazol-3-yl]-2,6-dimethyl-phenoxy}-2-hydroxy-propyl)-2-hydroxy-acetamide 1160956-68-2 C21H23N3O6S
(2S)-N-(3-{4-[5-(5-formyl-4-methyl-thiophen-2-yl)-[1,2,4]oxadiazol-3-yl]-2,6-dimethyl-phenoxy}-2-hydroxy-propyl)-2-hydroxy-acetamide
—— 5-amino-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-nitro-3-trifluoromethylpyrazole 111246-88-9 C11H4Cl2F6N4O2
5-amino-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-nitro-3-trifluoromethylpyrazole
—— 6-[6-(4-fluorophenyl)-imidazo[2,1-b]oxazol-5-yl]-1-isopropyl-1H-benzotriazole 1029524-78-4 C20H16FN5O
6-[6-(4-fluorophenyl)-imidazo[2,1-b]oxazol-5-yl]-1-isopropyl-1H-benzotriazole
—— 5-amino-4-chlorodifluoromethylthio-3-cyano-1-(2,6-dichloro-4-trifluoromethylphenyl) pyrazole 120067-96-1 C12H4Cl3F5N4S
5-amino-4-chlorodifluoromethylthio-3-cyano-1-(2,6-dichloro-4-trifluoromethylphenyl) pyrazole
—— 2-(5-fluoropyridin-3-yl)-9-(2-methoxyphenyl)-8-oxo-8,9-dihydro-7H-purine-6-carboxamide 1022155-46-9 C18H13FN6O3
2-(5-fluoropyridin-3-yl)-9-(2-methoxyphenyl)-8-oxo-8,9-dihydro-7H-purine-6-carboxamide
—— 4-{2-[3-(2,6-Dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazolo [1,5-a]pyrimidin-7-ylamino]-ethylamino}-cyclohexanol 332178-52-6 C23H29Cl2N5O2
4-{2-[3-(2,6-Dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazolo [1,5-a]pyrimidin-7-ylamino]-ethylamino}-cyclohexanol
—— 3-[4-chloro-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]-1-[1-(4-fluorophenyl)-5-propylpyrazol-4-yl]pyrrolidin-2-one 1613395-00-8 C21H20ClF4N5O
3-[4-chloro-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]-1-[1-(4-fluorophenyl)-5-propylpyrazol-4-yl]pyrrolidin-2-one
—— 5-[4-(1H-tetrazol-5-yl)phenyl]-1H-naphtho[1,2-b][1,4]diazepin-2,4(3H,5H)-dione 1239578-67-6 C20H14N6O2
5-[4-(1H-tetrazol-5-yl)phenyl]-1H-naphtho[1,2-b][1,4]diazepin-2,4(3H,5H)-dione
—— 3-(2-fluoro-phenyl)-2-oxo-2,3-dihydro-1<i>H</i>-imidazo[4,5-<i>b</i>]pyridine-6-carboxylic acid methyl ester 67482-01-3 C14H10FN3O3
3-(2-fluoro-phenyl)-2-oxo-2,3-dihydro-1<i>H</i>-imidazo[4,5-<i>b</i>]pyridine-6-carboxylic acid methyl ester
—— US9216962, Cfh407-C 1408235-25-5 C18H22N4O3S2
US9216962, Cfh407-C
—— (S)-5-amino-N-(5-(5-amino-3,3-difluoroazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(3-fluoropyridin-2-yl)thiazole-4-carboxamide 1428571-08-7 C19H21F3N8OS
(S)-5-amino-N-(5-(5-amino-3,3-difluoroazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(3-fluoropyridin-2-yl)thiazole-4-carboxamide
—— ethyl 2-(2-(3-bromophenyl)imidazo[1,2-a]pyridin-3-yl)acetate 1394867-25-4 C17H15BrN2O2
ethyl 2-(2-(3-bromophenyl)imidazo[1,2-a]pyridin-3-yl)acetate
—— 5-(chloromethyl)-1-phenyl-1H-1,2,3-triazole 1338664-01-9 C9H8ClN3
5-(chloromethyl)-1-phenyl-1H-1,2,3-triazole
—— 1-methyl-4-phenyl-N-(trideuteriomethyl)tetrazol-5-imine 97990-73-3 C9H11N5
1-methyl-4-phenyl-N-(trideuteriomethyl)tetrazol-5-imine
—— 3-phenyl-1-ethyl-1H-thieno[2,3-c]pyrazole-5-carboxylic acid 924645-44-3 C14H12N2O2S
3-phenyl-1-ethyl-1H-thieno[2,3-c]pyrazole-5-carboxylic acid