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中文名称 英文名称 CAS号 化学式 结构式图片
—— N'-(5-cyano-1-methyl-6-oxo-4-phenylpyrimidin-2-yl)-4-(4-methoxyphenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carbohydrazide 1311274-12-0 C25H23N7O4
N'-(5-cyano-1-methyl-6-oxo-4-phenylpyrimidin-2-yl)-4-(4-methoxyphenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carbohydrazide
—— 3-CD3-Aminopyrin 68229-56-1 C13H17N3O
3-CD3-Aminopyrin
—— 5-chloropentanoic acid (1-{4-[3-(2-methylpyrrolidin-1-yl)propoxy]phenyl}-1H-pyrazol-4-yl)amide 1152748-40-7 C22H31ClN4O2
5-chloropentanoic acid (1-{4-[3-(2-methylpyrrolidin-1-yl)propoxy]phenyl}-1H-pyrazol-4-yl)amide
—— <i>N</i>-carbamimidoyl-4-(3-methyl-1-phenyl-5-<i>p</i>-tolyl-1<i>H</i>-pyrazol-4-ylazo)-benzenesulfonamide 62352-73-2 C24H23N7O2S
<i>N</i>-carbamimidoyl-4-(3-methyl-1-phenyl-5-<i>p</i>-tolyl-1<i>H</i>-pyrazol-4-ylazo)-benzenesulfonamide
—— 2-(1-ethylpiperidin-4-yl)-1-[2-(4-fluorophenyl)-3-[(4-methylphenyl)amino]-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl]ethan-1-one 1261112-00-8 C28H34FN5O
2-(1-ethylpiperidin-4-yl)-1-[2-(4-fluorophenyl)-3-[(4-methylphenyl)amino]-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl]ethan-1-one
—— 4-[4-(butylcarbamoyl-sulfamoyl)-phenylazo]-5-(4-ethyl-phenyl)-3-methyl-pyrazole-1-carbothioic acid amide 62353-27-9 C24H29N7O3S2
4-[4-(butylcarbamoyl-sulfamoyl)-phenylazo]-5-(4-ethyl-phenyl)-3-methyl-pyrazole-1-carbothioic acid amide
—— (5-methyl-isoxazol-3-yl)-(1-phenyl-1<i>H</i>-imidazol-2-yl)-methanone 32902-35-5 C14H11N3O2
(5-methyl-isoxazol-3-yl)-(1-phenyl-1<i>H</i>-imidazol-2-yl)-methanone
—— N-ethyl-5-[4-[(2S)-piperidin-2-yl]-2-pyridin-3-yl-1,3-thiazol-5-yl]-1H-pyrazole-3-carboxamide 1232031-35-4 C19H22N6OS
N-ethyl-5-[4-[(2S)-piperidin-2-yl]-2-pyridin-3-yl-1,3-thiazol-5-yl]-1H-pyrazole-3-carboxamide
—— (5-phenyl-[1,2,4]oxadiazol-3-ylmethyl)-(1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amine 1056991-29-7 C19H25N3O
(5-phenyl-[1,2,4]oxadiazol-3-ylmethyl)-(1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amine
—— 1160954-65-3 C25H32N4O5S
—— US9216962, Cfh409-C 1408235-14-2 C18H24N4O3S2
US9216962, Cfh409-C
—— 2-chloro-4-(7-cyano-4-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}imidazo[1,2-a]quinoxalin-1-yl)-N-cyclopropylbenzamide 1254196-19-4 C26H21ClN8O
2-chloro-4-(7-cyano-4-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}imidazo[1,2-a]quinoxalin-1-yl)-N-cyclopropylbenzamide
—— 1-(4-cyano-3-(cyanomethyl)-1-phenyl-1H-pyrazol-5-yl)-3-((3S,4R)-4-(3,4-difluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)urea 1414552-08-1 C26H25F2N7O2
1-(4-cyano-3-(cyanomethyl)-1-phenyl-1H-pyrazol-5-yl)-3-((3S,4R)-4-(3,4-difluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)urea
—— 4-[6-amino-8-(oxan-4-ylmethylamino)imidazo[1,2-b]pyridazin-3-yl]-N-cyclopropylbenzamide 1263423-76-2 C22H26N6O2
4-[6-amino-8-(oxan-4-ylmethylamino)imidazo[1,2-b]pyridazin-3-yl]-N-cyclopropylbenzamide
—— 3-[5-(4-Fluorophenyl)-2-phenylpyrazol-3-yl]chromen-2-one 1415931-19-9 C24H15FN2O2
3-[5-(4-Fluorophenyl)-2-phenylpyrazol-3-yl]chromen-2-one
—— 1-(3-(2-cyanopropan-2-yl)-1-phenyl-1H-pyrazol-5-yl)-3-((3S,4R)-4-(3,4-difluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)urea 1414552-10-5 C27H30F2N6O2
1-(3-(2-cyanopropan-2-yl)-1-phenyl-1H-pyrazol-5-yl)-3-((3S,4R)-4-(3,4-difluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)urea
—— 5-{2-[2-(4-chloro-phenyl)-5,6-difluoro-benzoimidazol-1-yl]-2-cyclohexyl-ethoxy}-4-methyl-pyrimidine-2-carboxylic acid ethyl ester 1214878-39-3 C29H29ClF2N4O3
5-{2-[2-(4-chloro-phenyl)-5,6-difluoro-benzoimidazol-1-yl]-2-cyclohexyl-ethoxy}-4-methyl-pyrimidine-2-carboxylic acid ethyl ester
—— ethyl 2-(dimethylamino)-4-[(2R)-tetrahydrofuran-2-yl]thiazole-5-carboxylate 1547490-66-3 C12H18N2O3S
ethyl 2-(dimethylamino)-4-[(2R)-tetrahydrofuran-2-yl]thiazole-5-carboxylate
—— 1-phenyl-4-(4-nitrophenyl)imidazole 97814-19-2 C15H11N3O2
1-phenyl-4-(4-nitrophenyl)imidazole
—— [4-(4-Hydroxy-phenylazo)-3,5-diphenyl-pyrazol-1-yl]-pyridin-2-yl-methanone 98407-88-6 C27H19N5O2
[4-(4-Hydroxy-phenylazo)-3,5-diphenyl-pyrazol-1-yl]-pyridin-2-yl-methanone
—— 5,5'-bis-benzylsulfanyl-4,4'-di-<i>p</i>-tolyl-4<i>H</i>,4'<i>H</i>-3,3'-methanediyl-bis-[1,2,4]triazole 62575-68-2 C33H30N6S2
5,5'-bis-benzylsulfanyl-4,4'-di-<i>p</i>-tolyl-4<i>H</i>,4'<i>H</i>-3,3'-methanediyl-bis-[1,2,4]triazole
—— 2-Methyl-5-<4-aethoxy-phenyl>-2.4-dihydro-<1.2.4>triazol-3-on 59812-25-8 C11H13N3O2
2-Methyl-5-<4-aethoxy-phenyl>-2.4-dihydro-<1.2.4>triazol-3-on
—— 4-chloro-3,5,5-trimethyl-1-phenyl-1,4,5,6-tetrahydro-cyclopentapyrazole-4-carboxylic acid <i>tert</i>-butylamide 63006-33-7 C20H26ClN3O
4-chloro-3,5,5-trimethyl-1-phenyl-1,4,5,6-tetrahydro-cyclopentapyrazole-4-carboxylic acid <i>tert</i>-butylamide
—— 1-N-[4-(4-fluorobenzyl)piperazin-1-yl]carbonylethyl-4-phenylimidazole 1202777-91-0 C23H25FN4O
1-N-[4-(4-fluorobenzyl)piperazin-1-yl]carbonylethyl-4-phenylimidazole
—— 2-(7-{[4-Methoxy-7-(3-methyl-1H-1,2,4-triazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl](oxo)acetyl}-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyrazin-3-yl)benzamide 1202800-01-8 C25H22N10O4
2-(7-{[4-Methoxy-7-(3-methyl-1H-1,2,4-triazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl](oxo)acetyl}-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyrazin-3-yl)benzamide
—— 3-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(3-methoxyphenyl)propan-2-yl]imidazolidine-2,4-dione 1034152-53-8 C26H23FN4O4
3-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(3-methoxyphenyl)propan-2-yl]imidazolidine-2,4-dione
—— 2-Isopropyl-5-(6-methyl-1,2,5,6-tetrahydro-3-pyridyl)-2H-tetrazole, hydrobromide 120241-44-3 BrH*C10H17N5
2-Isopropyl-5-(6-methyl-1,2,5,6-tetrahydro-3-pyridyl)-2H-tetrazole, hydrobromide
—— 6-phenyl-1H-pyrazolo[5,1-c]-1,2,4-triazole-3,7-dicarboxylic acid diethyl ester 1649479-43-5 C16H16N4O4
6-phenyl-1H-pyrazolo[5,1-c]-1,2,4-triazole-3,7-dicarboxylic acid diethyl ester
—— 3-(1-methyl-1H-indol-3-yl)-1-phenyl-4-(1H-1,2,4-triazol-1-yl)-1H-pyrrole-2,5-dione 1654013-98-5 C21H15N5O2
3-(1-methyl-1H-indol-3-yl)-1-phenyl-4-(1H-1,2,4-triazol-1-yl)-1H-pyrrole-2,5-dione
—— 1-(2,4-dichlorophenyl)-3-(5-bromoindol-3-yl)-3-(2-phenyl-1,2,3-triazol-4-yl)propan-1-one 1257533-03-1 C25H17BrCl2N4O
1-(2,4-dichlorophenyl)-3-(5-bromoindol-3-yl)-3-(2-phenyl-1,2,3-triazol-4-yl)propan-1-one
—— N-tert-butyl-1-methyl-5-phenylpyrazol-3-amine 116545-27-8 C14H19N3
N-tert-butyl-1-methyl-5-phenylpyrazol-3-amine
—— 4-benzylamino-3,5,5-trimethyl-1-phenyl-1,4,5,6-tetrahydro-cyclopentapyrazole-4-carboxylic acid benzylamide 63006-37-1 C30H32N4O
4-benzylamino-3,5,5-trimethyl-1-phenyl-1,4,5,6-tetrahydro-cyclopentapyrazole-4-carboxylic acid benzylamide
—— <i>N</i>-(5-bromo-4-phenethyl-thiazol-2-yl)-3,5-dichloro-2-mercapto-benzamide 61954-68-5 C18H13BrCl2N2OS2
<i>N</i>-(5-bromo-4-phenethyl-thiazol-2-yl)-3,5-dichloro-2-mercapto-benzamide
—— 1-(4-hydroxy-phenyl)-4'-methyl-2,1',2',6',7'-pentaphenyl-1',4',6',7'-tetrahydro-2'<i>H</i>-spiro[pyrazolidine-4,8'-pyrazolo[4,3-<i>f</i>]indazole]-3,5,3',5'-tetraone 55138-20-0 C47H34N6O5
1-(4-hydroxy-phenyl)-4'-methyl-2,1',2',6',7'-pentaphenyl-1',4',6',7'-tetrahydro-2'<i>H</i>-spiro[pyrazolidine-4,8'-pyrazolo[4,3-<i>f</i>]indazole]-3,5,3',5'-tetraone
—— 5-amino-1-(4-nitro-phenyl)-3-<i>p</i>-tolyl-1<i>H</i>-pyrazole-4-carboxylic acid ethyl ester 61457-27-0 C19H18N4O4
5-amino-1-(4-nitro-phenyl)-3-<i>p</i>-tolyl-1<i>H</i>-pyrazole-4-carboxylic acid ethyl ester
—— 5-amino-3-cyano-1-(2,6-dichloro-4-trifluoromethoxyphenyl)-4-ethylsulfinylpyrazole 192808-16-5 C13H9Cl2F3N4O2S
5-amino-3-cyano-1-(2,6-dichloro-4-trifluoromethoxyphenyl)-4-ethylsulfinylpyrazole
—— 5-amino-1-(4-fluorophenyl)-N-(3,3,3-trifluoro-2-((2-fluoroethyl)(2-trifluorophenylcarbonyl)aminomethyl)-2-hydroxypropyl)-1H-pyrazole-4-carboxamide 1034141-62-2 C24H21F8N5O3
5-amino-1-(4-fluorophenyl)-N-(3,3,3-trifluoro-2-((2-fluoroethyl)(2-trifluorophenylcarbonyl)aminomethyl)-2-hydroxypropyl)-1H-pyrazole-4-carboxamide
—— 4-isobutyl-5-(2,2,2-trifluoro-ethyl)-1-(2-trifluoromethyl-phenyl)-1,3-dihydro-imidazol-2-one 1021389-90-1 C16H16F6N2O
4-isobutyl-5-(2,2,2-trifluoro-ethyl)-1-(2-trifluoromethyl-phenyl)-1,3-dihydro-imidazol-2-one
—— 5-[4-[(4-chlorophenyl)thio]-1-(4-fluorophenyl)-1H-pyrazol-3-yl]-2-methoxypyridine 1199802-94-2 C21H15ClFN3OS
5-[4-[(4-chlorophenyl)thio]-1-(4-fluorophenyl)-1H-pyrazol-3-yl]-2-methoxypyridine
—— N1-(2,4,5-triphenylimidazol-1-ylethanoyl)-N4-(4-fluorophenyl)thiosemicarbazide 1296625-57-4 C30H24FN5OS
N1-(2,4,5-triphenylimidazol-1-ylethanoyl)-N4-(4-fluorophenyl)thiosemicarbazide
—— 4-(5-isopropyl-2,4-dimethoxyphenyl)-1-(3,4-dimethoxyphenyl)-1H-1,2,3-triazole 1155371-53-1 C21H25N3O4
4-(5-isopropyl-2,4-dimethoxyphenyl)-1-(3,4-dimethoxyphenyl)-1H-1,2,3-triazole
—— 3-[(5-hydroxy-1-phenyl-1H-pyrazole-3-carbonyl)-amino]-3-(4-trifluoromethyl-phenyl)-propionic acid 1318781-78-0 C20H16F3N3O4
3-[(5-hydroxy-1-phenyl-1H-pyrazole-3-carbonyl)-amino]-3-(4-trifluoromethyl-phenyl)-propionic acid
—— (S)-3-{[1-(2,4-difluoro-phenyl)-5-hydroxy-1H-pyrazole-3-carbonyl]-amino}-3-(4-methoxy-phenyl)-propionic acid 1318784-86-9 C20H17F2N3O5
(S)-3-{[1-(2,4-difluoro-phenyl)-5-hydroxy-1H-pyrazole-3-carbonyl]-amino}-3-(4-methoxy-phenyl)-propionic acid
—— (S)-3-[(5-hydroxy-1-phenyl-1H-pyrazole-3-carbonyl)-amino]-3-(4-methoxy-phenyl)-propionic acid 1318784-78-9 C20H19N3O5
(S)-3-[(5-hydroxy-1-phenyl-1H-pyrazole-3-carbonyl)-amino]-3-(4-methoxy-phenyl)-propionic acid
—— 940872-32-2 C30H37N7O2S
—— 500143-56-6 C19H19Cl2N3
—— 1193355-54-2 C17H12BrClF2N2O
—— 5-(3-dimethylaminoprop-2-en-1-oyl)-1-(1-cyclopropylethyl)-2-methylimidazole 600699-73-8 C14H21N3O
5-(3-dimethylaminoprop-2-en-1-oyl)-1-(1-cyclopropylethyl)-2-methylimidazole
—— (3-(4-chlorophenyl)-1,2,4-thiadiazol-5-yl)(4-((2R,3R)-3-(2,4-difluorophenyl)-3-hydroxy-4-(1H-1,2,4-triazol-1-yl)butan-2-yl)piperazin-1-yl)methanone 1092849-27-8 C25H24ClF2N7O2S
(3-(4-chlorophenyl)-1,2,4-thiadiazol-5-yl)(4-((2R,3R)-3-(2,4-difluorophenyl)-3-hydroxy-4-(1H-1,2,4-triazol-1-yl)butan-2-yl)piperazin-1-yl)methanone
—— 4-[({4-[3-(3-carbamoylphenyl)-7-morpholin-4-yl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]phenyl}carbamoyl)amino]-N-[2-(dimethylamino)ethyl]benzamide 1173207-56-1 C33H35N11O4
4-[({4-[3-(3-carbamoylphenyl)-7-morpholin-4-yl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]phenyl}carbamoyl)amino]-N-[2-(dimethylamino)ethyl]benzamide