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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 3'-[4-difluoromethyl-6-(6-trifluoromethylpyridin-3-yl)pyrimidin-2-yl]biphenyl-3-sulfonic acid amide 1068107-27-6 C23H15F5N4O2S
3'-[4-difluoromethyl-6-(6-trifluoromethylpyridin-3-yl)pyrimidin-2-yl]biphenyl-3-sulfonic acid amide
—— 4-(3,4-dichlorophenyl)-N-(4-((7-(methyloxy)-1,5-naphthyridin-4-yl)oxy)phenyl)-1-phthalazinamine 1071531-88-8 C29H19Cl2N5O2
4-(3,4-dichlorophenyl)-N-(4-((7-(methyloxy)-1,5-naphthyridin-4-yl)oxy)phenyl)-1-phthalazinamine
—— 10-[(tert-butoxycarbonyl)(methyl)amino]-2-{[(4-fluoro-3-methylbenzyl)amino]carbonyl}-7-methoxy-7-methyl-4-oxo-4,6,7,8,9,10-hexahydropyrimido[1,2-a]azepin-3-yl methanesulfonate 1220510-71-3 C27H37FN4O8S
10-[(tert-butoxycarbonyl)(methyl)amino]-2-{[(4-fluoro-3-methylbenzyl)amino]carbonyl}-7-methoxy-7-methyl-4-oxo-4,6,7,8,9,10-hexahydropyrimido[1,2-a]azepin-3-yl methanesulfonate
—— O3'-acetyl-2'-bromo-5'-chloro-2',5'-dideoxy-uridine 65591-45-9 C11H12BrClN2O5
O3'-acetyl-2'-bromo-5'-chloro-2',5'-dideoxy-uridine
—— N-cyclopropyl-2-[6-(3-hydroxyphenyl)-2-morpholin-4-ylpurin-9-yl]acetamide 1138158-66-3 C20H22N6O3
N-cyclopropyl-2-[6-(3-hydroxyphenyl)-2-morpholin-4-ylpurin-9-yl]acetamide
—— 3-hydroxy-4-oxo-10-(2-piperidin-1-yl-ethyl)-4,10-dihydro-benzo[4,5]imidazo[1,2-a]pyrimidine-2-carboxylic acid 3,4-dichloro-benzylamide 1036646-81-7 C25H25Cl2N5O3
3-hydroxy-4-oxo-10-(2-piperidin-1-yl-ethyl)-4,10-dihydro-benzo[4,5]imidazo[1,2-a]pyrimidine-2-carboxylic acid 3,4-dichloro-benzylamide
—— 1-(2-Methoxy-6-methyl-pyrimidinyl-(4))-2,3-dimethyl-pyrazolinon-(5) 23906-06-1 C11H14N4O2
1-(2-Methoxy-6-methyl-pyrimidinyl-(4))-2,3-dimethyl-pyrazolinon-(5)
—— 6-chloro-2-n-propylimidazo[1,2-b]pyridazin-3-ylsulfonamide 570416-41-0 C9H11ClN4O2S
6-chloro-2-n-propylimidazo[1,2-b]pyridazin-3-ylsulfonamide
—— N-(5-fluoro-4-methylpyrimidin-2-yl)-4-(1H-pyrazol-4-yl)thiazol-2-amine 1235313-39-9 C11H9FN6S
N-(5-fluoro-4-methylpyrimidin-2-yl)-4-(1H-pyrazol-4-yl)thiazol-2-amine
—— 5-(2-methylpiperidin-1-yl)-6-(2-chloro-6-fluorophenyl)-7-chloroimidazo[1,2-a]pyrimidine 502501-61-3 C18H17Cl2FN4
5-(2-methylpiperidin-1-yl)-6-(2-chloro-6-fluorophenyl)-7-chloroimidazo[1,2-a]pyrimidine
—— 405222-98-2 C20H22F2N6O
—— 1313913-56-2 C23H26N6O3
—— 5-[6-Chloro-1-(oxan-4-yl)pyrazolo[3,4-d]pyrimidin-4-yl]-4-methylpyrimidin-2-amine 1227062-27-2 C15H16ClN7O
5-[6-Chloro-1-(oxan-4-yl)pyrazolo[3,4-d]pyrimidin-4-yl]-4-methylpyrimidin-2-amine
—— 1,3-Dimethyl-6-o-hydroxyphenyl-7-azalumazin 30561-29-6 C13H11N5O3
1,3-Dimethyl-6-o-hydroxyphenyl-7-azalumazin
—— 4-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-N-ethyl-3,6-dihydro-2H-pyridine-1-carboxamide 1207350-39-7 C20H23N7O
4-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-N-ethyl-3,6-dihydro-2H-pyridine-1-carboxamide
—— ethyl 2-(1-(2-fluorobenzyl)-5-(isoxazol-3-yl)-1H-pyrazol-3-yl)-4-hydroxypyrimidine-5-carboxylate 1354041-67-0 C20H16FN5O4
ethyl 2-(1-(2-fluorobenzyl)-5-(isoxazol-3-yl)-1H-pyrazol-3-yl)-4-hydroxypyrimidine-5-carboxylate
—— 3-[2-chloro-9-(4-nitro-benzyl)-9H-purin-6-yl]-phenol 1138159-26-8 C18H12ClN5O3
3-[2-chloro-9-(4-nitro-benzyl)-9H-purin-6-yl]-phenol
—— 1161076-25-0 C20H22FN5O2
—— 1161076-45-4 C19H21N5
—— 2-(4-fluoro-3-(pyrrolidine-1-carboxamido)phenylamino)-4-(2-fluorobenzylamino)pyrimidine-5-carboxamide 1254216-59-5 C23H23F2N7O2
2-(4-fluoro-3-(pyrrolidine-1-carboxamido)phenylamino)-4-(2-fluorobenzylamino)pyrimidine-5-carboxamide
—— 3-[4-(2-amino-pyrimidin-5-yl)-2-morpholin-4-yl-5,6-dihydro-pyrrolo[2,3-d]pyrimidin-7-yl]-N-(2-dimethylamino-ethyl)-benzamide 1007208-64-1 C25H31N9O2
3-[4-(2-amino-pyrimidin-5-yl)-2-morpholin-4-yl-5,6-dihydro-pyrrolo[2,3-d]pyrimidin-7-yl]-N-(2-dimethylamino-ethyl)-benzamide
—— 4-[4-(2-amino-pyrimidin-5-yl)-2-morpholin-4-yl-5,6-dihydro-pyrrolo[2,3-d]pyrimidin-7-yl]-4-oxo-butyric acid methyl ester 1007207-84-2 C19H23N7O4
4-[4-(2-amino-pyrimidin-5-yl)-2-morpholin-4-yl-5,6-dihydro-pyrrolo[2,3-d]pyrimidin-7-yl]-4-oxo-butyric acid methyl ester
—— 5-[(3S)-3-amino-3,4-dihydro-2H-chromen-5-yl]-N,N-dimethylpyrimidine-2-carboxamide 1072855-15-2 C16H18N4O2
5-[(3S)-3-amino-3,4-dihydro-2H-chromen-5-yl]-N,N-dimethylpyrimidine-2-carboxamide
—— 5-[7-(5-bromo-pyridin-2-yl)-2-morpholin-4-yl-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl]-pyrimidin-2-ylamine 1007208-32-3 C19H19BrN8O
5-[7-(5-bromo-pyridin-2-yl)-2-morpholin-4-yl-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl]-pyrimidin-2-ylamine
—— 4-chloro-5-[<i>N</i>-(2-hydroxy-ethyl)-hydrazino]-2-(3-trifluoromethyl-phenyl)-2<i>H</i>-pyridazin-3-one 41933-21-5 C13H12ClF3N4O2
4-chloro-5-[<i>N</i>-(2-hydroxy-ethyl)-hydrazino]-2-(3-trifluoromethyl-phenyl)-2<i>H</i>-pyridazin-3-one
—— 3-(4-(1-(2,2-difluoroethyl)-3-iodo-1H-pyrazol-4-yl)pyrimidin-2-ylamino)propanenitrile 1111638-19-7 C12H11F2IN6
3-(4-(1-(2,2-difluoroethyl)-3-iodo-1H-pyrazol-4-yl)pyrimidin-2-ylamino)propanenitrile
—— 632343-06-7 C17H13Cl2F3N4
—— 5-(Pent-2-en-2-yl)-5-propyldihydropyrimidine-2,4(1H,3H)-dione 831220-20-3 C12H20N2O2
5-(Pent-2-en-2-yl)-5-propyldihydropyrimidine-2,4(1H,3H)-dione
—— 3-(4-Iodo-3-oxo-butyl)-1,5,5-trimethyl-imidazolidine-2,4-dione 220615-38-3 C10H15IN2O3
3-(4-Iodo-3-oxo-butyl)-1,5,5-trimethyl-imidazolidine-2,4-dione
—— 4-Methyl-5-[2-(3-methylimidazol-4-yl)ethynyl]-6-pyridin-3-ylpyrimidin-2-amine 1207346-87-9 C16H14N6
4-Methyl-5-[2-(3-methylimidazol-4-yl)ethynyl]-6-pyridin-3-ylpyrimidin-2-amine
—— 3-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-5-fluoro-N,N-dimethylbenzamide 1207350-47-7 C21H19FN6O
3-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-5-fluoro-N,N-dimethylbenzamide
—— 6-hydroxy-2-morpholin-4-ylmethyl-5-oxo-5H-thiazolo[3,2-a]pyrimidine-7-carboxylic acid 3,4-dichloro-benzylamide 1036647-15-0 C19H18Cl2N4O4S
6-hydroxy-2-morpholin-4-ylmethyl-5-oxo-5H-thiazolo[3,2-a]pyrimidine-7-carboxylic acid 3,4-dichloro-benzylamide
—— 9-(2-Aminopyrimidin-5-yl)-1-(4-fluorophenyl)benzo[h][1,6]naphthyridin-2-one 1223001-25-9 C22H14FN5O
9-(2-Aminopyrimidin-5-yl)-1-(4-fluorophenyl)benzo[h][1,6]naphthyridin-2-one
—— 4-Methyl-6-(4-methylsulfonylphenyl)-5-(2-pyridin-3-ylethynyl)pyrimidin-2-amine 1207347-12-3 C19H16N4O2S
4-Methyl-6-(4-methylsulfonylphenyl)-5-(2-pyridin-3-ylethynyl)pyrimidin-2-amine
—— [4-[2-Amino-6-methyl-5-[2-[6-(methylamino)pyridin-3-yl]ethynyl]pyrimidin-4-yl]-2-chlorophenyl]-morpholin-4-ylmethanone 1207349-00-5 C24H23ClN6O2
[4-[2-Amino-6-methyl-5-[2-[6-(methylamino)pyridin-3-yl]ethynyl]pyrimidin-4-yl]-2-chlorophenyl]-morpholin-4-ylmethanone
—— 4-(2-Fluoro-4-methylsulfonylphenyl)-6-methyl-5-[2-[6-(methylamino)pyridin-3-yl]ethynyl]pyrimidin-2-amine 1207349-21-0 C20H18FN5O2S
4-(2-Fluoro-4-methylsulfonylphenyl)-6-methyl-5-[2-[6-(methylamino)pyridin-3-yl]ethynyl]pyrimidin-2-amine
—— 855528-25-5 C18H15Cl2FN4O
—— 1001190-42-6 C14H14N8O
—— 2-(2,4-dichlorobenzylidene)-7-methyl-5-(4-nitrophenyl)-3-oxo-2,3-dihydro-5H-thiazolo[3,2-a]pyrimidine-6-carboxylic acid (4-fluorophenyl)amide 1198746-67-6 C27H17Cl2FN4O4S
2-(2,4-dichlorobenzylidene)-7-methyl-5-(4-nitrophenyl)-3-oxo-2,3-dihydro-5H-thiazolo[3,2-a]pyrimidine-6-carboxylic acid (4-fluorophenyl)amide
—— 855528-34-6 C19H19Cl2FN4O
—— [3-(6-trifluoromethylpyridazin-3-yl)benzyl]carbamic acid tert-butyl ester 1590398-11-0 C17H18F3N3O2
[3-(6-trifluoromethylpyridazin-3-yl)benzyl]carbamic acid tert-butyl ester
—— 2-Iodamino-4,6-dimethyl-pyrimidin 3005-25-2 C6H8IN3
2-Iodamino-4,6-dimethyl-pyrimidin
—— [trans-4-(4-{4-amino-2-[(2,2-dimethylpropyl)amino]-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl}phenyl)cyclohexyl]acetic acid 1434905-59-5 C26H35N5O4
[trans-4-(4-{4-amino-2-[(2,2-dimethylpropyl)amino]-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl}phenyl)cyclohexyl]acetic acid
—— 6-(3,4-dimethoxy-phenyl)-3-[1-(4-methoxy-benzenesulfonyl)-1H-pyrazol-3-yl]-2-methyl-imidazo[1,2-b]pyridazine 1083428-90-3 C25H23N5O5S
6-(3,4-dimethoxy-phenyl)-3-[1-(4-methoxy-benzenesulfonyl)-1H-pyrazol-3-yl]-2-methyl-imidazo[1,2-b]pyridazine
—— (4-{4-[(R)-amino(4-fluorophenyl)-methyl]piperidin-1-ylsulphonyl}phenyl)-[4-(4-(trifluoromethyl)-phenyl)-pyrimidin-2-yl]amine 1049105-22-7 C29H27F4N5O2S
(4-{4-[(R)-amino(4-fluorophenyl)-methyl]piperidin-1-ylsulphonyl}phenyl)-[4-(4-(trifluoromethyl)-phenyl)-pyrimidin-2-yl]amine
—— 1-[4-(3-hydroxyphenyl)-2-morpholin-4-yl-5,6-dihydropyrrolo[2,3-d]pyrimidin-7-yl]-2,2-dimethyl-propan-1-one 1007207-03-5 C21H26N4O3
1-[4-(3-hydroxyphenyl)-2-morpholin-4-yl-5,6-dihydropyrrolo[2,3-d]pyrimidin-7-yl]-2,2-dimethyl-propan-1-one
—— 2-amino-4-(4-bromo-2-chloro-5-methoxyphenyl)-N-(4-cyanophenyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide 1046858-98-3 C21H16BrClN6O2
2-amino-4-(4-bromo-2-chloro-5-methoxyphenyl)-N-(4-cyanophenyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
—— 2-(((S)-2-N-Glycylamino-3-phenylpropyl)-amino)-3-methyl-5-(3-methylphenyl)-6-(4-pyridyl)-4-(3H)-pyrimidinone 208654-59-5 C28H30N6O2
2-(((S)-2-N-Glycylamino-3-phenylpropyl)-amino)-3-methyl-5-(3-methylphenyl)-6-(4-pyridyl)-4-(3H)-pyrimidinone
—— 3-Methoxymethyl-4-oxo-3,4-dihydro-benzo<b>thieno<2,3-d>pyridazin 24049-68-1 C12H10N2O2S
3-Methoxymethyl-4-oxo-3,4-dihydro-benzo<b>thieno<2,3-d>pyridazin
—— N2-(trans-4-aminocyclohexyl)-6-[(methyloxy)methyl]-N4-[1,3]thiazolo[5,4-b]pyridin-2-yl-2,4-pyrimidinediamine 1365838-60-3 C18H23N7OS
N2-(trans-4-aminocyclohexyl)-6-[(methyloxy)methyl]-N4-[1,3]thiazolo[5,4-b]pyridin-2-yl-2,4-pyrimidinediamine