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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (7R)-7-[(Z)-2-phenylethenyl]-2-(4-pyrimidin-2-ylpiperazin-1-yl)-7,8-dihydro-6H-quinazolin-5-one —— C24H24N6O
(7R)-7-[(Z)-2-phenylethenyl]-2-(4-pyrimidin-2-ylpiperazin-1-yl)-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-7-[(Z)-2-phenylethenyl]-2-(4-pyrimidin-2-ylpiperazin-1-yl)-7,8-dihydro-6H-quinazolin-5-one —— C24H24N6O
(7S)-7-[(Z)-2-phenylethenyl]-2-(4-pyrimidin-2-ylpiperazin-1-yl)-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-4-methyl-7-[(Z)-2-phenylethenyl]-2-(4-pyrimidin-2-ylpiperazin-1-yl)-7,8-dihydro-6H-quinazolin-5-one —— C25H26N6O
(7R)-4-methyl-7-[(Z)-2-phenylethenyl]-2-(4-pyrimidin-2-ylpiperazin-1-yl)-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-2-[4-(2-hydroxyethyl)piperazin-1-yl]-7-[(Z)-2-phenylethenyl]-7,8-dihydro-6H-quinazolin-5-one —— C22H26N4O2
(7R)-2-[4-(2-hydroxyethyl)piperazin-1-yl]-7-[(Z)-2-phenylethenyl]-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-2-[4-(2-hydroxyethyl)piperazin-1-yl]-4-methyl-7-[(Z)-2-phenylethenyl]-7,8-dihydro-6H-quinazolin-5-one —— C23H28N4O2
(7S)-2-[4-(2-hydroxyethyl)piperazin-1-yl]-4-methyl-7-[(Z)-2-phenylethenyl]-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-4-methyl-7-[(Z)-2-phenylethenyl]-2-(4-pyrimidin-2-ylpiperazin-1-yl)-7,8-dihydro-6H-quinazolin-5-one —— C25H26N6O
(7S)-4-methyl-7-[(Z)-2-phenylethenyl]-2-(4-pyrimidin-2-ylpiperazin-1-yl)-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-2-[4-(2-hydroxyethyl)piperazin-1-yl]-4-methyl-7-[(Z)-2-phenylethenyl]-7,8-dihydro-6H-quinazolin-5-one —— C23H28N4O2
(7R)-2-[4-(2-hydroxyethyl)piperazin-1-yl]-4-methyl-7-[(Z)-2-phenylethenyl]-7,8-dihydro-6H-quinazolin-5-one
—— (3R)-4-methyl-N-[3-(methylsulfamoyl)phenyl]-3-phenylpiperazine-1-carboxamide —— C19H24N4O3S
(3R)-4-methyl-N-[3-(methylsulfamoyl)phenyl]-3-phenylpiperazine-1-carboxamide
—— (3S)-4-methyl-N-[3-(methylsulfamoyl)phenyl]-3-phenylpiperazine-1-carboxamide —— C19H24N4O3S
(3S)-4-methyl-N-[3-(methylsulfamoyl)phenyl]-3-phenylpiperazine-1-carboxamide
—— N-[(2R)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-4-oxo-4-(5-phenyl-3,4-dihydropyrazol-2-yl)butanamide —— C23H35N5O2
N-[(2R)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-4-oxo-4-(5-phenyl-3,4-dihydropyrazol-2-yl)butanamide
—— N-[(2R)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-4-[methyl(thiophen-2-ylsulfonyl)amino]butanamide —— C19H34N4O3S2
N-[(2R)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-4-[methyl(thiophen-2-ylsulfonyl)amino]butanamide
—— N-[(2S)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-4-oxo-4-(5-phenyl-3,4-dihydropyrazol-2-yl)butanamide —— C23H35N5O2
N-[(2S)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-4-oxo-4-(5-phenyl-3,4-dihydropyrazol-2-yl)butanamide
—— N-[(2S)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-4-[methyl(thiophen-2-ylsulfonyl)amino]butanamide —— C19H34N4O3S2
N-[(2S)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-4-[methyl(thiophen-2-ylsulfonyl)amino]butanamide
—— 2-[4-[2,5-dimethyl-1-[(1S)-1-phenylethyl]pyrrole-3-carbonyl]piperazin-1-yl]-1-morpholin-4-ylethanone —— C25H34N4O3
2-[4-[2,5-dimethyl-1-[(1S)-1-phenylethyl]pyrrole-3-carbonyl]piperazin-1-yl]-1-morpholin-4-ylethanone
—— 2-[4-[2,5-dimethyl-1-[(1R)-1-phenylethyl]pyrrole-3-carbonyl]piperazin-1-yl]-1-morpholin-4-ylethanone —— C25H34N4O3
2-[4-[2,5-dimethyl-1-[(1R)-1-phenylethyl]pyrrole-3-carbonyl]piperazin-1-yl]-1-morpholin-4-ylethanone
—— N-[(1S)-1-(4-bromophenyl)ethyl]-4-(2-cyano-3-fluorophenyl)piperazine-1-carboxamide —— C20H20BrFN4O
N-[(1S)-1-(4-bromophenyl)ethyl]-4-(2-cyano-3-fluorophenyl)piperazine-1-carboxamide
—— 4-(2-cyano-3-fluorophenyl)-N-[(1S)-1-(7-ethoxy-1-benzofuran-2-yl)ethyl]piperazine-1-carboxamide —— C24H25FN4O3
4-(2-cyano-3-fluorophenyl)-N-[(1S)-1-(7-ethoxy-1-benzofuran-2-yl)ethyl]piperazine-1-carboxamide
—— 2-[4-[2,5-dimethyl-1-[(1R)-1-phenylethyl]pyrrole-3-carbonyl]piperazin-1-yl]-N,N-diethylacetamide —— C25H36N4O2
2-[4-[2,5-dimethyl-1-[(1R)-1-phenylethyl]pyrrole-3-carbonyl]piperazin-1-yl]-N,N-diethylacetamide
—— 1-[[2-[(4-phenylpiperazin-1-yl)methyl]phenyl]methyl]-3-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]urea —— C27H32N4O2
1-[[2-[(4-phenylpiperazin-1-yl)methyl]phenyl]methyl]-3-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]urea
—— 2-[4-[2,5-dimethyl-1-[(1S)-1-phenylethyl]pyrrole-3-carbonyl]piperazin-1-yl]-N,N-diethylacetamide —— C25H36N4O2
2-[4-[2,5-dimethyl-1-[(1S)-1-phenylethyl]pyrrole-3-carbonyl]piperazin-1-yl]-N,N-diethylacetamide
—— 1-[(2S)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]urea —— C24H34N4O2
1-[(2S)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]urea
—— 1-[(2R)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-(4-nitrophenyl)urea —— C22H29N5O3
1-[(2R)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-(4-nitrophenyl)urea
—— 4-(5-bromopyridin-2-yl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]piperazine-1-carboxamide —— C18H21BrN4O2
4-(5-bromopyridin-2-yl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]piperazine-1-carboxamide
—— 1-[(2S)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]urea —— C24H34N4O2
1-[(2S)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]urea
—— 4-(2-cyano-3-fluorophenyl)-N-[(1R)-1-(7-ethoxy-1-benzofuran-2-yl)ethyl]piperazine-1-carboxamide —— C24H25FN4O3
4-(2-cyano-3-fluorophenyl)-N-[(1R)-1-(7-ethoxy-1-benzofuran-2-yl)ethyl]piperazine-1-carboxamide
—— N-[(1R)-1-(4-bromophenyl)ethyl]-4-(2-cyano-3-fluorophenyl)piperazine-1-carboxamide —— C20H20BrFN4O
N-[(1R)-1-(4-bromophenyl)ethyl]-4-(2-cyano-3-fluorophenyl)piperazine-1-carboxamide
—— 4-(5-bromopyridin-2-yl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]piperazine-1-carboxamide —— C18H21BrN4O2
4-(5-bromopyridin-2-yl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]piperazine-1-carboxamide
—— 1-[(2S)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-(4-nitrophenyl)urea —— C22H29N5O3
1-[(2S)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-(4-nitrophenyl)urea
—— 1-[(2R)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]urea —— C24H34N4O2
1-[(2R)-4-[4-(3-methylphenyl)piperazin-1-yl]butan-2-yl]-3-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]urea
—— (2R)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-cyclohexyl-N-(1,3-thiazol-2-yl)propanamide —— C23H28FN5OS
(2R)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-cyclohexyl-N-(1,3-thiazol-2-yl)propanamide
—— (2R)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methylpropanamide —— C24H27FN4O3
(2R)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methylpropanamide
—— (2R)-2-[4-(5-bromopyridin-2-yl)piperazin-1-yl]-N-prop-2-ynylpropanamide —— C15H19BrN4O
(2R)-2-[4-(5-bromopyridin-2-yl)piperazin-1-yl]-N-prop-2-ynylpropanamide
—— (2R)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methylpropanamide —— C24H27FN4O3
(2R)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methylpropanamide
—— 1-[(2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-1-oxopropan-2-yl]-N-methyl-N-propan-2-ylpiperidine-4-carboxamide —— C23H35FN4O2
1-[(2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-1-oxopropan-2-yl]-N-methyl-N-propan-2-ylpiperidine-4-carboxamide
—— 1-[(2S)-1-[4-(4-fluorophenyl)piperazin-1-yl]-1-oxopropan-2-yl]-N-methyl-N-propan-2-ylpiperidine-4-carboxamide —— C23H35FN4O2
1-[(2S)-1-[4-(4-fluorophenyl)piperazin-1-yl]-1-oxopropan-2-yl]-N-methyl-N-propan-2-ylpiperidine-4-carboxamide
—— (2S)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methylpropanamide —— C24H27FN4O3
(2S)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methylpropanamide
—— (2S)-2-[4-(5-bromopyridin-2-yl)piperazin-1-yl]-N-prop-2-ynylpropanamide —— C15H19BrN4O
(2S)-2-[4-(5-bromopyridin-2-yl)piperazin-1-yl]-N-prop-2-ynylpropanamide
—— (2S)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-cyclohexyl-N-(1,3-thiazol-2-yl)propanamide —— C23H28FN5OS
(2S)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-cyclohexyl-N-(1,3-thiazol-2-yl)propanamide
—— (2R)-2-[4-(5-bromopyridin-2-yl)piperazin-1-yl]-N-(1-cyano-4-methylcyclohexyl)-N-methylpropanamide —— C21H30BrN5O
(2R)-2-[4-(5-bromopyridin-2-yl)piperazin-1-yl]-N-(1-cyano-4-methylcyclohexyl)-N-methylpropanamide
—— (2S)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-(1-cyano-4-methylcyclohexyl)-N-methylpropanamide —— C23H30FN5O
(2S)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-(1-cyano-4-methylcyclohexyl)-N-methylpropanamide
—— N-methyl-1-[(2R)-1-oxo-1-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-yl]-N-propan-2-ylpiperidine-4-carboxamide —— C21H34N6O2
N-methyl-1-[(2R)-1-oxo-1-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-yl]-N-propan-2-ylpiperidine-4-carboxamide
—— N-methyl-1-[(2S)-1-oxo-1-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-yl]-N-propan-2-ylpiperidine-4-carboxamide —— C21H34N6O2
N-methyl-1-[(2S)-1-oxo-1-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-yl]-N-propan-2-ylpiperidine-4-carboxamide
—— (2S)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methylpropanamide —— C24H27FN4O3
(2S)-2-[4-(2-cyano-3-fluorophenyl)piperazin-1-yl]-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methylpropanamide
—— 1-[(4R)-4-ethyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-(4-pyridin-3-ylsulfonylpiperazin-1-yl)ethanone —— C20H26N4O3S2
1-[(4R)-4-ethyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-(4-pyridin-3-ylsulfonylpiperazin-1-yl)ethanone
—— (2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-2-[methyl-[(5-methyl-1,2-oxazol-3-yl)methyl]amino]propan-1-one —— C19H25FN4O2
(2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-2-[methyl-[(5-methyl-1,2-oxazol-3-yl)methyl]amino]propan-1-one
—— (2S)-2-[4-(5-bromopyridin-2-yl)piperazin-1-yl]-N-(1-cyano-4-methylcyclohexyl)-N-methylpropanamide —— C21H30BrN5O
(2S)-2-[4-(5-bromopyridin-2-yl)piperazin-1-yl]-N-(1-cyano-4-methylcyclohexyl)-N-methylpropanamide
—— (2S)-1-[4-(4-fluorophenyl)piperazin-1-yl]-2-[methyl-[(5-methyl-1,2-oxazol-3-yl)methyl]amino]propan-1-one —— C19H25FN4O2
(2S)-1-[4-(4-fluorophenyl)piperazin-1-yl]-2-[methyl-[(5-methyl-1,2-oxazol-3-yl)methyl]amino]propan-1-one
—— N-[(1R)-1-(4-fluorophenyl)ethyl]-N-methyl-2-[4-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazin-1-yl]acetamide —— C21H26FN7O
N-[(1R)-1-(4-fluorophenyl)ethyl]-N-methyl-2-[4-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazin-1-yl]acetamide
—— (2S)-N-(1-cyano-4-methylcyclohexyl)-N-methyl-2-[4-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazin-1-yl]propanamide —— C22H32N8O
(2S)-N-(1-cyano-4-methylcyclohexyl)-N-methyl-2-[4-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazin-1-yl]propanamide
—— (2S)-N-(2-cyanoethyl)-2-[4-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazin-1-yl]-N-phenylpropanamide —— C22H26N8O
(2S)-N-(2-cyanoethyl)-2-[4-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazin-1-yl]-N-phenylpropanamide