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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(4-chlorophenyl)-1-[4-[2-oxo-2-[(3S)-3-(trifluoromethyl)piperidin-1-yl]ethyl]piperazin-1-yl]ethanone —— C20H25ClF3N3O2
2-(4-chlorophenyl)-1-[4-[2-oxo-2-[(3S)-3-(trifluoromethyl)piperidin-1-yl]ethyl]piperazin-1-yl]ethanone
—— N-[(1S)-1-(3,4-difluorophenyl)ethyl]-N-methyl-2-[4-(2-oxo-2-pyrrolidin-1-ylacetyl)piperazin-1-yl]acetamide —— C21H28F2N4O3
N-[(1S)-1-(3,4-difluorophenyl)ethyl]-N-methyl-2-[4-(2-oxo-2-pyrrolidin-1-ylacetyl)piperazin-1-yl]acetamide
—— 2-[4-[2-(4-chlorophenyl)acetyl]piperazin-1-yl]-N-[(1R)-1-(3,4-difluorophenyl)ethyl]-N-methylacetamide —— C23H26ClF2N3O2
2-[4-[2-(4-chlorophenyl)acetyl]piperazin-1-yl]-N-[(1R)-1-(3,4-difluorophenyl)ethyl]-N-methylacetamide
—— 1-[4-[[2-(2,4-dichlorophenyl)-2-(imidazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]-4-[(Z)-1,3,3,3-tetrafluoro-2-[4-(trifluoromethyl)phenyl]prop-1-enyl]piperazine —— C34H29Cl2F7N4O3
1-[4-[[2-(2,4-dichlorophenyl)-2-(imidazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]-4-[(Z)-1,3,3,3-tetrafluoro-2-[4-(trifluoromethyl)phenyl]prop-1-enyl]piperazine
—— N-ethyl-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[4-(2-oxo-2-pyrrolidin-1-ylacetyl)piperazin-1-yl]acetamide —— C22H31FN4O3
N-ethyl-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[4-(2-oxo-2-pyrrolidin-1-ylacetyl)piperazin-1-yl]acetamide
—— copper;1-[4-[4-[[(2R,4S)-2-(2,4-dichlorophenyl)-2-(imidazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]piperazin-1-yl]ethanone;N-methyl-N-oxidomethanethioamide —— C30H36Cl2CuN6O6S2
copper;1-[4-[4-[[(2R,4S)-2-(2,4-dichlorophenyl)-2-(imidazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]piperazin-1-yl]ethanone;N-methyl-N-oxidomethanethioamide
—— N-[(1R)-1-(3,4-difluorophenyl)ethyl]-N-methyl-2-[4-(2-oxo-2-pyrrolidin-1-ylacetyl)piperazin-1-yl]acetamide —— C21H28F2N4O3
N-[(1R)-1-(3,4-difluorophenyl)ethyl]-N-methyl-2-[4-(2-oxo-2-pyrrolidin-1-ylacetyl)piperazin-1-yl]acetamide
—— 2-[4-[2-(4-chlorophenyl)acetyl]piperazin-1-yl]-N-[(1S)-1-(3,4-difluorophenyl)ethyl]-N-methylacetamide —— C23H26ClF2N3O2
2-[4-[2-(4-chlorophenyl)acetyl]piperazin-1-yl]-N-[(1S)-1-(3,4-difluorophenyl)ethyl]-N-methylacetamide
—— 1-[(4R)-4-ethyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-[4-(3-methyl-1,2-oxazole-5-carbonyl)piperazin-1-yl]ethanone —— C20H26N4O3S
1-[(4R)-4-ethyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-[4-(3-methyl-1,2-oxazole-5-carbonyl)piperazin-1-yl]ethanone
—— 1-N,3-N-dibenzyl-1-N,3-N-dimethyl-4-(4-methylpiperazin-1-yl)-6-(3-phenylpropylamino)benzene-1,3-disulfonamide —— C36H45N5O4S2
1-N,3-N-dibenzyl-1-N,3-N-dimethyl-4-(4-methylpiperazin-1-yl)-6-(3-phenylpropylamino)benzene-1,3-disulfonamide
—— 1-[2-(3,4-Dichlorophenyl)-4-(3,5-dimethylbenzoyl)piperazin-1-yl]-3-[5-(thiophen-2-ylmethylsulfonyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]propan-1-one —— C32H36Cl2N4O4S2
1-[2-(3,4-Dichlorophenyl)-4-(3,5-dimethylbenzoyl)piperazin-1-yl]-3-[5-(thiophen-2-ylmethylsulfonyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]propan-1-one
—— 2-[4-[4-[4-[[2-(4-Chlorophenyl)-2-[(4-methyl-1,2,4-triazol-3-yl)methyl]-1,3-dioxolan-4-yl]methoxy]phenyl]piperazin-1-yl]phenyl]-4-ethyl-1,2,4-triazol-3-one —— C34H37ClN8O4
2-[4-[4-[4-[[2-(4-Chlorophenyl)-2-[(4-methyl-1,2,4-triazol-3-yl)methyl]-1,3-dioxolan-4-yl]methoxy]phenyl]piperazin-1-yl]phenyl]-4-ethyl-1,2,4-triazol-3-one
—— 4-[5-(Oxan-4-yl)-2-oxo-4-(4-pyridin-2-ylpiperazin-1-yl)pyrimidin-1-yl]-3-(phenylmethoxycarbonylamino)butanoic acid —— C30H36N6O6
4-[5-(Oxan-4-yl)-2-oxo-4-(4-pyridin-2-ylpiperazin-1-yl)pyrimidin-1-yl]-3-(phenylmethoxycarbonylamino)butanoic acid
—— (2S)-2-(dimethylamino)-N-[(2S)-7,7-dimethyl-1-[[4-(2-methylphenyl)piperazin-1-yl]sulfonylmethyl]-2-bicyclo[2.2.1]heptanyl]-4-methylsulfonylbutanamide —— C28H46N4O5S2
(2S)-2-(dimethylamino)-N-[(2S)-7,7-dimethyl-1-[[4-(2-methylphenyl)piperazin-1-yl]sulfonylmethyl]-2-bicyclo[2.2.1]heptanyl]-4-methylsulfonylbutanamide
—— 2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-[(1S,3R)-3-(trifluoromethyl)cyclohexyl]acetamide —— C19H27F3N4O3S
2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-[(1S,3R)-3-(trifluoromethyl)cyclohexyl]acetamide
—— 1-N,3-N-dimethyl-4-(4-methylpiperazin-1-yl)-1-N,3-N-diphenyl-6-(3-phenylpropylamino)benzene-1,3-disulfonamide —— C34H41N5O4S2
1-N,3-N-dimethyl-4-(4-methylpiperazin-1-yl)-1-N,3-N-diphenyl-6-(3-phenylpropylamino)benzene-1,3-disulfonamide
—— (2S)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]propan-1-one —— C23H28FN3O3S
(2S)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]propan-1-one
—— 4-[4-[(2S)-1-oxo-1-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]propan-2-yl]piperazin-1-yl]benzenesulfonamide —— C21H28N4O3S2
4-[4-[(2S)-1-oxo-1-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]propan-2-yl]piperazin-1-yl]benzenesulfonamide
—— N-[(2R)-2-cyanopropyl]-N-ethyl-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]acetamide —— C20H27FN4O3
N-[(2R)-2-cyanopropyl]-N-ethyl-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]acetamide
—— (2R)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]propan-1-one —— C23H28FN3O3S
(2R)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]propan-1-one
—— (2R)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]propan-1-one —— C23H28FN3O3S
(2R)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]propan-1-one
—— (2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-2-[4-(pyridine-4-carbonyl)-1,4-diazepan-1-yl]propan-1-one —— C24H30FN5O2
(2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-2-[4-(pyridine-4-carbonyl)-1,4-diazepan-1-yl]propan-1-one
—— 2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(3S)-3-(trifluoromethyl)piperidin-1-yl]ethanone —— C20H25F4N3O3
2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(3S)-3-(trifluoromethyl)piperidin-1-yl]ethanone
—— 2-[4-[4-[4-[[2-(4-Fluorophenyl)-2-[(4-methyl-1,2,4-triazol-3-yl)methyl]-1,3-dioxolan-4-yl]methoxy]phenyl]piperazin-1-yl]phenyl]-4-propan-2-yl-1,2,4-triazol-3-one —— C35H39FN8O4
2-[4-[4-[4-[[2-(4-Fluorophenyl)-2-[(4-methyl-1,2,4-triazol-3-yl)methyl]-1,3-dioxolan-4-yl]methoxy]phenyl]piperazin-1-yl]phenyl]-4-propan-2-yl-1,2,4-triazol-3-one
—— N-ethyl-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]acetamide —— C22H29FN4O3S
N-ethyl-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]acetamide
—— 4-[4-[(2S)-1-oxo-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]propan-2-yl]piperazin-1-yl]benzenesulfonamide —— C21H28N4O3S2
4-[4-[(2S)-1-oxo-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]propan-2-yl]piperazin-1-yl]benzenesulfonamide
—— N-[(S)-cyclopropyl(phenyl)methyl]-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]acetamide —— C22H28N4O3S
N-[(S)-cyclopropyl(phenyl)methyl]-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]acetamide
—— N-ethyl-N-[(1S)-1-(4-fluorophenyl)ethyl]-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]acetamide —— C22H29FN4O3S
N-ethyl-N-[(1S)-1-(4-fluorophenyl)ethyl]-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]acetamide
—— 4-[2-aminoethyl(ethyl)amino]-1-N,3-N-bis(3-methoxypropyl)-6-(4-phenylpiperazin-1-yl)benzene-1,3-disulfonamide —— C28H46N6O6S2
4-[2-aminoethyl(ethyl)amino]-1-N,3-N-bis(3-methoxypropyl)-6-(4-phenylpiperazin-1-yl)benzene-1,3-disulfonamide
—— (2S)-1-[4-(4-fluorophenyl)piperazin-1-yl]-2-[4-(pyridine-4-carbonyl)-1,4-diazepan-1-yl]propan-1-one —— C24H30FN5O2
(2S)-1-[4-(4-fluorophenyl)piperazin-1-yl]-2-[4-(pyridine-4-carbonyl)-1,4-diazepan-1-yl]propan-1-one
—— 2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-[(1R,3S)-3-(trifluoromethyl)cyclohexyl]acetamide —— C19H27F3N4O3S
2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-[(1R,3S)-3-(trifluoromethyl)cyclohexyl]acetamide
—— (2R)-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-(2,4,6-trimethylphenyl)propanamide —— C22H30N4O3S
(2R)-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-(2,4,6-trimethylphenyl)propanamide
—— N-[(2S)-2-cyanopropyl]-N-ethyl-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]acetamide —— C20H27FN4O3
N-[(2S)-2-cyanopropyl]-N-ethyl-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]acetamide
—— 4-[4-[2-oxo-2-[(3R)-3-(trifluoromethyl)piperidin-1-yl]ethyl]piperazin-1-yl]benzenesulfonamide —— C18H25F3N4O3S
4-[4-[2-oxo-2-[(3R)-3-(trifluoromethyl)piperidin-1-yl]ethyl]piperazin-1-yl]benzenesulfonamide
—— 4-[4-[(2R)-1-oxo-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]propan-2-yl]piperazin-1-yl]benzenesulfonamide —— C21H28N4O3S2
4-[4-[(2R)-1-oxo-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]propan-2-yl]piperazin-1-yl]benzenesulfonamide
—— N-[(1R)-1-(3,4-difluorophenyl)ethyl]-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-N-methylacetamide —— C23H26F3N3O3
N-[(1R)-1-(3,4-difluorophenyl)ethyl]-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-N-methylacetamide
—— 4-[4-[2-oxo-2-[(3S)-3-(trifluoromethyl)piperidin-1-yl]ethyl]piperazin-1-yl]benzenesulfonamide —— C18H25F3N4O3S
4-[4-[2-oxo-2-[(3S)-3-(trifluoromethyl)piperidin-1-yl]ethyl]piperazin-1-yl]benzenesulfonamide
—— (2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]propan-1-one —— C22H26FN3O3S
(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]propan-1-one
—— 2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-[(1S,3S)-3-(trifluoromethyl)cyclohexyl]acetamide —— C19H27F3N4O3S
2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-[(1S,3S)-3-(trifluoromethyl)cyclohexyl]acetamide
—— (2S)-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-(2,4,6-trimethylphenyl)propanamide —— C22H30N4O3S
(2S)-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]-N-(2,4,6-trimethylphenyl)propanamide
—— 2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(3R)-3-(trifluoromethyl)piperidin-1-yl]ethanone —— C20H25F4N3O3
2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(3R)-3-(trifluoromethyl)piperidin-1-yl]ethanone
—— N-[(R)-cyclopropyl(phenyl)methyl]-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]acetamide —— C22H28N4O3S
N-[(R)-cyclopropyl(phenyl)methyl]-2-[4-(4-sulfamoylphenyl)piperazin-1-yl]acetamide
—— 1-[(2R)-2-(4-methoxyphenyl)azepan-1-yl]-2-[4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]ethanone —— C23H33N5O3
1-[(2R)-2-(4-methoxyphenyl)azepan-1-yl]-2-[4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]ethanone
—— (2S)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]propan-1-one —— C23H28FN3O3S
(2S)-2-[4-[2-(4-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]propan-1-one
—— 4-[3-cyano-6-methoxy-7-(3-piperidin-1-ylpropoxy)quinolin-4-yl]-N-(4-propan-2-yloxyphenyl)piperazine-1-carboxamide —— C33H42N6O4
4-[3-cyano-6-methoxy-7-(3-piperidin-1-ylpropoxy)quinolin-4-yl]-N-(4-propan-2-yloxyphenyl)piperazine-1-carboxamide
—— 1-[(2R)-2-(3,4-dichlorophenyl)-4-(3,5-dimethylbenzoyl)piperazin-1-yl]-3-[(1S,4S)-5-(thiophen-2-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]propan-1-one —— C32H36Cl2N4O2S
1-[(2R)-2-(3,4-dichlorophenyl)-4-(3,5-dimethylbenzoyl)piperazin-1-yl]-3-[(1S,4S)-5-(thiophen-2-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]propan-1-one
—— N-(cyclohexanecarbonyl)-N-[1-(4-methoxyphenyl)-3-[4-(2-methoxyphenyl)piperazin-1-yl]propan-2-yl]cyclohexanecarboxamide —— C35H49N3O4
N-(cyclohexanecarbonyl)-N-[1-(4-methoxyphenyl)-3-[4-(2-methoxyphenyl)piperazin-1-yl]propan-2-yl]cyclohexanecarboxamide
—— 3-(2-chlorophenyl)-5-methyl-N-[3-[4-[2-(1,1,2,2,2-pentafluoroethoxy)phenyl]piperazin-1-yl]propyl]-1,2-oxazole-4-carboxamide —— C26H26ClF5N4O3
3-(2-chlorophenyl)-5-methyl-N-[3-[4-[2-(1,1,2,2,2-pentafluoroethoxy)phenyl]piperazin-1-yl]propyl]-1,2-oxazole-4-carboxamide
—— 2-Carbamoyl-8-<3-{4-[2-methoxy-5-(2,2,2-trifluoroethoxy)-phenyl]-1-piperazinyl}-propylcarbamoyl>-3-methyl-4-oxo-4H-1-benzopyran 335087-23-5 C28H31F3N4O6
2-Carbamoyl-8-<3-{4-[2-methoxy-5-(2,2,2-trifluoroethoxy)-phenyl]-1-piperazinyl}-propylcarbamoyl>-3-methyl-4-oxo-4H-1-benzopyran
—— (2S)-2-methyl-1,4-bis(3-methylbutyl)piperazine —— C15H32N2
(2S)-2-methyl-1,4-bis(3-methylbutyl)piperazine