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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl 4-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate —— C31H38N4O6S
ethyl 4-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate
—— 4-chloro-N-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]butanamide —— C29H35ClN4O4S
4-chloro-N-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]butanamide
—— 4-chloro-N-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]butanamide —— C29H35ClN4O4S
4-chloro-N-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]butanamide
—— [(2S)-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl] 3-methyl-4-oxophthalazine-1-carboxylate —— C23H24N4O4
[(2S)-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl] 3-methyl-4-oxophthalazine-1-carboxylate
—— (4aR,5S)-9-chloro-3-(3-chlorophenyl)-5'-methyl-2'-phenylspiro[2,4,4a,6-tetrahydro-1H-pyrazino[1,2-a]quinoline-5,4'-pyrazole]-3'-one —— C27H24Cl2N4O
(4aR,5S)-9-chloro-3-(3-chlorophenyl)-5'-methyl-2'-phenylspiro[2,4,4a,6-tetrahydro-1H-pyrazino[1,2-a]quinoline-5,4'-pyrazole]-3'-one
—— [(2R)-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl] 4-propan-2-yloxybenzoate —— C23H28N2O4
[(2R)-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl] 4-propan-2-yloxybenzoate
—— (2S)-N-benzyl-4-[3-(2-fluorophenyl)-[1,2,4]triazolo[4,3-c]quinazolin-5-yl]-2-methylpiperazine-1-carboxamide —— C28H26FN7O
(2S)-N-benzyl-4-[3-(2-fluorophenyl)-[1,2,4]triazolo[4,3-c]quinazolin-5-yl]-2-methylpiperazine-1-carboxamide
—— 4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]-3-[4-[2-(trifluoromethoxy)benzoyl]piperazin-1-yl]benzenesulfonamide —— C24H28F3N3O6S
4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]-3-[4-[2-(trifluoromethoxy)benzoyl]piperazin-1-yl]benzenesulfonamide
—— [(2S)-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl] 4-(2-methylpropoxy)benzoate —— C24H30N2O4
[(2S)-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl] 4-(2-methylpropoxy)benzoate
—— (2S)-2-[(5-methyl-4-phenyl-1,2,4-triazol-3-yl)sulfanyl]-1-(4-phenylpiperazin-1-yl)propan-1-one —— C22H25N5OS
(2S)-2-[(5-methyl-4-phenyl-1,2,4-triazol-3-yl)sulfanyl]-1-(4-phenylpiperazin-1-yl)propan-1-one
—— 3-[4-(3-chloro-4-fluorophenyl)sulfonylpiperazin-1-yl]-4-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzenesulfonamide —— C22H27ClFN3O6S2
3-[4-(3-chloro-4-fluorophenyl)sulfonylpiperazin-1-yl]-4-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzenesulfonamide
—— [(1S)-2-[4-[2-methoxy-5-[methyl(2-phenylethyl)sulfamoyl]phenyl]piperazin-1-yl]-2-oxo-1-phenylethyl] acetate —— C30H35N3O6S
[(1S)-2-[4-[2-methoxy-5-[methyl(2-phenylethyl)sulfamoyl]phenyl]piperazin-1-yl]-2-oxo-1-phenylethyl] acetate
—— 2-(4-fluorophenyl)-1-[(2S)-4-[3-(2-fluorophenyl)-[1,2,4]triazolo[4,3-c]quinazolin-5-yl]-2-methylpiperazin-1-yl]ethanone —— C28H24F2N6O
2-(4-fluorophenyl)-1-[(2S)-4-[3-(2-fluorophenyl)-[1,2,4]triazolo[4,3-c]quinazolin-5-yl]-2-methylpiperazin-1-yl]ethanone
—— [(2S)-4-[3-(2-fluorophenyl)-[1,2,4]triazolo[4,3-c]quinazolin-5-yl]-2-methylpiperazin-1-yl]-(2-methoxyphenyl)methanone —— C28H25FN6O2
[(2S)-4-[3-(2-fluorophenyl)-[1,2,4]triazolo[4,3-c]quinazolin-5-yl]-2-methylpiperazin-1-yl]-(2-methoxyphenyl)methanone
—— 3-[4-(3-chloro-4-fluorophenyl)sulfonylpiperazin-1-yl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzenesulfonamide —— C22H27ClFN3O6S2
3-[4-(3-chloro-4-fluorophenyl)sulfonylpiperazin-1-yl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzenesulfonamide
—— (1R,2S,4R)-N-[3-[4-(3-methylphenyl)piperazin-1-yl]propyl]bicyclo[2.2.1]heptane-2-carboxamide —— C22H33N3O
(1R,2S,4R)-N-[3-[4-(3-methylphenyl)piperazin-1-yl]propyl]bicyclo[2.2.1]heptane-2-carboxamide
—— (1R,2R,4R)-N-[3-[4-(3-methylphenyl)piperazin-1-yl]propyl]bicyclo[2.2.1]heptane-2-carboxamide —— C22H33N3O
(1R,2R,4R)-N-[3-[4-(3-methylphenyl)piperazin-1-yl]propyl]bicyclo[2.2.1]heptane-2-carboxamide
—— (7S)-4-[4-(4-methoxyphenyl)sulfonylpiperazin-1-yl]-7-methyl-2-(2-phenylethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine —— C30H34N4O3S2
(7S)-4-[4-(4-methoxyphenyl)sulfonylpiperazin-1-yl]-7-methyl-2-(2-phenylethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine
—— (5E)-3-(3-ethoxypropyl)-5-[[2-[4-(4-methoxyphenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H33N5O4S2
(5E)-3-(3-ethoxypropyl)-5-[[2-[4-(4-methoxyphenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-3-hexyl-5-[[2-[4-(2-methoxyphenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H35N5O3S2
(5E)-3-hexyl-5-[[2-[4-(2-methoxyphenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[(4-bromophenyl)sulfonylamino]-2-(4-ethylpiperazin-1-yl)-N-[(1R)-1-phenylethyl]benzenesulfonamide —— C26H31BrN4O4S2
5-[(4-bromophenyl)sulfonylamino]-2-(4-ethylpiperazin-1-yl)-N-[(1R)-1-phenylethyl]benzenesulfonamide
—— 4-chloro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]butanamide —— C29H35ClN4O4S
4-chloro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]butanamide
—— ethyl 4-[4-oxo-3-[(E)-[4-oxo-3-(3-phenylpropyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyrido[1,2-a]pyrimidin-2-yl]piperazine-1-carboxylate —— C28H29N5O4S2
ethyl 4-[4-oxo-3-[(E)-[4-oxo-3-(3-phenylpropyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyrido[1,2-a]pyrimidin-2-yl]piperazine-1-carboxylate
—— (2S)-4-[6-chloro-2-[2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide —— C24H31Cl2N7O2S
(2S)-4-[6-chloro-2-[2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide
—— 2-chloro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]acetamide —— C27H31ClN4O4S
2-chloro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]acetamide
—— (1R,2R,4R)-N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]bicyclo[2.2.1]heptane-2-carboxamide —— C22H33N3O
(1R,2R,4R)-N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]bicyclo[2.2.1]heptane-2-carboxamide
—— 2-chloro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]acetamide —— C27H31ClN4O4S
2-chloro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]acetamide
—— (2S)-4-[6-chloro-2-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide —— C24H31ClFN7O2S
(2S)-4-[6-chloro-2-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide
—— (5E)-5-[[5-(4-methylphenyl)furan-2-yl]methylidene]-2-[4-(4-nitrophenyl)piperazin-1-yl]-1,3-thiazol-4-one —— C25H22N4O4S
(5E)-5-[[5-(4-methylphenyl)furan-2-yl]methylidene]-2-[4-(4-nitrophenyl)piperazin-1-yl]-1,3-thiazol-4-one
—— (2R)-4-[6-chloro-2-[2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide —— C24H31Cl2N7O2S
(2R)-4-[6-chloro-2-[2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide
—— 4-chloro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]butanamide —— C29H35ClN4O4S
4-chloro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]butanamide
—— (E)-3-(2,3-dimethoxyphenyl)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]prop-2-enenitrile —— C22H22FN3O3
(E)-3-(2,3-dimethoxyphenyl)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]prop-2-enenitrile
—— (2R)-4-[6-chloro-2-[2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-(3-chlorophenyl)-2-methylpiperazine-1-carboxamide —— C29H33Cl2N7O2S
(2R)-4-[6-chloro-2-[2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-(3-chlorophenyl)-2-methylpiperazine-1-carboxamide
—— (E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3-(4-morpholin-4-ylphenyl)prop-2-enenitrile —— C24H25FN4O2
(E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3-(4-morpholin-4-ylphenyl)prop-2-enenitrile
—— (5E)-5-[[2-[4-(2-fluorophenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(3-methylbutyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C28H30FN5O2S2
(5E)-5-[[2-[4-(2-fluorophenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(3-methylbutyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— (2E,4E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-phenylpenta-2,4-dienenitrile —— C22H20FN3O
(2E,4E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-phenylpenta-2,4-dienenitrile
—— 2-[2-[(E)-2-cyano-3-[4-(2-fluorophenyl)piperazin-1-yl]-3-oxoprop-1-enyl]phenoxy]acetate —— C22H19FN3O4-
2-[2-[(E)-2-cyano-3-[4-(2-fluorophenyl)piperazin-1-yl]-3-oxoprop-1-enyl]phenoxy]acetate
—— (E)-3-(3-fluorophenyl)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]prop-2-enenitrile —— C20H17F2N3O
(E)-3-(3-fluorophenyl)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]prop-2-enenitrile
—— (E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3-(4-hydroxy-3,5-dimethoxyphenyl)prop-2-enenitrile —— C22H22FN3O4
(E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3-(4-hydroxy-3,5-dimethoxyphenyl)prop-2-enenitrile
—— (2R)-4-[6-chloro-2-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide —— C24H31ClFN7O2S
(2R)-4-[6-chloro-2-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide
—— 5-[(4-bromophenyl)sulfonylamino]-2-(4-ethylpiperazin-1-yl)-N-[(1S)-1-phenylethyl]benzenesulfonamide —— C26H31BrN4O4S2
5-[(4-bromophenyl)sulfonylamino]-2-(4-ethylpiperazin-1-yl)-N-[(1S)-1-phenylethyl]benzenesulfonamide
—— (5E)-3-(furan-2-ylmethyl)-5-[[2-[4-(2-methoxyphenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H27N5O4S2
(5E)-3-(furan-2-ylmethyl)-5-[[2-[4-(2-methoxyphenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (2R)-N-tert-butyl-4-[6-chloro-2-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-2-methylpiperazine-1-carboxamide —— C26H35ClFN7O2S
(2R)-N-tert-butyl-4-[6-chloro-2-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-2-methylpiperazine-1-carboxamide
—— (2S)-N-tert-butyl-4-[6-chloro-2-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-2-methylpiperazine-1-carboxamide —— C26H35ClFN7O2S
(2S)-N-tert-butyl-4-[6-chloro-2-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-2-methylpiperazine-1-carboxamide
—— (E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3-(4-hydroxy-3-nitrophenyl)prop-2-enenitrile —— C20H17FN4O4
(E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3-(4-hydroxy-3-nitrophenyl)prop-2-enenitrile
—— (2S)-4-[2-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]sulfanyl-6-chloropyrimidin-4-yl]-N-tert-butyl-2-methylpiperazine-1-carboxamide —— C27H38ClN7O2S
(2S)-4-[2-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]sulfanyl-6-chloropyrimidin-4-yl]-N-tert-butyl-2-methylpiperazine-1-carboxamide
—— (2S)-4-[6-chloro-2-[2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-(3-chlorophenyl)-2-methylpiperazine-1-carboxamide —— C29H33Cl2N7O2S
(2S)-4-[6-chloro-2-[2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl]sulfanylpyrimidin-4-yl]-N-(3-chlorophenyl)-2-methylpiperazine-1-carboxamide
—— (2R)-4-[6-chloro-2-[2-oxo-2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide —— C25H31ClF3N7O2S
(2R)-4-[6-chloro-2-[2-oxo-2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide
—— (2S)-4-[6-chloro-2-[2-oxo-2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide —— C25H31ClF3N7O2S
(2S)-4-[6-chloro-2-[2-oxo-2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]sulfanylpyrimidin-4-yl]-N-ethyl-2-methylpiperazine-1-carboxamide
—— (2R)-4-[2-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]sulfanyl-6-chloropyrimidin-4-yl]-N-tert-butyl-2-methylpiperazine-1-carboxamide —— C27H38ClN7O2S
(2R)-4-[2-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]sulfanyl-6-chloropyrimidin-4-yl]-N-tert-butyl-2-methylpiperazine-1-carboxamide