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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(2-naphthylthio)benzo[b]thiophene 1453485-43-2 C18H12S2
3-(2-naphthylthio)benzo[b]thiophene
—— ethyl 6-(3,4,5-trimethoxyphenyl)-2-naphthoate 1334137-90-4 C22H22O5
ethyl 6-(3,4,5-trimethoxyphenyl)-2-naphthoate
—— 1-(4-methylphenyl)-4-(2-phenylethynyl)[1,2,4]triazolo[4,3-a]quinoxaline 1435938-57-0 C24H16N4
1-(4-methylphenyl)-4-(2-phenylethynyl)[1,2,4]triazolo[4,3-a]quinoxaline
—— 2-{[3-((R)-2-Acetylamino-2-methylcarbamoyl-ethylsulfanylmethyl)-2-hydroxy-tetrahydro-furan-2-carbonyl]-amino}-3,4-dihydroxy-4-methyl-tetrahydro-furan-2-carboxylic acid amide 126503-36-4 C18H30N4O9S
2-{[3-((R)-2-Acetylamino-2-methylcarbamoyl-ethylsulfanylmethyl)-2-hydroxy-tetrahydro-furan-2-carbonyl]-amino}-3,4-dihydroxy-4-methyl-tetrahydro-furan-2-carboxylic acid amide
—— 1-(2,3,4,6-tetra-O-acetyl-β-D-galactopyranosyl)-3,3-bis(4-methylphenyl)indolin-2-one 1629138-85-7 C36H37NO10
1-(2,3,4,6-tetra-O-acetyl-β-D-galactopyranosyl)-3,3-bis(4-methylphenyl)indolin-2-one
—— 4-(2-amino-acetyl)-piperazine-1-carboxylic acid tert-butyl ester acetate 1021522-67-7 C2H4O2*C11H21N3O3
4-(2-amino-acetyl)-piperazine-1-carboxylic acid tert-butyl ester acetate
—— 3-(2-cyclohex-1-enyl-pyridin-4-yl)-7-pyridin-3-yl-imidazo[1,2-a]pyridine 1146612-67-0 C23H20N4
3-(2-cyclohex-1-enyl-pyridin-4-yl)-7-pyridin-3-yl-imidazo[1,2-a]pyridine
—— (+/-)-5-(4-fluorophenoxy)-2-methyl-8-(1H-pyrazol-4-yl)-2,3,4,5-tetrahydro-1H-benzo[c]azepine 1084809-83-5 C20H20FN3O
(+/-)-5-(4-fluorophenoxy)-2-methyl-8-(1H-pyrazol-4-yl)-2,3,4,5-tetrahydro-1H-benzo[c]azepine
—— 4-({(S)-3-methyl-2-[4-(2-phenoxy-phenylsulfamoyl)-benzoylamino]-butyrylamino}-methyl)-piperidine-1-carboxylic acid tert-butyl ester 1021522-93-9 C35H44N4O7S
4-({(S)-3-methyl-2-[4-(2-phenoxy-phenylsulfamoyl)-benzoylamino]-butyrylamino}-methyl)-piperidine-1-carboxylic acid tert-butyl ester
—— N-(4-((3R,4S)-4-(4-chlorophenyl)-3,4-dihydroxy-3-methylpiperidin-1-yl)-2-methyl-4-oxobutan-2-yl)benzamide 1108154-32-0 C24H29ClN2O4
N-(4-((3R,4S)-4-(4-chlorophenyl)-3,4-dihydroxy-3-methylpiperidin-1-yl)-2-methyl-4-oxobutan-2-yl)benzamide
—— 2-chloro-N-cyclopropyl-5-(3-methoxy-propyl)-benzamide 1007392-83-7 C14H18ClNO2
2-chloro-N-cyclopropyl-5-(3-methoxy-propyl)-benzamide
—— 6-[5-(2-methoxy-4-trifluoromethylbenzoylamino)pyridin-2-yloxy]-1-methyl-1H-indole-2-carboxylic acid 1150744-87-8 C24H18F3N3O5
6-[5-(2-methoxy-4-trifluoromethylbenzoylamino)pyridin-2-yloxy]-1-methyl-1H-indole-2-carboxylic acid
—— 2-benzyl-3-[(4-isobutylphenylsulfonyl)amino]-3-oxopropionic acid 1094201-52-1 C20H23NO5S
2-benzyl-3-[(4-isobutylphenylsulfonyl)amino]-3-oxopropionic acid
—— 6-{3-[(4-cyclobutyl-3-methyl-5-oxopiperazin-1-yl)carbonyl]-4-fluorobenzyl}-4,5-dimethylpyridazin-3(2H)-one 1154872-20-4 C23H27FN4O3
6-{3-[(4-cyclobutyl-3-methyl-5-oxopiperazin-1-yl)carbonyl]-4-fluorobenzyl}-4,5-dimethylpyridazin-3(2H)-one
—— 6-{2-bromo-5-[(4-cyclopentyl-3-oxopiperazin-1-yl)carbonyl]-4-fluorobenzyl}-4,5-dimethylpyridazin-3(2H)-one 1154870-79-7 C23H26BrFN4O3
6-{2-bromo-5-[(4-cyclopentyl-3-oxopiperazin-1-yl)carbonyl]-4-fluorobenzyl}-4,5-dimethylpyridazin-3(2H)-one
—— 4-[1-methyl-5-(5-nitropyrimidin-2-yloxy)-1H-indole-2-carbonyl]piperazine-1-carboxylic acid tert-butyl ester 1150742-95-2 C23H26N6O6
4-[1-methyl-5-(5-nitropyrimidin-2-yloxy)-1H-indole-2-carbonyl]piperazine-1-carboxylic acid tert-butyl ester
—— 6-bromo-2-(5-bromopyridin-3-yl)-1-cyclopropyl-1H-benzimidazole 1356481-16-7 C15H11Br2N3
6-bromo-2-(5-bromopyridin-3-yl)-1-cyclopropyl-1H-benzimidazole
—— 5-bromo-1-(propan-2-yloxy)-2-(pyridin-3-yl)-1H-benzimidazole 1356482-85-3 C15H14BrN3O
5-bromo-1-(propan-2-yloxy)-2-(pyridin-3-yl)-1H-benzimidazole
—— [(R)-2-(5-(dimethylamino)methyl-7-cyclopentylamino-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-methanol 1120342-46-2 C20H28N4OS
[(R)-2-(5-(dimethylamino)methyl-7-cyclopentylamino-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-methanol
—— (S)-tert-butyl 2-(8-(2H-tetrazol-5-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoate 1080642-28-9 C22H25N5O5S
(S)-tert-butyl 2-(8-(2H-tetrazol-5-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoate
—— {3-[3-(2-cyclopent-1-enyl-pyridin-4-yl)-imidazo[1,2-a]pyridin-7-yl]-benzyl}-isopropyl-amine 1146613-55-9 C27H28N4
{3-[3-(2-cyclopent-1-enyl-pyridin-4-yl)-imidazo[1,2-a]pyridin-7-yl]-benzyl}-isopropyl-amine
—— 4-iodo-N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide 1150463-56-1 C34H31F3IN5O5S
4-iodo-N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide
—— N-{[6-(benzoylamino)-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-4-fluorobenzamide 1141878-76-3 C24H17F4N3O4
N-{[6-(benzoylamino)-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-4-fluorobenzamide
—— 4-cyano-N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide 1150463-79-8 C35H31F3N6O5S
4-cyano-N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide
—— phenylmethyl 4-[(2-hydroxy-2-methylpropyl)amino]-1-piperidinecarboxylate 1237840-92-4 C17H26N2O3
phenylmethyl 4-[(2-hydroxy-2-methylpropyl)amino]-1-piperidinecarboxylate
—— 4-[((S)-2-{4-[2-(2,4-dichloro-phenoxy)-phenylsulfamoyl]-benzoylamino}-propionylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester 1021522-45-1 C33H38Cl2N4O7S
4-[((S)-2-{4-[2-(2,4-dichloro-phenoxy)-phenylsulfamoyl]-benzoylamino}-propionylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester
—— 3,4-dichloro-N-{2-[1-methyl-2-(piperazine-1-carbonyl)-1H-indol-5-yloxy]pyrimidin-5-yl}benzamide 1150746-34-1 C25H22Cl2N6O3
3,4-dichloro-N-{2-[1-methyl-2-(piperazine-1-carbonyl)-1H-indol-5-yloxy]pyrimidin-5-yl}benzamide
—— N-methyl-3-{3-[2-(3-methyl-pyrazol-1-yl)-pyridin-4-yl]-imidazo[1,2-a]pyridin-7-yl}-benzamide 1146612-48-7 C24H20N6O
N-methyl-3-{3-[2-(3-methyl-pyrazol-1-yl)-pyridin-4-yl]-imidazo[1,2-a]pyridin-7-yl}-benzamide
—— 3-[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]-N-(6-methylpyridin-3-yl)propanamide 1141877-36-2 C18H15ClF3N3O3
3-[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]-N-(6-methylpyridin-3-yl)propanamide
—— (4-benzo[1,3]dioxol-5-ylmethylpiperazin-1-yl)[1-methyl-5-(5-methylaminopyridin-2-yloxy)-1H-indol-2-yl]methanone 1150745-02-0 C28H29N5O4
(4-benzo[1,3]dioxol-5-ylmethylpiperazin-1-yl)[1-methyl-5-(5-methylaminopyridin-2-yloxy)-1H-indol-2-yl]methanone
—— N-(benzothiazole-6-yl)-2-chloro-N-[1-(4-trifluoromethylbenzoyl)piperidin-4-yl]acetamide 1186213-37-5 C22H19ClF3N3O2S
N-(benzothiazole-6-yl)-2-chloro-N-[1-(4-trifluoromethylbenzoyl)piperidin-4-yl]acetamide
—— 2-ethylsulfanyl-4,6-dimethyl-quinoline-3-carboxylic acid 1242555-56-1 C14H15NO2S
2-ethylsulfanyl-4,6-dimethyl-quinoline-3-carboxylic acid
—— 3-(5-tert-butylbenzoxazol-2-yl)-5-(2-chlorophenoxymethyl)phenylamine 1033803-22-3 C24H23ClN2O2
3-(5-tert-butylbenzoxazol-2-yl)-5-(2-chlorophenoxymethyl)phenylamine
—— (R)-3-methyl-2-(7-(5-methyl-1,3,4-thiadiazol-2-yl)dibenzo[b,d]furan-2-sulfonamido)butanoic acid 1080640-57-8 C20H19N3O5S2
(R)-3-methyl-2-(7-(5-methyl-1,3,4-thiadiazol-2-yl)dibenzo[b,d]furan-2-sulfonamido)butanoic acid
—— tert-butyl 4-(6-(cyclopentyloxy)pyridin-2-yl)piperazine-1-carboxylate 1092848-24-2 C19H29N3O3
tert-butyl 4-(6-(cyclopentyloxy)pyridin-2-yl)piperazine-1-carboxylate
—— 2-(7-bromo-5-fluoro-2-oxo-1,2-dihydro-indol-3-ylidenemethyl)-5-(2-diethylamino-ethyl)-3-methyl-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one 1082988-28-0 C24H28BrFN4O2
2-(7-bromo-5-fluoro-2-oxo-1,2-dihydro-indol-3-ylidenemethyl)-5-(2-diethylamino-ethyl)-3-methyl-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one
—— 1-(3,4-dichlorobenzyl)-1,3-dimethyl-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)urea hydrochloride 1227095-82-0 C20H24Cl2N4O*ClH
1-(3,4-dichlorobenzyl)-1,3-dimethyl-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)urea hydrochloride
—— N-(1-methylethyl)-4-(4,5,6,7-tetrahydro-2-phenylpyrazolo[1,5-a]pyridin-3-yl)-2-aminopyrimidine 1161075-27-9 C20H23N5
N-(1-methylethyl)-4-(4,5,6,7-tetrahydro-2-phenylpyrazolo[1,5-a]pyridin-3-yl)-2-aminopyrimidine
—— 5-Methylisoindoline hydrochloride 1204600-16-7 C9H12ClN
5-Methylisoindoline hydrochloride
—— (2-methoxy-1-oxy-pyridin-3-yl)carbamic acid benzyl ester 1009121-41-8 C14H14N2O4
(2-methoxy-1-oxy-pyridin-3-yl)carbamic acid benzyl ester
—— methyl 4-(2-{5-bromo-3-chloro-6-[(3-methoxyphenoxy)methyl]-2-oxopyridin-1(2H)-yl}ethyl)benzoate 1091600-13-3 C23H21BrClNO5
methyl 4-(2-{5-bromo-3-chloro-6-[(3-methoxyphenoxy)methyl]-2-oxopyridin-1(2H)-yl}ethyl)benzoate
—— 4-[2-(4-fluorophenyl)-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]thiazin-3-yl]-N-(1-methylethyl)-2-pyrimidinamine 1161076-12-5 C19H20FN5S
4-[2-(4-fluorophenyl)-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]thiazin-3-yl]-N-(1-methylethyl)-2-pyrimidinamine
—— N,N-diethyl-2-{4-[(4-methoxybenzoyl)amino]benzyl}-N'-(2-naphthylsulfonyl)malonamide 1094194-80-5 C32H33N3O6S
N,N-diethyl-2-{4-[(4-methoxybenzoyl)amino]benzyl}-N'-(2-naphthylsulfonyl)malonamide
—— 1-(1-tert-butoxycarbonyl-piperidin-4-yl)-1H-benzotriazole-5-carboxylic acid allyl ester 1067718-05-1 C20H26N4O4
1-(1-tert-butoxycarbonyl-piperidin-4-yl)-1H-benzotriazole-5-carboxylic acid allyl ester
—— 2-methyl-2-(1,3,3-trimethyl-butyl)-tetrahydrofuran 1103676-17-0 C12H24O
2-methyl-2-(1,3,3-trimethyl-butyl)-tetrahydrofuran
—— 4-[(acetyl-phenyl-amino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester 199105-13-0 C19H28N2O3
4-[(acetyl-phenyl-amino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester
—— 1-[(S)-2-amino-4-oxo-4-(2-thiophen-3-yl-4-trifluoromethyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-butyl]-3-methyl-piperidine-2,6-dione hydrochloride 1173175-42-2 C22H24F3N5O3S*ClH
1-[(S)-2-amino-4-oxo-4-(2-thiophen-3-yl-4-trifluoromethyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-butyl]-3-methyl-piperidine-2,6-dione hydrochloride
—— 5-[4-(4-morpholinyl)-6-quinazolinyl]-3-pyridinamine 1093819-55-6 C17H17N5O
5-[4-(4-morpholinyl)-6-quinazolinyl]-3-pyridinamine
—— [(S)-1-(3,3-difluoro-2-hydroxy-6-oxo-piperidin-1-ylmethyl)-3-(2-furan-2-yl-4-trifluoromethyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-3-oxo-propyl]-carbamic acid t-butyl ester 1173175-56-8 C26H30F5N5O6
[(S)-1-(3,3-difluoro-2-hydroxy-6-oxo-piperidin-1-ylmethyl)-3-(2-furan-2-yl-4-trifluoromethyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-3-oxo-propyl]-carbamic acid t-butyl ester
—— (2R,4S)-methyl 2-(3,4-difluorophenyl)-4-(3-oxo-2,3-dihydroisoxazol-5-yl)piperidine-1-carboxylate 1251845-97-2 C16H16F2N2O4
(2R,4S)-methyl 2-(3,4-difluorophenyl)-4-(3-oxo-2,3-dihydroisoxazol-5-yl)piperidine-1-carboxylate