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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[1-(3-chloro-2,6-difluorophenyl)ethoxy]aniline 1146854-14-9 C14H12ClF2NO
4-[1-(3-chloro-2,6-difluorophenyl)ethoxy]aniline
—— ethyl 2-[4-(benzoylamino)benzyl]-3-[(2-naphthylsulfonyl)amino]-3-oxopropionate 1094201-80-5 C29H26N2O6S
ethyl 2-[4-(benzoylamino)benzyl]-3-[(2-naphthylsulfonyl)amino]-3-oxopropionate
—— N-[2-hydroxy-1-(2-methoxy-phenyl)-ethyl]-2-methoxy-4-pyridin-4-yl-benzamide 1127309-13-0 C22H22N2O4
N-[2-hydroxy-1-(2-methoxy-phenyl)-ethyl]-2-methoxy-4-pyridin-4-yl-benzamide
—— 7-{[(3-piperidin-1-ylpropyl)amino]methyl}pyrrolo[1,2-a]quinoxalin-4(5H)-one 1036726-74-5 C20H26N4O
7-{[(3-piperidin-1-ylpropyl)amino]methyl}pyrrolo[1,2-a]quinoxalin-4(5H)-one
—— 2-(biphenyl-4-ylmethyl)-3-chloro-7-isobutyl-5-methyl-2H-pyrazolo[3,4-d]pyrimidine-4,6(5H,7H)-dione 1160490-76-5 C23H23ClN4O2
2-(biphenyl-4-ylmethyl)-3-chloro-7-isobutyl-5-methyl-2H-pyrazolo[3,4-d]pyrimidine-4,6(5H,7H)-dione
—— Methyl 2-amino-2-(pyridin-4-yl)acetate hydrochloride 1427475-14-6 C8H11ClN2O2
Methyl 2-amino-2-(pyridin-4-yl)acetate hydrochloride
—— 4-(3-methyl-pyridin-4-yl)-N-[(R)-1-(3-trifluoromethyl-phenyl)-ethyl]-benzamide 1127309-52-7 C22H19F3N2O
4-(3-methyl-pyridin-4-yl)-N-[(R)-1-(3-trifluoromethyl-phenyl)-ethyl]-benzamide
—— N,N-diethyl-N'-(2-naphthylsulfonyl)-2-[4-(pivaloylamino)benzyl]malonamide 1094194-65-6 C29H35N3O5S
N,N-diethyl-N'-(2-naphthylsulfonyl)-2-[4-(pivaloylamino)benzyl]malonamide
—— methyl 3-{4-[(6-butyl-8-quinolinyl)oxy]-1-piperidinyl}propanoate 1145873-32-0 C22H30N2O3
methyl 3-{4-[(6-butyl-8-quinolinyl)oxy]-1-piperidinyl}propanoate
—— 2-isopropylamino-6-methyl-pyrimidine-4-carboxylic acid ethyl ester 1150644-96-4 C11H17N3O2
2-isopropylamino-6-methyl-pyrimidine-4-carboxylic acid ethyl ester
—— {5-[6-(4-chloro-2-fluorophenyl)-imidazo[2,1-b]oxazol-5-yl]-pyridin-2-yl}-hydrazine 1033041-18-7 C16H11ClFN5O
{5-[6-(4-chloro-2-fluorophenyl)-imidazo[2,1-b]oxazol-5-yl]-pyridin-2-yl}-hydrazine
—— 4-(2,5-difluorobenzoyl)piperazine-1-carboxylic acid tert-butyl ester 1071521-84-0 C16H20F2N2O3
4-(2,5-difluorobenzoyl)piperazine-1-carboxylic acid tert-butyl ester
—— (R)-2-(8-(4,4-dimethyl-2-oxo-2,4-dihydro-1H-benzo[d][1,3]oxazin-6-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoic acid 1080637-55-3 C27H26N2O7S
(R)-2-(8-(4,4-dimethyl-2-oxo-2,4-dihydro-1H-benzo[d][1,3]oxazin-6-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoic acid
—— 3-but-2-yn-1-yl-8-[(2R)-1-(2H-1,2,3-triazol-2-yl)propan-2-yl]-3,8-dihydrobenzo[1,2-d:4,5-d']bis[1,2,3]triazine-4,9-dione 1134101-31-7 C17H15N9O2
3-but-2-yn-1-yl-8-[(2R)-1-(2H-1,2,3-triazol-2-yl)propan-2-yl]-3,8-dihydrobenzo[1,2-d:4,5-d']bis[1,2,3]triazine-4,9-dione
—— 1,3-dichloro-2-[1-(4-nitrophenoxy)propyl]benzene 1173240-95-3 C15H13Cl2NO3
1,3-dichloro-2-[1-(4-nitrophenoxy)propyl]benzene
—— 4-(tert-butyldimethylsilyloxy)-methyl-2-chloro-5-(2,3-difluoro-6-methoxybenzyloxy)-1-nitrobenzene 1073437-94-1 C21H26ClF2NO5Si
4-(tert-butyldimethylsilyloxy)-methyl-2-chloro-5-(2,3-difluoro-6-methoxybenzyloxy)-1-nitrobenzene
—— 3-bromo-6-chloromethyl-2-propyl-pyridine 1149593-14-5 C9H11BrClN
3-bromo-6-chloromethyl-2-propyl-pyridine
—— isopropyl N-acetyl-tyrosinate 1003591-92-1 C14H19NO4
isopropyl N-acetyl-tyrosinate
—— 1-(4-benzo[1,3]dioxol-5-ylmethylpiperazin-1-yl)-2-[5-(5-bromopyridin-2-yloxy)indol-1-yl]ethanone 1150745-04-2 C27H25BrN4O4
1-(4-benzo[1,3]dioxol-5-ylmethylpiperazin-1-yl)-2-[5-(5-bromopyridin-2-yloxy)indol-1-yl]ethanone
—— (4-fluorophenyl)(2-piperidin-1-ylthiazol-5-ylmethyl)carbamic acid tert-butyl ester 1033619-95-2 C20H26FN3O2S
(4-fluorophenyl)(2-piperidin-1-ylthiazol-5-ylmethyl)carbamic acid tert-butyl ester
—— (3,4-dichlorobenzyl)-[2-methyl-8-(2-pyrazol-1-yl-ethoxy)-quinolin-4-yl]-amine hydrochloride 1121528-24-2 C22H20Cl2N4O*ClH
(3,4-dichlorobenzyl)-[2-methyl-8-(2-pyrazol-1-yl-ethoxy)-quinolin-4-yl]-amine hydrochloride
—— 2-phenylamino-N-(2-piperidin-1-yl-ethyl)-6-[4-(3-pyridin-3-ylmethyl-ureido)-phenyl]-nicotinamide 1138321-63-7 C32H35N7O2
2-phenylamino-N-(2-piperidin-1-yl-ethyl)-6-[4-(3-pyridin-3-ylmethyl-ureido)-phenyl]-nicotinamide
—— 6-(3-{[4-(3,3-difluorocyclobutyl)-3-methyl-5-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethylpyridazin-3(2H)-one 1154872-45-3 C23H25F3N4O3
6-(3-{[4-(3,3-difluorocyclobutyl)-3-methyl-5-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethylpyridazin-3(2H)-one
—— N-methyl-N-[1-[1-[5-methyl-6-[[6-[5-(trifluoromethyl)furan-2-yl]oxan-2-yl]methylamino]pyrimidine-4-carbonyl]piperidin-4-yl]piperidin-4-yl]methanesulfonamide 1312779-13-7 C29H41F3N6O5S
N-methyl-N-[1-[1-[5-methyl-6-[[6-[5-(trifluoromethyl)furan-2-yl]oxan-2-yl]methylamino]pyrimidine-4-carbonyl]piperidin-4-yl]piperidin-4-yl]methanesulfonamide
—— N-{2-chloro-4-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-ylsulfamoyl]phenyl}acetamide 1150463-81-2 C36H34ClF3N6O6S
N-{2-chloro-4-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-ylsulfamoyl]phenyl}acetamide
—— [4-(1-methylpiperidin-4-ylidene)-10-oxo-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]carboxylic acid 1176737-28-2 C20H19NO3S
[4-(1-methylpiperidin-4-ylidene)-10-oxo-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]carboxylic acid
—— N-(2-{[4-(1H-benzimidazol-5-yl)phenyl]oxy}ethyl)-4,4-dimethylcyclohexanamine trifluoroacetate 1008357-75-2 C2HF3O2*C23H29N3O
N-(2-{[4-(1H-benzimidazol-5-yl)phenyl]oxy}ethyl)-4,4-dimethylcyclohexanamine trifluoroacetate
—— 4-bromo-N-cyclobutyl-3-fluorobenzenesulfonamide 1055995-86-2 C10H11BrFNO2S
4-bromo-N-cyclobutyl-3-fluorobenzenesulfonamide
—— N,N-diethyl-2-{4-[(3-methyl-2-furoyl)amino]benzyl}-N'-(2-naphthylsulfonyl)malonamide 1094195-25-1 C30H31N3O6S
N,N-diethyl-2-{4-[(3-methyl-2-furoyl)amino]benzyl}-N'-(2-naphthylsulfonyl)malonamide
—— 1-methyl-6-[5-(4-trifluoromethylbenzoylamino)pyrimidin-2-yloxy]-1H-indole-2-carboxylic acid ethyl ester 1150743-93-3 C24H19F3N4O4
1-methyl-6-[5-(4-trifluoromethylbenzoylamino)pyrimidin-2-yloxy]-1H-indole-2-carboxylic acid ethyl ester
—— 4-({(S)-3-hydroxy-2-[4-(2-phenoxy-phenylsulfamoyl)-benzoylamino]-propionylamino}-methyl)-piperidine-1-carboxylic acid tert-butyl ester 1021524-00-4 C33H40N4O8S
4-({(S)-3-hydroxy-2-[4-(2-phenoxy-phenylsulfamoyl)-benzoylamino]-propionylamino}-methyl)-piperidine-1-carboxylic acid tert-butyl ester
—— {4-[2-(2-chloro-4-fluoro-phenoxy)-phenylsulfamoyl]-benzoylamino}-acetic acid ethyl ester 1021524-13-9 C23H20ClFN2O6S
{4-[2-(2-chloro-4-fluoro-phenoxy)-phenylsulfamoyl]-benzoylamino}-acetic acid ethyl ester
—— 6-(4-fluoro-2-(trifluoromethyl)phenyl)-5-(6-hydrazinylpyridin-3-yl)imidazo[2,1-b]oxazole 1033041-10-9 C17H11F4N5O
6-(4-fluoro-2-(trifluoromethyl)phenyl)-5-(6-hydrazinylpyridin-3-yl)imidazo[2,1-b]oxazole
—— 4-(4-aminopiperidin-1-yl)-N-methyl-2-pyrimidin-5-yloxy-9H-pyrimido[4,5-b]indol-8-amine 1400803-10-2 C20H22N8O
4-(4-aminopiperidin-1-yl)-N-methyl-2-pyrimidin-5-yloxy-9H-pyrimido[4,5-b]indol-8-amine
—— {(3S,4S)-4-[4-((S)-3-methoxy-2-methyl-propoxymethyl)-phenyl]-3-[4-(3-methoxy-propyl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethoxy]-piperidin-4-yloxy}-acetonitrile 1146170-03-7 C32H45N3O6
{(3S,4S)-4-[4-((S)-3-methoxy-2-methyl-propoxymethyl)-phenyl]-3-[4-(3-methoxy-propyl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethoxy]-piperidin-4-yloxy}-acetonitrile
—— 4-{4-[3-(tert-butyl-dimethyl-silanyloxy)-propyl]-phenyl}-3-[cyclopropyl-(2,3-dimethyl-benzyl)-carbamoyl]-piperidine-1-carboxylic acid tert-butyl ester 1007393-56-7 C38H58N2O4Si
4-{4-[3-(tert-butyl-dimethyl-silanyloxy)-propyl]-phenyl}-3-[cyclopropyl-(2,3-dimethyl-benzyl)-carbamoyl]-piperidine-1-carboxylic acid tert-butyl ester
—— 2-(2,6-difluorophenyl)-5-(4-(2-(dimethylamino)ethylamino)phenyl)oxazole-4-carboxamide 1082441-31-3 C20H20F2N4O2
2-(2,6-difluorophenyl)-5-(4-(2-(dimethylamino)ethylamino)phenyl)oxazole-4-carboxamide
—— 3-nitro-2-(pentylthio)quinoline 1242431-18-0 C14H16N2O2S
3-nitro-2-(pentylthio)quinoline
—— 6-(3-{[4-(4,4-dimethylcyclohexyl)-3-methyl-5-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethylpyridazin-3(2H)-one trifluoroacetate 1154871-72-3 C2HF3O2*C27H35FN4O3
6-(3-{[4-(4,4-dimethylcyclohexyl)-3-methyl-5-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethylpyridazin-3(2H)-one trifluoroacetate
—— N-{4-(6-fluoro-3'-methyl-2-biphenylyl)-4-hydroxy-4-[(3R)-1-({4-[(methylamino)methyl]phenyl}carbonyl)-3-piperidinyl]butyl}acetamide 1070870-14-2 C33H40FN3O3
N-{4-(6-fluoro-3'-methyl-2-biphenylyl)-4-hydroxy-4-[(3R)-1-({4-[(methylamino)methyl]phenyl}carbonyl)-3-piperidinyl]butyl}acetamide
—— 2-(4-methoxyphenyl)-5-methyl-1-((1-tosyl-indol-3-yl)methyl)benzimidazole 1234802-39-1 C31H27N3O3S
2-(4-methoxyphenyl)-5-methyl-1-((1-tosyl-indol-3-yl)methyl)benzimidazole
—— 8-({[t-butyl(dimethyl)silyl]oxy}methyl)-3-[2-chloro-4-(pyrrolidin-1-yl)phenyl]-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1035929-50-0 C24H37ClN4OSSi
8-({[t-butyl(dimethyl)silyl]oxy}methyl)-3-[2-chloro-4-(pyrrolidin-1-yl)phenyl]-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— 1-cyclopropyl-2-[5-(3,5-difluorophenyl)pyridin-3-yl]-5,6-difluoro-1H-benzimidazole 1356481-64-5 C21H13F4N3
1-cyclopropyl-2-[5-(3,5-difluorophenyl)pyridin-3-yl]-5,6-difluoro-1H-benzimidazole
—— 1-{[2-(aminomethyl)-6-(4-chlorophenyl)-5-(2,4-dichlorophenyl)pyrid-3-yl]-methyl}-3-(2-fluorobenzyl)urea 1173144-23-4 C27H22Cl3FN4O
1-{[2-(aminomethyl)-6-(4-chlorophenyl)-5-(2,4-dichlorophenyl)pyrid-3-yl]-methyl}-3-(2-fluorobenzyl)urea
—— 1-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-ethanone 1150646-90-4 C10H15N3O
1-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-ethanone
—— 2-[5-fluoro-6-(4-fluoro-benzylamino)-2-oxo-1,2-dihydro-indol-3-ylidenemethyl]-3-methyl-5-(2-morpholin-4-yl-ethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one 1082988-58-6 C31H33F2N5O3
2-[5-fluoro-6-(4-fluoro-benzylamino)-2-oxo-1,2-dihydro-indol-3-ylidenemethyl]-3-methyl-5-(2-morpholin-4-yl-ethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one
—— 8-(((2-ethoxyethyl)(methyl)amino)methyl)-5,6-dihydro-4H-pyrrolo[1,2-a][1,4]benzodiazepin-4-one 1036726-30-3 C18H23N3O2
8-(((2-ethoxyethyl)(methyl)amino)methyl)-5,6-dihydro-4H-pyrrolo[1,2-a][1,4]benzodiazepin-4-one
—— 3-(2-ethoxyphenyl)-8,8-dimethyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1035927-48-0 C16H21N3OS
3-(2-ethoxyphenyl)-8,8-dimethyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— 1-{2-ethyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}ethanol 1150220-54-4 C15H15F3O2
1-{2-ethyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}ethanol
—— 2-{4-[(2-amino-3-methylbenzoyl)amino]benzyl}-N, N-diethyl-N'-(2-naphthylsulfonyl)malonamide 1094195-00-2 C32H34N4O5S
2-{4-[(2-amino-3-methylbenzoyl)amino]benzyl}-N, N-diethyl-N'-(2-naphthylsulfonyl)malonamide