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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-fluorobenzyl 4-[3-oxo-3-(2-oxo-2,3-dihydrobenzoxazol-6-yl)propyl]piperazine-1-carboxylate 1144036-51-0 C22H22FN3O5
2-fluorobenzyl 4-[3-oxo-3-(2-oxo-2,3-dihydrobenzoxazol-6-yl)propyl]piperazine-1-carboxylate
—— 8-{2-[(3R,4S)-4-amino-3-hydroxy-1-piperidinyl]ethyl}-7-chloro-1-methyl-1,5-naphthyridin-2(1H)-one 1002108-51-1 C16H21ClN4O2
8-{2-[(3R,4S)-4-amino-3-hydroxy-1-piperidinyl]ethyl}-7-chloro-1-methyl-1,5-naphthyridin-2(1H)-one
—— 4-(4-fluorophenyl)-3-methyl-5-oxo-piperazine-1-carboxylic acid tert-butyl ester 1154870-52-6 C16H21FN2O3
4-(4-fluorophenyl)-3-methyl-5-oxo-piperazine-1-carboxylic acid tert-butyl ester
—— 6-{3-[(4-cyclohexyl-3-ethyl-5-oxopiperazin-1-yl)carbonyl]-4-fluorobenzyl}-4,5-dimethylpyridazin-3(2H)-one 1154872-41-9 C26H33FN4O3
6-{3-[(4-cyclohexyl-3-ethyl-5-oxopiperazin-1-yl)carbonyl]-4-fluorobenzyl}-4,5-dimethylpyridazin-3(2H)-one
—— [4-(1-methylpiperidin-4-ylidene)-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]carboxylic acid-N-(2-methoxyethyl)amide hydrochloride 1176737-06-6 C23H28N2O2S*ClH
[4-(1-methylpiperidin-4-ylidene)-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]carboxylic acid-N-(2-methoxyethyl)amide hydrochloride
—— (2S,4S)-methyl 2-methyl-4-(3-oxo-2,3-dihydroisoxazol-5-yl)piperidine-1-carboxylate 1251845-81-4 C11H16N2O4
(2S,4S)-methyl 2-methyl-4-(3-oxo-2,3-dihydroisoxazol-5-yl)piperidine-1-carboxylate
—— 4-(1-methyl-5-{5-[methyl(toluene-4-sulfonyl)amino]pyridin-2-yloxy}-1H-indole-2-carbonyl)piperazine-1-carboxylic acid tert-butyl ester 1150745-95-1 C32H37N5O6S
4-(1-methyl-5-{5-[methyl(toluene-4-sulfonyl)amino]pyridin-2-yloxy}-1H-indole-2-carbonyl)piperazine-1-carboxylic acid tert-butyl ester
—— 2-{4-[(2-amino-4, 5-difluorobenzoyl)amino]benzyl}-N, N-diethyl-N'-(2-naphthylsulfonyl)malonamide 1094195-08-0 C31H30F2N4O5S
2-{4-[(2-amino-4, 5-difluorobenzoyl)amino]benzyl}-N, N-diethyl-N'-(2-naphthylsulfonyl)malonamide
—— N-methyl-N-[1-[1-[5-methyl-6-[[(2S,6R)-6-(4-methylphenyl)oxan-2-yl]methylamino]pyrimidine-4-carbonyl]piperidin-4-yl]piperidin-4-yl]methanesulfonamide 1312779-02-4 C31H46N6O4S
N-methyl-N-[1-[1-[5-methyl-6-[[(2S,6R)-6-(4-methylphenyl)oxan-2-yl]methylamino]pyrimidine-4-carbonyl]piperidin-4-yl]piperidin-4-yl]methanesulfonamide
—— 4-fluoro-N-{[6-methyl-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}benzamide 1141878-18-3 C18H14F4N2O3
4-fluoro-N-{[6-methyl-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}benzamide
—— 2-[[(2S)-4-(4-fluorophenyl)-2-methylpiperazin-1-yl]methyl]-7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-5-amine 1616597-34-2 C22H24FN7O
2-[[(2S)-4-(4-fluorophenyl)-2-methylpiperazin-1-yl]methyl]-7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-5-amine
—— 4-(1-cyclopropyl-4,6-difluoro-1H-benzimidazol-2-yl)isoquinoline 1356482-35-3 C19H13F2N3
4-(1-cyclopropyl-4,6-difluoro-1H-benzimidazol-2-yl)isoquinoline
—— N-(2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)acrylamide 1957235-52-7 C16H15N3O4
N-(2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)acrylamide
—— N-[[4-[3-(3,5-dichlorophenyl)-2-hydroxy-3-(trifluoromethyl)pyrrolidin-1-yl]-2-(trifluoromethyl)phenyl]methyl]cyclopropanecarboxamide 1365067-94-2 C23H20Cl2F6N2O2
N-[[4-[3-(3,5-dichlorophenyl)-2-hydroxy-3-(trifluoromethyl)pyrrolidin-1-yl]-2-(trifluoromethyl)phenyl]methyl]cyclopropanecarboxamide
—— (5-methyl-2-{(S)-4-[2-oxopiperazin-4-ylethyl]-4,5-dihydrothiazol-2-yl}-1H-indol-7-yl)-(tetrahydropyran-4-ylmethyl)amine 1120344-68-4 C24H33N5O2S
(5-methyl-2-{(S)-4-[2-oxopiperazin-4-ylethyl]-4,5-dihydrothiazol-2-yl}-1H-indol-7-yl)-(tetrahydropyran-4-ylmethyl)amine
—— 6-cyano-4-(1-methylpiperidin-4-ylidene)-4,10-dihydro-9-oxa-3-thiabenzo[f]azulene 1176736-90-5 C19H18N2OS
6-cyano-4-(1-methylpiperidin-4-ylidene)-4,10-dihydro-9-oxa-3-thiabenzo[f]azulene
—— 3-benzyl-6-(2-nitrobenzyl)-1,3,4-trimethylpiperazine-2,5-dione 1092584-28-5 C21H23N3O4
3-benzyl-6-(2-nitrobenzyl)-1,3,4-trimethylpiperazine-2,5-dione
—— [4-(1-ethoxycarbonylpiperidin-4-ylidene)-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]carboxylic acid 1176737-69-1 C22H23NO4S
[4-(1-ethoxycarbonylpiperidin-4-ylidene)-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]carboxylic acid
—— [3-(3-dimethylaminophenylamino)phenyl]-bis-[2-(tert-butyldimethylsilanyloxy)ethyl]amine 1138888-92-2 C30H53N3O2Si2
[3-(3-dimethylaminophenylamino)phenyl]-bis-[2-(tert-butyldimethylsilanyloxy)ethyl]amine
—— 3-[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]-N-pyridin-4-ylpropanamide 1141877-29-3 C17H13ClF3N3O3
3-[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]-N-pyridin-4-ylpropanamide
—— [2-(4-methyl-piperazine-1-yl)-ethyl]-{4-[3-(3-pyrazol-1-yl-phenyl)-imidazo[1,2-a]pyridin-7-yl]-benzyl}-amine 1146613-44-6 C30H33N7
[2-(4-methyl-piperazine-1-yl)-ethyl]-{4-[3-(3-pyrazol-1-yl-phenyl)-imidazo[1,2-a]pyridin-7-yl]-benzyl}-amine
—— 2-ethylamino-N-methyl-6-[4-((E)-3-pyridin-3-yl-acryloylamino)-phenyl]-nicotinamide 1138321-98-8 C23H23N5O2
2-ethylamino-N-methyl-6-[4-((E)-3-pyridin-3-yl-acryloylamino)-phenyl]-nicotinamide
—— {4-[3-(2-furan-3-yl-pyridin-4-yl)-imidazo[1,2-a]pyridin-6-yl]-pyrazol-1-yl}-acetic acid 1146614-78-9 C21H15N5O3
{4-[3-(2-furan-3-yl-pyridin-4-yl)-imidazo[1,2-a]pyridin-6-yl]-pyrazol-1-yl}-acetic acid
—— (S)-3-hydroxy-2-[4-(2-phenoxy-phenylsulfamoyl)-benzoylamino]-propionic acid 1021523-99-8 C22H20N2O7S
(S)-3-hydroxy-2-[4-(2-phenoxy-phenylsulfamoyl)-benzoylamino]-propionic acid
—— 4-fluoro-N-{[2-oxo-6-(1H-pyrazol-4-yl)-4-(trifluoromethyl)-1,2,3,4-tetrahydroquinazolin-4-yl]methyl}benzamide 1141879-10-8 C20H15F4N5O2
4-fluoro-N-{[2-oxo-6-(1H-pyrazol-4-yl)-4-(trifluoromethyl)-1,2,3,4-tetrahydroquinazolin-4-yl]methyl}benzamide
—— N-{[4-(4-methyl-1H-benzimidazol-5-yl)phenyl]methyl}-2,3-dihydro-1H-inden-2-amine trifluoroacetate 1008358-48-2 C2HF3O2*C24H23N3
N-{[4-(4-methyl-1H-benzimidazol-5-yl)phenyl]methyl}-2,3-dihydro-1H-inden-2-amine trifluoroacetate
—— 2-(4-fluoro-phenylamino)-N-(2-piperidin-1-yl-ethyl)-6-[4-(3-pyridin-3-ylmethyl-ureido)-phenyl]-nicotinamide 1138321-69-3 C32H34FN7O2
2-(4-fluoro-phenylamino)-N-(2-piperidin-1-yl-ethyl)-6-[4-(3-pyridin-3-ylmethyl-ureido)-phenyl]-nicotinamide
—— N-[(1S,2R)-1-benzyl-2-hydroxy-3-{[3-(trifluoromethyl)benzyl]amino}propyl]-1-oxo-2-(1-propylbutyl)-2,3,4,5-tetrahydro-1H-pyrrolo[1,2-a][1,4]diazepine-7-carboxamide hydrochloride 1108235-09-1 C34H43F3N4O3*ClH
N-[(1S,2R)-1-benzyl-2-hydroxy-3-{[3-(trifluoromethyl)benzyl]amino}propyl]-1-oxo-2-(1-propylbutyl)-2,3,4,5-tetrahydro-1H-pyrrolo[1,2-a][1,4]diazepine-7-carboxamide hydrochloride
—— tert-butyl 4-(4-chlorophenyl)-5-methyl-5,6-dihydropyridine-1(2H)-carboxylate 1293995-05-7 C17H22ClNO2
tert-butyl 4-(4-chlorophenyl)-5-methyl-5,6-dihydropyridine-1(2H)-carboxylate
—— 2-{3-[5-chloro-7-(tetrahydropyran-4-ylmethyl)amino-1H-indole-2-yl]-phenyl}-acetic acid 1120333-69-8 C22H23ClN2O3
2-{3-[5-chloro-7-(tetrahydropyran-4-ylmethyl)amino-1H-indole-2-yl]-phenyl}-acetic acid
—— (S)-1-(5-nitropyridin-2-ylamino)-1-oxo-3-phenylpropan-2-ylcarbamic acid tert-butyl ester 1094107-67-1 C19H22N4O5
(S)-1-(5-nitropyridin-2-ylamino)-1-oxo-3-phenylpropan-2-ylcarbamic acid tert-butyl ester
—— N-({4-chloro-3-[(3-chloro-5-cyanophenyl)oxy]-2-fluorophenyl}methyl)-5-{[(2R)-2-morpholinylmethyl]oxy}-1H-indole-2-carboxamide hydrochloride 1093254-41-1 C28H23Cl2FN4O4*ClH
N-({4-chloro-3-[(3-chloro-5-cyanophenyl)oxy]-2-fluorophenyl}methyl)-5-{[(2R)-2-morpholinylmethyl]oxy}-1H-indole-2-carboxamide hydrochloride
—— 5-hydroxy-2-methyl-4-[5-methyl-3-[4-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl]-3(2H)-pyridazinone 1164163-95-4 C16H13F3N4O2
5-hydroxy-2-methyl-4-[5-methyl-3-[4-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl]-3(2H)-pyridazinone
—— rac-2-methoxy-6-methylsulfanyl-N-[1-methyl-3-(3-thiazol-2-yl-phenyl)-piperidin-3-yl]-4-trifluoromethyl-benzamide formic acid 1236304-21-4 CH2O2*C25H26F3N3O2S2
rac-2-methoxy-6-methylsulfanyl-N-[1-methyl-3-(3-thiazol-2-yl-phenyl)-piperidin-3-yl]-4-trifluoromethyl-benzamide formic acid
—— N-{[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-2-ethylbutanamide 1141877-03-3 C16H18ClF3N2O3
N-{[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-2-ethylbutanamide
—— (S)-3-{4-[5-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-methoxy-6-methyl-phenoxy}-propane-1,2-diol 1150646-10-8 C21H27N5O5
(S)-3-{4-[5-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-methoxy-6-methyl-phenoxy}-propane-1,2-diol
—— N-{[2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}benzamide 1141876-51-8 C17H13F3N2O3
N-{[2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}benzamide
—— 2-methoxy-N-[(R)-1-(4-methoxy-phenyl)-ethyl]-4-pyridin-4-yl-benzamide 1127308-99-9 C22H22N2O3
2-methoxy-N-[(R)-1-(4-methoxy-phenyl)-ethyl]-4-pyridin-4-yl-benzamide
—— tert-butyl 4-[3-(4-{4-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperazin-1-yl}phenoxy)propyl]piperazine-1-carboxylate 1240300-15-5 C28H39F3N8O3
tert-butyl 4-[3-(4-{4-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperazin-1-yl}phenoxy)propyl]piperazine-1-carboxylate
—— (1-hydroxy-2-oxo-1,2-dihydro-pyridin-3-yl)carbamic acid benzyl ester 1009121-42-9 C13H12N2O4
(1-hydroxy-2-oxo-1,2-dihydro-pyridin-3-yl)carbamic acid benzyl ester
—— cyclohexyl{2-methyl-5-[4-(trifluoromethoxy)phenyl]-3-furyl}methanol 1150221-97-8 C19H21F3O3
cyclohexyl{2-methyl-5-[4-(trifluoromethoxy)phenyl]-3-furyl}methanol
—— 2-(N<sup>6</sup>-benzoyladenin-9-yl)ethanal 123156-36-5 C14H11N5O2
2-(N<sup>6</sup>-benzoyladenin-9-yl)ethanal
—— bis[methyl N-(dithiocarboxy-κS,κS')-N-methylglycinato]-copper(II) 1040751-28-7 C10H16CuN2O4S4
bis[methyl N-(dithiocarboxy-κS,κS')-N-methylglycinato]-copper(II)
—— (1R,4R)-7,7-dimethyl-1-((R)-4-phenyl-4,5-dihydrooxazol-2-yl)bicyclo[2.2.1]heptan-2-one 1000304-16-4 C18H21NO2
(1R,4R)-7,7-dimethyl-1-((R)-4-phenyl-4,5-dihydrooxazol-2-yl)bicyclo[2.2.1]heptan-2-one
—— N-[(2-bromo-4,6-dimethylphenyl)diazenyl]-4-methoxy-N-methylaniline 1295605-58-1 C16H18BrN3O
N-[(2-bromo-4,6-dimethylphenyl)diazenyl]-4-methoxy-N-methylaniline
—— 2-Cyano-2-(1-pyrrolidino)carbonyl-5-isopropylthio-1,3-dithiane 126832-96-0 C14H22N2OS3
2-Cyano-2-(1-pyrrolidino)carbonyl-5-isopropylthio-1,3-dithiane
—— 7,8-dihydro-9-chloro-12-methylbenzo[a]pyridine[3,2,1-de]phenanthridin-5-one 1330074-76-4 C21H16ClNO
7,8-dihydro-9-chloro-12-methylbenzo[a]pyridine[3,2,1-de]phenanthridin-5-one
—— 5-(2,4-difluorophenoxy)-1,3-dimethyl-1H-pyrazole-4-carbaldehyde O-(4-((2-chlorothiazol-5-yl)methoxy)benzyl) oxime 1620883-71-7 C23H19ClF2N4O3S
5-(2,4-difluorophenoxy)-1,3-dimethyl-1H-pyrazole-4-carbaldehyde O-(4-((2-chlorothiazol-5-yl)methoxy)benzyl) oxime
—— 4-ethynyl-2,6-di(thiophen-2-yl)pyridine 1629603-35-5 C15H9NS2
4-ethynyl-2,6-di(thiophen-2-yl)pyridine
—— 4,6-dimethoxy-4,9,9-trimethylbenzo[f][2]benzofuran-1,3-dione 107828-81-9 C17H18O5
4,6-dimethoxy-4,9,9-trimethylbenzo[f][2]benzofuran-1,3-dione