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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-chloro-6-cyclobutyl-8-(trifluoromethyl)imidazo[1,2-a]pyridine-2-carboxylic acid 1237839-23-4 C13H10ClF3N2O2
3-chloro-6-cyclobutyl-8-(trifluoromethyl)imidazo[1,2-a]pyridine-2-carboxylic acid
—— 2-ethylamino-N-methyl-6-{-4-[3-(2-pyridin-3-yl-ethyl)-ureido]-phenyl}-nicotinamide 1138321-54-6 C23H26N6O2
2-ethylamino-N-methyl-6-{-4-[3-(2-pyridin-3-yl-ethyl)-ureido]-phenyl}-nicotinamide
—— (4-benzylpiperazin-1-yl)[5-(5-ethylaminopyridin-2-yloxy)-1-methyl-1H-indol-2-yl]methanone 1150460-19-7 C28H31N5O2
(4-benzylpiperazin-1-yl)[5-(5-ethylaminopyridin-2-yloxy)-1-methyl-1H-indol-2-yl]methanone
—— 2-[N-(8-dimethylamino-10H-phenothiazin-2-yl)-N-(2-hydroxyethyl)amino]ethanol 1132109-98-8 C18H23N3O2S
2-[N-(8-dimethylamino-10H-phenothiazin-2-yl)-N-(2-hydroxyethyl)amino]ethanol
—— [4-(1-methylpiperidin-4-ylidene)-4,10-dihydro-9-oxa-3-thiabenzo[f]azulen-2-yl]carboxylic acid-N-(2-hydroxyethyl)amide 1176737-32-8 C21H24N2O3S
[4-(1-methylpiperidin-4-ylidene)-4,10-dihydro-9-oxa-3-thiabenzo[f]azulen-2-yl]carboxylic acid-N-(2-hydroxyethyl)amide
—— 6-{3-[(4-cyclohexyl-3-oxopiperazin-1-yl)carbonyl]-4-fluorobenzyl}-4-ethylpyridazin-3(2H)-one trifluoroacetate 1154868-80-0 C2HF3O2*C24H29FN4O3
6-{3-[(4-cyclohexyl-3-oxopiperazin-1-yl)carbonyl]-4-fluorobenzyl}-4-ethylpyridazin-3(2H)-one trifluoroacetate
—— 5-(4-(methylsulfonyl)phenyl)-3-(6-(trifluoromethyl)-1H-benzo[d]imidazol-2-yl)pyrazin-2-ylamine 1232410-85-3 C19H14F3N5O2S
5-(4-(methylsulfonyl)phenyl)-3-(6-(trifluoromethyl)-1H-benzo[d]imidazol-2-yl)pyrazin-2-ylamine
—— 1-methyl-6-(5-nitropyridin-2-yloxy)-1H-indole-2-carboxylic acid ethyl ester 1150743-00-2 C17H15N3O5
1-methyl-6-(5-nitropyridin-2-yloxy)-1H-indole-2-carboxylic acid ethyl ester
—— N-{6-[2-(4-benzo[1,3]dioxol-5-ylmethylpiperazine-1-carbonyl)-1H-indol-5-yloxy]pyridin-3-yl}-3,4-dichlorobenzamide 1150342-82-7 C33H27Cl2N5O5
N-{6-[2-(4-benzo[1,3]dioxol-5-ylmethylpiperazine-1-carbonyl)-1H-indol-5-yloxy]pyridin-3-yl}-3,4-dichlorobenzamide
—— {4-[2-(4-bromo-phenoxy)-5-fluoro-phenylsulfamoyl]-benzoylamino}-acetic acid 1021522-31-5 C21H16BrFN2O6S
{4-[2-(4-bromo-phenoxy)-5-fluoro-phenylsulfamoyl]-benzoylamino}-acetic acid
—— (4-dimethylamino-phenyl)-(3-(1H-pyrrolo[2,3-b]pyridin-3-yl)-pyrrolidin-1-yl)-methanone 1151768-68-1 C20H22N4O
(4-dimethylamino-phenyl)-(3-(1H-pyrrolo[2,3-b]pyridin-3-yl)-pyrrolidin-1-yl)-methanone
—— [2-methoxy-5-methyl-6-[[(2R,6S)-6-[4-(trifluoromethoxy)phenyl]oxan-2-yl]methylamino]pyrimidin-4-yl]-[4-[[(3S,4S)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]methanone 1312779-80-8 C31H42F3N5O6
[2-methoxy-5-methyl-6-[[(2R,6S)-6-[4-(trifluoromethoxy)phenyl]oxan-2-yl]methylamino]pyrimidin-4-yl]-[4-[[(3S,4S)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]methanone
—— 2-(2,4-dimethoxybenzyl)-1,2,3,4-tetrahydroisoquinolin-6-ol 1064206-19-4 C18H21NO3
2-(2,4-dimethoxybenzyl)-1,2,3,4-tetrahydroisoquinolin-6-ol
—— 4-{[(4-fluorobenzoyl)amino]methyl}-2-oxo-N-((3R)-tetrahydrofuran-3-yl)-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazine-6-carboxamide 1141878-67-2 C22H19F4N3O5
4-{[(4-fluorobenzoyl)amino]methyl}-2-oxo-N-((3R)-tetrahydrofuran-3-yl)-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazine-6-carboxamide
—— N-(5-chloro-pyridin-2-yl)-N-piperidin-4-ylmethyl-propionamide trifluoroacetate 1112990-92-7 C2HF3O2*C14H20ClN3O
N-(5-chloro-pyridin-2-yl)-N-piperidin-4-ylmethyl-propionamide trifluoroacetate
—— 1-((S)-1-(2,3-dihydrobenzo[1,4]dioxin-2-yl)methyl)-3-(3-fluorophenyl)piperidine 1107177-66-1 C20H22FNO2
1-((S)-1-(2,3-dihydrobenzo[1,4]dioxin-2-yl)methyl)-3-(3-fluorophenyl)piperidine
—— 5-methyl-6-[[(2S,6R)-6-(3-methylphenyl)oxan-2-yl]methylamino]pyrimidine-4-carboxylic acid 1312780-72-5 C19H23N3O3
5-methyl-6-[[(2S,6R)-6-(3-methylphenyl)oxan-2-yl]methylamino]pyrimidine-4-carboxylic acid
—— 4-(2-benzoyl-phenylsulfamoyl)-N-cyclohexylcarbamoylmethyl-benzamide 1021523-53-4 C28H29N3O5S
4-(2-benzoyl-phenylsulfamoyl)-N-cyclohexylcarbamoylmethyl-benzamide
—— 2-(3-fluoropropoxy)-5-bromopyridine 1248622-88-9 C8H9BrFNO
2-(3-fluoropropoxy)-5-bromopyridine
—— phenyl N-(5-indanyl)-3-(3-trifluoromethylphenylthio)acrylimidate 1107009-92-6 C25H20F3NOS
phenyl N-(5-indanyl)-3-(3-trifluoromethylphenylthio)acrylimidate
—— N-{[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-5-ethylisoxazole-3-carboxamide 1141877-11-3 C16H13ClF3N3O4
N-{[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-5-ethylisoxazole-3-carboxamide
—— 1-Ethyl-3-[1-methyl-2-oxo-5-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-1,2-dihydro-pyridin-3-yl]-urea 1178884-82-6 C15H24BN3O4
1-Ethyl-3-[1-methyl-2-oxo-5-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-1,2-dihydro-pyridin-3-yl]-urea
—— ethyl 5-methyl-7-(2-(pyridin-4-yl)phenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate 1099637-33-8 C19H18N6O2
ethyl 5-methyl-7-(2-(pyridin-4-yl)phenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— N-{[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-6-fluoronicotinamide 1141876-75-6 C16H10ClF4N3O3
N-{[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-6-fluoronicotinamide
—— 4-(6-fluoropyridine-3-yl)-4-methoxy-1-phenylcyclohexanecarbonitrile 1092532-08-5 C19H19FN2O
4-(6-fluoropyridine-3-yl)-4-methoxy-1-phenylcyclohexanecarbonitrile
—— (S)-1-[3-(3-chloro-phenylamino)-5-(2-ethylamino-pyridin-4-yl)-[1,2,4]triazol-1-yl]-butan-2-ol 1145355-41-4 C19H23ClN6O
(S)-1-[3-(3-chloro-phenylamino)-5-(2-ethylamino-pyridin-4-yl)-[1,2,4]triazol-1-yl]-butan-2-ol
—— 1-(3-bromo-4-chloro-benzenesulfonyl)-1,2,3,4-tetrahydro-benzo[b]azepin-5-one 1070972-87-0 C16H13BrClNO3S
1-(3-bromo-4-chloro-benzenesulfonyl)-1,2,3,4-tetrahydro-benzo[b]azepin-5-one
—— 6-{-4-[3-(6-amino-pyridin-3-ylmethyl)-ureido]-phenyl}-2-ethylamino-N-(2-methoxy-ethyl)-nicotinamide 1161014-41-0 C24H29N7O3
6-{-4-[3-(6-amino-pyridin-3-ylmethyl)-ureido]-phenyl}-2-ethylamino-N-(2-methoxy-ethyl)-nicotinamide
—— (E)-3-(2-Hydroxy-phenyl)-acrylic acid 2-ethyl-4-(2,2,3-trimethyl-cyclopent-3-enyl)-but-2-enyl ester 1097692-84-6 C23H30O3
(E)-3-(2-Hydroxy-phenyl)-acrylic acid 2-ethyl-4-(2,2,3-trimethyl-cyclopent-3-enyl)-but-2-enyl ester
—— 3-(1-chloro-3-methylbutyl)-2-methyl-5-[4-(trifluoromethyl)phenyl]furan 1150221-42-3 C17H18ClF3O
3-(1-chloro-3-methylbutyl)-2-methyl-5-[4-(trifluoromethyl)phenyl]furan
—— 3-fluoro-N-((R)-1-naphthalen-1-yl-ethyl)-4-pyridin-4-yl-benzamide 1127309-88-9 C24H19FN2O
3-fluoro-N-((R)-1-naphthalen-1-yl-ethyl)-4-pyridin-4-yl-benzamide
—— 3-[cyclopropyl-(2,3-dimethyl-benzyl)-carbamoyl]-4-[4-(3-hydroxy-propyl)-phenyl]-piperidine-1-carboxylic acid tert-butyl ester 1007393-58-9 C32H44N2O4
3-[cyclopropyl-(2,3-dimethyl-benzyl)-carbamoyl]-4-[4-(3-hydroxy-propyl)-phenyl]-piperidine-1-carboxylic acid tert-butyl ester
—— 1-methyl-4-(5-nitropyridin-2-yloxy)-1H-indole-2-carboxylic acid ethyl ester 1150743-04-6 C17H15N3O5
1-methyl-4-(5-nitropyridin-2-yloxy)-1H-indole-2-carboxylic acid ethyl ester
—— 4-{[(5-tert-butyl-2-methyl-3-furyl)(cyclohexyl)methyl]amino}benzoic acid 1150222-59-5 C23H31NO3
4-{[(5-tert-butyl-2-methyl-3-furyl)(cyclohexyl)methyl]amino}benzoic acid
—— ethyl 3-[3-(4-bromo-2-tert-butylphenoxy)azetidin-1-yl]-3-oxopropanoate 1146956-99-1 C18H24BrNO4
ethyl 3-[3-(4-bromo-2-tert-butylphenoxy)azetidin-1-yl]-3-oxopropanoate
—— 4-{[cyclohexyl(2-methyl-5-phenyl-3-furyl)methyl]amino}benzoic acid 1150221-62-7 C25H27NO3
4-{[cyclohexyl(2-methyl-5-phenyl-3-furyl)methyl]amino}benzoic acid
—— 6-ethoxy-N-(1-methyl-piperidin-4-yl)-N'-(3-trifluoromethyl-phenyl)-[1,3,5]triazine-2,4-diamine hydrochloride 1174126-54-5 C18H23F3N6O*ClH
6-ethoxy-N-(1-methyl-piperidin-4-yl)-N'-(3-trifluoromethyl-phenyl)-[1,3,5]triazine-2,4-diamine hydrochloride
—— rac-2-hydroxy-N-(2-hydroxy-2-{4-[5-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-phenyl}-ethyl)-acetamide 1150646-85-7 C20H24N6O4
rac-2-hydroxy-N-(2-hydroxy-2-{4-[5-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-phenyl}-ethyl)-acetamide
—— N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzylsulfonamide 1150342-44-1 C35H34F3N5O5S
N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzylsulfonamide
—— 6-(3-{[4-(4-chlorophenyl)-3-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethyl-3-oxo-2,3-dihydropyridazin-1-ium trifluoroacetate 1154868-94-6 C2HF3O2*C24H22ClFN4O3
6-(3-{[4-(4-chlorophenyl)-3-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethyl-3-oxo-2,3-dihydropyridazin-1-ium trifluoroacetate
—— (3R)-1-(cyclopropylmethyl)-6-fluoro-3-{4-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one 1093978-97-2 C27H27FN6O2
(3R)-1-(cyclopropylmethyl)-6-fluoro-3-{4-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one
—— N-[1-(3,4-diethoxy-phenyl)-ethyl]-2-methoxy-4-pyridin-4-yl-benzamide 1127309-04-9 C25H28N2O4
N-[1-(3,4-diethoxy-phenyl)-ethyl]-2-methoxy-4-pyridin-4-yl-benzamide
—— 4-(2-benzoyl-phenylsulfamoyl)-N-[(2-piperidin-4-yl-ethylcarbamoyl)-methyl]-benzamide hydrochloride 1021524-06-0 C29H32N4O5S*ClH
4-(2-benzoyl-phenylsulfamoyl)-N-[(2-piperidin-4-yl-ethylcarbamoyl)-methyl]-benzamide hydrochloride
—— 8-(((cyclohexylmethyl)amino)methyl)-5,6-dihydro-4H-pyrrolo[1,2-a][1,4]benzodiazepin4-one 1036726-31-4 C20H25N3O
8-(((cyclohexylmethyl)amino)methyl)-5,6-dihydro-4H-pyrrolo[1,2-a][1,4]benzodiazepin4-one
—— N-(2-aminophenyl)-4-((3-(4-carbmethoxyphenyl)-2-(3-chlorophenyl)acrylamido)methyl)benzamide 1141445-43-3 C31H26ClN3O4
N-(2-aminophenyl)-4-((3-(4-carbmethoxyphenyl)-2-(3-chlorophenyl)acrylamido)methyl)benzamide
—— [2-(4-chloro-3-hydroxymethyl-phenyl)-ethyl]-methyl-carbamic acid tert-butyl ester 1007392-94-0 C15H22ClNO3
[2-(4-chloro-3-hydroxymethyl-phenyl)-ethyl]-methyl-carbamic acid tert-butyl ester
—— 6-[4-fluoro-3-({3-oxo-4-[(3S)-tetrahydro-2H-pyran-3-yl]piperazin-1-yl}carbonyl)benzyl]-4,5-dimethylpyridazin-3(2H)-one 1154871-31-4 C23H27FN4O4
6-[4-fluoro-3-({3-oxo-4-[(3S)-tetrahydro-2H-pyran-3-yl]piperazin-1-yl}carbonyl)benzyl]-4,5-dimethylpyridazin-3(2H)-one
—— 6-(3-fluoropropoxy)benzothiophene-2-boronic acid 1248622-80-1 C11H12BFO3S
6-(3-fluoropropoxy)benzothiophene-2-boronic acid
—— N-[2-amino-1-(4-methoxyphenyl)ethyl]-4-pyridin-4-ylbenzamide 1127308-09-1 C21H21N3O2
N-[2-amino-1-(4-methoxyphenyl)ethyl]-4-pyridin-4-ylbenzamide
—— [1-methyl-5-(5-nitropyridin-2-yloxy)-1H-indol-2-yl]{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazin-1-yl}methanone 1150460-70-0 C28H26F3N5O5
[1-methyl-5-(5-nitropyridin-2-yloxy)-1H-indol-2-yl]{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazin-1-yl}methanone