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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(3-bromo-8-ethyl-quinolin-6-yloxy)-N-(1,1-dimethyl-but-2-ynyl)-2-methylsulfanyl-acetamide 1126434-43-2 C20H23BrN2O2S
2-(3-bromo-8-ethyl-quinolin-6-yloxy)-N-(1,1-dimethyl-but-2-ynyl)-2-methylsulfanyl-acetamide
—— 4-[1-(2,6-dichlorophenyl)ethoxy]-2-nitroaniline 1146852-81-4 C14H12Cl2N2O3
4-[1-(2,6-dichlorophenyl)ethoxy]-2-nitroaniline
—— 3-{4-[1-(2-methanesulfonylaminoethyl)piperidin-4-ylidene]-4,10-dihydro-9-oxa-3-thiabenzo[f]azulen-6-yl}propionic acid 1176739-25-5 C23H28N2O5S2
3-{4-[1-(2-methanesulfonylaminoethyl)piperidin-4-ylidene]-4,10-dihydro-9-oxa-3-thiabenzo[f]azulen-6-yl}propionic acid
—— 6-(3-{[(3R)-4-(5-chloro-2-fluorophenyl)-3-methyl-5-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethylpyridazin-3(2H)-one 1154872-61-3 C25H23ClF2N4O3
6-(3-{[(3R)-4-(5-chloro-2-fluorophenyl)-3-methyl-5-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethylpyridazin-3(2H)-one
—— 7-{[(2-piperidin-1-ylethyl)amino]methyl}pyrrolo(1,2-a]quinoxalin-4(5H)-one 1036726-76-7 C19H24N4O
7-{[(2-piperidin-1-ylethyl)amino]methyl}pyrrolo(1,2-a]quinoxalin-4(5H)-one
—— 4-{1-methyl-5-[5-(toluene-4-sulfonylamino)pyridin-2-yloxy]-1H-indole-2-carbonyl}piperazine-1-carboxylic acid tert-butyl ester 1150744-34-5 C31H35N5O6S
4-{1-methyl-5-[5-(toluene-4-sulfonylamino)pyridin-2-yloxy]-1H-indole-2-carbonyl}piperazine-1-carboxylic acid tert-butyl ester
—— 4-[2-(4-fluoro-phenoxy)-phenylsulfamoyl]-benzoic acid 1021522-57-5 C19H14FNO5S
4-[2-(4-fluoro-phenoxy)-phenylsulfamoyl]-benzoic acid
—— 4-amino-6-(3-(benzyloxymethyl)-3H-benzo[d]imidazol-5-yl)-2-methoxy-7,8-dihydropyrido[4,3-d]pyrimidin-5(6H)-one 1236410-67-5 C23H22N6O3
4-amino-6-(3-(benzyloxymethyl)-3H-benzo[d]imidazol-5-yl)-2-methoxy-7,8-dihydropyrido[4,3-d]pyrimidin-5(6H)-one
—— N-(5-indanyl)-3-(phenylthio)acrylamide 1107010-27-4 C18H17NOS
N-(5-indanyl)-3-(phenylthio)acrylamide
—— N,N-diethyl-2-{4-[(4-fluorobenzoyl)amino]benzyl}-N'-(2-naphthylsulfonyl)malonamide 1094194-74-7 C31H30FN3O5S
N,N-diethyl-2-{4-[(4-fluorobenzoyl)amino]benzyl}-N'-(2-naphthylsulfonyl)malonamide
—— 3-[2-(trifluoromethyl)phenyl]pyrazine-2,6-diamine 1076245-86-7 C11H9F3N4
3-[2-(trifluoromethyl)phenyl]pyrazine-2,6-diamine
—— 3-(1H-benzo[d]imidazol-2-yl)-5-(2-(piperazin-1-yl)pyridin-4-yl)pyrazin-2-ylamine 1232411-03-8 C20H20N8
3-(1H-benzo[d]imidazol-2-yl)-5-(2-(piperazin-1-yl)pyridin-4-yl)pyrazin-2-ylamine
—— N,N-diethyl-2-{4-[(3-fluorobenzoyl)amino]benzyl}-N'-(2-naphthylsulfonyl)malonamide 1094194-75-8 C31H30FN3O5S
N,N-diethyl-2-{4-[(3-fluorobenzoyl)amino]benzyl}-N'-(2-naphthylsulfonyl)malonamide
—— methyl 3-{(3R)-3-[(6-butyl-8-quinolinyl)oxy]-1-pyrrolidinyl}propanoate 1145873-34-2 C21H28N2O3
methyl 3-{(3R)-3-[(6-butyl-8-quinolinyl)oxy]-1-pyrrolidinyl}propanoate
—— 3-isopropyl-5-(5-methylpyridin-2-yl)benzoic acid 1150263-26-5 C16H17NO2
3-isopropyl-5-(5-methylpyridin-2-yl)benzoic acid
—— [4-[[(3R,4R)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]-[2-methoxy-6-[[(2R,6S)-6-[4-(trifluoromethoxy)phenyl]oxan-2-yl]methylamino]pyrimidin-4-yl]methanone 1312779-66-0 C30H40F3N5O6
[4-[[(3R,4R)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]-[2-methoxy-6-[[(2R,6S)-6-[4-(trifluoromethoxy)phenyl]oxan-2-yl]methylamino]pyrimidin-4-yl]methanone
—— 2-[2-chloro-4-(difluoromethoxy)phenyl]-3,7-dimethyl-5-(1-propylbutyl)pyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079355-36-4 C22H26ClF2N3O2
2-[2-chloro-4-(difluoromethoxy)phenyl]-3,7-dimethyl-5-(1-propylbutyl)pyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— 3-{1-[4-(3-hydroxypropoxy)phenyl]-3-(2-phenylethyl)-1H-indol-5-yl}propanoic acid 2-amino-2-(hydroxymethyl)propane-1,3-diol salt 1069050-66-3 C4H11NO3*C28H29NO4
3-{1-[4-(3-hydroxypropoxy)phenyl]-3-(2-phenylethyl)-1H-indol-5-yl}propanoic acid 2-amino-2-(hydroxymethyl)propane-1,3-diol salt
—— 3-ethyl-5-isopropyl-7-methyl-2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]pyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079356-31-2 C22H25N5O
3-ethyl-5-isopropyl-7-methyl-2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]pyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— 1-cyclohexyl-4-methoxy-2-isopropyl-benzene 1058159-81-1 C16H24O
1-cyclohexyl-4-methoxy-2-isopropyl-benzene
—— 2-(2-chloro-4-phenoxyphenyl)-5-(1-ethylpropyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079352-01-4 C25H26ClN3O2
2-(2-chloro-4-phenoxyphenyl)-5-(1-ethylpropyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— N-[(1S)-1-benzyl-2-hydroxyethyl]-2-fluoro-4-pyridin-4-ylbenzamide 1127307-69-0 C21H19FN2O2
N-[(1S)-1-benzyl-2-hydroxyethyl]-2-fluoro-4-pyridin-4-ylbenzamide
—— (4-chloro-3-cyclopropylaminomethyl-benzyl)-methyl-carbamic acid tert-butyl ester 1007393-01-2 C17H25ClN2O2
(4-chloro-3-cyclopropylaminomethyl-benzyl)-methyl-carbamic acid tert-butyl ester
—— 3-(3-(4-(6-aminopyrimidin-4-yl)phenyl)ureido)-N-isopropylbenzamide 1219727-32-8 C21H22N6O2
3-(3-(4-(6-aminopyrimidin-4-yl)phenyl)ureido)-N-isopropylbenzamide
—— 2-(4-cyanophenyl)-5-(4-methoxyphenyl)oxazole-4-carboxamide 1082441-91-5 C18H13N3O3
2-(4-cyanophenyl)-5-(4-methoxyphenyl)oxazole-4-carboxamide
—— N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-pyridin-4-ylbenzamide 1127307-99-6 C23H20N4O
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-pyridin-4-ylbenzamide
—— N-{4-[5-(3,5-dichlorophenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-yl]-2-nitrobenzyl}acetamide 1067924-95-1 C19H14Cl2F3N3O4
N-{4-[5-(3,5-dichlorophenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-yl]-2-nitrobenzyl}acetamide
—— N-(3-(2-cyano-1-hydroxyethyl)phenyl)butane-1-sulfonamide 1222165-56-1 C13H18N2O3S
N-(3-(2-cyano-1-hydroxyethyl)phenyl)butane-1-sulfonamide
—— 4-[[3,4-bis(difluoromethoxy)phenyl](pyrimidin-5-ylmethyl)amino]benzoic acid tert-butyl ester 1203596-86-4 C24H23F4N3O4
4-[[3,4-bis(difluoromethoxy)phenyl](pyrimidin-5-ylmethyl)amino]benzoic acid tert-butyl ester
—— N-diphenylmethyl-N'-(2-naphthylsulfonyl)-2-(4-nitrobenzyl)malonamide 1094197-15-5 C33H27N3O6S
N-diphenylmethyl-N'-(2-naphthylsulfonyl)-2-(4-nitrobenzyl)malonamide
—— 2-acetamido-N-[4-[4-(methylsulfonylmethyl)-6-morpholin-4-yl-pyrimidin-2-yl]phenyl]propanamide 1099774-03-4 C21H27N5O5S
2-acetamido-N-[4-[4-(methylsulfonylmethyl)-6-morpholin-4-yl-pyrimidin-2-yl]phenyl]propanamide
—— N-[(1S)-2-hydroxy-1-(4-hydroxybenzyl)ethyl]-4-pyridin-4-ylbenzamide 1127307-76-9 C21H20N2O3
N-[(1S)-2-hydroxy-1-(4-hydroxybenzyl)ethyl]-4-pyridin-4-ylbenzamide
—— 6-(4-fluoro-3-{[4-(4-methoxybenzyl)-3-methyl-5-oxopiperazin-1-yl]carbonyl}benzyl)-4,5-dimethyl-3-oxo-2,3-dihydropyridazin-1-ium trifluoroacetate 1154871-92-7 C2HF3O2*C27H29FN4O4
6-(4-fluoro-3-{[4-(4-methoxybenzyl)-3-methyl-5-oxopiperazin-1-yl]carbonyl}benzyl)-4,5-dimethyl-3-oxo-2,3-dihydropyridazin-1-ium trifluoroacetate
—— rac-2-(2-Hydroxy-ethylamino)-1-{4-[5-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-phenyl}-ethanol 1150646-80-2 C20H26N6O3
rac-2-(2-Hydroxy-ethylamino)-1-{4-[5-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-phenyl}-ethanol
—— 2-(5-fluoro-2-oxo-1,2-dihydro-indol-3-ylidenemethyl)-3-methyl-5-(2-pyrrolidin-1-yl-ethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one 1082989-15-8 C24H27FN4O2
2-(5-fluoro-2-oxo-1,2-dihydro-indol-3-ylidenemethyl)-3-methyl-5-(2-pyrrolidin-1-yl-ethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one
—— 4-[2-(4-bromophenoxy)-5-fluorophenylsulfamoyl]-N-[2-(4-pyrimidin-2-ylpiperazin-1-yl)ethyl]benzamide 1021362-41-3 C29H28BrFN6O4S
4-[2-(4-bromophenoxy)-5-fluorophenylsulfamoyl]-N-[2-(4-pyrimidin-2-ylpiperazin-1-yl)ethyl]benzamide
—— 3-[(3R)-3-hydroxypyrrolidin-1-yl]benzoic acid 1000016-89-6 C11H13NO3
3-[(3R)-3-hydroxypyrrolidin-1-yl]benzoic acid
—— 4-(6,7-dihydro-2-phenyl-4H-pyrazolo[5,1-c][1,4]oxaazin-3-yl)-N-(1-methylethyl)-2-aminopyrimidine 1161076-18-1 C19H21N5O
4-(6,7-dihydro-2-phenyl-4H-pyrazolo[5,1-c][1,4]oxaazin-3-yl)-N-(1-methylethyl)-2-aminopyrimidine
—— 1-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-3-(3-methylbenzyl)urea 1219727-34-0 C21H19N5O
1-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-3-(3-methylbenzyl)urea
—— 1-(4-(5-cyclopropyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2-fluorophenyl)-1-(2-hydroxyethyl)-3-(pyridin-3-yl)urea 1219728-08-1 C23H21FN6O2
1-(4-(5-cyclopropyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2-fluorophenyl)-1-(2-hydroxyethyl)-3-(pyridin-3-yl)urea
—— 4-(cyclohexyl{2-methyl-5-[4-(trifluoromethoxy)phenyl]-3-furyl}methoxy)benzoic acid 1150221-99-0 C26H25F3O5
4-(cyclohexyl{2-methyl-5-[4-(trifluoromethoxy)phenyl]-3-furyl}methoxy)benzoic acid
—— 2-[4-(cyclopropylcarbonylamino)benzyl]-N, N-diethyl-N'-(2-naphthylsulfonyl)malonamide 1094194-68-9 C28H31N3O5S
2-[4-(cyclopropylcarbonylamino)benzyl]-N, N-diethyl-N'-(2-naphthylsulfonyl)malonamide
—— 3-chloro-4-fluoro-N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide 1150463-95-8 C34H30ClF4N5O5S
3-chloro-4-fluoro-N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide
—— N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-4-pyridin-4-ylbenzamide 1127308-32-0 C21H23N5O
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-4-pyridin-4-ylbenzamide
—— 5-sec-butyl-2-(2-chloro-4-methoxy-5-methylphenyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079355-03-5 C20H24ClN3O2
5-sec-butyl-2-(2-chloro-4-methoxy-5-methylphenyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— 2-(1-adamantyl)-5-methyl-1-(3,4,5-trimethoxybenzyl)benzimidazole 1234802-15-3 C28H34N2O3
2-(1-adamantyl)-5-methyl-1-(3,4,5-trimethoxybenzyl)benzimidazole
—— 3-methyl-2-[[(2R,6S)-6-phenyloxan-2-yl]methylamino]pyridine-4-carboxylic acid 1312780-92-9 C19H22N2O3
3-methyl-2-[[(2R,6S)-6-phenyloxan-2-yl]methylamino]pyridine-4-carboxylic acid
—— 1-[(S)-2-amino-4-oxo-4-(2-thiophen-3-yl-4-trifluoromethyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-butyl]-5-fluoro-6-hydroxy-piperidin-2-one hydrochloride 1173175-36-4 C21H23F4N5O3S*ClH
1-[(S)-2-amino-4-oxo-4-(2-thiophen-3-yl-4-trifluoromethyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-butyl]-5-fluoro-6-hydroxy-piperidin-2-one hydrochloride
—— N-(2-morpholino-2-oxoethyl)-4-oxo4,5-dihydropyrrolo[1,2-a]quinoxaline-7-carboxamide 1036726-68-7 C18H18N4O4
N-(2-morpholino-2-oxoethyl)-4-oxo4,5-dihydropyrrolo[1,2-a]quinoxaline-7-carboxamide
—— 5-methyl-2-(thiophen-2-yl)-1-((1-tosyl-indol-3-yl)methyl)benzimidazole 1234802-53-9 C28H23N3O2S2
5-methyl-2-(thiophen-2-yl)-1-((1-tosyl-indol-3-yl)methyl)benzimidazole