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中文名称 英文名称 CAS号 化学式 结构式图片
—— (1S,4S,5R,8R,10S,13R,14R,16R,17S,18R,19S,20R)-16-fluoro-10-hydroxy-4,5,9,9,13,19,20-heptamethyl-24-oxahexacyclo[15.5.2.01,18.04,17.05,14.08,13]tetracosan-23-one 1402830-16-3 C30H47FO3
(1S,4S,5R,8R,10S,13R,14R,16R,17S,18R,19S,20R)-16-fluoro-10-hydroxy-4,5,9,9,13,19,20-heptamethyl-24-oxahexacyclo[15.5.2.01,18.04,17.05,14.08,13]tetracosan-23-one
—— (4R,6S)-4-cyclopropyl-7,7-difluoro-6-(4-fluorophenyl)-2-(4-methylphenyl)sulfonyl-5-[6-(trifluoromethyl)pyridin-3-yl]sulfonyl-4,6-dihydropyrazolo[4,3-c]pyridine 1415916-35-6 C28H22F6N4O4S2
(4R,6S)-4-cyclopropyl-7,7-difluoro-6-(4-fluorophenyl)-2-(4-methylphenyl)sulfonyl-5-[6-(trifluoromethyl)pyridin-3-yl]sulfonyl-4,6-dihydropyrazolo[4,3-c]pyridine
—— 2-[2-(5-methoxy-1H-indol-3-yl)ethylamino]-6-(2-methyl-1H-indol-5-ylamino)pyrimidine-4-carboxamide 1400890-39-2 C25H25N7O2
2-[2-(5-methoxy-1H-indol-3-yl)ethylamino]-6-(2-methyl-1H-indol-5-ylamino)pyrimidine-4-carboxamide
—— 3-(4-amino-[1]benzothiolo[3,2-d]pyrimidin-7-yl)-N-(3-amino-3-oxopropyl)benzamide 1401531-05-2 C20H17N5O2S
3-(4-amino-[1]benzothiolo[3,2-d]pyrimidin-7-yl)-N-(3-amino-3-oxopropyl)benzamide
—— 2-(2,4-dimethylthiophen-3-yl)-3-(2-fluoro-4-hydroxyphenyl)-N'-hydroxy-5,6-dihydrocyclopenta[b]pyrrole-1(4H)-carboximidamide 1402652-22-5 C20H20FN3O2S
2-(2,4-dimethylthiophen-3-yl)-3-(2-fluoro-4-hydroxyphenyl)-N'-hydroxy-5,6-dihydrocyclopenta[b]pyrrole-1(4H)-carboximidamide
—— 4-[4-[5-amino-6-(3-phenylisoxazol-5-yl)pyrazin-2-yl]pyridin-2-yl]piperidine-4-carbonitrile 1402389-01-8 C24H21N7O
4-[4-[5-amino-6-(3-phenylisoxazol-5-yl)pyrazin-2-yl]pyridin-2-yl]piperidine-4-carbonitrile
—— 3-(4-methoxyphenyl)-1-phenyl-2-thia-3-azabicyclo[3.1.0]hexane 2,2-dioxide 1417156-32-1 C17H17NO3S
3-(4-methoxyphenyl)-1-phenyl-2-thia-3-azabicyclo[3.1.0]hexane 2,2-dioxide
—— (6Z,9Z,12Z)-tetradecatrien-14-olide 1394847-28-9 C14H20O2
(6Z,9Z,12Z)-tetradecatrien-14-olide
—— (R)-7-[3-((R)-3-amino-6,6-difluoro-5,7,7-trimethyl-2,5,6,7-tetrahydro-[1,4]oxazepin-5-yl)-4-fluoro-phenylamino]-6,7-dihydro-5H-[1]pyrindine-3-carbonitrile 1400682-73-6 C23H24F3N5O
(R)-7-[3-((R)-3-amino-6,6-difluoro-5,7,7-trimethyl-2,5,6,7-tetrahydro-[1,4]oxazepin-5-yl)-4-fluoro-phenylamino]-6,7-dihydro-5H-[1]pyrindine-3-carbonitrile
—— 1-[(1S,3R)-3-(2-fluorophenyl)cyclopentyl]-3-[(2S)-2-hydroxy-2,3-dihydro-1H-inden-4-yl]urea 1401076-45-6 C21H23FN2O2
1-[(1S,3R)-3-(2-fluorophenyl)cyclopentyl]-3-[(2S)-2-hydroxy-2,3-dihydro-1H-inden-4-yl]urea
—— (2-Methoxy-5-(trifluoromethyl)pyridin-3-yl)methanamine hydrochloride 1095321-10-0 C8H9F3N2O*ClH
(2-Methoxy-5-(trifluoromethyl)pyridin-3-yl)methanamine hydrochloride
—— 1,4,7-Tri-tert-butyl-10-oxabicyclo[5.2.1]decan-4-ol 1415841-55-2 C21H40O2
1,4,7-Tri-tert-butyl-10-oxabicyclo[5.2.1]decan-4-ol
—— [3-[4-[(4-oxo-3H-quinazolin-2-yl)methyl]piperazin-1-yl]phenyl] 2-methylpropanoate 1403240-36-7 C23H26N4O3
[3-[4-[(4-oxo-3H-quinazolin-2-yl)methyl]piperazin-1-yl]phenyl] 2-methylpropanoate
—— N-[(2S)-2-[2-iodo-3-[(2S)-1-[[4-(trifluoromethyl)benzoyl]amino]propan-2-yl]oxyphenoxy]propyl]-4-(trifluoromethyl)benzamide 1399008-19-5 C28H25F6IN2O4
N-[(2S)-2-[2-iodo-3-[(2S)-1-[[4-(trifluoromethyl)benzoyl]amino]propan-2-yl]oxyphenoxy]propyl]-4-(trifluoromethyl)benzamide
—— (4aS,4bR,5S,6aS,6bR,9aS,10aS,10bS,12S)-4b,12-difluoro-5-hydroxy-6b-(2-hydroxy-acetyl)-4a,6a-dimethyl-8-[4-(4-hydroxy-phenylsulfanylmethyl)-benzyl]-4a,4b,5,6,6a,6b,8,9,9a,10,10a,10b,11,12-tetradecahydro-7-oxa-8-aza-pentaleno[2,1-a]phenanthren-2-one 1399259-54-1 C36H39F2NO6S
(4aS,4bR,5S,6aS,6bR,9aS,10aS,10bS,12S)-4b,12-difluoro-5-hydroxy-6b-(2-hydroxy-acetyl)-4a,6a-dimethyl-8-[4-(4-hydroxy-phenylsulfanylmethyl)-benzyl]-4a,4b,5,6,6a,6b,8,9,9a,10,10a,10b,11,12-tetradecahydro-7-oxa-8-aza-pentaleno[2,1-a]phenanthren-2-one
—— 4-[3-(3-fluoro-4-morpholin-4-ylphenyl)isoxazol-5-yl]-N-hydroxy-2-methyl-2-(methylsulfonyl)butanamide 1402353-67-6 C19H24FN3O6S
4-[3-(3-fluoro-4-morpholin-4-ylphenyl)isoxazol-5-yl]-N-hydroxy-2-methyl-2-(methylsulfonyl)butanamide
—— 1-(3',4'-dimethoxybiphenyl-3-yl)-6-(2H-tetrazol-5-yl)-1H-benzimidazole 1401321-19-4 C22H18N6O2
1-(3',4'-dimethoxybiphenyl-3-yl)-6-(2H-tetrazol-5-yl)-1H-benzimidazole
—— (2S)-2-({[7-(1-methyl-1H-pyrazol-4-yl)pyrido[3,4-b]pyrazin-5-yl]oxy}methyl)-1-(2,2,2-trifluoroethyl)piperazine 1400587-41-8 C18H20F3N7O
(2S)-2-({[7-(1-methyl-1H-pyrazol-4-yl)pyrido[3,4-b]pyrazin-5-yl]oxy}methyl)-1-(2,2,2-trifluoroethyl)piperazine
—— 3-Benzyl-3-(iodomethyl)-1-(4-methylphenyl)sulfonylpyrrolidine 1395474-22-2 C19H22INO2S
3-Benzyl-3-(iodomethyl)-1-(4-methylphenyl)sulfonylpyrrolidine
—— N-cyclopropyl-2-methyl-4-{6-[3-(trifluoromethoxy)phenoxy]-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyridin-3-yl}benzamide 1402594-08-4 C28H24F6N4O3
N-cyclopropyl-2-methyl-4-{6-[3-(trifluoromethoxy)phenoxy]-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyridin-3-yl}benzamide
—— 8-(2-fluoroethyl)-3-methyl-4-{[7-(trifluoromethyl)-3,4-dihydroisoquinolin-2(1H)-yl]carbonyl}-1-oxa-8-azaspiro[4.5]dec-3-en-2-one 1401993-30-3 C22H24F4N2O3
8-(2-fluoroethyl)-3-methyl-4-{[7-(trifluoromethyl)-3,4-dihydroisoquinolin-2(1H)-yl]carbonyl}-1-oxa-8-azaspiro[4.5]dec-3-en-2-one
—— N-(2,4-dichlorophenyI)-2-[6,7-methylenedioxy-3-(2-naphthoyl)-4-oxo-1-quinolinyl]acetamide 1401169-61-6 C29H18Cl2N2O5
N-(2,4-dichlorophenyI)-2-[6,7-methylenedioxy-3-(2-naphthoyl)-4-oxo-1-quinolinyl]acetamide
—— 4'-((1H-indole-2-sulfonamido)methyl)biphenyl-4-carboxamide 1394431-41-4 C22H19N3O3S
4'-((1H-indole-2-sulfonamido)methyl)biphenyl-4-carboxamide
—— N-[3-(4-amino-[1]benzothiolo[3,2-d]pyrimidin-7-yl)phenyl]-4-methylpiperazine-1-carboxamide 1378233-79-4 C22H22N6OS
N-[3-(4-amino-[1]benzothiolo[3,2-d]pyrimidin-7-yl)phenyl]-4-methylpiperazine-1-carboxamide
—— (4aS,4bR,5S,6aS,6bR,9aS,10aS,10bS,12S)-4b,12-difluoro-5-hydroxy-4a,6a-dimethyl-2-oxo-8-(2-(phenylsulfanyl)ethyl)-2,4a,4b,5,6,6a,8,9,9a,10,10a,10b,11,12-tetradecahydro-7-oxa-8-azapentaleno[2,1-a]phenanthrene-6b-carbothioic acid S-fluoromethyl ester 1400571-68-7 C30H34F3NO4S2
(4aS,4bR,5S,6aS,6bR,9aS,10aS,10bS,12S)-4b,12-difluoro-5-hydroxy-4a,6a-dimethyl-2-oxo-8-(2-(phenylsulfanyl)ethyl)-2,4a,4b,5,6,6a,8,9,9a,10,10a,10b,11,12-tetradecahydro-7-oxa-8-azapentaleno[2,1-a]phenanthrene-6b-carbothioic acid S-fluoromethyl ester
—— N,2-dimethyl-4-{6-phenoxy-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyridin-3-yl}benzamide 1402593-94-5 C25H23F3N4O2
N,2-dimethyl-4-{6-phenoxy-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyridin-3-yl}benzamide
—— 4-[2-(difluoromethoxy)-4-fluorophenyl]-N-{3-[(methylsulfonyl)methyl]phenyl}-1,3,5-triazin-2-amine 1403987-76-7 C18H15F3N4O3S
4-[2-(difluoromethoxy)-4-fluorophenyl]-N-{3-[(methylsulfonyl)methyl]phenyl}-1,3,5-triazin-2-amine
—— 1-[4-(3-carbamoylphenoxy)phenyl]-1H-benzimidazole-6-carboxylic acid 1401320-97-5 C21H15N3O4
1-[4-(3-carbamoylphenoxy)phenyl]-1H-benzimidazole-6-carboxylic acid
—— N-cyclopropyl-4-{6-(2-hydroxyphenoxy)-4-[(3,3,3-trifluoropropyl)amino]-1H-benzimidazol-1-yl}-2-methylbenzamide 1401450-37-0 C27H25F3N4O3
N-cyclopropyl-4-{6-(2-hydroxyphenoxy)-4-[(3,3,3-trifluoropropyl)amino]-1H-benzimidazol-1-yl}-2-methylbenzamide
—— (R)-2-(4-chloro-3,5-diphenyl-1H-pyrazolo[3,4-c]pyridazin-hydroxypropyl)acetamide 1404506-09-7 C22H20ClN5O2
(R)-2-(4-chloro-3,5-diphenyl-1H-pyrazolo[3,4-c]pyridazin-hydroxypropyl)acetamide
—— N-(4-fluorophenyl)-N-(((2R)-4-(2-thiophenylsulfonyl)-1-(4-(2,2,2-trifluoro-1-hydroxy-1-methylethyl)phenyl)-2 piperazinyl)methyl)methanesulfonamide 1361224-97-6 C25H27F4N3O5S3
N-(4-fluorophenyl)-N-(((2R)-4-(2-thiophenylsulfonyl)-1-(4-(2,2,2-trifluoro-1-hydroxy-1-methylethyl)phenyl)-2 piperazinyl)methyl)methanesulfonamide
—— 2-[2-fluoro-4-[2-[(1S,2R)-2-[1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]cyclopropyl]ethoxy]phenyl]-N-methyl-N-(oxan-4-yl)acetamide 1402553-40-5 C29H41FN4O4
2-[2-fluoro-4-[2-[(1S,2R)-2-[1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]cyclopropyl]ethoxy]phenyl]-N-methyl-N-(oxan-4-yl)acetamide
—— 2-(3-(allylthio)-5-ethyl-4H-1,2,4-triazol-4-yl)isoindoline-1,3-dione 1394017-09-4 C15H14N4O2S
2-(3-(allylthio)-5-ethyl-4H-1,2,4-triazol-4-yl)isoindoline-1,3-dione
—— 2-[3,5-dimethyl-1-[[4-[6-(trifluoromethyl)-1H-indol-2-yl]phenyl]methyl]pyrazol-4-yl]acetic acid 1401963-35-6 C23H20F3N3O2
2-[3,5-dimethyl-1-[[4-[6-(trifluoromethyl)-1H-indol-2-yl]phenyl]methyl]pyrazol-4-yl]acetic acid
—— 3-(4-hydroxyphenyl)-4-(4-hydroxyphenyl)-8-methylchroman-7-ol 1374524-55-6 C22H20O4
3-(4-hydroxyphenyl)-4-(4-hydroxyphenyl)-8-methylchroman-7-ol
—— 2-acetylamino-N-[3-(3-ethyl-ureido)-isoquinolin-8-ylmethyl]-acetamide 1401308-20-0 C17H21N5O3
2-acetylamino-N-[3-(3-ethyl-ureido)-isoquinolin-8-ylmethyl]-acetamide
—— 2-(3-methyl-5-(2-oxo-2-phenylethylthio)-4H-1,2,4-triazol-4-yl)isoindoline-1,3-dione 1394017-00-5 C19H14N4O3S
2-(3-methyl-5-(2-oxo-2-phenylethylthio)-4H-1,2,4-triazol-4-yl)isoindoline-1,3-dione
—— 1-(4'-{3-methyl-4-[(2-phenylthiazol-5-ylmethyl)amino]isoxazol-5-yl}biphenyl-4-yl)cyclopropanecarboxylic acid ethyl ester 1280734-12-4 C32H29N3O3S
1-(4'-{3-methyl-4-[(2-phenylthiazol-5-ylmethyl)amino]isoxazol-5-yl}biphenyl-4-yl)cyclopropanecarboxylic acid ethyl ester
—— 2-(3-chloro-7-((5-fluoropyrimidin-2-yl)(propyl)amino)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid 1403367-42-9 C21H22ClFN4O2
2-(3-chloro-7-((5-fluoropyrimidin-2-yl)(propyl)amino)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
—— (7aS,9R,11aS)-11a-benzyl-9-ethoxymethyl-9-hydroxy-6,7,7a,8,9,10,11,11a-octahydro-5H-dibenzo[a,c]cycloheptene-3-carboxylic acid (2-methyl-pyridin-3-yl)-amide 1400925-51-0 C32H38N2O3
(7aS,9R,11aS)-11a-benzyl-9-ethoxymethyl-9-hydroxy-6,7,7a,8,9,10,11,11a-octahydro-5H-dibenzo[a,c]cycloheptene-3-carboxylic acid (2-methyl-pyridin-3-yl)-amide
—— 1-(4'-{3-methyl-4-[6-(4-methylphenyl)pyridin-2-ylamino]isoxazol-5-yl}biphenyl-4-yl)cyclopropanecarboxylic acid 1402207-77-5 C32H27N3O3
1-(4'-{3-methyl-4-[6-(4-methylphenyl)pyridin-2-ylamino]isoxazol-5-yl}biphenyl-4-yl)cyclopropanecarboxylic acid
—— 2-ethylphenyl 3-(3-(2-chloroacetyl)ureido)benzenesulfonate 1403940-05-5 C17H17ClN2O5S
2-ethylphenyl 3-(3-(2-chloroacetyl)ureido)benzenesulfonate
—— N-(2,6-diethylphenyl)-5-{2-[(2-methoxyphenyl)amino]pyrimidin-4-yl}-1-methyl-1H-pyrazole-3-carboxamide 1403332-18-2 C26H28N6O2
N-(2,6-diethylphenyl)-5-{2-[(2-methoxyphenyl)amino]pyrimidin-4-yl}-1-methyl-1H-pyrazole-3-carboxamide
—— 3-(1-(5-bromo-4-(4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl)oxazol-2-yl)-2-hydroxyethoxy)-2,6-difluorobenzamide 1403881-39-9 C21H15BrF2N4O5
3-(1-(5-bromo-4-(4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl)oxazol-2-yl)-2-hydroxyethoxy)-2,6-difluorobenzamide
—— tert-butyl N-[(2S)-1-[[(3R,4S,5S)-1-[[(2R,3R,4S,5R)-5-(benzylcarbamoyl)-3,4-dimethoxyoxolan-2-yl]methylamino]-3-hydroxy-5-methyl-1-oxoheptan-4-yl]-methylamino]-3-methyl-1-oxobutan-2-yl]carbamate 1400435-92-8 C34H56N4O9
tert-butyl N-[(2S)-1-[[(3R,4S,5S)-1-[[(2R,3R,4S,5R)-5-(benzylcarbamoyl)-3,4-dimethoxyoxolan-2-yl]methylamino]-3-hydroxy-5-methyl-1-oxoheptan-4-yl]-methylamino]-3-methyl-1-oxobutan-2-yl]carbamate
—— 1-[(1S,3R)-3-(2-fluorophenyl)cyclopentyl]-3-(1H-indazol-4-yl)urea 1401075-75-9 C19H19FN4O
1-[(1S,3R)-3-(2-fluorophenyl)cyclopentyl]-3-(1H-indazol-4-yl)urea
—— 4-{6-(5-fluoro-2-methylphenoxy)-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyridin-3-yl}-N,2-dimethylbenzamide 1402593-58-1 C26H24F4N4O2
4-{6-(5-fluoro-2-methylphenoxy)-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyridin-3-yl}-N,2-dimethylbenzamide
—— (3S)-3-[({7-[4-(propan-2-yloxy)phenyl]pyrido[3,4-b]pyrazin-5-yl}oxy)methyl]piperidine 1400586-95-9 C22H26N4O2
(3S)-3-[({7-[4-(propan-2-yloxy)phenyl]pyrido[3,4-b]pyrazin-5-yl}oxy)methyl]piperidine
—— 5-(3-fluoro-phenylethynyl)-3-methyl-pyridine-2-carboxylic acid tert-butyl-methyl-amide 1403770-60-4 C20H21FN2O
5-(3-fluoro-phenylethynyl)-3-methyl-pyridine-2-carboxylic acid tert-butyl-methyl-amide
—— ethyl 3-((1R,2R)-2-heptylcyclopropyl)propanoate 1394818-60-0 C15H28O2
ethyl 3-((1R,2R)-2-heptylcyclopropyl)propanoate