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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[4-[4-[[methyl[(1R)-1,2,3,4-tetrahydro-1-naphthalenyl]amino]methyl]-2-thiazolyl]-1-piperidinyl]-2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethanone 1041436-99-0 C27H32F3N5OS
1-[4-[4-[[methyl[(1R)-1,2,3,4-tetrahydro-1-naphthalenyl]amino]methyl]-2-thiazolyl]-1-piperidinyl]-2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethanone
—— 1-[3-methyl-5-(morpholin-4-yl)-2-thienyl]ethanone 1203509-26-5 C11H15NO2S
1-[3-methyl-5-(morpholin-4-yl)-2-thienyl]ethanone
—— (S)-3-t-butoxycarbonylamino-4-(3-methyl-2,6-dioxo-piperidin-1-yl)-butyric acid benzyl ester 1173175-74-0 C22H30N2O6
(S)-3-t-butoxycarbonylamino-4-(3-methyl-2,6-dioxo-piperidin-1-yl)-butyric acid benzyl ester
—— tert-butyl 3-(3-(tert-butoxycarbonyl(cyclohexylmethyl)amino)phenyl)-3-oxopropylcarbamate 1222167-96-5 C26H40N2O5
tert-butyl 3-(3-(tert-butoxycarbonyl(cyclohexylmethyl)amino)phenyl)-3-oxopropylcarbamate
—— N-{4-(3'-ethyl-6-fluoro-2-biphenylyl)-4-hydroxy-4-[(3R)-1-({4-[(methylamino)methyl]phenyl}carbonyl)-3-piperidinyl]butyl}acetamide 1070870-16-4 C34H42FN3O3
N-{4-(3'-ethyl-6-fluoro-2-biphenylyl)-4-hydroxy-4-[(3R)-1-({4-[(methylamino)methyl]phenyl}carbonyl)-3-piperidinyl]butyl}acetamide
—— N-benzyl-N-(2-methoxy-1-oxy-pyridin-3-yl)-4-phenoxy-benzenesulfonamide 1009121-39-4 C25H22N2O5S
N-benzyl-N-(2-methoxy-1-oxy-pyridin-3-yl)-4-phenoxy-benzenesulfonamide
—— cyclohexyl{2-methyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}methanol 1150221-23-0 C19H21F3O2
cyclohexyl{2-methyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}methanol
—— 3-(4-(2-aminopyrimidin-4-yl)phenyl)-1-cyclopropyl-1-(3-fluorobenzyl)urea 1219727-24-8 C21H20FN5O
3-(4-(2-aminopyrimidin-4-yl)phenyl)-1-cyclopropyl-1-(3-fluorobenzyl)urea
—— tert-butyl 4-(6-butoxypyridin-2-yl)piperazine-1-carboxylate 1092848-30-0 C18H29N3O3
tert-butyl 4-(6-butoxypyridin-2-yl)piperazine-1-carboxylate
—— (9aR)-2-(2-fluoro-5-{[6-oxo-5-(trifluoromethyl)-1,6-dihydropyridazin-3-yl]methyl}benzoyl)octahydro-4H-pyrido[1,2-a]pyrazin-4-one 1154871-10-9 C21H20F4N4O3
(9aR)-2-(2-fluoro-5-{[6-oxo-5-(trifluoromethyl)-1,6-dihydropyridazin-3-yl]methyl}benzoyl)octahydro-4H-pyrido[1,2-a]pyrazin-4-one
—— 6-{-4-[3-(6-Amino-pyridin-3-ylmethyl)-ureido]-phenyl}-2-cyclopropylamino-N-(2-piperidin-1-yl-ethyl)-nicotinamide 1161014-19-2 C29H36N8O2
6-{-4-[3-(6-Amino-pyridin-3-ylmethyl)-ureido]-phenyl}-2-cyclopropylamino-N-(2-piperidin-1-yl-ethyl)-nicotinamide
—— N,N-diethyl-N'-2-{4-[(4,5-dimethyl-2-furoyl)amino]benzyl}-(2-naphthylsulfonyl)malonamide 1094195-28-4 C31H33N3O6S
N,N-diethyl-N'-2-{4-[(4,5-dimethyl-2-furoyl)amino]benzyl}-(2-naphthylsulfonyl)malonamide
—— 2-[4-(1-ethylpiperidin-4-ylidene)-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]-2-methylpropionic acid 1176738-52-5 C24H29NO2S
2-[4-(1-ethylpiperidin-4-ylidene)-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]-2-methylpropionic acid
—— 2-hydroxy-N-((S)-2-hydroxy-3-{4-[5-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-methoxy-6-methyl-phenoxy}-propyl)-acetamide 1150645-82-1 C23H30N6O6
2-hydroxy-N-((S)-2-hydroxy-3-{4-[5-(2-isopropylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-methoxy-6-methyl-phenoxy}-propyl)-acetamide
—— 3-[4-(1-methylpiperidin-4-ylidene)-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]acrylic acid hydrochloride 1176736-66-5 C22H23NO2S*ClH
3-[4-(1-methylpiperidin-4-ylidene)-9,10-dihydro-4H-1-thiabenzo[f]azulen-2-yl]acrylic acid hydrochloride
—— 3-(3-{[4-(2,4-dimethyl-1,3-thiazol-5-yl)-3-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethyl-6-oxo-1,6-dihydropyridazin-1-ium trifluoroacetate 1154871-50-7 C2HF3O2*C23H24FN5O3S
3-(3-{[4-(2,4-dimethyl-1,3-thiazol-5-yl)-3-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethyl-6-oxo-1,6-dihydropyridazin-1-ium trifluoroacetate
—— N-(2-hydroxyethyl)-N-methyl-4-(4-{1-[3-(trifluoromethyl)[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl}phenoxy)butanamide 1240300-13-3 C24H29F3N6O3
N-(2-hydroxyethyl)-N-methyl-4-(4-{1-[3-(trifluoromethyl)[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl}phenoxy)butanamide
—— tert-butyl 4-cyclohexyl-3-oxopiperazine-1-carboxylate 1154869-42-7 C15H26N2O3
tert-butyl 4-cyclohexyl-3-oxopiperazine-1-carboxylate
—— 5-(4-tert-butyl-2-methyl-phenoxymethyl)-4,5-dihydro-oxazol-2-ylamine 1058159-55-9 C15H22N2O2
5-(4-tert-butyl-2-methyl-phenoxymethyl)-4,5-dihydro-oxazol-2-ylamine
—— (4R)-1-{[3-(4-{[4-[5-fluoro-2-(methyloxy)phenyl]-2-hydroxy-4-methyl-2-(trifluoromethyl)pentyl]amino}-6-methyl-1H-indazol-1-yl)phenyl]carbonyl}-4-hydroxy-D-proline 1020169-27-0 C34H36F4N4O6
(4R)-1-{[3-(4-{[4-[5-fluoro-2-(methyloxy)phenyl]-2-hydroxy-4-methyl-2-(trifluoromethyl)pentyl]amino}-6-methyl-1H-indazol-1-yl)phenyl]carbonyl}-4-hydroxy-D-proline
—— N-[2-(4-pyrimidin-2-ylpiperazin-1-yl)ethyl]-4-[2-(4-trifluoromethylphenoxy)phenylsulfamoyl]benzamide 1021362-63-9 C30H29F3N6O4S
N-[2-(4-pyrimidin-2-ylpiperazin-1-yl)ethyl]-4-[2-(4-trifluoromethylphenoxy)phenylsulfamoyl]benzamide
—— N-{(2S)-2-[N-(3-Chloropropyl)-N-methylamino]-2-hydroxycarbonylethyl}-N-[4-(4-trifluoromethylphenoxy)phenyl]methanesulfonamide 1020105-08-1 C21H24ClF3N2O5S
N-{(2S)-2-[N-(3-Chloropropyl)-N-methylamino]-2-hydroxycarbonylethyl}-N-[4-(4-trifluoromethylphenoxy)phenyl]methanesulfonamide
—— 5-(4-methylbenzoyl)imidazo[2,1-b]thiazol-2-carboxylic acid 1092849-38-1 C14H10N2O3S
5-(4-methylbenzoyl)imidazo[2,1-b]thiazol-2-carboxylic acid
—— 2-chloro-2-methyl-N-phenyl-N-[1-(4-trifluoromethylbenzoyl)piperidin-4-yl]acetamide 1186213-41-1 C22H22ClF3N2O2
2-chloro-2-methyl-N-phenyl-N-[1-(4-trifluoromethylbenzoyl)piperidin-4-yl]acetamide
—— 5-sec-butyl-3,7-dimethyl-2-[2-methyl-4-(trifluoromethoxy)phenyl]pyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079355-14-8 C20H22F3N3O2
5-sec-butyl-3,7-dimethyl-2-[2-methyl-4-(trifluoromethoxy)phenyl]pyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— N-((1R,2R)-2-hydroxy-indan-1-yl)-2-methoxy-4-pyridin-4-yl-benzamide 1127308-89-7 C22H20N2O3
N-((1R,2R)-2-hydroxy-indan-1-yl)-2-methoxy-4-pyridin-4-yl-benzamide
—— N-{3-[3-methyl-4-oxo-5-(2-pyrrolidin-1-yl-ethyl)-1,4,5,6,7,8-hexahydro-pyrrolo[3,2-c]azepin-2-ylmethylene]-2-oxo-2,3-dihydro-1H-indol-5-yl}-acetamide 1082988-80-4 C26H31N5O3
N-{3-[3-methyl-4-oxo-5-(2-pyrrolidin-1-yl-ethyl)-1,4,5,6,7,8-hexahydro-pyrrolo[3,2-c]azepin-2-ylmethylene]-2-oxo-2,3-dihydro-1H-indol-5-yl}-acetamide
—— 4-(4-chloro-benzyl)-5-hydroxy-5-methyl-3-(2,4,6-trifluoro-phenyl)-5H-furan-2-one 1164101-23-8 C18H12ClF3O3
4-(4-chloro-benzyl)-5-hydroxy-5-methyl-3-(2,4,6-trifluoro-phenyl)-5H-furan-2-one
—— 3-[(4-ethoxy-3-methoxyphenyl)(1,3-oxazol-5-ylmethyl)amino]benzoic acid tert-butyl ester 1203598-27-9 C24H28N2O5
3-[(4-ethoxy-3-methoxyphenyl)(1,3-oxazol-5-ylmethyl)amino]benzoic acid tert-butyl ester
—— Isonicotinsaeure-m-tolylhydrazid 10517-75-6 C13H13N3O
Isonicotinsaeure-m-tolylhydrazid
—— 4-pyridin-4-yl-N-{(1R)-1-[2-(trifluoromethyl)phenyl]ethyl}benzamide 1127308-54-6 C21H17F3N2O
4-pyridin-4-yl-N-{(1R)-1-[2-(trifluoromethyl)phenyl]ethyl}benzamide
—— 1-{6-[(2,6-dichlorobenzyl)oxy]-1H-benzimidazol-2-yl}-3-(2-morpholin-4-ylethyl)urea 1146852-73-4 C21H23Cl2N5O3
1-{6-[(2,6-dichlorobenzyl)oxy]-1H-benzimidazol-2-yl}-3-(2-morpholin-4-ylethyl)urea
—— 3-(4-bromo-benzenesulfonyl)-1-trityloxy-azepan-2-one 1009373-05-0 C31H28BrNO4S
3-(4-bromo-benzenesulfonyl)-1-trityloxy-azepan-2-one
—— methyl 4-oxo-1-phenyl-1,4,5,6,7,8-hexahydrocycloheptapyrazole-5-carboxylate 1195073-38-1 C16H16N2O3
methyl 4-oxo-1-phenyl-1,4,5,6,7,8-hexahydrocycloheptapyrazole-5-carboxylate
—— 3-(2-methoxy-4-(1H-pyrazol-4-yl)phenyl)-1-(3-methoxybenzyl)-1-(2-(piperidin-1-yl)ethyl)urea 1219726-57-4 C26H33N5O3
3-(2-methoxy-4-(1H-pyrazol-4-yl)phenyl)-1-(3-methoxybenzyl)-1-(2-(piperidin-1-yl)ethyl)urea
—— (2S,5S)-2-tert-butyl-5-[2-fluoro-5-(tetrahydro-2H-pyrane-2-yloxymethyl)-benzyl]-3-methyl-4-oxoimidazoline-1-carboxylic acid tert-butyl ester 1159894-75-3 C26H39FN2O5
(2S,5S)-2-tert-butyl-5-[2-fluoro-5-(tetrahydro-2H-pyrane-2-yloxymethyl)-benzyl]-3-methyl-4-oxoimidazoline-1-carboxylic acid tert-butyl ester
—— 2,2-dimethyl-5-[4-(phenylethynyl)benzyl]-1,3-dioxane-4,6-dione 1094201-07-6 C21H18O4
2,2-dimethyl-5-[4-(phenylethynyl)benzyl]-1,3-dioxane-4,6-dione
—— 4-(4-Bromo-6H-dibenz[b,e]oxepin-11-ylidene)-1-methylpiperidine 1017796-07-4 C20H20BrNO
4-(4-Bromo-6H-dibenz[b,e]oxepin-11-ylidene)-1-methylpiperidine
—— 4-benzyloxy-3-ethyl-5-methyl-benzonitrile 1150644-92-0 C17H17NO
4-benzyloxy-3-ethyl-5-methyl-benzonitrile
—— (3S)-4-(6-amino-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)-3-methyl-N-(1-methyl-1H-benzotriazol-4-yl)piperazine-1-carboxamide 1616414-97-1 C19H23N11O
(3S)-4-(6-amino-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)-3-methyl-N-(1-methyl-1H-benzotriazol-4-yl)piperazine-1-carboxamide
—— methyl 2-(7-(benzyl(methyl)amino)-2-methoxy-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetate 1403368-06-8 C24H28N2O3
methyl 2-(7-(benzyl(methyl)amino)-2-methoxy-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetate
—— (3S)-4-(6-amino-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)-3-methyl-N-(1-methyl-1H-pyrazolo[4,3-c]pyridin-4-yl)piperazine-1-carboxamide 1616415-00-9 C19H23N11O
(3S)-4-(6-amino-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)-3-methyl-N-(1-methyl-1H-pyrazolo[4,3-c]pyridin-4-yl)piperazine-1-carboxamide
—— 2,6-Naphthyridine-2(1H)-carboxylic acid, 3,4-dihydro-7-methyl-, 1,1-dimethylethyl ester 1279822-51-3 C14H20N2O2
2,6-Naphthyridine-2(1H)-carboxylic acid, 3,4-dihydro-7-methyl-, 1,1-dimethylethyl ester
—— Gramicidin J, mono-N-methanesulfonate 101563-92-2 C45H69N9O10S
Gramicidin J, mono-N-methanesulfonate
—— —— 1055781-81-1 C25H27NO5
—— 6-hydroxy-6-(pyridin-3-yl)hexane-2,4-dione 1221016-25-6 C11H13NO3
6-hydroxy-6-(pyridin-3-yl)hexane-2,4-dione
—— (1S,2S,3R,4R)-3-Pyridin-3-yl-bicyclo[2.2.1]heptane-2-carboxylic acid methyl ester 133870-53-8 C14H17NO2
(1S,2S,3R,4R)-3-Pyridin-3-yl-bicyclo[2.2.1]heptane-2-carboxylic acid methyl ester
—— (R)-tert-butyl 5-amino-5-oxo-1-(4-(trifluoromethyl)phenyl)pentan-2-ylcarbamate 1236031-45-0 C17H23F3N2O3
(R)-tert-butyl 5-amino-5-oxo-1-(4-(trifluoromethyl)phenyl)pentan-2-ylcarbamate
—— 6-chloro-3-(2-(1-methoxynaphthalen-2-yl)-2-oxoethyl)quinazolin-4(3H)-one 1323954-02-4 C21H15ClN2O3
6-chloro-3-(2-(1-methoxynaphthalen-2-yl)-2-oxoethyl)quinazolin-4(3H)-one
—— 4-(9,10-Diethoxy-2-imino-6,7-dihydro-2H-pyrimido[6,1-a]isoquinolin-4-yl)-phenol; hydrochloride 107301-53-1 C22H23N3O3*ClH
4-(9,10-Diethoxy-2-imino-6,7-dihydro-2H-pyrimido[6,1-a]isoquinolin-4-yl)-phenol; hydrochloride