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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(3-cyclopropylimidazo[1,2-a]pyridin-2-yl)-N-[[4-(trifluoromethoxy)phenyl]methyl]benzenesulfonamide 1381784-82-2 C24H20F3N3O3S
N-(3-cyclopropylimidazo[1,2-a]pyridin-2-yl)-N-[[4-(trifluoromethoxy)phenyl]methyl]benzenesulfonamide
—— Tert-butyl 2-(hydroxymethyl)-1,4-diazepane-1-carboxylate 1381946-91-3 C11H22N2O3
Tert-butyl 2-(hydroxymethyl)-1,4-diazepane-1-carboxylate
—— N-[2-(2-oxopyrrolidin-1-yl)ethyl]-2-(4-{3-[3-({[(2,2,2-trifluoroethyl)amino]carbonyl]amino)phenyl]imidazo[1,2-b]pyridazin-7-yl}-1H-pyrazol-1-yl)propanamide 1383480-54-3 C27H28F3N9O3
N-[2-(2-oxopyrrolidin-1-yl)ethyl]-2-(4-{3-[3-({[(2,2,2-trifluoroethyl)amino]carbonyl]amino)phenyl]imidazo[1,2-b]pyridazin-7-yl}-1H-pyrazol-1-yl)propanamide
—— ethyl 8-allyl-5-ethyl-7-hydroxy-2,2-dimethyl-4-oxo-4H-benzo[d][1,3]dioxine-6-carboxylate 1370334-62-5 C18H22O6
ethyl 8-allyl-5-ethyl-7-hydroxy-2,2-dimethyl-4-oxo-4H-benzo[d][1,3]dioxine-6-carboxylate
—— (S)-7-(2-(3,4-dimethylpiperazin-1-yl)ethoxy)-N-(1-((5-fluoro-6-isopropylpyridin-2-yl)methyl)-3-methyl-1H-indazol-4-yl)imidazo[1,2-a]pyridine-3-carboxamide 1383471-79-1 C33H39FN8O2
(S)-7-(2-(3,4-dimethylpiperazin-1-yl)ethoxy)-N-(1-((5-fluoro-6-isopropylpyridin-2-yl)methyl)-3-methyl-1H-indazol-4-yl)imidazo[1,2-a]pyridine-3-carboxamide
—— 5-methyl-[1,3,4]oxadiazole-2-carboxylic acid [3-((R)-1-{5-[5-chloro-3-fluoro-2-(5-methyl-[1,2,4]oxadiazol-3-yl)-phenyl]-3-fluoro-pyridin-2-yl}-ethylcarbamoyl)-oxetan-3-yl]-amide 1384171-11-2 C24H20ClF2N7O5
5-methyl-[1,3,4]oxadiazole-2-carboxylic acid [3-((R)-1-{5-[5-chloro-3-fluoro-2-(5-methyl-[1,2,4]oxadiazol-3-yl)-phenyl]-3-fluoro-pyridin-2-yl}-ethylcarbamoyl)-oxetan-3-yl]-amide
—— 5-benzyl-7-(4-methoxyphenyl)-2,3-dihydrofuro[3,2-c]pyridin-4(5H)-one 1350743-57-5 C21H19NO3
5-benzyl-7-(4-methoxyphenyl)-2,3-dihydrofuro[3,2-c]pyridin-4(5H)-one
—— 3-(4-allyl-3-(trifluoromethyl)phenyl)-5-(1-methyl-5-phenyl-1H-pyrazol-3-yl)-1,2,4-oxadiazole 1350825-35-2 C22H17F3N4O
3-(4-allyl-3-(trifluoromethyl)phenyl)-5-(1-methyl-5-phenyl-1H-pyrazol-3-yl)-1,2,4-oxadiazole
—— 2-[2-[(6-methoxynaphthalen-2-yl)sulfonyl]-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-1-yl]-N-[6-(morpholin-4-ylmethyl)-1,2,3,4-tetrahydronaphthalen-2-yl]acetamide 1242848-46-9 C35H40N4O5S
2-[2-[(6-methoxynaphthalen-2-yl)sulfonyl]-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-1-yl]-N-[6-(morpholin-4-ylmethyl)-1,2,3,4-tetrahydronaphthalen-2-yl]acetamide
—— 3-(4'-hydroxy-3',4',5',6'-tetrahydro-2'H-[3,4']bipyridinyl-1'-ylmethyl)-1-oxo-2-phenyl-1,2-dihydro-isoquinoline-4-carboxylic acid ((S)-1-phenyl-propyl)-amide 1075712-17-2 C36H36N4O3
3-(4'-hydroxy-3',4',5',6'-tetrahydro-2'H-[3,4']bipyridinyl-1'-ylmethyl)-1-oxo-2-phenyl-1,2-dihydro-isoquinoline-4-carboxylic acid ((S)-1-phenyl-propyl)-amide
—— N-[(1-benzylpyrrolidin-3-yl)methyl]-2-[2-[(4-methoxy-2,6-dimethylphenyl)sulfonyl]-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-1-yl]acetamide 1242848-78-7 C30H38N4O4S
N-[(1-benzylpyrrolidin-3-yl)methyl]-2-[2-[(4-methoxy-2,6-dimethylphenyl)sulfonyl]-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-1-yl]acetamide
—— N-tert-butoxycarbonyl-1-i-propyl-L-tryptophan 1219040-06-8 C19H26N2O4
N-tert-butoxycarbonyl-1-i-propyl-L-tryptophan
—— 1-methyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl}-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-3-carboxamide 1227409-36-0 C19H24N6O2
1-methyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl}-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
—— 2-ethylsulfanyl-7-fluoro-N-[(4-fluorophenyl)-methyl]-4-methyl-quinoline-3-carboxamide 1242554-05-7 C20H18F2N2OS
2-ethylsulfanyl-7-fluoro-N-[(4-fluorophenyl)-methyl]-4-methyl-quinoline-3-carboxamide
—— 5-(3-chlorophenyl)-6-methy-5-azaspiro[2.3]hexan-4-one 1353889-62-9 C12H12ClNO
5-(3-chlorophenyl)-6-methy-5-azaspiro[2.3]hexan-4-one
—— 2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-3-(3-ethynylphenyl)-2-methylpropanenitrile 1056887-37-6 C23H20N2O
2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-3-(3-ethynylphenyl)-2-methylpropanenitrile
—— 6-(5-bromomethylnaphthalen-1-yloxy)nicotinonitrile 1087351-36-7 C17H11BrN2O
6-(5-bromomethylnaphthalen-1-yloxy)nicotinonitrile
—— N-(cyclobutylmethyl)-N-[4-(1H-imidazol-5-ylmethyl)-3,4-dihydro-2H-chromen-6-yl]acetamide 1049633-45-5 C20H25N3O2
N-(cyclobutylmethyl)-N-[4-(1H-imidazol-5-ylmethyl)-3,4-dihydro-2H-chromen-6-yl]acetamide
—— 3-[2-Cyano-2-(3-ethyl-2-methoxyquinolin-7-yl)propyl]benzoic acid 1056892-25-1 C23H22N2O3
3-[2-Cyano-2-(3-ethyl-2-methoxyquinolin-7-yl)propyl]benzoic acid
—— 2-[(3S,4R)-4-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-ethoxypiperidin-1-yl]-4-{5-[(3R)-3-methylpiperazin-1-yl]pyrazin-2-yl}-1,3-thiazole-5-carboxylic acid 1229572-24-0 C26H32Cl2N8O4S
2-[(3S,4R)-4-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-ethoxypiperidin-1-yl]-4-{5-[(3R)-3-methylpiperazin-1-yl]pyrazin-2-yl}-1,3-thiazole-5-carboxylic acid
—— 4-{[(Tert-butoxy)carbonyl]amino}oxepane-4-carboxylicacid 1498717-02-4 C12H21NO5
4-{[(Tert-butoxy)carbonyl]amino}oxepane-4-carboxylicacid
—— Ethyl 7-[3-bromo-2-(bromomethyl)-6-oxopyridin-1-yl]heptanoate 1091600-34-8 C15H21Br2NO3
Ethyl 7-[3-bromo-2-(bromomethyl)-6-oxopyridin-1-yl]heptanoate
—— [9-(2,6-Diethyl-4-methylphenyl)-10-oxo-3-oxaspiro[5.5]undec-8-en-8-yl] propane-1-sulfonate 1058730-92-9 C24H34O5S
[9-(2,6-Diethyl-4-methylphenyl)-10-oxo-3-oxaspiro[5.5]undec-8-en-8-yl] propane-1-sulfonate
—— 4-(1-acetyl-piperidin-3-yl)-N-[2-methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenyl]-benzamide 1146700-52-8 C30H40N4O2
4-(1-acetyl-piperidin-3-yl)-N-[2-methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenyl]-benzamide
—— 3-(1H-indol-2-yl)-2-(2-methoxy-3-methylquinolin-7-yl)-2-methylpropanenitrile 1056894-25-7 C23H21N3O
3-(1H-indol-2-yl)-2-(2-methoxy-3-methylquinolin-7-yl)-2-methylpropanenitrile
—— Nα-[3-(2-fluorophenyl)acryloyl]-d-tryptophan 1219039-61-8 C20H17FN2O3
Nα-[3-(2-fluorophenyl)acryloyl]-d-tryptophan
—— [(3S)-6-{[(3S)-7-(2-ethoxy-1H-benzimidazol-1-yl)-2,3-dihydro-1-benzofuran-3-yl]amino}-2,3-dihydro-1-benzofuran-3-yl]acetic acid 1258396-02-9 C27H25N3O5
[(3S)-6-{[(3S)-7-(2-ethoxy-1H-benzimidazol-1-yl)-2,3-dihydro-1-benzofuran-3-yl]amino}-2,3-dihydro-1-benzofuran-3-yl]acetic acid
—— N-((R)-2-[4-(2,5-dimethyl-phenyl)-piperazin-1-yl]-1-hydroxymethyl-2-oxo-ethyl)-benzenesulfonamide 1065143-21-6 C21H27N3O4S
N-((R)-2-[4-(2,5-dimethyl-phenyl)-piperazin-1-yl]-1-hydroxymethyl-2-oxo-ethyl)-benzenesulfonamide
—— N-(1-(5-(3-chloro-4-cyanophenyl)pyridin-3-yl)butyl)ethanesulfonamide 1255872-03-7 C18H20ClN3O2S
N-(1-(5-(3-chloro-4-cyanophenyl)pyridin-3-yl)butyl)ethanesulfonamide
—— 2-amino-4-(2,4-dimethylphenyl)phthalazin-1(2H)-one 1309196-09-5 C16H15N3O
2-amino-4-(2,4-dimethylphenyl)phthalazin-1(2H)-one
—— 9-cyclopentyl-2-({2-ethoxy-4-[(1-methylpiperidin-4-yl)-oxy]-phenyl}amino)-7-methyl-7,9-dihydro-8H-purin-8-one 1124329-35-6 C25H34N6O3
9-cyclopentyl-2-({2-ethoxy-4-[(1-methylpiperidin-4-yl)-oxy]-phenyl}amino)-7-methyl-7,9-dihydro-8H-purin-8-one
—— 6-(2-chlorophenyl)-7-(4-chlorophenyl)-3-[N-(cyclohexylmethyl)carbamoyl]-2-sulfamoylpyrazolo[1,5-a]pyrimidine 1001425-48-4 C26H25Cl2N5O3S
6-(2-chlorophenyl)-7-(4-chlorophenyl)-3-[N-(cyclohexylmethyl)carbamoyl]-2-sulfamoylpyrazolo[1,5-a]pyrimidine
—— cis-2-Benzyltetrahydropyrrolo[3,4-c]pyrrole-1,3(2H,3aH)-dione 189348-40-1 C13H14N2O2
cis-2-Benzyltetrahydropyrrolo[3,4-c]pyrrole-1,3(2H,3aH)-dione
—— 9-cyclopentyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)-phenyl]amino}-7-methyl-7,9-dihydro-8H-purin-8-one 1124329-13-0 C23H31N7O2
9-cyclopentyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)-phenyl]amino}-7-methyl-7,9-dihydro-8H-purin-8-one
—— N-(5-(2-aminophenylcarbamoyl)pentyl)-3-methyl-4-(3-pyridinyl)-benzamide 1255951-52-0 C25H28N4O2
N-(5-(2-aminophenylcarbamoyl)pentyl)-3-methyl-4-(3-pyridinyl)-benzamide
—— 6-(3-amino-6-(1-methyl-1H-pyrazol-4-yl)pyrazin-2-yl)-3,4-dihydroisoquinolin-1(2H)-one 1396772-98-7 C17H16N6O
6-(3-amino-6-(1-methyl-1H-pyrazol-4-yl)pyrazin-2-yl)-3,4-dihydroisoquinolin-1(2H)-one
—— 2-amino-4-(2,5-difluorophenyl)-1,3-thiazol-5-carbonitrile 1139743-04-6 C10H5F2N3S
2-amino-4-(2,5-difluorophenyl)-1,3-thiazol-5-carbonitrile
—— 3-((5-chloro-1-(4-fluorobutyl)-1H-benzo[d]imidazol-2-yl)methyl)-1-(methylsulfonyl)-1H-imidazo[4,5-c]pyridin-2(3H)-one 1383423-07-1 C19H19ClFN5O3S
3-((5-chloro-1-(4-fluorobutyl)-1H-benzo[d]imidazol-2-yl)methyl)-1-(methylsulfonyl)-1H-imidazo[4,5-c]pyridin-2(3H)-one
—— 4-{8-[(2-amino-2-oxoethyl)amino]-6-phenylimidazo[1,2-a]pyrazin-3-yl}-N-cyclopropylbenzamide 1382479-36-8 C24H22N6O2
4-{8-[(2-amino-2-oxoethyl)amino]-6-phenylimidazo[1,2-a]pyrazin-3-yl}-N-cyclopropylbenzamide
—— N-[N'-[(3-chloro-4-fluorophenyl)methyl]-N-[5-(trifluoromethyl)-1H-pyrazol-3-yl]carbamimidoyl]-3,4-difluorobenzamide 1381805-06-6 C19H12ClF6N5O
N-[N'-[(3-chloro-4-fluorophenyl)methyl]-N-[5-(trifluoromethyl)-1H-pyrazol-3-yl]carbamimidoyl]-3,4-difluorobenzamide
—— 3-amino-4-bromo-5-fluorobenzoic acid 1340341-79-8 C7H5BrFNO2
3-amino-4-bromo-5-fluorobenzoic acid
—— N-(6-fluoro-3-methylimidazo[1,2-a]pyridin-2-yl)-N-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]benzenesulfonamide 1381784-31-1 C22H16F5N3O2S
N-(6-fluoro-3-methylimidazo[1,2-a]pyridin-2-yl)-N-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]benzenesulfonamide
—— 5-(3-fluoro-phenyl)-2-methyl-oxazole-4-carboxylic acid {2-[4-(1-hydroxy-1-methyl-ethyl)-oxazol-2-ylmethyl]-2H-[1,2,3]triazol-4-yl}-amide 1380665-91-7 C20H19FN6O4
5-(3-fluoro-phenyl)-2-methyl-oxazole-4-carboxylic acid {2-[4-(1-hydroxy-1-methyl-ethyl)-oxazol-2-ylmethyl]-2H-[1,2,3]triazol-4-yl}-amide
—— 2-(2-(2-(4-benzhydrylpiperazin-1-yl)-2-oxoethoxy)acetamido)-5-(pyridin-4-yl)benzoic acid sodium salt 1103927-13-4 C33H31N4O5*Na
2-(2-(2-(4-benzhydrylpiperazin-1-yl)-2-oxoethoxy)acetamido)-5-(pyridin-4-yl)benzoic acid sodium salt
—— methyl 4-(4-((4'-chlorobiphenyl-2-yl)methyl)piperazin-1-yl)-2-(phenylsulfonyl)benzoate 1228780-15-1 C31H29ClN2O4S
methyl 4-(4-((4'-chlorobiphenyl-2-yl)methyl)piperazin-1-yl)-2-(phenylsulfonyl)benzoate
—— 1-({1-(3-chlorophenyl)-5-[3-(3-(ethylamino)propoxy)phenyl]-1H-pyrazol-3-yl}carbonyl)imidazolidin-4-one formate 1187917-61-8 CH2O2*C24H26ClN5O3
1-({1-(3-chlorophenyl)-5-[3-(3-(ethylamino)propoxy)phenyl]-1H-pyrazol-3-yl}carbonyl)imidazolidin-4-one formate
—— 3-((2-methoxy-acetyl)amino)-oxetane-3-carboxylic acid ((R)-1-{5-[3,5-dichloro-2-(2,2-difluoro-ethoxy)-phenyl]-3-fluoro-pyridin-2-yl}-ethyl)-amide 1384171-34-9 C22H22Cl2F3N3O5
3-((2-methoxy-acetyl)amino)-oxetane-3-carboxylic acid ((R)-1-{5-[3,5-dichloro-2-(2,2-difluoro-ethoxy)-phenyl]-3-fluoro-pyridin-2-yl}-ethyl)-amide
—— N-cyclopropyl-4-{8-[(2-hydroxybenzyl)amino]imidazo[1,2-a]pyrazin-3-yl}-2-methylbenzamide 1383102-89-3 C24H23N5O2
N-cyclopropyl-4-{8-[(2-hydroxybenzyl)amino]imidazo[1,2-a]pyrazin-3-yl}-2-methylbenzamide
—— N-benzyl-2-(4-(dimethylamino)benzamido)isonicotinamide 1202926-64-4 C22H22N4O2
N-benzyl-2-(4-(dimethylamino)benzamido)isonicotinamide
—— 2-(5-fluoro-3-(3-(3-fluoro-4-(trifluoromethyl)benzyl)-4-oxo-3,4-dihydrophthalazin-1-yl)-2-methyl-1H-indol-1-yl)acetic acid 1297275-28-5 C27H18F5N3O3
2-(5-fluoro-3-(3-(3-fluoro-4-(trifluoromethyl)benzyl)-4-oxo-3,4-dihydrophthalazin-1-yl)-2-methyl-1H-indol-1-yl)acetic acid