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—— (Z)-3-(4-methoxyphenyl)-N-[[(3S)-1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl]methyl]-N-methylprop-2-en-1-amine —— C26H36N2O2
(Z)-3-(4-methoxyphenyl)-N-[[(3S)-1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl]methyl]-N-methylprop-2-en-1-amine
—— (Z)-3-(3,4-dimethoxyphenyl)-N-[(1R)-1-(5-methyl-1-pyridin-2-ylpyrazol-4-yl)ethyl]prop-2-enamide —— C22H24N4O3
(Z)-3-(3,4-dimethoxyphenyl)-N-[(1R)-1-(5-methyl-1-pyridin-2-ylpyrazol-4-yl)ethyl]prop-2-enamide
—— (Z)-1-[(4aS,9bR)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-3-(3-nitrophenyl)prop-2-en-1-one —— C22H23N3O3
(Z)-1-[(4aS,9bR)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-3-(3-nitrophenyl)prop-2-en-1-one
—— (Z)-3-[4-(dimethylamino)phenyl]-2-(6-ethyl-4-oxo-3H-quinazolin-2-yl)prop-2-enenitrile —— C21H20N4O
(Z)-3-[4-(dimethylamino)phenyl]-2-(6-ethyl-4-oxo-3H-quinazolin-2-yl)prop-2-enenitrile
—— (Z)-3-(2-methoxyphenyl)-N-[(1R)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]prop-2-en-1-amine —— C22H24N4O
(Z)-3-(2-methoxyphenyl)-N-[(1R)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]prop-2-en-1-amine
—— (Z)-3-[1-(4-bromophenyl)-2,5-dimethylpyrrol-3-yl]-2-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]prop-2-enenitrile —— C23H22BrN3S
(Z)-3-[1-(4-bromophenyl)-2,5-dimethylpyrrol-3-yl]-2-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]prop-2-enenitrile
—— (Z)-N-methyl-N-[[(3S)-1-[2-(2-methylphenyl)ethyl]piperidin-3-yl]methyl]-3-pyridin-3-ylprop-2-enamide —— C24H31N3O
(Z)-N-methyl-N-[[(3S)-1-[2-(2-methylphenyl)ethyl]piperidin-3-yl]methyl]-3-pyridin-3-ylprop-2-enamide
—— (Z)-1-[4-[4-(2-aminopropan-2-yl)triazol-1-yl]piperidin-1-yl]-3-phenylprop-2-en-1-one —— C19H25N5O
(Z)-1-[4-[4-(2-aminopropan-2-yl)triazol-1-yl]piperidin-1-yl]-3-phenylprop-2-en-1-one
—— (Z)-2-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-3-(3-phenoxyphenyl)prop-2-enenitrile —— C23H20N2OS
(Z)-2-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-3-(3-phenoxyphenyl)prop-2-enenitrile
—— (Z)-3-(2-chloroquinolin-3-yl)-2-(6,7-dimethoxy-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile —— C22H15ClN4O3
(Z)-3-(2-chloroquinolin-3-yl)-2-(6,7-dimethoxy-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile
—— (Z)-1-[(4aS,9bS)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-3-(3-nitrophenyl)prop-2-en-1-one —— C22H23N3O3
(Z)-1-[(4aS,9bS)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-3-(3-nitrophenyl)prop-2-en-1-one
—— (Z)-3-[5-(4-chloro-3-nitrophenyl)furan-2-yl]-2-(morpholine-4-carbonyl)prop-2-enenitrile —— C18H14ClN3O5
(Z)-3-[5-(4-chloro-3-nitrophenyl)furan-2-yl]-2-(morpholine-4-carbonyl)prop-2-enenitrile
—— (Z)-N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-(1H-imidazol-5-yl)prop-2-enamide —— C21H23N5O
(Z)-N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-(1H-imidazol-5-yl)prop-2-enamide
—— (Z)-3-(3-nitrophenyl)-N-[4-nitro-3-(trifluoromethyl)phenyl]prop-2-enamide —— C16H10F3N3O5
(Z)-3-(3-nitrophenyl)-N-[4-nitro-3-(trifluoromethyl)phenyl]prop-2-enamide
—— (Z)-N-[(4R)-6,6-dimethyl-1-(4-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]-3-(1H-imidazol-5-yl)prop-2-enamide —— C22H25N5O
(Z)-N-[(4R)-6,6-dimethyl-1-(4-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]-3-(1H-imidazol-5-yl)prop-2-enamide
—— (Z)-3-(2-chloro-7,8-dimethylquinolin-3-yl)-2-(6-methyl-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile —— C23H17ClN4O
(Z)-3-(2-chloro-7,8-dimethylquinolin-3-yl)-2-(6-methyl-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile
—— (Z)-3-(4-fluorophenyl)-N-[(1S)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]prop-2-en-1-amine —— C21H21FN4
(Z)-3-(4-fluorophenyl)-N-[(1S)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]prop-2-en-1-amine
—— (Z)-3-(2-chloro-8-methylquinolin-3-yl)-2-(6-methyl-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile —— C22H15ClN4O
(Z)-3-(2-chloro-8-methylquinolin-3-yl)-2-(6-methyl-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile
—— (Z)-3-(1H-imidazol-5-yl)-1-[(3S)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]prop-2-en-1-one —— C21H25N3O3
(Z)-3-(1H-imidazol-5-yl)-1-[(3S)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]prop-2-en-1-one
—— (Z)-N-(3-amino-4-chlorophenyl)sulfonyl-3-(5-bromofuran-2-yl)-N-(4-methoxyphenyl)prop-2-enamide —— C20H16BrClN2O5S
(Z)-N-(3-amino-4-chlorophenyl)sulfonyl-3-(5-bromofuran-2-yl)-N-(4-methoxyphenyl)prop-2-enamide
—— (Z)-3-(1H-imidazol-5-yl)-1-[(3R)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]prop-2-en-1-one —— C21H25N3O3
(Z)-3-(1H-imidazol-5-yl)-1-[(3R)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]prop-2-en-1-one
—— (Z)-3-[1-(4-bromophenyl)-2,5-dimethylpyrrol-3-yl]-2-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]prop-2-enenitrile —— C23H22BrN3S
(Z)-3-[1-(4-bromophenyl)-2,5-dimethylpyrrol-3-yl]-2-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]prop-2-enenitrile
—— (Z)-3-(2-chloroquinolin-3-yl)-2-(6-methyl-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile —— C21H13ClN4O
(Z)-3-(2-chloroquinolin-3-yl)-2-(6-methyl-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile
—— (Z)-1-[3-(3-methylbutyl)-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl]-3-(1-methylpyrazol-4-yl)prop-2-en-1-one —— C18H25N5O
(Z)-1-[3-(3-methylbutyl)-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl]-3-(1-methylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-1-[(3R)-3-(6-morpholin-4-ylpyrimidin-4-yl)piperidin-1-yl]pent-3-en-1-one —— C18H26N4O2
(Z)-1-[(3R)-3-(6-morpholin-4-ylpyrimidin-4-yl)piperidin-1-yl]pent-3-en-1-one
—— (Z)-3-(4-chlorophenyl)sulfonyl-2-methylprop-2-enoic acid —— C10H9ClO4S
(Z)-3-(4-chlorophenyl)sulfonyl-2-methylprop-2-enoic acid
—— (Z)-3-(2-methoxyphenyl)-N-[(1S)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]prop-2-en-1-amine —— C22H24N4O
(Z)-3-(2-methoxyphenyl)-N-[(1S)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]prop-2-en-1-amine
—— (Z)-2-methyl-3-(4-methylphenyl)sulfonylprop-2-enoic acid —— C11H12O4S
(Z)-2-methyl-3-(4-methylphenyl)sulfonylprop-2-enoic acid
—— (Z)-3-(4-chlorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]prop-2-en-1-one —— C19H26ClN3O2
(Z)-3-(4-chlorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]prop-2-en-1-one
—— (Z)-3-(3,4-dimethoxyphenyl)-N-[(1S)-1-(5-methyl-1-pyridin-2-ylpyrazol-4-yl)ethyl]prop-2-enamide —— C22H24N4O3
(Z)-3-(3,4-dimethoxyphenyl)-N-[(1S)-1-(5-methyl-1-pyridin-2-ylpyrazol-4-yl)ethyl]prop-2-enamide
—— (Z)-N-[(4-chlorophenyl)methyl]-3-[2-(difluoromethoxy)-5-nitrophenyl]prop-2-enamide —— C17H13ClF2N2O4
(Z)-N-[(4-chlorophenyl)methyl]-3-[2-(difluoromethoxy)-5-nitrophenyl]prop-2-enamide
—— (Z)-N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-(1H-imidazol-5-yl)prop-2-enamide —— C21H23N5O
(Z)-N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-(1H-imidazol-5-yl)prop-2-enamide
—— (Z)-1-[(3R)-3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-(4-methoxyphenyl)prop-2-en-1-one —— C25H31NO3
(Z)-1-[(3R)-3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-(4-methoxyphenyl)prop-2-en-1-one
—— (Z)-1-(4-chlorophenyl)-3-(9-methylcarbazol-3-yl)prop-2-en-1-one —— C22H16ClNO
(Z)-1-(4-chlorophenyl)-3-(9-methylcarbazol-3-yl)prop-2-en-1-one
—— (Z)-N-[(2R,4S)-1-acetyl-2-methyl-3,4-dihydro-2H-quinolin-4-yl]-N,3-diphenylprop-2-enamide —— C27H26N2O2
(Z)-N-[(2R,4S)-1-acetyl-2-methyl-3,4-dihydro-2H-quinolin-4-yl]-N,3-diphenylprop-2-enamide
—— (Z)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(4-methoxyphenyl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-en-1-amine —— C26H40N2O2
(Z)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(4-methoxyphenyl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-en-1-amine
—— (Z)-N-[(4S)-6,6-dimethyl-1-(4-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]-3-(1H-imidazol-5-yl)prop-2-enamide —— C22H25N5O
(Z)-N-[(4S)-6,6-dimethyl-1-(4-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]-3-(1H-imidazol-5-yl)prop-2-enamide
—— (Z)-1-[(5R)-9-(cyclohexylmethyl)-2,9-diazaspiro[4.5]decan-2-yl]-2-methylbut-2-en-1-one —— C20H34N2O
(Z)-1-[(5R)-9-(cyclohexylmethyl)-2,9-diazaspiro[4.5]decan-2-yl]-2-methylbut-2-en-1-one
—— (Z)-1-[(5S)-9-(cyclohexylmethyl)-2,9-diazaspiro[4.5]decan-2-yl]-2-methylbut-2-en-1-one —— C20H34N2O
(Z)-1-[(5S)-9-(cyclohexylmethyl)-2,9-diazaspiro[4.5]decan-2-yl]-2-methylbut-2-en-1-one
—— (Z)-3-(3,4-dimethoxyphenyl)-N-[(3S)-1-(1-methylpiperidin-4-yl)piperidin-3-yl]prop-2-enamide —— C22H33N3O3
(Z)-3-(3,4-dimethoxyphenyl)-N-[(3S)-1-(1-methylpiperidin-4-yl)piperidin-3-yl]prop-2-enamide
—— (Z)-N-ethyl-N-[[1-[2-(2-methylphenyl)ethyl]piperidin-4-yl]methyl]-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C24H34N4O
(Z)-N-ethyl-N-[[1-[2-(2-methylphenyl)ethyl]piperidin-4-yl]methyl]-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— (Z)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(2-methoxyphenyl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-en-1-amine —— C26H40N2O2
(Z)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(2-methoxyphenyl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-en-1-amine
—— (Z)-1-[(5R)-9-(cyclohexylmethyl)-2,9-diazaspiro[4.5]decan-2-yl]-3-pyridin-4-ylprop-2-en-1-one —— C23H33N3O
(Z)-1-[(5R)-9-(cyclohexylmethyl)-2,9-diazaspiro[4.5]decan-2-yl]-3-pyridin-4-ylprop-2-en-1-one
—— (Z)-3-pyridin-2-yl-N-[(3S)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]prop-2-enamide —— C19H19F3N4O
(Z)-3-pyridin-2-yl-N-[(3S)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]prop-2-enamide
—— (Z)-2-Cyano-3-[4-(difluoromethoxy)phenyl]-N-(3-sulfamoylphenyl)prop-2-enamide —— C17H13F2N3O4S
(Z)-2-Cyano-3-[4-(difluoromethoxy)phenyl]-N-(3-sulfamoylphenyl)prop-2-enamide
—— (Z)-3-[3-(5-methylfuran-2-yl)-1-phenylpyrazol-4-yl]-1-thiophen-2-ylprop-2-en-1-one —— C21H16N2O2S
(Z)-3-[3-(5-methylfuran-2-yl)-1-phenylpyrazol-4-yl]-1-thiophen-2-ylprop-2-en-1-one
—— (Z)-N-[(2S,4S)-1-acetyl-2-methyl-3,4-dihydro-2H-quinolin-4-yl]-N,3-diphenylprop-2-enamide —— C27H26N2O2
(Z)-N-[(2S,4S)-1-acetyl-2-methyl-3,4-dihydro-2H-quinolin-4-yl]-N,3-diphenylprop-2-enamide
—— (Z)-3-(2-chloro-6,8-dimethylquinolin-3-yl)-2-(6-methyl-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile —— C23H17ClN4O
(Z)-3-(2-chloro-6,8-dimethylquinolin-3-yl)-2-(6-methyl-4-oxo-1H-quinazolin-2-yl)prop-2-enenitrile
—— (Z)-2-cyano-N-(1,3-dioxoisoindol-4-yl)-3-(4-methoxyphenyl)prop-2-enamide —— C19H13N3O4
(Z)-2-cyano-N-(1,3-dioxoisoindol-4-yl)-3-(4-methoxyphenyl)prop-2-enamide
—— (Z)-3-pyridin-2-yl-N-[(3R)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]prop-2-enamide —— C19H19F3N4O
(Z)-3-pyridin-2-yl-N-[(3R)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]prop-2-enamide