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—— (S)-N-(6-hydroxypyridin-3-yl)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide 1616085-05-2 C23H28N8O2
(S)-N-(6-hydroxypyridin-3-yl)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide
—— spiro[3H-1,2-dioxine-6,5'-3aH-furo[2,3-d][1,3]dioxole]-3,6'-diol —— C8H8O7
spiro[3H-1,2-dioxine-6,5'-3aH-furo[2,3-d][1,3]dioxole]-3,6'-diol
—— (S)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-methylpyrrolidine-2-carboxamide 1616083-89-6 C19H27N7O
(S)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-methylpyrrolidine-2-carboxamide
—— (S)-2,4-diamino-6-((1-(5-chloro-3-(3-(difluoromethyl)-5-fluorophenyl)-6-fluoro-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)amino)pyrimidine-5-carbonitrile 1615253-04-7 C22H15ClF4N8O
(S)-2,4-diamino-6-((1-(5-chloro-3-(3-(difluoromethyl)-5-fluorophenyl)-6-fluoro-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)amino)pyrimidine-5-carbonitrile
—— (S)-tert-butyl 1-(3-(3,5-difluorophenyl)-8-ethyl-4-oxo-3,4-dihydroquinazolin-2-yl)ethylcarbamate 1615254-40-4 C23H25F2N3O3
(S)-tert-butyl 1-(3-(3,5-difluorophenyl)-8-ethyl-4-oxo-3,4-dihydroquinazolin-2-yl)ethylcarbamate
—— (S)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((R)-piperidin-3-yl)pyrrolidine-2-carboxamide 1616084-09-3 C23H34N8O
(S)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((R)-piperidin-3-yl)pyrrolidine-2-carboxamide
—— (S)-tert-butyl 1-(5-(difluoromethyl)-3-(3,5-difluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)propylcarbamate 1615253-82-1 C23H23F4N3O3
(S)-tert-butyl 1-(5-(difluoromethyl)-3-(3,5-difluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)propylcarbamate
—— (S)-3-(2-(1-aminoethyl)-5-fluoro-4-oxoquinazolin-3(4H)-yl)benzonitrile 1615255-64-5 C17H13FN4O
(S)-3-(2-(1-aminoethyl)-5-fluoro-4-oxoquinazolin-3(4H)-yl)benzonitrile
—— (S)-2-(1-aminoethyl)-5-(difluoromethyl)-3-phenylquinazolin-4(3H)-one 1615255-75-8 C17H15F2N3O
(S)-2-(1-aminoethyl)-5-(difluoromethyl)-3-phenylquinazolin-4(3H)-one
—— (S)-2-(1-aminoethyl)-5,8-difluoro-3-phenylquinazolin-4(3H)-one 1615255-17-8 C16H13F2N3O
(S)-2-(1-aminoethyl)-5,8-difluoro-3-phenylquinazolin-4(3H)-one
—— spiro[3,5,7,12-tetraoxatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-triene-11,5'-3aH-furo[2,3-d][1,3]dioxole]-6'-ol —— C12H8O8
spiro[3,5,7,12-tetraoxatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-triene-11,5'-3aH-furo[2,3-d][1,3]dioxole]-6'-ol
—— (S)-2-(1-aminoethyl)-8-fluoro-3-phenylquinazolin-4(3H)-one 1615255-13-4 C16H14FN3O
(S)-2-(1-aminoethyl)-8-fluoro-3-phenylquinazolin-4(3H)-one
—— (S)-2-(1-aminopropyl)-5-fluoro-3-(3,5-difluorophenyl)quinazolin-4(3H)-one 1615255-20-3 C17H14F3N3O
(S)-2-(1-aminopropyl)-5-fluoro-3-(3,5-difluorophenyl)quinazolin-4(3H)-one
—— (S)-tert-butyl 2-(5-chloro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)piperidine-1-carboxylate 1615680-14-2 C24H26ClN3O3
(S)-tert-butyl 2-(5-chloro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)piperidine-1-carboxylate
—— (S)-2-(1-aminoethyl)-4-oxo-3-phenyl-3,4-dihydroquinazoline-5-carbonitrile 1615255-80-5 C17H14N4O
(S)-2-(1-aminoethyl)-4-oxo-3-phenyl-3,4-dihydroquinazoline-5-carbonitrile
—— (S)-5-(azetidin-1-yl)-4-(4-cyclopropyl-1H-imidazol-1-yl)-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide —— C23H22F3N9OS
(S)-5-(azetidin-1-yl)-4-(4-cyclopropyl-1H-imidazol-1-yl)-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide
—— (S)-4-(4-cyclopropyl-1H-imidazol-1-yl)-5-morpholino-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide —— C24H24F3N9O2S
(S)-4-(4-cyclopropyl-1H-imidazol-1-yl)-5-morpholino-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide
—— (S)-ethyl 2-ethoxy-3-(4-((R)-2-hydroxy-2-(3-methoxyphenyl)ethoxy)phenyl)propanoate 1416821-44-7 C22H28O6
(S)-ethyl 2-ethoxy-3-(4-((R)-2-hydroxy-2-(3-methoxyphenyl)ethoxy)phenyl)propanoate
—— [(S)-1-((S)-2-{(2S,4S)-4-amino-2-[(S)-(1,2,3,4-tetrahydro-naphthalen-1-yl)carbamoyl]-pyrrolidin-1-yl}-1-cyclohexyl-2-oxo-ethylcarbamoyl)-ethyl]-methyl-carbamic acid tert-butyl ester 1613552-11-6 C32H49N5O5
[(S)-1-((S)-2-{(2S,4S)-4-amino-2-[(S)-(1,2,3,4-tetrahydro-naphthalen-1-yl)carbamoyl]-pyrrolidin-1-yl}-1-cyclohexyl-2-oxo-ethylcarbamoyl)-ethyl]-methyl-carbamic acid tert-butyl ester
—— (S)-N-[4-(4-acetyl-piperazin-1-yl)-benzyl]-N-{1-benzyl-2-[4-(4-{[2-(tert-butyl-dimethyl-silanyloxy)-ethyl]-methyl-amino}-benzyl)-piperazin-1-yl]-2-oxo-ethyl}-3-(6-methoxy-pyridin-3-yl)-acrylamide 1314144-10-9 C51H69N7O5Si
(S)-N-[4-(4-acetyl-piperazin-1-yl)-benzyl]-N-{1-benzyl-2-[4-(4-{[2-(tert-butyl-dimethyl-silanyloxy)-ethyl]-methyl-amino}-benzyl)-piperazin-1-yl]-2-oxo-ethyl}-3-(6-methoxy-pyridin-3-yl)-acrylamide
—— (S)-4-amino-5-chloro-N-{[4-{[1-((S)-2-methoxypropionyl)-4-piperidinyl]methyl}-2-morpholinyl]methyl}-2-methoxybenzamide 1184661-38-8 C23H35ClN4O5
(S)-4-amino-5-chloro-N-{[4-{[1-((S)-2-methoxypropionyl)-4-piperidinyl]methyl}-2-morpholinyl]methyl}-2-methoxybenzamide
—— Sodium;1-bromoethenesulfonate —— C2H2BrNaO3S
Sodium;1-bromoethenesulfonate
—— (S)-4-(4-chloro-6-cyclopropylpyrimidin-2-yl)-3-methylmorpholine —— C12H16ClN3O
(S)-4-(4-chloro-6-cyclopropylpyrimidin-2-yl)-3-methylmorpholine
—— [(S)-1-(2-methoxy-naphthalen-1-ylmethyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl]-carbamic acid tert-butyl ester 1613551-79-3 C26H29N3O4
[(S)-1-(2-methoxy-naphthalen-1-ylmethyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl]-carbamic acid tert-butyl ester
—— ((S)-1-{(S)-1-[1-(2-cyano-phenyl)-1H-indazol-3-ylmethyl]-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-ylcarbamoyl}-ethyl)-methyl-carbamic acid tert-butyl ester 1613551-89-5 C33H35N7O4
((S)-1-{(S)-1-[1-(2-cyano-phenyl)-1H-indazol-3-ylmethyl]-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-ylcarbamoyl}-ethyl)-methyl-carbamic acid tert-butyl ester
—— (S)-2-(3-((5-bromo-2-((4-(4-(2-hydroxyethyl)piperazin-1-yl)phenyl)amino)pyrimidin-4-yl)amino)-2-oxopyridin-1(2H)-yl)propanenitrile 1614217-55-8 C24H27BrN8O2
(S)-2-(3-((5-bromo-2-((4-(4-(2-hydroxyethyl)piperazin-1-yl)phenyl)amino)pyrimidin-4-yl)amino)-2-oxopyridin-1(2H)-yl)propanenitrile
—— S-(phosphanylmethyl) ethanethioate —— C3H7OPS
S-(phosphanylmethyl) ethanethioate
—— Suc-Tyr-Lys(1)-NH2.Suc-Tyr-(1) —— C32H41N5O11
Suc-Tyr-Lys(1)-NH2.Suc-Tyr-(1)
—— (S)-tert-butyl (2-(((7-(3,4-dimethoxyphenyl)pyrido[3,4-b]pyrazin-5-yl)oxy)methyl)morpholino)sulfonylcarbamate —— C25H31N5O8S
(S)-tert-butyl (2-(((7-(3,4-dimethoxyphenyl)pyrido[3,4-b]pyrazin-5-yl)oxy)methyl)morpholino)sulfonylcarbamate
—— (S)-N-(5-chloro-2-methyl-3-((3-methylpiperazin-1-yl)methyl)phenyl)-2-methylpyrimidine-5-carboxamide —— C19H24ClN5O
(S)-N-(5-chloro-2-methyl-3-((3-methylpiperazin-1-yl)methyl)phenyl)-2-methylpyrimidine-5-carboxamide
—— (S)-2-methyl-N-[(2R)-pent-4-en-2-yl]propane-2-sulfinamide —— C9H19NOS
(S)-2-methyl-N-[(2R)-pent-4-en-2-yl]propane-2-sulfinamide
—— (S)-N-(5-fluoro-2-methyl-3-((3-methylpiperazin-1-yl)methyl)phenyl)-6-methylnicotinamide —— C20H25FN4O
(S)-N-(5-fluoro-2-methyl-3-((3-methylpiperazin-1-yl)methyl)phenyl)-6-methylnicotinamide
—— [(S)-[3-[[4-[[[2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-3-methoxyphenyl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C34H33N3O7
[(S)-[3-[[4-[[[2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-3-methoxyphenyl]methoxy]phenyl]-phenylmethyl]carbamic acid
—— [(S)-[3-[[4-[4-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]piperidine-1-carbonyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C38H38N4O7
[(S)-[3-[[4-[4-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]piperidine-1-carbonyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid
—— [(S)-[3-[[3-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C33H31N3O6
[(S)-[3-[[3-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid
—— (S)-tert-butyl 2-((7-(3,4-dimethoxyphenyl)pyrido[4,3-b]pyrazin-5-yloxy)methyl)morpholine-4-carboxylate —— C25H30N4O6
(S)-tert-butyl 2-((7-(3,4-dimethoxyphenyl)pyrido[4,3-b]pyrazin-5-yloxy)methyl)morpholine-4-carboxylate
—— [(S)-[3-[[4-[[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]phenyl]methylcarbamoyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C41H38N4O7
[(S)-[3-[[4-[[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]phenyl]methylcarbamoyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid
—— (S)-N-(5-fluoro-3-((4-(3-fluoro-3-methylcyclobutanecarbonyl)-3-methylpiperazin-1-yl)methyl)-2-methylphenyl)-6-methylnicotinamide —— C26H32F2N4O2
(S)-N-(5-fluoro-3-((4-(3-fluoro-3-methylcyclobutanecarbonyl)-3-methylpiperazin-1-yl)methyl)-2-methylphenyl)-6-methylnicotinamide
—— [(S)-[3-[[5-[4-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]butylcarbamoyl]-2-methylpyrazol-3-yl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C35H38N6O7
[(S)-[3-[[5-[4-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]butylcarbamoyl]-2-methylpyrazol-3-yl]methoxy]phenyl]-phenylmethyl]carbamic acid
—— S-(3-methoxy-2-nitrophenyl)thiohydroxylamine —— C7H8N2O3S
S-(3-methoxy-2-nitrophenyl)thiohydroxylamine
—— [(S)-[3-[[4-[(4-chlorophenyl)methyl-[3-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]propyl]carbamoyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C43H41ClN4O7
[(S)-[3-[[4-[(4-chlorophenyl)methyl-[3-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]propyl]carbamoyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid
—— [(S)-[3-[[4-[(4-fluorophenyl)methyl-[3-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]propyl]carbamoyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C43H41FN4O7
[(S)-[3-[[4-[(4-fluorophenyl)methyl-[3-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]propyl]carbamoyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid
—— sodium;5-[2-(2,3,4-trimethoxyanilino)ethyl]-1H-1,2,4-triazole-3-carboxylate —— C14H17N4NaO5
sodium;5-[2-(2,3,4-trimethoxyanilino)ethyl]-1H-1,2,4-triazole-3-carboxylate
—— ((S)-2-(((7-chloropyrido[3,4-b]pyrazin-5-yl)oxy)methyl)morpholino)((S)-pyrrolidin-3-yl)methanone 1613260-21-1 C17H20ClN5O3
((S)-2-(((7-chloropyrido[3,4-b]pyrazin-5-yl)oxy)methyl)morpholino)((S)-pyrrolidin-3-yl)methanone
—— [(S)-[3-[[4-[3-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]propyl-[(3-methoxyphenyl)methyl]carbamoyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C44H44N4O8
[(S)-[3-[[4-[3-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]propyl-[(3-methoxyphenyl)methyl]carbamoyl]phenyl]methoxy]phenyl]-phenylmethyl]carbamic acid
—— [(S)-[3-[[1-(4-formylbenzoyl)piperidin-4-yl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C28H28N2O5
[(S)-[3-[[1-(4-formylbenzoyl)piperidin-4-yl]methoxy]phenyl]-phenylmethyl]carbamic acid
—— S-[carbamoyl(pentyl)amino] 4-ethoxybenzenecarbothioate —— C15H22N2O3S
S-[carbamoyl(pentyl)amino] 4-ethoxybenzenecarbothioate
—— (S)-N-(3-((4-(3,3-dimethylcyclobutanecarbonyl)-3-methylpiperazin-1-yl)methyl)-5-fluoro-2-methylphenyl)-6-methylnicotinamide —— C27H35FN4O2
(S)-N-(3-((4-(3,3-dimethylcyclobutanecarbonyl)-3-methylpiperazin-1-yl)methyl)-5-fluoro-2-methylphenyl)-6-methylnicotinamide
—— [(S)-[3-[2-[2-chloro-4-[[[2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-5-methoxyanilino]-2-oxoethoxy]phenyl]-phenylmethyl]carbamic acid —— C35H33ClN4O8
[(S)-[3-[2-[2-chloro-4-[[[2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-5-methoxyanilino]-2-oxoethoxy]phenyl]-phenylmethyl]carbamic acid
—— [(S)-[3-[[4-[3-(1,3-dioxolan-2-ylmethyl)benzoyl]piperidin-4-yl]methoxy]phenyl]-phenylmethyl]carbamic acid —— C31H34N2O6
[(S)-[3-[[4-[3-(1,3-dioxolan-2-ylmethyl)benzoyl]piperidin-4-yl]methoxy]phenyl]-phenylmethyl]carbamic acid