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—— (S)-4'-(3-amino-2-(4-(tert-butoxycarbonylamino)tetrahydro-2H-pyran-4-carboxamido)-3-oxopropyl)biphenyl-3-yl methanesulfonate 1254319-19-1 C27H35N3O8S
(S)-4'-(3-amino-2-(4-(tert-butoxycarbonylamino)tetrahydro-2H-pyran-4-carboxamido)-3-oxopropyl)biphenyl-3-yl methanesulfonate
—— (S)-tert-butyl 4-(1-amino-3-(4-(4-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]thiazin-7-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-47-5 C29H36N4O6S
(S)-tert-butyl 4-(1-amino-3-(4-(4-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]thiazin-7-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-amino-3-(4-(3-(3-methoxypropyl)-2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-17-9 C31H40N4O8
(S)-tert-butyl 4-(1-amino-3-(4-(3-(3-methoxypropyl)-2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-cyano-2-(4-(1-methyl-2-oxoindolin-6-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-35-1 C29H34N4O5
(S)-tert-butyl 4-(1-cyano-2-(4-(1-methyl-2-oxoindolin-6-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-cyano-2-(4-(3-(2-methoxyethyl)-2-oxo-2,3-dihydrobenzo[d]thiazol-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-12-4 C30H36N4O6S
(S)-tert-butyl 4-(1-cyano-2-(4-(3-(2-methoxyethyl)-2-oxo-2,3-dihydrobenzo[d]thiazol-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-cyano-2-(3'-cyano-4'-methylbiphenyl-4-yl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-30-6 C28H32N4O4
(S)-tert-butyl 4-(1-cyano-2-(3'-cyano-4'-methylbiphenyl-4-yl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-amino-3-(4-(2-methyl-1-oxoisoindolin-5-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-53-3 C29H36N4O6
(S)-tert-butyl 4-(1-amino-3-(4-(2-methyl-1-oxoisoindolin-5-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 1-(1-cyano-2-(4-(6-methyl-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-3-yl)phenyl)ethylcarbamoyl)cyclohexylcarbamate 1254319-57-7 C28H33N5O5
(S)-tert-butyl 1-(1-cyano-2-(4-(6-methyl-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-3-yl)phenyl)ethylcarbamoyl)cyclohexylcarbamate
—— (S)-2-tert-butoxycarbonylamino-3-(4-{(R)-4-[1-(5-chloropyrimidin-2-yl)-piperidin-4-yl]pent-1-ynyl}-2-fluorophenyl)propionic acid methyl ester 1131872-63-3 C29H36ClFN4O4
(S)-2-tert-butoxycarbonylamino-3-(4-{(R)-4-[1-(5-chloropyrimidin-2-yl)-piperidin-4-yl]pent-1-ynyl}-2-fluorophenyl)propionic acid methyl ester
—— (S)-3-(tert-butyl-dimethyl-silanyloxy)-2-(8-carbamoyl-4-oxo-imidazo[5,1-d][1,2,3,5]tetrazin-3-yl)-2-methyl-propionic acid methyl ester 1161826-11-4 C16H26N6O5Si
(S)-3-(tert-butyl-dimethyl-silanyloxy)-2-(8-carbamoyl-4-oxo-imidazo[5,1-d][1,2,3,5]tetrazin-3-yl)-2-methyl-propionic acid methyl ester
—— [(S)-1-(4-{3-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)piperidin-4-yl]propoxy}-benzyl)-2-oxo-2-pyrrolidin-1-ylethyl]carbamic acid tert-butyl ester 1131870-77-3 C31H47N5O5
[(S)-1-(4-{3-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)piperidin-4-yl]propoxy}-benzyl)-2-oxo-2-pyrrolidin-1-ylethyl]carbamic acid tert-butyl ester
—— (S)-4'-(2-(4-aminotetrahydro-2H-pyran-4-carboxamido)-2-cyanoethyl)biphenyl-4-ylmethanesulfonate 1254318-47-2 C22H25N3O5S
(S)-4'-(2-(4-aminotetrahydro-2H-pyran-4-carboxamido)-2-cyanoethyl)biphenyl-4-ylmethanesulfonate
—— (S)-tert-butyl 4-(1-cyano-2-(4'-(trifluoromethyl)biphenyl-4-yl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254318-94-9 C27H30F3N3O4
(S)-tert-butyl 4-(1-cyano-2-(4'-(trifluoromethyl)biphenyl-4-yl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-amino-3-(4-(3-(2-methoxyethyl)-2-oxo-2,3-dihydrobenzo[d]thiazol-5-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-11-3 C30H38N4O7S
(S)-tert-butyl 4-(1-amino-3-(4-(3-(2-methoxyethyl)-2-oxo-2,3-dihydrobenzo[d]thiazol-5-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-amino-3-(4-(3-(2-methoxyethyl)-2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)-1-oxopropan-2-ylcarbalnoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-40-8 C30H38N4O8
(S)-tert-butyl 4-(1-amino-3-(4-(3-(2-methoxyethyl)-2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)-1-oxopropan-2-ylcarbalnoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(2-(4'-carbamoyl-3'-fluorobiphenyl-4-yl)-1-cyanoethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-42-0 C27H31FN4O5
(S)-tert-butyl 4-(2-(4'-carbamoyl-3'-fluorobiphenyl-4-yl)-1-cyanoethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-cyano-2-(4-(1-oxoisoindolin-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-23-7 C28H32N4O5
(S)-tert-butyl 4-(1-cyano-2-(4-(1-oxoisoindolin-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 3-(piperidin-1-ylmethyl)piperidine-1-carboxylate 1100155-50-7 C16H30N2O2
(S)-tert-butyl 3-(piperidin-1-ylmethyl)piperidine-1-carboxylate
—— (S)-tert-butyl 4-(1-cyano-2-(4-(2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-59-9 C27H30N4O6
(S)-tert-butyl 4-(1-cyano-2-(4-(2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-4'-(2-(4-(tert-butoxycarbonylamino)tetrahydro-2H-pyran-4-carboxamido)-2-cyanoethyl)biphenyl-4-yl methanesulfonate 1254319-05-5 C27H33N3O7S
(S)-4'-(2-(4-(tert-butoxycarbonylamino)tetrahydro-2H-pyran-4-carboxamido)-2-cyanoethyl)biphenyl-4-yl methanesulfonate
—— (S)-tert-butyl 4-(1-cyano-2-(4-(2-methyl-1-oxoisoindolin-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-54-4 C29H34N4O5
(S)-tert-butyl 4-(1-cyano-2-(4-(2-methyl-1-oxoisoindolin-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-cyano-2-(4'-(4-methylpiperazin-1-ylsulfonyl)biphenyl-4-yl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-50-0 C31H41N5O6S
(S)-tert-butyl 4-(1-cyano-2-(4'-(4-methylpiperazin-1-ylsulfonyl)biphenyl-4-yl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-amino-1-oxo-3-(4'-(trifluoromethyl)biphenyl-4-yl)propan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254318-92-7 C27H32F3N3O5
(S)-tert-butyl 4-(1-amino-1-oxo-3-(4'-(trifluoromethyl)biphenyl-4-yl)propan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-Butyl 4-(1-cyano-2-(4-(3-(3-methoxypropyl)-2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-18-0 C31H38N4O7
(S)-tert-Butyl 4-(1-cyano-2-(4-(3-(3-methoxypropyl)-2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-2-((R)-2-(4-fluorophenyl)-2-methoxyethyl)-N-hydroxyhexanamide 1100154-94-6 C15H22FNO3
(S)-2-((R)-2-(4-fluorophenyl)-2-methoxyethyl)-N-hydroxyhexanamide
—— (S)-tert-butyl 4-(1-cyano-2-(4-(3-methyl-2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-28-2 C28H32N4O6
(S)-tert-butyl 4-(1-cyano-2-(4-(3-methyl-2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-cyano-2-(4-(4-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]thiazin-7-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-48-6 C29H34N4O5S
(S)-tert-butyl 4-(1-cyano-2-(4-(4-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]thiazin-7-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-amino-3-(4'-fluorobiphenyl-4-yl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-00-0 C26H32FN3O5
(S)-tert-butyl 4-(1-amino-3-(4'-fluorobiphenyl-4-yl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-amino-3-(4'-(4-methylpiperazin-1-ylsulfonyl)biphenyl-4-yl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-49-7 C31H43N5O7S
(S)-tert-butyl 4-(1-amino-3-(4'-(4-methylpiperazin-1-ylsulfonyl)biphenyl-4-yl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-amino-3-(4'-(ethylsulfonyl)biphenyl-4-yl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254318-93-8 C28H37N3O7S
(S)-tert-butyl 4-(1-amino-3-(4'-(ethylsulfonyl)biphenyl-4-yl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-cyano-2-(4-(4-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-14-6 C29H34N4O6
(S)-tert-butyl 4-(1-cyano-2-(4-(4-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)phenyl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-cyano-2-(4'-(morpholinosulfonyl)biphenyl-4-yl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-45-3 C30H38N4O7S
(S)-tert-butyl 4-(1-cyano-2-(4'-(morpholinosulfonyl)biphenyl-4-yl)ethylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-tert-butyl 4-(1-amino-3-(4-(4-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate 1254319-13-5 C29H36N4O7
(S)-tert-butyl 4-(1-amino-3-(4-(4-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)phenyl)-1-oxopropan-2-ylcarbamoyl)tetrahydro-2H-pyran-4-ylcarbamate
—— (S)-2-((R)-2-(4-fluorophenyl)-2-hydroxyethyl)hexanoic acid 1100154-88-8 C14H19FO3
(S)-2-((R)-2-(4-fluorophenyl)-2-hydroxyethyl)hexanoic acid
—— (S)-4-(3-hydroxy-2-oxopyrrolidin-1-yl)-N-(thiazol-2-yl)benzenesulfonamide 1203587-11-4 C13H13N3O4S2
(S)-4-(3-hydroxy-2-oxopyrrolidin-1-yl)-N-(thiazol-2-yl)benzenesulfonamide
—— (S)-tert-butyl 2-(5-formyl-1-{{2-(trimethylsilyl)ethoxy}methyl}-1H-imidazol-2-yl)pyrrolidine-1-carboxylate 1251998-80-7 C19H33N3O4Si
(S)-tert-butyl 2-(5-formyl-1-{{2-(trimethylsilyl)ethoxy}methyl}-1H-imidazol-2-yl)pyrrolidine-1-carboxylate
—— (S)-3-((S)-2-(benzyloxy)-2,2-d2-1-hydroxyethyl)-4,4,5,5-d4-dihydrofuran-2(3H)-one 1254047-66-9 C13H16O4
(S)-3-((S)-2-(benzyloxy)-2,2-d2-1-hydroxyethyl)-4,4,5,5-d4-dihydrofuran-2(3H)-one
—— (S,S)-3,9-bis(2-(pyrrolidin-2-yl)-3H-imidazol-4-yl)-5,7-dihydrodibenzo[c,e]oxepine 1256384-26-5 C28H30N6O
(S,S)-3,9-bis(2-(pyrrolidin-2-yl)-3H-imidazol-4-yl)-5,7-dihydrodibenzo[c,e]oxepine
—— (S)-2-(1-((2-(2-ethyl-1H-benzo[d]imidazol-1-yl)-9-methyl-6-(3-methylmorpholino)-9H-purin-8-yl)methyl)piperidin-4-yl)propan-2-ol 1257384-97-6 C29H40N8O2
(S)-2-(1-((2-(2-ethyl-1H-benzo[d]imidazol-1-yl)-9-methyl-6-(3-methylmorpholino)-9H-purin-8-yl)methyl)piperidin-4-yl)propan-2-ol
—— (S)-4-(2-(1-tert-butoxycarbonylpyrrolidin-2-yl)-3H-imidazol-4-yl)piperidine-1-carboxylic acid benzyl ester 1256386-49-8 C25H34N4O4
(S)-4-(2-(1-tert-butoxycarbonylpyrrolidin-2-yl)-3H-imidazol-4-yl)piperidine-1-carboxylic acid benzyl ester
—— (S)-2-tert-butoxycarbonylamino-4-(4-chloro-phenyl)-butyric acid 157683-99-3 C15H20ClNO4
(S)-2-tert-butoxycarbonylamino-4-(4-chloro-phenyl)-butyric acid
—— (S)-2-tert-butoxycarbonylamino-4-(4-chloro-phenyl)-butyric acid methyl ester 1257614-37-1 C16H22ClNO4
(S)-2-tert-butoxycarbonylamino-4-(4-chloro-phenyl)-butyric acid methyl ester
—— (S)-4-(2-(1-tert-butoxycarbonylpyrrolidin-2-yl)-3-(2-trimethylsilanylethoxymethyl)-3H-imidazol-4-yl)piperidine-1-carboxylic acid benzyl ester 1256386-50-1 C31H48N4O5Si
(S)-4-(2-(1-tert-butoxycarbonylpyrrolidin-2-yl)-3-(2-trimethylsilanylethoxymethyl)-3H-imidazol-4-yl)piperidine-1-carboxylic acid benzyl ester
—— (S)-(1-(2-(5-(4'-(2-(3-amino-2-oxopiperidin-1-ylmethyl)-3H-imidazol-4-yl)biphenyl-4-yl)-1H-imidazol-2-yl)pyrrolidine-1-carbonyl)-2-methylpropyl)carbamic acid methyl ester 1256385-99-5 C35H42N8O4
(S)-(1-(2-(5-(4'-(2-(3-amino-2-oxopiperidin-1-ylmethyl)-3H-imidazol-4-yl)biphenyl-4-yl)-1H-imidazol-2-yl)pyrrolidine-1-carbonyl)-2-methylpropyl)carbamic acid methyl ester
—— (S)-tert-butyl 2-benzyl-3-((3R,4R)-4-(3-carbamoylphenyl)-3,4-dimethylpiperidin-1-yl)propanoate 1257642-52-6 C28H38N2O3
(S)-tert-butyl 2-benzyl-3-((3R,4R)-4-(3-carbamoylphenyl)-3,4-dimethylpiperidin-1-yl)propanoate
—— [(S)-1-(2-cyclohexyl-ethyl)-2-hydroxy-propyl]-carbamic acid tert-butyl ester 1257614-29-1 C16H31NO3
[(S)-1-(2-cyclohexyl-ethyl)-2-hydroxy-propyl]-carbamic acid tert-butyl ester
—— (S)-1-((S)-1-(4-bromophenyl)ethyl)-4-(2-hydroxy-2-methylpropyl)-4-phenyltetrahydropyrimidin-2(1H)-one 1151796-50-7 C22H27BrN2O2
(S)-1-((S)-1-(4-bromophenyl)ethyl)-4-(2-hydroxy-2-methylpropyl)-4-phenyltetrahydropyrimidin-2(1H)-one
—— (S)-3-[(5-chloro-thiophen-2-yl)-carbonylamino]-N-((R)-3,5-dimethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-tetrahydro-furan-3-carboxylic acid amide 1037301-39-5 C22H26ClN3O3S
(S)-3-[(5-chloro-thiophen-2-yl)-carbonylamino]-N-((R)-3,5-dimethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-tetrahydro-furan-3-carboxylic acid amide
—— (S)-1-((S)-1-(2',4'-difluorobiphenyl-4-yl)ethyl)-4-(4-fluorophenyl)-4-(2-hydroxyethyl)tetrahydropyrimidin-2(1H)-one 1151796-23-4 C26H25F3N2O2
(S)-1-((S)-1-(2',4'-difluorobiphenyl-4-yl)ethyl)-4-(4-fluorophenyl)-4-(2-hydroxyethyl)tetrahydropyrimidin-2(1H)-one
—— (S)-3-[(5-chloro-thiophene-2-carbonyl)-amino]-tetrahydro-furan-3-carboxylic acid ((S)-3,5-dimethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 1037301-25-9 C22H26ClN3O3S
(S)-3-[(5-chloro-thiophene-2-carbonyl)-amino]-tetrahydro-furan-3-carboxylic acid ((S)-3,5-dimethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide