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—— (7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5OS
(7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-chlorophenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26ClN5OS
(7R)-2-benzylsulfanyl-7-(4-chlorophenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(4-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25F2N5OS
(7R)-N-(2,3-dimethylphenyl)-7-(4-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-tert-butylphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C31H33N5OS
(7S)-2-benzylsulfanyl-7-(4-tert-butylphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-(dimethylamino)phenyl]-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29FN6OS
(7S)-7-[4-(dimethylamino)phenyl]-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-5-methyl-N-phenyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2S
(7R)-2-benzylsulfanyl-5-methyl-N-phenyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26FN5OS
(7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5OS
(7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5OS
(7S)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24FN5OS
(7S)-2-benzylsulfanyl-7-(4-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-ethoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2S
(7R)-2-benzylsulfanyl-7-(4-ethoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-N-(2-ethoxyphenyl)-7-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O3S
(7R)-2-benzylsulfanyl-N-(2-ethoxyphenyl)-7-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-5-methyl-N-(3-methylphenyl)-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O2S
(7R)-2-benzylsulfanyl-5-methyl-N-(3-methylphenyl)-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H30N6OS
(7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-5-methyl-N-(3-methylphenyl)-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O2S
(7R)-2-benzylsulfanyl-5-methyl-N-(3-methylphenyl)-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-N-(2-ethoxyphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O2S
(7S)-2-benzylsulfanyl-N-(2-ethoxyphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H30N6O2S
(7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-5-methyl-7-(4-propan-2-ylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C31H33N5OS
(7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-5-methyl-7-(4-propan-2-ylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5OS
(7S)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-chlorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24ClN5OS
(7S)-2-benzylsulfanyl-7-(4-chlorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26FN5OS
(7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H24FN5OS2
(7S)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26FN5OS
(7R)-N-(2,4-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-N-(2-ethoxyphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O2S
(7R)-2-benzylsulfanyl-N-(2-ethoxyphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26FN5O2S
(7R)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-5-methyl-N-(2-methylphenyl)-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O2S
(7S)-2-benzylsulfanyl-5-methyl-N-(2-methylphenyl)-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-(dimethylamino)phenyl]-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29FN6OS
(7S)-7-[4-(dimethylamino)phenyl]-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24FN5OS
(7R)-2-benzylsulfanyl-7-(4-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-chlorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClFN5OS
(7S)-7-(4-chlorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H30FN5OS
(7S)-N-(2,3-dimethylphenyl)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O2S
(7R)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2S
(7S)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28FN5OS
(7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-5-methyl-N-(3-methylphenyl)-7-(4-propan-2-ylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5OS
(7S)-2-benzylsulfanyl-5-methyl-N-(3-methylphenyl)-7-(4-propan-2-ylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H30N6OS
(7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-methyl-6,6a,8,9,10,10a-hexahydro-4H-indolo[4,3-fg]quinoline —— C15H18N2
7-methyl-6,6a,8,9,10,10a-hexahydro-4H-indolo[4,3-fg]quinoline
—— (7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28FN5OS
(7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23F2N5OS
(7S)-7-(4-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H30FN5OS
(7S)-N-(2,4-dimethylphenyl)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26FN5OS
(7S)-2-benzylsulfanyl-N-(2,3-dimethylphenyl)-7-(4-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-fluoro-2-methyl-N-[[6-(2-methylimidazol-1-yl)pyridin-3-yl]methyl]quinoline-4-carboxamide —— C21H18FN5O
7-fluoro-2-methyl-N-[[6-(2-methylimidazol-1-yl)pyridin-3-yl]methyl]quinoline-4-carboxamide
—— (7R)-2-[(2-chlorophenyl)methylsulfanyl]-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClFN5OS
(7R)-2-[(2-chlorophenyl)methylsulfanyl]-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26ClN5OS
(7S)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-(3,5-dichloroanilino)-pyridin-4-ylmethyl]-2-methylquinolin-8-ol —— C22H17Cl2N3O
7-[(R)-(3,5-dichloroanilino)-pyridin-4-ylmethyl]-2-methylquinolin-8-ol
—— 7-[(R)-(2-methyl-4-nitroanilino)-pyridin-4-ylmethyl]quinolin-8-ol —— C22H18N4O3
7-[(R)-(2-methyl-4-nitroanilino)-pyridin-4-ylmethyl]quinolin-8-ol
—— 7-[(R)-(4-chloro-2-methylanilino)-thiophen-2-ylmethyl]-2-methylquinolin-8-ol —— C22H19ClN2OS
7-[(R)-(4-chloro-2-methylanilino)-thiophen-2-ylmethyl]-2-methylquinolin-8-ol
—— (7R)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24ClN5OS
(7R)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-(2,4-dichloroanilino)-(4-fluorophenyl)methyl]-2-methylquinolin-8-ol —— C23H17Cl2FN2O
7-[(R)-(2,4-dichloroanilino)-(4-fluorophenyl)methyl]-2-methylquinolin-8-ol
—— 7-[(R)-(3,4-dichloroanilino)-(furan-2-yl)methyl]-2-methylquinolin-8-ol —— C21H16Cl2N2O2
7-[(R)-(3,4-dichloroanilino)-(furan-2-yl)methyl]-2-methylquinolin-8-ol
—— 7-[(S)-furan-2-yl-(2-methoxy-5-methylanilino)methyl]quinolin-8-ol —— C22H20N2O3
7-[(S)-furan-2-yl-(2-methoxy-5-methylanilino)methyl]quinolin-8-ol