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—— (6E)-6-{[5-(4-chlorophenyl)furan-2-yl]methylidene}-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C18H13ClN4O2S
(6E)-6-{[5-(4-chlorophenyl)furan-2-yl]methylidene}-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[(5-bromofuran-2-yl)methylidene]-3-(4-fluorophenyl)-5-imino-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C17H9BrFN3O2S
(6Z)-6-[(5-bromofuran-2-yl)methylidene]-3-(4-fluorophenyl)-5-imino-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C18H15ClN6OS
(6Z)-6-[(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[4-(dimethylamino)phenyl]methylidene]-5-imino-2-(phenoxymethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H19N5O2S
(6E)-6-[[4-(dimethylamino)phenyl]methylidene]-5-imino-2-(phenoxymethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-5-imino-6-(1H-indol-3-ylmethylidene)-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H15N5O2S
(6E)-5-imino-6-(1H-indol-3-ylmethylidene)-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-(1,3-benzodioxol-5-ylmethylidene)-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H14N4O4S
(6Z)-6-(1,3-benzodioxol-5-ylmethylidene)-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-chloro-N-[(1R,2S)-2-cyanocyclopentyl]pyridazine-3-carboxamide —— C11H11ClN4O
6-chloro-N-[(1R,2S)-2-cyanocyclopentyl]pyridazine-3-carboxamide
—— 6-chloro-N-[(1S,2R)-2-cyanocyclopentyl]pyridine-3-sulfonamide —— C11H12ClN3O2S
6-chloro-N-[(1S,2R)-2-cyanocyclopentyl]pyridine-3-sulfonamide
—— 6-chloro-N-[(1R,2R)-2-cyanocyclopentyl]pyridazine-3-carboxamide —— C11H11ClN4O
6-chloro-N-[(1R,2R)-2-cyanocyclopentyl]pyridazine-3-carboxamide
—— 6-bromo-N-[(Z)-(2,4-dimethoxyphenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C18H17BrN4O3
6-bromo-N-[(Z)-(2,4-dimethoxyphenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— 6-chloro-N-[(1S,2S)-2-cyanocyclopentyl]pyridine-3-sulfonamide —— C11H12ClN3O2S
6-chloro-N-[(1S,2S)-2-cyanocyclopentyl]pyridine-3-sulfonamide
—— 6-bromo-N-[(Z)-(4-ethoxyphenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C18H17BrN4O2
6-bromo-N-[(Z)-(4-ethoxyphenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— 6-[[(1R,2S)-2-cyanocyclopentyl]amino]-6-oxohexanoic acid —— C12H18N2O3
6-[[(1R,2S)-2-cyanocyclopentyl]amino]-6-oxohexanoic acid
—— 6-methyl-N-[(Z)-[5-[[(4-methylphenyl)methyl-(4-methylphenyl)sulfonylamino]methyl]furan-2-yl]methylideneamino]imidazo[2,1-b][1,3]thiazole-5-carboxamide —— C28H27N5O4S2
6-methyl-N-[(Z)-[5-[[(4-methylphenyl)methyl-(4-methylphenyl)sulfonylamino]methyl]furan-2-yl]methylideneamino]imidazo[2,1-b][1,3]thiazole-5-carboxamide
—— 6-chloro-N-[(1S,2S)-2-cyanocyclopentyl]pyridazine-3-carboxamide —— C11H11ClN4O
6-chloro-N-[(1S,2S)-2-cyanocyclopentyl]pyridazine-3-carboxamide
—— 6-[[(1S,2S)-2-cyanocyclopentyl]amino]-6-oxohexanoic acid —— C12H18N2O3
6-[[(1S,2S)-2-cyanocyclopentyl]amino]-6-oxohexanoic acid
—— 6-[[(1S,2R)-2-cyanocyclopentyl]amino]-6-oxohexanoic acid —— C12H18N2O3
6-[[(1S,2R)-2-cyanocyclopentyl]amino]-6-oxohexanoic acid
—— 6-[[(1R,2R)-2-cyanocyclopentyl]amino]-6-oxohexanoic acid —— C12H18N2O3
6-[[(1R,2R)-2-cyanocyclopentyl]amino]-6-oxohexanoic acid
—— 6-chloro-N-[(1S,2R)-2-cyanocyclopentyl]pyridazine-3-carboxamide —— C11H11ClN4O
6-chloro-N-[(1S,2R)-2-cyanocyclopentyl]pyridazine-3-carboxamide
—— 6-chloro-N-[(1R,2S)-2-cyanocyclopentyl]pyridine-3-sulfonamide —— C11H12ClN3O2S
6-chloro-N-[(1R,2S)-2-cyanocyclopentyl]pyridine-3-sulfonamide
—— 6-chloro-N-[(1R,2R)-2-cyanocyclopentyl]pyridine-3-sulfonamide —— C11H12ClN3O2S
6-chloro-N-[(1R,2R)-2-cyanocyclopentyl]pyridine-3-sulfonamide
—— (6S,7S,8S)-7-methyl-N-(2-phenylethyl)-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine —— C28H31NO6
(6S,7S,8S)-7-methyl-N-(2-phenylethyl)-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine
—— (6S,7R,8R)-7-methyl-N-(2-phenylethyl)-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine —— C28H31NO6
(6S,7R,8R)-7-methyl-N-(2-phenylethyl)-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine
—— (6S,7S,8R)-N-benzyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine —— C27H29NO6
(6S,7S,8R)-N-benzyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine
—— (6R,7R,8R)-N,N-diethyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine —— C24H31NO6
(6R,7R,8R)-N,N-diethyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine
—— (6S,7R,8R)-N-benzyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine —— C27H29NO6
(6S,7R,8R)-N-benzyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine
—— (6S,7S,8R)-7-methyl-N-(2-phenylethyl)-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine —— C28H31NO6
(6S,7S,8R)-7-methyl-N-(2-phenylethyl)-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine
—— (6S,7S,8S)-N-benzyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine —— C27H29NO6
(6S,7S,8S)-N-benzyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine
—— (6S,7R,8R)-N,N-diethyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine —— C24H31NO6
(6S,7R,8R)-N,N-diethyl-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-amine
—— (6R)-N-[(Z)-1,3-benzodioxol-5-ylmethylideneamino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C21H24N2O3S
(6R)-N-[(Z)-1,3-benzodioxol-5-ylmethylideneamino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-N-[(Z)-1,3-benzodioxol-5-ylmethylideneamino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C21H24N2O3S
(6S)-N-[(Z)-1,3-benzodioxol-5-ylmethylideneamino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-6-tert-butyl-N-[(Z)-(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C21H23N3O5S
(6R)-6-tert-butyl-N-[(Z)-(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-chloro-N'-[(Z)-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-2-methylimidazo[1,2-a]pyridine-3-carbohydrazide —— C17H15ClN4O3
6-chloro-N'-[(Z)-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-2-methylimidazo[1,2-a]pyridine-3-carbohydrazide
—— (6E)-2,4-dibromo-6-[[(5-methyl-1,3,4-thiadiazol-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C10H7Br2N3OS
(6E)-2,4-dibromo-6-[[(5-methyl-1,3,4-thiadiazol-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6,7-dimethyl-2-[4-(4-morpholinyl)benzylidene][1,3]thiazolo[3,2-a]benzimidazol-3(2H)-one —— C22H21N3O2S
6,7-dimethyl-2-[4-(4-morpholinyl)benzylidene][1,3]thiazolo[3,2-a]benzimidazol-3(2H)-one
—— (6S)-6-tert-butyl-N-[(Z)-(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C21H23N3O5S
(6S)-6-tert-butyl-N-[(Z)-(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(2S,6S)-2,6-diphenyl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one —— C22H20N2O
6-[(2S,6S)-2,6-diphenyl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(2R,6S)-2,6-diphenyl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one —— C22H20N2O
6-[(2R,6S)-2,6-diphenyl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(2S,6R)-2,6-diphenyl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one —— C22H20N2O
6-[(2S,6R)-2,6-diphenyl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-6-[[4-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H21FN4O3S
(6Z)-6-[[4-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-{4-[(4-fluorobenzyl)oxy]-3-methoxybenzylidene}-5-imino-2-isopropyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H21FN4O3S
6-{4-[(4-fluorobenzyl)oxy]-3-methoxybenzylidene}-5-imino-2-isopropyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-5-imino-6-[(5-phenylfuran-2-yl)methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C19H16N4O2S
(6E)-5-imino-6-[(5-phenylfuran-2-yl)methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(2R,6R)-2,6-diphenyl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one —— C22H20N2O
6-[(2R,6R)-2,6-diphenyl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one
—— (6E)-6-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C19H15ClN4O2S
(6E)-6-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-5-imino-2-propyl-6-[(3,4,5-trimethoxyphenyl)methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C18H20N4O4S
(6Z)-5-imino-2-propyl-6-[(3,4,5-trimethoxyphenyl)methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[(3-bromophenyl)methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C15H13BrN4OS
(6Z)-6-[(3-bromophenyl)methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-chloro-2-methyl-N'-[(Z)-(2-oxonaphthalen-1-ylidene)methyl]imidazo[1,2-a]pyridine-3-carbohydrazide —— C20H15ClN4O2
6-chloro-2-methyl-N'-[(Z)-(2-oxonaphthalen-1-ylidene)methyl]imidazo[1,2-a]pyridine-3-carbohydrazide
—— (6E)-6-[[1-(1,3-benzodioxol-5-ylmethyl)indol-3-yl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H19N5O3S
(6E)-6-[[1-(1,3-benzodioxol-5-ylmethyl)indol-3-yl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[5-(4-fluorophenyl)furan-2-yl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C19H15FN4O2S
(6E)-6-[[5-(4-fluorophenyl)furan-2-yl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-5-imino-6-({1-[2-(3-methoxyphenoxy)ethyl]-1H-indol-3-yl}methylidene)-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H25N5O3S
(6E)-5-imino-6-({1-[2-(3-methoxyphenoxy)ethyl]-1H-indol-3-yl}methylidene)-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one