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—— 6-[4-[3-[(4R,6S)-2-amino-4-methyl-6-(trifluoromethyl)-5,6-dihydro-1,3-oxazin-4-yl]-4-fluorophenyl]triazol-1-yl]pyridine-3-carbonitrile —— C20H15F4N7O
6-[4-[3-[(4R,6S)-2-amino-4-methyl-6-(trifluoromethyl)-5,6-dihydro-1,3-oxazin-4-yl]-4-fluorophenyl]triazol-1-yl]pyridine-3-carbonitrile
—— (6E)-4-[[4-(2,4-dinitrophenoxy)phenyl]methylideneamino]-6-(5-methyl-3H-1,3-benzoxazol-2-ylidene)cyclohexa-2,4-dien-1-one —— C27H18N4O7
(6E)-4-[[4-(2,4-dinitrophenoxy)phenyl]methylideneamino]-6-(5-methyl-3H-1,3-benzoxazol-2-ylidene)cyclohexa-2,4-dien-1-one
—— 6-[(4-Fluorophenyl)methyl]-3-methoxy-2-(3-methylphenyl)aniline —— C21H20FNO
6-[(4-Fluorophenyl)methyl]-3-methoxy-2-(3-methylphenyl)aniline
—— (6E)-6-[[4-[(1S,2S)-2-(dimethylamino)-1,3-dihydroxypropyl]anilino]methylidene]cyclohexa-2,4-dien-1-one —— C18H22N2O3
(6E)-6-[[4-[(1S,2S)-2-(dimethylamino)-1,3-dihydroxypropyl]anilino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-(ethylsulfonylamino)-5-[15-fluoro-9-(2-hydroxyethyl)-8-oxa-3,10-diazatetracyclo[8.7.0.02,7.011,16]heptadeca-1(17),2(7),3,5,11(16),12,14-heptaen-4-yl]-2-(4-fluorophenyl)-N-methyl-1-benzofuran-3-carboxamide —— C34H28F2N4O6S
6-(ethylsulfonylamino)-5-[15-fluoro-9-(2-hydroxyethyl)-8-oxa-3,10-diazatetracyclo[8.7.0.02,7.011,16]heptadeca-1(17),2(7),3,5,11(16),12,14-heptaen-4-yl]-2-(4-fluorophenyl)-N-methyl-1-benzofuran-3-carboxamide
—— 6-Methoxy-1-oxo-3-pyridin-3-yl-2,9-dihydropyrrolo[2,3-h]isoquinoline-4-carbonitrile —— C18H12N4O2
6-Methoxy-1-oxo-3-pyridin-3-yl-2,9-dihydropyrrolo[2,3-h]isoquinoline-4-carbonitrile
—— (6S)-N-[(2-bromo-4,6-dichlorophenyl)methyl]-5,6-dihydrofuro[2,3-d][1,3]thiazole-6-carboxamide —— C13H9BrCl2N2O2S
(6S)-N-[(2-bromo-4,6-dichlorophenyl)methyl]-5,6-dihydrofuro[2,3-d][1,3]thiazole-6-carboxamide
—— 6,7-dichloro-3,5-dihydro-1H-imidazo[2,1-b]quinazolin-2-one;[(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-piperidin-1-ylpiperidine-1-carboxylate;4-[(2S)-2-(3,5-dioxopiperazin-1-yl)propyl]piperazine-2,6-dione —— C54H61Cl2N11O11
6,7-dichloro-3,5-dihydro-1H-imidazo[2,1-b]quinazolin-2-one;[(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-piperidin-1-ylpiperidine-1-carboxylate;4-[(2S)-2-(3,5-dioxopiperazin-1-yl)propyl]piperazine-2,6-dione
—— 6-[2-[5-[(4R,6S)-2-[[bis(4-methoxyphenyl)-phenylmethyl]amino]-4-methyl-6-(trifluoromethyl)-5,6-dihydro-1,3-oxazin-4-yl]thiophen-3-yl]ethynyl]pyridine-3-carbonitrile —— C39H31F3N4O3S
6-[2-[5-[(4R,6S)-2-[[bis(4-methoxyphenyl)-phenylmethyl]amino]-4-methyl-6-(trifluoromethyl)-5,6-dihydro-1,3-oxazin-4-yl]thiophen-3-yl]ethynyl]pyridine-3-carbonitrile
—— 6-(Ethylsulfonylamino)-5-(15-fluoro-8-oxa-3,10-diazatetracyclo[8.7.0.02,7.011,16]heptadeca-1(17),2(7),3,5,11(16),12,14-heptaen-4-yl)-2-(4-fluorophenyl)-1-benzofuran-3-carboxamide —— C31H22F2N4O5S
6-(Ethylsulfonylamino)-5-(15-fluoro-8-oxa-3,10-diazatetracyclo[8.7.0.02,7.011,16]heptadeca-1(17),2(7),3,5,11(16),12,14-heptaen-4-yl)-2-(4-fluorophenyl)-1-benzofuran-3-carboxamide
—— 6-[2-[5-[(4S,6S)-2-amino-6-methyl-4-(trifluoromethyl)-4,5-dihydro-1,3-oxazin-6-yl]-4-fluoro-2-methylphenyl]ethynyl]pyridine-3-carbonitrile —— C21H16F4N4O
6-[2-[5-[(4S,6S)-2-amino-6-methyl-4-(trifluoromethyl)-4,5-dihydro-1,3-oxazin-6-yl]-4-fluoro-2-methylphenyl]ethynyl]pyridine-3-carbonitrile
—— 6-((5-((4S,6S)-2-(bis(4-methoxyphenyl)(phenyl)methylamino)-4-methyl-6-(trifluoromethyl)-5,6-dihydro-4H-1,3-oxazin-4-yl)thiophen-3-yl)ethynyl)nicotinonitrile 1620828-97-8 C39H31F3N4O3S
6-((5-((4S,6S)-2-(bis(4-methoxyphenyl)(phenyl)methylamino)-4-methyl-6-(trifluoromethyl)-5,6-dihydro-4H-1,3-oxazin-4-yl)thiophen-3-yl)ethynyl)nicotinonitrile
—— 6-(ethylsulfonylamino)-2-(4-fluorophenyl)-N-methyl-5-(6-oxoindolo[1,2-c][1,3]benzoxazin-2-yl)-1-benzofuran-3-carboxamide —— C33H24FN3O6S
6-(ethylsulfonylamino)-2-(4-fluorophenyl)-N-methyl-5-(6-oxoindolo[1,2-c][1,3]benzoxazin-2-yl)-1-benzofuran-3-carboxamide
—— 6-(ethylsulfonylamino)-2-(4-fluorophenyl)-N-methyl-5-(6-phenyl-6,11-dihydrochromeno[4,3-b]indol-2-yl)-1-benzofuran-3-carboxamide —— C39H30FN3O5S
6-(ethylsulfonylamino)-2-(4-fluorophenyl)-N-methyl-5-(6-phenyl-6,11-dihydrochromeno[4,3-b]indol-2-yl)-1-benzofuran-3-carboxamide
—— (6-Methyl-2-methylsulfonyloxyhept-5-en-2-yl) methanesulfonate —— C10H20O6S2
(6-Methyl-2-methylsulfonyloxyhept-5-en-2-yl) methanesulfonate
—— 6-(ethylsulfonylamino)-2-(4-fluorophenyl)-N-methyl-5-(8-oxa-11,17-diazatetracyclo[8.7.0.02,7.011,16]heptadeca-1(10),2(7),3,5,12,14,16-heptaen-4-yl)-1-benzofuran-3-carboxamide —— C32H25FN4O5S
6-(ethylsulfonylamino)-2-(4-fluorophenyl)-N-methyl-5-(8-oxa-11,17-diazatetracyclo[8.7.0.02,7.011,16]heptadeca-1(10),2(7),3,5,12,14,16-heptaen-4-yl)-1-benzofuran-3-carboxamide
—— 6-methyl-4-oxo-1,2,3,4-tetrahydrocyclopenta[c]chromen-7-yl N-(tert-butoxycarbonyl)-L-alaninate —— C21H25NO6
6-methyl-4-oxo-1,2,3,4-tetrahydrocyclopenta[c]chromen-7-yl N-(tert-butoxycarbonyl)-L-alaninate
—— 6-(3,3-difluoropropylsulfonylamino)-2-(4-fluorophenyl)-N-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-benzofuran-3-carboxamide —— C25H28BF3N2O6S
6-(3,3-difluoropropylsulfonylamino)-2-(4-fluorophenyl)-N-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-benzofuran-3-carboxamide
—— 6-Cyclopropyl-5-isoquinolin-5-yl-2-[4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]-4-methylpyridine-3-carbonitrile —— C28H31N5O2
6-Cyclopropyl-5-isoquinolin-5-yl-2-[4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]-4-methylpyridine-3-carbonitrile
—— 6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-(3-hydroxybutanoyl)piperazin-1-yl]-5-(2-ethenylpyridin-4-yl)pyridine-3-carbonitrile —— C27H31N5O2
6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-(3-hydroxybutanoyl)piperazin-1-yl]-5-(2-ethenylpyridin-4-yl)pyridine-3-carbonitrile
—— 6-cyclopropyl-5-[(4-ethenylpyridin-2-yl)amino]-2-[(3R)-4-(3-hydroxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile —— C24H28N6O2
6-cyclopropyl-5-[(4-ethenylpyridin-2-yl)amino]-2-[(3R)-4-(3-hydroxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile
—— 6-cyclopropyl-2-[(3R)-4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]-5-(quinolin-4-ylamino)pyridine-3-carbonitrile —— C27H30N6O2
6-cyclopropyl-2-[(3R)-4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]-5-(quinolin-4-ylamino)pyridine-3-carbonitrile
—— 6-Cyclopropyl-5-(4-fluorophenyl)-2-[4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile —— C24H27FN4O2
6-Cyclopropyl-5-(4-fluorophenyl)-2-[4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile
—— 6-cyclopropyl-5-(2-ethenylpyridin-4-yl)-2-[(3R)-4-(2-methoxyacetyl)-3-propan-2-ylpiperazin-1-yl]pyridine-3-carbonitrile —— C26H31N5O2
6-cyclopropyl-5-(2-ethenylpyridin-4-yl)-2-[(3R)-4-(2-methoxyacetyl)-3-propan-2-ylpiperazin-1-yl]pyridine-3-carbonitrile
—— 6-cyclopropyl-5-[(2-ethenylpyridin-4-yl)amino]-2-[(3R)-4-(2-methoxyacetyl)-3-propan-2-ylpiperazin-1-yl]pyridine-3-carbonitrile —— C26H32N6O2
6-cyclopropyl-5-[(2-ethenylpyridin-4-yl)amino]-2-[(3R)-4-(2-methoxyacetyl)-3-propan-2-ylpiperazin-1-yl]pyridine-3-carbonitrile
—— 6-Cyclopropyl-5-isoquinolin-8-yl-2-[4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile —— C27H29N5O2
6-Cyclopropyl-5-isoquinolin-8-yl-2-[4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile
—— 6-Propan-2-yl-2-[3-propan-2-yl-4-(2-thiophen-2-ylacetyl)piperazin-1-yl]-5-[4-(trifluoromethyl)phenyl]pyridine-3-carbonitrile —— C29H31F3N4OS
6-Propan-2-yl-2-[3-propan-2-yl-4-(2-thiophen-2-ylacetyl)piperazin-1-yl]-5-[4-(trifluoromethyl)phenyl]pyridine-3-carbonitrile
—— 6-cyclopropyl-5-(6-methoxynaphthalen-2-yl)-2-[(3R)-4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]-4-methylpyridine-3-carbonitrile —— C30H34N4O3
6-cyclopropyl-5-(6-methoxynaphthalen-2-yl)-2-[(3R)-4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]-4-methylpyridine-3-carbonitrile
—— 6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-(3,3,3-trifluoropropanoyl)piperazin-1-yl]-5-(4-fluorophenyl)-4-methylpyridine-3-carbonitrile —— C26H26F4N4O
6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-(3,3,3-trifluoropropanoyl)piperazin-1-yl]-5-(4-fluorophenyl)-4-methylpyridine-3-carbonitrile
—— 6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-[2-(2-oxopyrrolidin-1-yl)acetyl]piperazin-1-yl]-5-(2-ethenylpyridin-4-yl)pyridine-3-carbonitrile —— C29H32N6O2
6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-[2-(2-oxopyrrolidin-1-yl)acetyl]piperazin-1-yl]-5-(2-ethenylpyridin-4-yl)pyridine-3-carbonitrile
—— 6-cyclopropyl-2-[(3R)-4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]-4-methyl-5-(4-methylsulfonylphenyl)pyridine-3-carbonitrile —— C26H32N4O4S
6-cyclopropyl-2-[(3R)-4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]-4-methyl-5-(4-methylsulfonylphenyl)pyridine-3-carbonitrile
—— 6-Cyclopropyl-2-[3-cyclopropyl-4-[2-(oxetan-2-yl)acetyl]piperazin-1-yl]-5-(6-ethenylpyridazin-4-yl)-4-methylpyridine-3-carbonitrile —— C28H32N6O2
6-Cyclopropyl-2-[3-cyclopropyl-4-[2-(oxetan-2-yl)acetyl]piperazin-1-yl]-5-(6-ethenylpyridazin-4-yl)-4-methylpyridine-3-carbonitrile
—— 6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-(4-oxobutanoyl)piperazin-1-yl]-5-isoquinolin-5-ylpyridine-3-carbonitrile —— C29H29N5O2
6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-(4-oxobutanoyl)piperazin-1-yl]-5-isoquinolin-5-ylpyridine-3-carbonitrile
—— 6-isopropyl-4-(2-methoxyphenyl)-2-(4-(2-phenylacetyl)piperazin-1-yl)nicotinonitrile 1416139-06-4 C28H30N4O2
6-isopropyl-4-(2-methoxyphenyl)-2-(4-(2-phenylacetyl)piperazin-1-yl)nicotinonitrile
—— 6-cyclopropyl-2-((R)-3-cyclopropyl-4-((1S,2S)-2-ethoxycyclopropanecarbonyl)piperazin-1-yl)-5-(4-fluorophenyl)nicotinonitrile 1416141-35-9 C28H31FN4O2
6-cyclopropyl-2-((R)-3-cyclopropyl-4-((1S,2S)-2-ethoxycyclopropanecarbonyl)piperazin-1-yl)-5-(4-fluorophenyl)nicotinonitrile
—— 6-cyclopropyl-5-[(6-ethenylpyrimidin-4-yl)amino]-2-[(3R)-4-(3-hydroxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile —— C23H27N7O2
6-cyclopropyl-5-[(6-ethenylpyrimidin-4-yl)amino]-2-[(3R)-4-(3-hydroxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile
—— 6-cyclopropyl-5-(2-ethenylquinolin-5-yl)-2-[(3R)-4-(3-hydroxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile —— C28H29N5O2
6-cyclopropyl-5-(2-ethenylquinolin-5-yl)-2-[(3R)-4-(3-hydroxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile
—— 6-cyclopropyl-5-(2-ethenylpyridin-4-yl)-2-[(3R)-4-[(E)-5-hydroxypent-2-enoyl]-3-propan-2-ylpiperazin-1-yl]-4-methylpyridine-3-carbonitrile —— C29H35N5O2
6-cyclopropyl-5-(2-ethenylpyridin-4-yl)-2-[(3R)-4-[(E)-5-hydroxypent-2-enoyl]-3-propan-2-ylpiperazin-1-yl]-4-methylpyridine-3-carbonitrile
—— 6-isopropyl-2-(3-methyl-4-(2-phenylacetyl)piperazin-1-yl)-4-phenylnicotinonitrile 1416138-91-4 C28H30N4O
6-isopropyl-2-(3-methyl-4-(2-phenylacetyl)piperazin-1-yl)-4-phenylnicotinonitrile
—— 6-cyclopropyl-5-[2-(3-hydroxyprop-1-en-2-yl)pyridin-4-yl]-2-[(3R)-4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile —— C26H31N5O3
6-cyclopropyl-5-[2-(3-hydroxyprop-1-en-2-yl)pyridin-4-yl]-2-[(3R)-4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile
—— 6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-[(E)-5-hydroxypent-2-enoyl]piperazin-1-yl]-5-(5-ethenylpyridazin-3-yl)-4-methylpyridine-3-carbonitrile —— C28H32N6O2
6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-[(E)-5-hydroxypent-2-enoyl]piperazin-1-yl]-5-(5-ethenylpyridazin-3-yl)-4-methylpyridine-3-carbonitrile
—— 6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-(3-methoxypropanoyl)piperazin-1-yl]-5-(2-ethenylpyridin-4-yl)-4-methylpyridine-3-carbonitrile —— C28H33N5O2
6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-(3-methoxypropanoyl)piperazin-1-yl]-5-(2-ethenylpyridin-4-yl)-4-methylpyridine-3-carbonitrile
—— 6-cyclopropyl-5-(1H-indol-5-yl)-2-[4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile —— C26H29N5O2
6-cyclopropyl-5-(1H-indol-5-yl)-2-[4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile
—— [(6S,7R)-7-(5-bromo-2-fluoropyridin-3-yl)-6-(2-hydroxyethyl)-7-methyl-5,5-dioxo-5lambda6-thia-8-azaspiro[3.5]non-8-en-9-yl]carbamic acid —— C16H19BrFN3O5S
[(6S,7R)-7-(5-bromo-2-fluoropyridin-3-yl)-6-(2-hydroxyethyl)-7-methyl-5,5-dioxo-5lambda6-thia-8-azaspiro[3.5]non-8-en-9-yl]carbamic acid
—— 6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-hexanoylpiperazin-1-yl]-5-[(4-ethenylpyridin-2-yl)amino]pyridine-3-carbonitrile —— C29H36N6O
6-cyclopropyl-2-[(3R)-3-cyclopropyl-4-hexanoylpiperazin-1-yl]-5-[(4-ethenylpyridin-2-yl)amino]pyridine-3-carbonitrile
—— 6-Cyclopropyl-2-[3-cyclopropyl-4-[2-(oxetan-2-yl)acetyl]piperazin-1-yl]-5-[(2-ethenylpyridin-4-yl)amino]pyridine-3-carbonitrile —— C28H32N6O2
6-Cyclopropyl-2-[3-cyclopropyl-4-[2-(oxetan-2-yl)acetyl]piperazin-1-yl]-5-[(2-ethenylpyridin-4-yl)amino]pyridine-3-carbonitrile
—— 6-cyclopropyl-5-[(2-ethenylpyridin-4-yl)amino]-2-[(3R)-4-(3-hydroxypropanoyl)-3-propan-2-ylpiperazin-1-yl]pyridine-3-carbonitrile —— C26H32N6O2
6-cyclopropyl-5-[(2-ethenylpyridin-4-yl)amino]-2-[(3R)-4-(3-hydroxypropanoyl)-3-propan-2-ylpiperazin-1-yl]pyridine-3-carbonitrile
—— 6-(2,5-difluorophenyl)-N-[[3-(methylsulfamoyl)phenyl]methyl]pyridine-3-carboxamide —— C20H17F2N3O3S
6-(2,5-difluorophenyl)-N-[[3-(methylsulfamoyl)phenyl]methyl]pyridine-3-carboxamide
—— 6-cyclopropyl-2-[4-[(1R,2R)-2-(hydroxymethyl)cyclopropanecarbonyl]-3-methylpiperazin-1-yl]-5-isoquinolin-5-ylpyridine-3-carbonitrile —— C28H29N5O2
6-cyclopropyl-2-[4-[(1R,2R)-2-(hydroxymethyl)cyclopropanecarbonyl]-3-methylpiperazin-1-yl]-5-isoquinolin-5-ylpyridine-3-carbonitrile
—— 6-Cyclopropyl-2-[3-cyclopropyl-4-(3-hydroxypropanoyl)piperazin-1-yl]-5-(2-ethenylquinolin-7-yl)pyridine-3-carbonitrile —— C30H31N5O2
6-Cyclopropyl-2-[3-cyclopropyl-4-(3-hydroxypropanoyl)piperazin-1-yl]-5-(2-ethenylquinolin-7-yl)pyridine-3-carbonitrile