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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-3-(4-methoxyphenyl)triazolo[4,5-d]pyrimidin-7-one —— C22H20N6O3
6-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-3-(4-methoxyphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-(sec-butylthio)-1-phenyl-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one —— C15H16N4OS
6-(sec-butylthio)-1-phenyl-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-(2-(4-benzylpiperidin-1-yl)-2-oxoethyl)-3-(4-methoxyphenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7(6H)-one —— C25H26N6O3
6-(2-(4-benzylpiperidin-1-yl)-2-oxoethyl)-3-(4-methoxyphenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7(6H)-one
—— 6-[4-(furan-2-carbonyl)piperazin-1-yl]-3-(2-methylphenyl)-1H-pyrimidine-2,4-dione —— C20H20N4O4
6-[4-(furan-2-carbonyl)piperazin-1-yl]-3-(2-methylphenyl)-1H-pyrimidine-2,4-dione
—— 6-(3-morpholin-4-yl-3-oxopropyl)-2H-1,2,4-triazine-3,5-dione —— C10H14N4O4
6-(3-morpholin-4-yl-3-oxopropyl)-2H-1,2,4-triazine-3,5-dione
—— 6-{[2-(2-Ethylpiperidin-1-YL)-2-oxoethyl]sulfanyl}-1-(4-methylphenyl)-1H,4H,5H-pyrazolo[3,4-D]pyrimidin-4-one —— C21H25N5O2S
6-{[2-(2-Ethylpiperidin-1-YL)-2-oxoethyl]sulfanyl}-1-(4-methylphenyl)-1H,4H,5H-pyrazolo[3,4-D]pyrimidin-4-one
—— 6-chloro-4-N-[(S)-(5-methyl-1H-1,2,4-triazol-3-yl)-phenylmethyl]pyrimidine-2,4-diamine —— C14H14ClN7
6-chloro-4-N-[(S)-(5-methyl-1H-1,2,4-triazol-3-yl)-phenylmethyl]pyrimidine-2,4-diamine
—— 6-(Isopropylthio)-1-(p-tolyl)-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one —— C15H16N4OS
6-(Isopropylthio)-1-(p-tolyl)-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-chloro-4-N-[(R)-(5-methyl-1H-1,2,4-triazol-3-yl)-phenylmethyl]pyrimidine-2,4-diamine —— C14H14ClN7
6-chloro-4-N-[(R)-(5-methyl-1H-1,2,4-triazol-3-yl)-phenylmethyl]pyrimidine-2,4-diamine
—— 6-(2,6-dimethylmorpholino)-3-(4-fluorobenzyl)pyrimidine-2,4(1H,3H)-dione —— C17H20FN3O3
6-(2,6-dimethylmorpholino)-3-(4-fluorobenzyl)pyrimidine-2,4(1H,3H)-dione
—— 6-[4-[(2R)-2-phenyl-2-pyrrolidin-1-ylacetyl]piperazin-1-yl]pyridine-3-carbonitrile —— C22H25N5O
6-[4-[(2R)-2-phenyl-2-pyrrolidin-1-ylacetyl]piperazin-1-yl]pyridine-3-carbonitrile
—— 6-tert-butyl-2-oxo-1-[[(3R)-piperidin-3-yl]methyl]pyridine-3-carbonitrile —— C16H23N3O
6-tert-butyl-2-oxo-1-[[(3R)-piperidin-3-yl]methyl]pyridine-3-carbonitrile
—— 6-((2-chlorobenzyl)thio)-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one —— C18H13ClN4OS
6-((2-chlorobenzyl)thio)-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one
—— (6E)-6-[3-(3,3,5-trimethyl-7-azabicyclo[3.2.1]octane-7-carbonyl)-2H-1,2-oxazol-5-ylidene]cyclohexa-2,4-dien-1-one —— C20H24N2O3
(6E)-6-[3-(3,3,5-trimethyl-7-azabicyclo[3.2.1]octane-7-carbonyl)-2H-1,2-oxazol-5-ylidene]cyclohexa-2,4-dien-1-one
—— 6-tert-butyl-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile —— C16H23N3O
6-tert-butyl-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile
—— 6-methyl-2-[2-[(2R)-piperidin-2-yl]ethylsulfanyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C14H19N3OS2
6-methyl-2-[2-[(2R)-piperidin-2-yl]ethylsulfanyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinolin-2-yl)-[5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]methanone —— C24H25F3N4O4
(6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinolin-2-yl)-[5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]methanone
—— 6-ethyl-3-[2-[(2R)-piperidin-2-yl]ethyl]thieno[2,3-d]pyrimidin-4-one —— C15H21N3OS
6-ethyl-3-[2-[(2R)-piperidin-2-yl]ethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-(3,4-Dimethylphenyl)-2-oxo-1-piperidin-4-ylpyridine-3-carbonitrile —— C19H21N3O
6-(3,4-Dimethylphenyl)-2-oxo-1-piperidin-4-ylpyridine-3-carbonitrile
—— 6-methyl-3-[2-[(2R)-piperidin-2-yl]ethyl]thieno[2,3-d]pyrimidin-4-one —— C14H19N3OS
6-methyl-3-[2-[(2R)-piperidin-2-yl]ethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-Bromo-1-(3-oxo-3-piperazin-1-ylpropyl)pyridin-2-one —— C12H16BrN3O2
6-Bromo-1-(3-oxo-3-piperazin-1-ylpropyl)pyridin-2-one
—— 6-tert-butyl-2-oxo-1-[2-[(2S)-piperidin-2-yl]ethyl]pyridine-3-carbonitrile —— C17H25N3O
6-tert-butyl-2-oxo-1-[2-[(2S)-piperidin-2-yl]ethyl]pyridine-3-carbonitrile
—— 6-ethyl-3-[2-[(2S)-piperidin-2-yl]ethyl]thieno[2,3-d]pyrimidin-4-one —— C15H21N3OS
6-ethyl-3-[2-[(2S)-piperidin-2-yl]ethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-tert-butyl-2-oxo-1-[2-[(2R)-piperidin-2-yl]ethyl]pyridine-3-carbonitrile —— C17H25N3O
6-tert-butyl-2-oxo-1-[2-[(2R)-piperidin-2-yl]ethyl]pyridine-3-carbonitrile
—— 6-(4-chlorophenyl)-1-[(2R)-2-cyanopropyl]-2-oxopyridine-3-carbonitrile —— C16H12ClN3O
6-(4-chlorophenyl)-1-[(2R)-2-cyanopropyl]-2-oxopyridine-3-carbonitrile
—— 6-methyl-3-[2-[(2S)-piperidin-2-yl]ethyl]thieno[2,3-d]pyrimidin-4-one —— C14H19N3OS
6-methyl-3-[2-[(2S)-piperidin-2-yl]ethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-[(Dimethylsulfamoylamino)methyl]-3-methylimidazo[2,1-b][1,3]thiazole —— C9H14N4O2S2
6-[(Dimethylsulfamoylamino)methyl]-3-methylimidazo[2,1-b][1,3]thiazole
—— 6-(4-fluorophenyl)-3-methyl-N-(pyridin-4-yl)imidazo[2,1-b]thiazole-2-carboxamide —— C18H13FN4OS
6-(4-fluorophenyl)-3-methyl-N-(pyridin-4-yl)imidazo[2,1-b]thiazole-2-carboxamide
—— 6-ethyl-2-(piperidin-4-ylmethylsulfanyl)-3H-thieno[2,3-d]pyrimidin-4-one —— C14H19N3OS2
6-ethyl-2-(piperidin-4-ylmethylsulfanyl)-3H-thieno[2,3-d]pyrimidin-4-one
—— 6-(3,4-dimethylphenyl)-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile —— C20H23N3O
6-(3,4-dimethylphenyl)-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile
—— 6-(4-methoxyphenyl)-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile —— C19H21N3O2
6-(4-methoxyphenyl)-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile
—— 6-bromo-1-[2-[(2S)-piperidin-2-yl]ethyl]pyridin-2-one —— C12H17BrN2O
6-bromo-1-[2-[(2S)-piperidin-2-yl]ethyl]pyridin-2-one
—— 6-(4-methylphenyl)-2-oxo-1-[[(3R)-piperidin-3-yl]methyl]pyridine-3-carbonitrile —— C19H21N3O
6-(4-methylphenyl)-2-oxo-1-[[(3R)-piperidin-3-yl]methyl]pyridine-3-carbonitrile
—— 6-(4-chlorophenyl)-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile —— C18H18ClN3O
6-(4-chlorophenyl)-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile
—— 6-bromo-1-[[(3R)-piperidin-3-yl]methyl]pyridin-2-one —— C11H15BrN2O
6-bromo-1-[[(3R)-piperidin-3-yl]methyl]pyridin-2-one
—— 6-methyl-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile —— C13H17N3O
6-methyl-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile
—— 6-ethyl-2-[[(3R)-piperidin-3-yl]methylsulfanyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C14H19N3OS2
6-ethyl-2-[[(3R)-piperidin-3-yl]methylsulfanyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 6-(3-methoxyphenyl)-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile —— C19H21N3O2
6-(3-methoxyphenyl)-2-oxo-1-[[(3S)-piperidin-3-yl]methyl]pyridine-3-carbonitrile
—— 6-(dimethylsulfamoyl)-1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxoquinoline-3-carboxamide —— C21H31N5O4S
6-(dimethylsulfamoyl)-1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxoquinoline-3-carboxamide
—— 6-methyl-3-[[(3S)-piperidin-3-yl]methyl]thieno[2,3-d]pyrimidin-4-one —— C13H17N3OS
6-methyl-3-[[(3S)-piperidin-3-yl]methyl]thieno[2,3-d]pyrimidin-4-one
—— 6-(4-methoxyphenyl)-2-oxo-1-[[(3R)-piperidin-3-yl]methyl]pyridine-3-carbonitrile —— C19H21N3O2
6-(4-methoxyphenyl)-2-oxo-1-[[(3R)-piperidin-3-yl]methyl]pyridine-3-carbonitrile
—— 6-bromo-1-[[(3S)-piperidin-3-yl]methyl]pyridin-2-one —— C11H15BrN2O
6-bromo-1-[[(3S)-piperidin-3-yl]methyl]pyridin-2-one
—— 6-ethyl-4-[2-[(2R)-piperidin-2-yl]ethylsulfanyl]thieno[2,3-d]pyrimidine —— C15H21N3S2
6-ethyl-4-[2-[(2R)-piperidin-2-yl]ethylsulfanyl]thieno[2,3-d]pyrimidine
—— 6-[(3,5-dimethylpiperidin-1-yl)sulfonyl]-3-(2-morpholin-4-yl-2-oxoethyl)-1,3-benzoxazol-2(3H)-one —— C20H27N3O6S
6-[(3,5-dimethylpiperidin-1-yl)sulfonyl]-3-(2-morpholin-4-yl-2-oxoethyl)-1,3-benzoxazol-2(3H)-one
—— 6-methyl-N-[(1S,2R)-2-phenylcyclopropyl]-2-pyridin-4-ylpyrimidin-4-amine —— C19H18N4
6-methyl-N-[(1S,2R)-2-phenylcyclopropyl]-2-pyridin-4-ylpyrimidin-4-amine
—— 6-[2-(4-Fluorophenyl)-2-oxoethyl]-2-methyl-[1,2,4]triazolo[1,5-c]quinazolin-5-one —— C18H13FN4O2
6-[2-(4-Fluorophenyl)-2-oxoethyl]-2-methyl-[1,2,4]triazolo[1,5-c]quinazolin-5-one
—— 6-[[4-(3-methoxyphenyl)-5-propylsulfanyl-1,2,4-triazol-3-yl]methyl]-1H-pyrimidine-2,4-dione —— C17H19N5O3S
6-[[4-(3-methoxyphenyl)-5-propylsulfanyl-1,2,4-triazol-3-yl]methyl]-1H-pyrimidine-2,4-dione
—— 6-(3-bromophenyl)-N-cyclopropyl-N-[(3R)-1,1-dioxothiolan-3-yl]-2-methylpyridine-3-carboxamide —— C20H21BrN2O3S
6-(3-bromophenyl)-N-cyclopropyl-N-[(3R)-1,1-dioxothiolan-3-yl]-2-methylpyridine-3-carboxamide
—— 6-{[2-(4-Phenylpiperazine-1-carbonyl)pyrrolidin-1-YL]sulfonyl}-1,2,3,4-tetrahydroquinolin-2-one —— C24H28N4O4S
6-{[2-(4-Phenylpiperazine-1-carbonyl)pyrrolidin-1-YL]sulfonyl}-1,2,3,4-tetrahydroquinolin-2-one
—— 6-[3-(1,2-Dihydroimidazo[1,2-a]benzimidazole-3-carbonyl)piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C23H23N5O5S
6-[3-(1,2-Dihydroimidazo[1,2-a]benzimidazole-3-carbonyl)piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one