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—— (6E)-2-methyl-6-[3-[methyl-(2,2,6,6-tetramethylpiperidin-4-yl)amino]-1H-pyridazin-6-ylidene]-4-morpholin-4-ylquinolin-7-one —— C28H38N6O2
(6E)-2-methyl-6-[3-[methyl-(2,2,6,6-tetramethylpiperidin-4-yl)amino]-1H-pyridazin-6-ylidene]-4-morpholin-4-ylquinolin-7-one
—— (6Z)-6-[3-[methyl-(2,2,6,6-tetramethylpiperidin-4-yl)amino]-1H-pyridazin-6-ylidene]-7-oxoquinoline-3-carbonitrile —— C24H28N6O
(6Z)-6-[3-[methyl-(2,2,6,6-tetramethylpiperidin-4-yl)amino]-1H-pyridazin-6-ylidene]-7-oxoquinoline-3-carbonitrile
—— 6,8-difluoro-2-[4-[4-(4-methoxy-3-methyl-benzoyl)-1-piperidyl]-4-oxo-butyl]-3H-quinazolin-4-one —— C26H27F2N3O4
6,8-difluoro-2-[4-[4-(4-methoxy-3-methyl-benzoyl)-1-piperidyl]-4-oxo-butyl]-3H-quinazolin-4-one
—— 6-fluoro-2-{4-[4-(6-methoxy-pyridine-3-carbonyl)-piperidin-1-yl]-4-oxo-butyl}-3H-quinazolin-4-one —— C24H25FN4O4
6-fluoro-2-{4-[4-(6-methoxy-pyridine-3-carbonyl)-piperidin-1-yl]-4-oxo-butyl}-3H-quinazolin-4-one
—— 6-fluoro-2-(4-{4-[4-(1-hydroxy-1-methyl-ethyl)-benzoyl]-piperidin-1-yl}-4-oxo-butyl)-3H-quinazolin-4-one —— C27H30FN3O4
6-fluoro-2-(4-{4-[4-(1-hydroxy-1-methyl-ethyl)-benzoyl]-piperidin-1-yl}-4-oxo-butyl)-3H-quinazolin-4-one
—— (6Z)-1-methyl-6-[3-[methyl-(2,2,6,6-tetramethylpiperidin-4-yl)amino]-1H-pyridazin-6-ylidene]isoquinolin-7-one —— C24H31N5O
(6Z)-1-methyl-6-[3-[methyl-(2,2,6,6-tetramethylpiperidin-4-yl)amino]-1H-pyridazin-6-ylidene]isoquinolin-7-one
—— (6Z)-3-ethyl-6-[3-[methyl-(2,2,6,6-tetramethylpiperidin-4-yl)amino]-1H-pyridazin-6-ylidene]quinolin-7-one —— C25H33N5O
(6Z)-3-ethyl-6-[3-[methyl-(2,2,6,6-tetramethylpiperidin-4-yl)amino]-1H-pyridazin-6-ylidene]quinolin-7-one
—— 6-fluoro-2-{4-[4-(4-methoxy-3-methyl-benzoyl)-piperidin-1-yl]-4-oxo-butyl}-3H-quinazolin-4-one —— C26H28FN3O4
6-fluoro-2-{4-[4-(4-methoxy-3-methyl-benzoyl)-piperidin-1-yl]-4-oxo-butyl}-3H-quinazolin-4-one
—— 6-fluoro-2-{4-[4-(3-fluoro-4-methoxy-benzoyl)-piperidin-1-yl]-4-oxo-butyl}-3H-quinazolin-4-one —— C25H25F2N3O4
6-fluoro-2-{4-[4-(3-fluoro-4-methoxy-benzoyl)-piperidin-1-yl]-4-oxo-butyl}-3H-quinazolin-4-one
—— (6Ar)-5-bromo-N-[(1S,4R)-2-hydroxy-7-(2-methylpropyl)-5,8-dioxo-4-propan-2-yl-3-oxa-6,9-diazatricyclo[7.3.0.02,6]dodecan-4-yl]-7-methyl-6,6a,8,9-tetrahydro-4H-indolo[4,3-fg]quinoline-9-carboxamide —— C32H40BrN5O5
(6Ar)-5-bromo-N-[(1S,4R)-2-hydroxy-7-(2-methylpropyl)-5,8-dioxo-4-propan-2-yl-3-oxa-6,9-diazatricyclo[7.3.0.02,6]dodecan-4-yl]-7-methyl-6,6a,8,9-tetrahydro-4H-indolo[4,3-fg]quinoline-9-carboxamide
—— [6-(diethylamino)-9-[4-[[6-[[(1S)-1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-3H-2-benzofuran-5-yl]methylamino]-6-oxohexyl]sulfamoyl]-2-sulfophenyl]xanthen-3-ylidene]-diethylazanium —— C53H65FN5O8S2+
[6-(diethylamino)-9-[4-[[6-[[(1S)-1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-3H-2-benzofuran-5-yl]methylamino]-6-oxohexyl]sulfamoyl]-2-sulfophenyl]xanthen-3-ylidene]-diethylazanium
—— (6R)-7-[(2-amino-2-cyclohexa-1,4-dien-1-ylacetyl)amino]-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C16H19N3O4S
(6R)-7-[(2-amino-2-cyclohexa-1,4-dien-1-ylacetyl)amino]-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-[[[(3R,4S)-3-fluoro-1-[2-(7-methoxy-2-oxo-1,5-naphthyridin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one —— C24H27FN6O4
6-[[[(3R,4S)-3-fluoro-1-[2-(7-methoxy-2-oxo-1,5-naphthyridin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one
—— 6-[(2R)-4-(4-benzylphthalazin-1-yl)-2-(hydroxymethyl)piperazin-1-yl]pyridine-3-carbonitrile —— C26H24N6O
6-[(2R)-4-(4-benzylphthalazin-1-yl)-2-(hydroxymethyl)piperazin-1-yl]pyridine-3-carbonitrile
—— 6-hydroxy-4-(3-((3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidine-1-carbonyl)pyridin-2(1H)-one —— C18H18N4O4S
6-hydroxy-4-(3-((3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidine-1-carbonyl)pyridin-2(1H)-one
—— 6-hydroxy-4-(3-((3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidine-1-carbonyl)pyridin-2(1H)-one —— C18H18N6O4
6-hydroxy-4-(3-((3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidine-1-carbonyl)pyridin-2(1H)-one
—— 6-amino-8-{4-[(2,4-dichlorobenzyl)oxy]phenyl}-8H-[1,3]dioxolo[4,5-g]chromene-7-carbonitrile —— C24H16Cl2N2O4
6-amino-8-{4-[(2,4-dichlorobenzyl)oxy]phenyl}-8H-[1,3]dioxolo[4,5-g]chromene-7-carbonitrile
—— (6E)-2-bromo-4-chloro-3,5-dimethyl-6-(phenylhydrazinylidene)cyclohexa-2,4-dien-1-one —— C14H12BrClN2O
(6E)-2-bromo-4-chloro-3,5-dimethyl-6-(phenylhydrazinylidene)cyclohexa-2,4-dien-1-one
—— (6E)-4-tert-butyl-2-[(E)-(2H-tetrazol-5-ylhydrazinylidene)methyl]-6-[[2-(2H-tetrazol-5-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C14H18N12O
(6E)-4-tert-butyl-2-[(E)-(2H-tetrazol-5-ylhydrazinylidene)methyl]-6-[[2-(2H-tetrazol-5-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-2,4-ditert-butyl-6-[[2-(4,5-dihydro-1H-imidazol-2-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C18H28N4O
(6Z)-2,4-ditert-butyl-6-[[2-(4,5-dihydro-1H-imidazol-2-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-(4-Benzylpiperidin-1-yl)-2-chloro-3-nitropyridine —— C17H18ClN3O2
6-(4-Benzylpiperidin-1-yl)-2-chloro-3-nitropyridine
—— (6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-2-yl)(3-((3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone —— C19H21N7O3
(6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-2-yl)(3-((3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone
—— (6-Methoxypyridin-3-yl)(3-((3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone —— C19H20N6O3
(6-Methoxypyridin-3-yl)(3-((3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone
—— (6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-2-yl)(3-((3-(o-tolyl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone —— C22H25N5O3
(6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-2-yl)(3-((3-(o-tolyl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone
—— (6-Ethoxypyridin-3-yl)(3-((3-(o-tolyl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone —— C23H26N4O3
(6-Ethoxypyridin-3-yl)(3-((3-(o-tolyl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone
—— (6-methoxy-1H-indol-2-yl)(3-((3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone —— C22H22N6O3
(6-methoxy-1H-indol-2-yl)(3-((3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl)methyl)piperidin-1-yl)methanone
—— 6-((1-((5-ethylthiophen-2-yl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C16H22N4O3S2
6-((1-((5-ethylthiophen-2-yl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((2,4-dimethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C18H24N4O5S
6-((1-((2,4-dimethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((4-fluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C16H19FN4O3S
6-((1-((4-fluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((4-ethoxy-3-fluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C18H23FN4O4S
6-((1-((4-ethoxy-3-fluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((4-(tert-butyl)phenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C20H28N4O3S
6-((1-((4-(tert-butyl)phenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((4-methoxy-3-methylphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C18H24N4O4S
6-((1-((4-methoxy-3-methylphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((3,5-difluorobenzyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C17H20F2N4O3S
6-((1-((3,5-difluorobenzyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((4-fluoro-2-methylphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C17H21FN4O3S
6-((1-((4-fluoro-2-methylphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((4-ethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C18H24N4O4S
6-((1-((4-ethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((2,5-difluorobenzyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C17H20F2N4O3S
6-((1-((2,5-difluorobenzyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((2-fluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C16H19FN4O3S
6-((1-((2-fluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((3-chloro-2-methylphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C17H21ClN4O3S
6-((1-((3-chloro-2-methylphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— 6-((1-((3-fluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine —— C16H19FN4O3S
6-((1-((3-fluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyridazin-3-amine
—— (6-Ethoxypyridin-3-yl)(3-(pyridazin-3-yloxy)pyrrolidin-1-yl)methanone —— C16H18N4O3
(6-Ethoxypyridin-3-yl)(3-(pyridazin-3-yloxy)pyrrolidin-1-yl)methanone
—— (6E)-6-[(morpholin-4-ylamino)methylidene]cyclohexa-2,4-dien-1-one —— C11H14N2O2
(6E)-6-[(morpholin-4-ylamino)methylidene]cyclohexa-2,4-dien-1-one
—— 6-((1-((3,4-difluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine —— C16H18F2N4O3S
6-((1-((3,4-difluorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine
—— 6-((1-((2,3-dihydrobenzofuran-5-yl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine —— C18H22N4O4S
6-((1-((2,3-dihydrobenzofuran-5-yl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine
—— 6-((1-((4-ethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine —— C18H24N4O4S
6-((1-((4-ethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine
—— 6-((1-((2,5-dimethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine —— C18H24N4O5S
6-((1-((2,5-dimethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine
—— 6-((1-((5-chlorothiophen-2-yl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine —— C14H17ClN4O3S2
6-((1-((5-chlorothiophen-2-yl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine
—— 6-((1-((2,4-dimethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine —— C18H24N4O5S
6-((1-((2,4-dimethoxyphenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine
—— 6-((1-((3-chlorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine —— C16H19ClN4O3S
6-((1-((3-chlorophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine
—— 6-((1-((1,2-dimethyl-1H-imidazol-4-yl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine —— C15H22N6O3S
6-((1-((1,2-dimethyl-1H-imidazol-4-yl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine
—— 6-((1-((4-bromophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine —— C16H19BrN4O3S
6-((1-((4-bromophenyl)sulfonyl)pyrrolidin-3-yl)oxy)-N,N-dimethylpyrazin-2-amine