中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
1-methyl-5-[1-methyl-4-(4-methylpiperazin-1-yl)sulfonylpyrrol-2-yl]-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-7-one |
260780-81-2 |
C19H27N7O3S |
|
—— |
[(3R)-3-(5-bromo-2-hydroxyphenyl)-5-(5-bromothiophen-2-yl)-3,4-dihydropyrazol-2-yl]-[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone |
—— |
C25H13Br2ClF3N5O2S2 |
|
—— |
[(3S)-3-(5-bromo-2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone |
—— |
C27H16BrClF3N5O2S |
|
—— |
[(3S)-3-(5-bromo-2-hydroxyphenyl)-5-(5-bromothiophen-2-yl)-3,4-dihydropyrazol-2-yl]-[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone |
—— |
C25H13Br2ClF3N5O2S2 |
|
—— |
3-bromo-N-[(6S)-6-tert-butyl-3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide |
—— |
C25H23BrF3N5O2S2 |
|
—— |
[(3R)-3-(5-bromo-2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone |
—— |
C27H16BrClF3N5O2S |
|
—— |
propan-2-yl (6S)-2-[[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-6-phenyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate |
—— |
C30H24ClF3N4O3S2 |
|
—— |
ethyl (6S)-2-[[3-bromo-5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate |
—— |
C27H26BrF3N4O3S2 |
|
—— |
(5S,7S)-N-[(Z)-[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylideneamino]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide |
—— |
C32H32F3N5O4 |
|
—— |
propan-2-yl (6R)-2-[[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-6-phenyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate |
—— |
C30H24ClF3N4O3S2 |
|
—— |
ethyl (6R)-2-[[3-bromo-5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate |
—— |
C27H26BrF3N4O3S2 |
|
—— |
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-5-(4-fluorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone |
—— |
C27H16ClF4N5O2S |
|
—— |
(5S,7R)-N-[(Z)-[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylideneamino]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide |
—— |
C32H32F3N5O4 |
|
—— |
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]methanone |
—— |
C28H19ClF3N5O2S |
|
—— |
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]methanone |
—— |
C28H19ClF3N5O2S |
|
—— |
[(3R)-5-(2-chlorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]-[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone |
—— |
C27H16Cl2F3N5O2S |
|
—— |
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]methanone |
—— |
C28H19ClF3N5O3S |
|
—— |
(5R,7S)-N-[(Z)-[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylideneamino]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide |
—— |
C32H32F3N5O4 |
|
—— |
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-5-(4-fluorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone |
—— |
C27H16ClF4N5O2S |
|
—— |
[(3S)-5-(2-chlorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]-[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone |
—— |
C27H16Cl2F3N5O2S |
|
—— |
3-(4-tert-butyl-benzenesulphonyl)-5-methyl-2-methylsulphanyl-pyrazolo[1,5-a]pyrimidin-7-ylamine |
—— |
C18H22N4O2S2 |
|
—— |
13-(difluoromethyl)-4-[(5S,7S)-7-(difluoromethyl)-5-phenyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-3-ylidene]-11-methyl-16-thia-3,5,6,8,14-pentazatetracyclo[7.7.0.02,6.010,15]hexadeca-1(9),2,7,10(15),11,13-hexaene |
—— |
C25H18F4N8S |
|
—— |
1-cyclopentyl-3-ethyl-6-(2-propoxyphenyl)-pyrazolo[3,4-d]pyrimidin-4-one |
—— |
C21H26N4O2 |
|
—— |
4-butyl-2-(3-chloro-propane-1-sulfonyl)-6-methyl-2,4-dihydro-pyrazolo[4,3-d]-pyrimidine-5,7-dione |
—— |
C13H19ClN4O4S |
|
—— |
13-(difluoromethyl)-4-[(5R,7R)-7-(difluoromethyl)-5-phenyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-3-ylidene]-11-methyl-16-thia-3,5,6,8,14-pentazatetracyclo[7.7.0.02,6.010,15]hexadeca-1(9),2,7,10(15),11,13-hexaene |
—— |
C25H18F4N8S |
|
—— |
13-(difluoromethyl)-4-[(5R,7S)-7-(difluoromethyl)-5-phenyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-3-ylidene]-11-methyl-16-thia-3,5,6,8,14-pentazatetracyclo[7.7.0.02,6.010,15]hexadeca-1(9),2,7,10(15),11,13-hexaene |
—— |
C25H18F4N8S |
|
—— |
13-(difluoromethyl)-4-[(5S,7R)-7-(difluoromethyl)-5-phenyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-3-ylidene]-11-methyl-16-thia-3,5,6,8,14-pentazatetracyclo[7.7.0.02,6.010,15]hexadeca-1(9),2,7,10(15),11,13-hexaene |
—— |
C25H18F4N8S |
|
—— |
5-Benzyl-4,8-dimethyl-11-propan-2-yl-1,3,4,8,10-pentazatricyclo[7.3.0.02,6]dodeca-2,5,9-trien-7-one |
—— |
C19H23N5O |
|
—— |
4-chloro-1-N-(3-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidin-7-yl)benzene-1,3-diamine |
—— |
C14H15ClN6 |
|
—— |
2-(2,6-dichlorobenzyl)pyrazolo[3,4-d]pyrimidin-4(5H)-one |
—— |
C12H8Cl2N4O |
|
—— |
5-(2-chloro-6-fluorobenzyl)-2-butyl-2,5-dihydropyrazolo[3,4-d]pyrimidin-4-one |
402570-88-1 |
C16H16ClFN4O |
|
—— |
2-[1-(2-chlorophenyl)cyclobutyl]-5-(hydroxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C17H16ClN3O2 |
|
—— |
6-[[[(1S)-1-(2-fluorophenyl)ethyl]-methylamino]methyl]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one |
—— |
C16H18FN5O |
|
—— |
5-(2-chlorobenzyl)-6-methyl-2,5-dihydropyrazolo[3,4-d]-pyrimidin-4-one |
402571-03-3 |
C13H11ClN4O |
|
—— |
5-(2,6-difluorobenzyl)-2,5-dihydropyrazolo[3,4-d]-pyrimidin-4-one |
402570-44-9 |
C12H8F2N4O |
|
—— |
N-[(2R)-2-hydroxy-2-thiophen-2-ylethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide |
—— |
C15H16N4O2S |
|
—— |
N-[(2S)-2-hydroxy-2-thiophen-2-ylethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide |
—— |
C15H16N4O2S |
|
—— |
N-[2-[[(3R,5S)-3,5-dimethyl-1-adamantyl]oxy]ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide |
—— |
C21H28N4O2 |
|
—— |
N-[(2S)-2-(hydroxymethyl)-3-thiophen-2-ylpropyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide |
—— |
C16H18N4O2S |
|
—— |
N-[(2R)-2-(hydroxymethyl)-3-thiophen-3-ylpropyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide |
—— |
C16H18N4O2S |
|
—— |
N-[(2S)-2-(hydroxymethyl)-3-thiophen-3-ylpropyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide |
—— |
C16H18N4O2S |
|
—— |
N-[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide |
—— |
C18H21N5O2 |
|
—— |
N-[(2R)-2-(hydroxymethyl)-3-thiophen-2-ylpropyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide |
—— |
C16H18N4O2S |
|
—— |
N-methyl-N-[(3-methylsulfonylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-2-[(2S)-oxan-2-yl]ethanamine |
—— |
C16H24N4O3S |
|
—— |
N-methyl-N-[(3-methylsulfonylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-2-[(2R)-oxan-2-yl]ethanamine |
—— |
C16H24N4O3S |
|
—— |
(7-methylpyrazolo[1,5-a]pyrimidin-6-yl)-[(3S)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone |
—— |
C19H24N6O |
|
—— |
(7-methylpyrazolo[1,5-a]pyrimidin-6-yl)-[(3R)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone |
—— |
C19H24N6O |
|
—— |
[(6S)-6-hydroxy-4-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)-1,4-diazepan-1-yl]-(1H-pyrazol-5-yl)methanone |
—— |
C16H19N7O2 |
|
—— |
[(6R)-6-hydroxy-4-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)-1,4-diazepan-1-yl]-(1H-pyrazol-5-yl)methanone |
—— |
C16H19N7O2 |
|
—— |
(2,7-dimethylpyrazolo[1,5-a]pyrimidin-5-yl)-[(2S)-2-(2-thiophen-2-ylethyl)piperidin-1-yl]methanone |
—— |
C20H24N4OS |
|